| Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559) |
|---|
| 05/13/2009 | EP1466174B1 Mutations in the bcr-abl tyrosine kinase associated with resistance to sti-571 |
| 05/13/2009 | EP1299388B1 Variolin derivatives as anti-cancer agents |
| 05/13/2009 | CN101432286A Novel 1,4-diaza-bicyclo[3.2.2]nonyl oxadiazolyl derivatives and their medical use |
| 05/13/2009 | CN101432285A Pyrazolo-tetrahydro pyridine derivatives as orexin receptor antagonists |
| 05/13/2009 | CN101432284A Dihydropyrazolopyrimidinone derivative |
| 05/13/2009 | CN101432278A Diketo-piperazine and piperidine derivatives as antiviral agents |
| 05/13/2009 | CN101429199A Process for producing racemic cis-8-benzyl-7, 9-dioxo-2, 8-diazabicyclo [4.3.0] nonyl hydride |
| 05/13/2009 | CN101429198A Banisterine derivant and uses thereof |
| 05/13/2009 | CN100486573C Nitrosated and nitrosylated cyclooxygenase-2 inhibitors, compositions and use |
| 05/12/2009 | US7531661 Such as N-methyl(1-{2-[(1R,5S)-3-(2-methyl-1H-benzimidazol-1-yl)-8-azabicyclo[3.2.1]oct-8-yl]ethyl}-2,3-dihydro-1H-inden-1-yl)methanamine; chemokine receptor antagonists; prevention or treatment of a human T-cell leukemia/lymphoma virus infection |
| 05/12/2009 | US7531553 Heterocyclic compounds and methods of use |
| 05/12/2009 | US7531552 antiviral for HIV and AIDS; N-(1-Benzoyl-pyrrolidin-3-ylmethyl)-2-(4-fluoro-1H-indol-3-yl)-2-oxo-acetamide; N-(1-Benzoyl-pyrrolidin-3-ylmethyl)-2-oxo-2-(1H-pyrrolo[2,3-b]pyridin-3-yl)-acetamide |
| 05/12/2009 | US7531549 2-[(2-Isopropylsulfanyl-3-oxo-spiro[3.5]non-1-en-1-yl)amino]-3-[4-([2,7]naphthyridin-1-ylamino)phenyl]propanoic acid; compounds can inhibit the binding of integrins to their ligands and are of use in the prophylaxis and treatment of immuno or inflammatory disorders |
| 05/12/2009 | US7531545 2-amino-3,4-dihydro-pyrido[3,4-d]pyrimidine derivatives useful as inhibitors of β-secretase (BACE) |
| 05/12/2009 | US7531536 Inhibitors of glycogen synthase kinase-3 (gsk-3) and aurora-2, both serine/threonine protein kinases; for treating diseases such as cancer, diabetes and alzheimer's disease |
| 05/12/2009 | US7531535 Lactam-containing compounds and derivatives thereof as factor Xa inhibitors |
| 05/12/2009 | US7531531 Method of treating diseases associated with altered kinase activity with bicyclo-pyrazoles |
| 05/12/2009 | US7531526 Boronic ester and acid compounds, synthesis and uses |
| 05/12/2009 | CA2517933C Novel fused heteroaromatic compounds as transforming growth factor (tgf) inhibitors |
| 05/12/2009 | CA2264005C Piperazino derivatives as neurokinin antagonists |
| 05/07/2009 | WO2009057668A1 Amide compound and plant disease control using the same |
| 05/07/2009 | WO2009057578A1 Utilization of novel compounds with amyloid affinity and method of producing the same |
| 05/07/2009 | WO2009057577A1 Use of novel compound having affinity for amyloid, and process for production of the same |
| 05/07/2009 | WO2009057576A1 Use of novel compound having affinity for amyloid, and process for production of the same |
| 05/07/2009 | WO2009057575A1 Use of novel compound having affinity for amyloid, and process for production of the same |
| 05/07/2009 | WO2009056990A2 Paliperidone polymorphs |
| 05/07/2009 | WO2009056934A1 1,4-dihydronaphthyridine derivatives |
| 05/07/2009 | WO2009056556A1 Substitute 1, 6-naphthyridines for use as scd inhibitors |
| 05/07/2009 | WO2009037001A3 Novel tetrahydrofusedpyridines as histone deacetylase inhibitors |
| 05/07/2009 | WO2009030952A3 Phenylcarboxamide derivatives as inhibitors and effectors of the hedgehog pathway |
| 05/07/2009 | WO2009021957A3 Tricyclic heterocyclic compounds as gaba a modulators |
| 05/07/2009 | WO2009018065A3 Novel glucokinase activators and methods of using same |
| 05/07/2009 | WO2009006389A3 Pyrimidine derivatives useful as raf kinase inhibitors |
| 05/07/2009 | WO2008157179A3 N-substituted azaindoles and methods of use |
| 05/07/2009 | WO2008152068A3 [1,10]-phenanthroline derivatives for the treatment of neurodegenerative or haematological diseases |
| 05/07/2009 | WO2008145225A3 Photocrosslinkable materials comprising alicyclic group |
| 05/07/2009 | US20090118512 Process for Preparing 6,7-Dihydro-5H-Imidazo[1,5-A]Pyridin-8-One |
