Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559) |
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08/04/1998 | US5789587 Heterocyclic-fused lactams promote release of growth hormone |
08/04/1998 | US5789434 Derivatives of substituted 4-biarylbutyric acid as matrix metalloprotease inhibitors |
08/04/1998 | US5789415 Azacyclic-heterocyclic compounds as angiotension II receptor antagonists |
08/04/1998 | US5789402 Compounds having effects on serotonin-related systems |
08/04/1998 | CA2119647C Heteroaryl amines as novel acetylcholinesterase inhibitors |
07/30/1998 | WO1998032802A1 Soluble chromophores having improved solubilising groups |
07/30/1998 | WO1998032754A1 Imino-aza-anthracyclinone derivatives for the treatment of amyloidosis |
07/30/1998 | WO1998032742A1 Novel amide derivatives and medicinal compositions thereof |
07/30/1998 | CA2275965A1 Soluble chromophores having improved solubilising groups |
07/29/1998 | EP0854869A1 Spiro compounds as inhibitors of fibrinogen-dependent platelet aggregation |
07/29/1998 | EP0740668B1 Tetracyclic derivatives, process of preparation and use |
07/29/1998 | EP0717732B1 Polyamidic acid derivatives with antigastrin activity, a method for their preparation, and their pharmaceutical use |
07/29/1998 | EP0693068B1 Phenylpyrrole derivatives and their use as antipsychotic agents |
07/29/1998 | EP0665846B1 Topoisomerase ii inhibitors and therapeutic uses therefor |
07/29/1998 | EP0663913B1 New substituted pyrazole derivatives, processes for their preparation and their use as herbicides |
07/29/1998 | CN1189165A Imidazo £1, 5 alpha| pyridine derived serine protease inhibitors |
07/29/1998 | CN1188766A New ellipticine achroalkali compounds, process for their preparation and pharmaceutical compositions containing them |
07/29/1998 | CN1039324C Substituted nitrogen heterocyclic pyrimidines compound preparation method of medicinal salt or N-oxide |
07/29/1998 | CN1039323C Preparation method of imidazopyriding derivatives |
07/28/1998 | US5786481 N-alkyl and N-acyl derivatives of 3,7-Diazabicyclo- 3.3.1!nonanes and selected salts thereof as multi-class antiarrhythmic agents |
07/28/1998 | US5786480 4-substituted pyrazoloquinoline derivatives |
07/28/1998 | US5786361 Antiatherosclerosic agents |
07/28/1998 | US5786358 Inhibitors of glycinamide ribonucleotide formyl transferase |
07/28/1998 | US5786353 Tricyclic benzazepine vasopressin antagonists |
07/28/1998 | US5786352 Cyclic compounds, their production and use |
07/28/1998 | CA2141563C Novel 2-substituted indane-2-mercaptoacetylamide tricyclic derivatives useful as inhibitors of enkephalinase |
07/28/1998 | CA2127561C 3-azabicyclohexane compound intermediates for producing antibacterial compounds |
07/23/1998 | WO1998031364A1 3,3-disubstituted piperidines as modulators of chemokine receptor activity |
07/23/1998 | WO1998031363A1 Anti-viral compounds |
07/23/1998 | WO1998031359A1 Integrin antagonists |
07/23/1998 | CA2278309A1 3,3-disubstituted piperidines as modulators of chemokine receptor activity |
07/22/1998 | EP0854145A2 Vitronectin receptor antagonists, their production and their use |
07/22/1998 | EP0854140A2 Vitronectin receptor antagonists, their production and their use |
07/22/1998 | EP0853622A1 PROCESS FOR PREPARING 1-ARYL-4-OXOPYRROLO 3,2-c]QUINOLINE DERIVATIVES |
07/22/1998 | EP0853477A1 At1-receptor antagonists for preventing and treating postischemic renal failure and for protecting ischemic kidneys |
07/22/1998 | EP0725775B1 Certain fused pyrrolecarboxanilides; a new class of gaba brain receptor ligands |
07/21/1998 | US5783723 Reacting an alkali metal alcoholate with an excess of dialkyl succinate under anhydrous conditions followed by isolation of the di(alkali metal) salt of the dialkyl succinylsuccinate; cyclization; neutralization |
07/21/1998 | US5783708 Hexahydroisoindole derivatives |
07/21/1998 | US5783594 Administering to treat glioma, colon cancer and immunological disordaers |
07/21/1998 | US5783585 Solid bulk compositions containing quinolone carboxylic acids or naphthyridine carboxylic acids in free base form |
07/21/1998 | US5783582 Piperidines and hexahydro-1H-azepines spiro substituted at the 4-position promote release of growth hormone |
07/21/1998 | US5783579 Spiro-substituted azacyclic-substituted piperazino derivatives as neurokinin antagonists |
07/16/1998 | WO1998030564A1 Sulfonamide derivatives |
07/16/1998 | WO1998030562A1 Novel amide derivatives and intermediates for the synthesis thereof |
07/16/1998 | WO1998030560A1 Quinoline and quinazoline compounds useful in therapy, particularly in the treatment of begnin prostatic hyperplasia |
07/16/1998 | WO1998030558A2 Tricyclic compounds useful for inhibition of farnesyl protein transferase |
07/15/1998 | EP0853085A1 Piperidine derivatives having anxiolytic effect |
07/15/1998 | CN1039119C Condensed heterocyclic ketone derivatives, their production and use |
07/14/1998 | US5780645 Procedure for alkylation of imides |
07/14/1998 | US5780634 Decarboxylation |
