Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
04/1998
04/23/1998WO1998016527A1 Benzoxepine derivatives which promote release of growth hormone
04/23/1998WO1998016526A1 Tetrahydro-6h-pyrazino[1,2-b]isoquinoline 1,4-diones as apoprotein b-100 inhibitors
04/23/1998WO1998016514A1 Ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
04/23/1998WO1998016228A1 USE OF AN H+, K+-ATPase INHIBITOR IN THE TREATMENT OF NASAL POLYPS
04/23/1998DE19643037A1 Neue Oxadiazole, Verfahren zu ihrer Herstellung sowie deren Verwendung als Arzneimittel New oxadiazoles, processes for their preparation and their use as medicaments
04/23/1998CA2218804A1 Process for the separation of a mixture of enantiomers
04/22/1998EP0836605A1 Pyrrolopyrimidines and processes for the preparation thereof
04/22/1998EP0836602A1 Fungicidal pyrimidinones
04/22/1998CN1038131C Pyrrolopyrimidines and its preparing intermediate and medicinal composition containing same and use
04/21/1998US5741909 Pharmaceutical compositions which act as antiviral agents, induce biosynthesis of interferon and inhibit tumor formation in animals
04/21/1998US5741908 Reacting a 6h-imidazolo(4,5-c)tetrazolo(1,5-a)quinoline with triphenylphosphine; hydrolysis
04/21/1998US5741907 Pharmacologically active enantiomers
04/21/1998US5741796 Pyridyl and naphthyridyl compounds for inhibiting osteoclast-mediated bone resorption
04/21/1998US5741794 Platelet activating factor
04/21/1998US5741789 Hetero-oxy alkanamines
04/21/1998US5741657 Measuring gene expression
04/16/1998WO1998015556A1 TRICYCLIC COMPOUNDS HAVING ACTIVITY AS Ras-FPT INHIBITORS
04/16/1998WO1998015554A1 Acridone derivatives and method of preparation of 8-hydroxy imidazoacridinone derivatives
04/16/1998WO1998015553A1 5-HETEROATOM-CONTAINING ALKYL SUBSTITUTED-3-OXO-PYRIDO(1,2-a) BENZIMIDAZOLE-4-CARBOXAMIDE DERIVATIVES USEFUL IN TREATING CENTRAL NERVOUS SYSTEM DISORDERS
04/16/1998WO1998015552A1 1H-PYRIDO[3,4-b]INDOLE-4-CARBOXAMIDE DERIVATIVES, PREPARATION AND APPLICATION THEREOF IN THERAPEUTICS
04/16/1998WO1998015533A1 Method for producing 1,8-diaminonaphthalines and their 2,3-dihydroperimidine derivatives
04/16/1998WO1998015525A1 Hydroxamic acids
04/16/1998DE19641689A1 Verfahren zur Herstellung von 1,8-Diaminonaphthalinen und ihrer Derivate der 2,3-Dihydroperimidine Process for the preparation of 1,8-diaminonaphthalenes and their derivatives of the 2,3-Dihydroperimidine
04/16/1998CA2267943A1 5-heteroatom-containing alkyl substituted-3-oxo-pyrido(1,2-a) benzimidazole-4-carboxamide derivatives useful in treating central nervous system disorders
04/16/1998CA2266376A1 1h-pyrido¬3,4-b|indole-4-carboxamide derivatives, preparation and application thereof in therapeutics
04/15/1998EP0835258A1 Novel camptothecin analogues, preparation methods therefor, use thereof as drugs, and pharmaceutical compositions containing said analogues
04/15/1998EP0835257A1 Novel intermediates and process for the manufacture of camptothecin derivatives (cpt-11) and related compounds
04/15/1998EP0835244A1 Diheterocyclic acrylonitriles as smooth muscle cell proliferation inhibitors
04/15/1998CN1179158A 4 -amino -3 -acylnaphthyridine derivatives
04/15/1998CN1179155A Heterocyclic compounds
04/14/1998US5739345 Intermediate compounds in the preparation of heterocyclic compounds having anti-diabetic activity
04/14/1998US5739340 Indolizine derivatives with pharmaceutical activity
04/14/1998US5739339 Bactericides, antiprotozoa agents
04/14/1998US5739336 1,3,8-triaza- and 3,8-diaza-1-oxaspiro 4,5! decane derivatives
04/14/1998US5739334 Alkyl derivatives of trazodone with CNS activity
04/14/1998US5739326 Heterobicyclic herbicides
04/14/1998US5739281 Subjecting proteins to a time sequence of multiple denaturing-renaturing cycles
04/14/1998US5739147 Cyclohexane derivatives, process for their preparation, and the use of the compounds for the treatment of diseases
04/14/1998US5739134 N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2h-benzopyran, dihydrobenzodioxin, benzodioxole, dihydrobenzodioxepin, or tetrahydrobenzoxepin)carboxamide derivatives
04/14/1998US5739133 Pyridazinedione compounds useful in treating neurological disorders
04/14/1998US5739128 Administering for treatment of diseases characterized by excess renal reabsorption of water
04/14/1998US5739127 2,4'-bridged bis-2,4-diaminoquinazolines
04/14/1998CA2138298C Pyridopyrimidinone antianginal agents
04/09/1998WO1998014448A1 Pyrazolopyridylpyridazinone derivatives and process for the preparation thereof
04/09/1998WO1998014447A1 Novel indole-2,3-dione-3-oxime derivatives
04/09/1998WO1998014446A1 Novel 3, 5, and/or 6 substituted analogues of swainsonine, processes for their preparation and their use as therapeutic agents
04/09/1998WO1998014445A2 Novel 6 or 7 substituted analogues of swainsonine, processes for their preparation and their use as therapeutic agents
04/09/1998WO1998014433A1 Aralkyl and aralkylidene heterocyclic lactams and imides
04/09/1998CA2268114A1 Novel 6 or 7 substituted analogues of swainsonine, processes for their preparation and their use as therapeutic agents
04/09/1998CA2267412A1 Novel 3, 5, and/or 6 substituted analogues of swainsonine, processes for their preparation and their use as therapeutic agents
04/08/1998EP0834315A1 Use of an imidazole derivative for the manufacture of a medicament for preventing and/or treating rhinitis
04/08/1998EP0833837A1 Process for preparing derivatives of azabicyclo naphthyridine carboxylic acid comprising a dipeptide
04/08/1998EP0833818A1 Cb 2? receptor agonist compounds
04/08/1998EP0833638A1 USE OF IMIDAZO 1,5-a]QUINOLONES AS NEUROPROTECTIVE AGENTS
04/08/1998EP0833635A1 Novel use for pyrrole derivatives
04/08/1998CN1037966C Production of 4 -(5, 6, 7, 8 -tetrahydroimidazo £1.5-a| pyridine -5 -group) benzonitrile acidified hemihydrate
04/07/1998US5736555 Hypotensive agents; fda orange book listed patent for azilsartan medoxomil
04/07/1998US5736554 Treating and/or preventing cardiovascular disorders
04/07/1998US5736550 Pyrimidine derivatives
04/07/1998US5736547 Resists pneumocystis carnii and toxoplasmosis gondii infections in immunocompromised patients; dihydrofolate reductase inhibitors; aids; antitumor agents; synergistic agent with sulfa drugs
04/07/1998US5736544 Naphthylpiperazinyl compounds useful for treating 5HT2B receptor mediated conditions
04/07/1998US5736538 Treats in mammal the disease characterized by excess renal reabsorption of water, is congestive heart failure, nephrotic syndrome, hyponatremia, coronary and renal vasospasm, cardiac ischemia, liver cirrhosis and brain edema
04/07/1998CA2130116C Aminoacetylmercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace
04/02/1998WO1998013368A1 New pharmaceutically active compounds
04/02/1998WO1998013367A1 N-([1,2,4] triazoloazinyl)benzenesulfonamide and pyridinesulfonamide compounds and their use as herbicides
04/02/1998WO1998013350A1 Qinoline derivatives inhibiting the effect of growth factors such as vegf
04/02/1998CA2265854A1 New pharmaceutically active compounds
04/02/1998CA2263479A1 Quinoline derivatives inhibiting the effect of growth factors such as vegf
04/01/1998EP0832084A1 Novel derivatives of swainsonine, processes for their preparation and their use as therapeutic agents
04/01/1998EP0831831A1 Protein tyrosine kinase aryl and heteroaryl quinazoline compounds having selective inhibition of her-2 autophosphorylation properties
04/01/1998EP0831829A1 Heterocyclic ring-fused pyrimidine derivatives
04/01/1998EP0625987B1 Aminoacetylmercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace
03/1998
03/31/1998US5734049 Processes for preparing intermediates of inhibitors of enkephalinase and angiotensin converting enzyme and intermediates thereof
03/31/1998US5733914 Pyrido 2, 3-d!pyrimidines for inhibiting protein tyrosine kinase mediated cellular proliferation
03/31/1998US5733913 Treating atherosclerosis, postsurgical restenosis
03/31/1998US5733910 Pyridazinedione compounds useful in the treating neurological disorders
03/31/1998CA1339783C Tetramethylpiperidino-s-triazines
03/26/1998DE19638886A1 Selective herbicidal composition, especially for weed control in crops
03/25/1998EP0831327A1 Redox active compounds and their use
03/25/1998EP0831094A1 Fused polycyclic heterocycle derivatives
03/25/1998EP0830371A1 IMIDAZO 1,5a]PYRIDINE DERIVED SERINE PROTEASE INHIBITORS
03/25/1998CN1177297A Medicament interded to the treatment of obsessive compulsive troubles, sleep apnoea, sexual dysfuctions emesa and transport sickness
03/25/1998CN1176978A Oxidation process for preparing quinacridone pigments
03/25/1998CN1176785A Tricyclic compounds, their production and use
03/24/1998USRE35754 Cephem derivatives
03/24/1998US5731340 Dietetics; antidiabetic agents
03/24/1998US5731322 Octahydro-1H-pyrrolo 3,2-g!and 2,3-g!isoquinoline derivatives
03/24/1998US5731316 Derivatives of camptothecin and methods of treating cancer using these derivatives
03/24/1998US5731307 Antipsychotic agents; reduces chemical dependancy
03/24/1998US5731028 Crystallized zilpaterol hydrochloride
03/24/1998CA2216105A1 Redox-active compounds and their use
03/19/1998WO1998011128A1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production
03/19/1998WO1998011112A1 Tricyclic indazole derivatives, preparation and therapeutic application thereof
03/19/1998WO1998011107A1 Bicyclic hydantoin derivatives, process for producing the same, and herbicides containing the same as active ingredient
03/19/1998WO1998011092A1 Tricyclic antitumor compounds being farnesyl protein transferase inhibitors
03/19/1998WO1998011091A2 Tricyclic compounds useful for inhibition of farnesyl protein transferase
03/19/1998WO1998010653A1 Piperidines, pyrrolidines and hexahydro-1h-azepines promote release of growth hormone
03/19/1998CA2266014A1 Tricyclic compounds useful for inhibition of farnesyl protein transferase
03/19/1998CA2262818A1 Modified amino acids, pharmaceuticals containing these compounds and methods for their production
03/18/1998EP0829523A2 Oxidation process for preparing quinacridone pigments