07/14/1998 | US5780633 Enzyme inhibitor of testosterone 5-alpha-reductase |
07/14/1998 | US5780503 Compounds and methods for the treatment of cardiovascular, inflammatory and immune disorders |
07/14/1998 | US5780493 Treating brain disorders |
07/14/1998 | US5780482 Condensed 4-aminopyridines with antirheumatic activity |
07/14/1998 | US5780480 Thrombolytic agents, anticoagulants |
07/14/1998 | US5780454 Boronic ester and acid compounds |
07/09/1998 | WO1998029119A1 Inhibitors of farnesyl-protein transferase |
07/09/1998 | CA2276150A1 Inhibitors of farnesyl-protein transferase |
07/08/1998 | EP0851860A1 4-thiocarbamoyl-1-(3-pyrazolyl)-pyrazoles and their use as herbicides |
07/08/1998 | EP0851756A1 5-ht 3? receptor antagonists for dyskinesia |
07/08/1998 | CN1187129A Protein tyrosine kinase aryl and heteroaryl quinazoline compounds having selective inhibition of HER-2 autophosphorylation properties |
07/08/1998 | CN1039010C Oxdiazolyl substituted naphthyridine derivatives, its intermediate, its preparation and its medicinal composition and its use in medicine |
07/08/1998 | CN1039008C Dual action inhibitors in angiotensin invertase and neutral endopeptidase |
07/07/1998 | USRE35840 Imidazo 1,5-a!quinolines for treatment of anxiety and sleep disorders |
07/07/1998 | US5777114 Spiro heterocycle-imidazo 1,2-a!indeno 1,2-e!pyrazine!-4'-ones, preparation thereof and drugs containing same |
07/07/1998 | US5776964 Hypotensive agents; anticholesterol agents; cardiovascular disorders |
07/07/1998 | US5776963 3-(heteroaryl)-1- (2,3-dihydro-1h-isoindol-2-yl)alkyl!pyrrolidines and 3-(heteroaryl)-1- (2,3-dihydro-1h-indol-1-yl)alkyl!pyrrolidines and related compounds and their therapeutic untility |
07/07/1998 | US5776949 2-(1H) quinolinone compounds |
07/07/1998 | US5776944 7-(4-aminomethyl-3-methyloxyiminopyrroplidin-1-yl)-1-cyclopropyl-6-flu oro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid and the process for the preparation thereof |
07/07/1998 | US5776942 Bronchodilating pyrido 2,3-d!pyrimidine derivatives |
07/07/1998 | US5776935 Antagonists of strychnine-insensitive glycine site of n-methylaspartic acid receptor |
07/07/1998 | US5776930 Pharmaceutical preparation |
07/02/1998 | WO1998028305A1 Novel counterparts of camptothecin, their application as medicine and pharmaceutical compositions containing them |
07/02/1998 | WO1998028304A1 Pro-drugs and counterparts of camptothecin, their application as medicines |
07/02/1998 | WO1998028297A1 Spiro-substituted azacyclic-substituted piperazino derivatives as neurokinin antagonists |
07/02/1998 | WO1998028296A1 Pyrazol-based organic electroluminescent compounds and their use in electroluminescent devices |
07/02/1998 | WO1998028281A1 Fused polycyclic 2-aminopyrimidine derivatives, their preparation and their use as protein tyrosine kinase inhibitors |
07/02/1998 | WO1998027979A1 Heterocyclic inhibitors of microsomal triglyceride transfer protein and method |
07/02/1998 | WO1998014445A3 Novel 6 or 7 substituted analogues of swainsonine, processes for their preparation and their use as therapeutic agents |
07/02/1998 | CA2275163A1 Spiro-substituted azacyclic-substituted piperazino derivatives as neurokinin antagonists |
07/01/1998 | EP0850940A1 Ellipticine derivatives, their preparation and pharmaceutical compositions containing them |
07/01/1998 | EP0850939A1 Ellipticine derivatives, their preparation and pharmaceutical compositions containing them |
07/01/1998 | EP0850236A1 Piperazino derivatives as neurokinin antagonists |
07/01/1998 | EP0850060A1 Zwitterionic forms of trovafloxacin |
07/01/1998 | EP0751945B1 PROCESS FOR PREPARING (1H-TETRAZOL-5-yl)TETRAZOLO 1,5-a] QUINOLINES AND NAPHTHYRIDINES |
07/01/1998 | CN1186492A Imidazo £1, 2-alpha| pyridine derivatives |
06/30/1998 | US5773618 Tricyclic compounds having fungicidal activity, their preparation and their use |
06/30/1998 | US5773530 Pyrazolopyridine adenosine antagonists |
06/30/1998 | US5773456 Emphysema, rheumatoid arthritis and pancreatitis |
06/30/1998 | US5773450 Fluoroalkoxybenzylamino derivatives of nitrogen containing heterocycles |
06/30/1998 | US5773449 Thioquinolone compounds which have useful pharmaceutical activity |
06/30/1998 | US5773436 Use of serotonin antagonists for treating fibromyalgia |
06/30/1998 | CA2227506A1 New ellipticine derivatives, their preparation process and the pharmaceutical compositions containing them |
06/25/1998 | WO1998027098A1 SUBSTITUTED NITROGEN CONTAINING HETEROCYCLES AS INHIBITORS OF p38 PROTEIN KINASE |
06/25/1998 | WO1998027087A1 Combinatorial process for preparing fused pyrimidine libraries |
06/25/1998 | WO1998027065A1 Modulators of proteins with phosphotyrosine recognition units |
06/25/1998 | CA2275610A1 Modulators of proteins with phosphotyrosine recognition units |
06/25/1998 | CA2274022A1 Combinatorial process for preparing fused pyrimidine libraries |
06/24/1998 | CN1185782A 2-azabicyclo £2,2,1| heptane derivatives, preparation and application thereof |
06/24/1998 | CN1185781A Fused polycyclic heterocycle derivatives |