| 05/07/2009 | US20090118499 6,6-Bicyclic Ring Substituted Heterobicyclic Protein Kinase Inhibitors |
| 05/07/2009 | US20090118325 5-Thioxylopyranose Compounds |
| 05/07/2009 | US20090118324 Mapk/erk kinase inhibitors |
| 05/07/2009 | US20090118323 Antitumor benzoylsulfonamides |
| 05/07/2009 | US20090118322 Agent for repairing corneal sensitivity containing amide compound |
| 05/07/2009 | US20090118319 Fused and Spirocycle Compounds and the Use Thereof |
| 05/07/2009 | US20090118305 Pyridine and pyrazine derivatives - 083 |
| 05/07/2009 | US20090118304 2-heteroaryl-substituted indole derivative |
| 05/07/2009 | US20090118282 Compounds and methods for treatment of amyloid-beta-peptide related disorders |
| 05/07/2009 | US20090118279 Compound containing basic group and use thereof |
| 05/07/2009 | US20090118278 Compositions useful as inhibitors of gsk-3 |
| 05/07/2009 | US20090118274 Monocyclic aminopropyl tetrahydro-pyrazolo-pyridine modulators of cathepsin s |
| 05/07/2009 | US20090118266 Novel 1,4-diaza-bicyclo[3.2.2]nonyl oxadiazolyl derivatives and their medical use |
| 05/07/2009 | US20090118265 Novel 1,4-diaza-bicyclo[3.2.2]nonane derivatives and their medical use |
| 05/07/2009 | US20090118261 Quinazolinone derivatives and their use as b-raf inhibitors |
| 05/07/2009 | US20090118233 Heterocyclic compounds having inhibitory activity against HIV integrase |
| 05/07/2009 | US20090118232 Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof |
| 05/07/2009 | US20090117125 Synthesis of 8h-3a-aza-cyclopenta[a]indenes and 5,10-dihydropyrrolo[1,2-b]isoquinolines derivatives and their use as antitumor therapeutic agents |
| 05/07/2009 | US20090115316 Organic electroluminescent device having an azatriphenylene derivative |
| 05/07/2009 | US20090114596 Nanofilm and membrane compositions |
| 05/07/2009 | CA2704172A1 Use of novel compound having affinity for amyloid, and process for production of the same |
| 05/07/2009 | CA2704168A1 Use of novel compound having affinity for amyloid, and process for production of the same |
| 05/07/2009 | CA2704139A1 Utilization of novel compounds with amyloid affinity and method of producing the same |
| 05/07/2009 | CA2704137A1 Use of novel compound having affinity for amyloid, and process for production of the same |
| 05/07/2009 | CA2703876A1 Enantioselective process for preparing a substituted alkanoic acid |
| 05/07/2009 | CA2703217A1 Antidiabetic tricyclic compounds |
| 05/06/2009 | EP2055705A1 Compound having cyclic group bound thereto through spiro binding and use thereof |
| 05/06/2009 | EP2054422A1 Acrylamide derivatives as fab i inhibitors |
| 05/06/2009 | EP2054414A2 Imidazole amines as inhibitors of beta-secretase |
| 05/06/2009 | EP2054413A2 Pyridobenzazepine compounds and methods for inhibiting mitotic progression |
| 05/06/2009 | EP2054412A2 Imino-imidazo-pyridine derivatives having antithrombotic activity |
| 05/06/2009 | EP2054405A1 Novel biaryl benzoimidazole derivatives and pharmaceutical composition comprising the same |
| 05/06/2009 | EP2054385A2 Phenyl, pyridine and quinoline derivatives |
| 05/06/2009 | EP2054060A1 Fluorinated ligands for targeting peripheral benzodiazepine receptors |
| 05/06/2009 | EP1973907B1 Imidazo (1,2-a)pyridin-3-yl-acetic acid hydrazides, processes for their preparation and pharmaceutical uses thereof |
| 05/06/2009 | EP1828185B1 2-pyrimidinyl pyrazolopyridine erbb kinase inhibitors |
| 05/06/2009 | EP1802621B1 Crf receptor antagonists and methods relating thereto |
| 05/06/2009 | EP1682544A4 Hydroxylamine substituted imidazo ring compounds |
| 05/06/2009 | EP1326865B1 Aza- and polyaza-naphthalenyl carboxamides useful as hiv integrase inhibitors |
| 05/06/2009 | EP1268421B1 Phenyl-substituted indoles as histamine h3-receptor antagonists |
| 05/06/2009 | CN101426790A Novel 1,4-diaza-bicyclo[3.2.2]nonyl oxadiazolyl derivatives and their medical use |
| 05/06/2009 | CN101426778A N-substituted-azacyclylamines as histamine-3 antagonists |
| 05/06/2009 | CN101426777A Phenoxypiperidines and analogs thereof useful as histamine h3 antagonists |
| 05/06/2009 | CN101426499A Modulators of muscarinic receptors |
| 05/06/2009 | CN101426486A Compounds for the treatment of inflammatory disorders and microbial diseases |
| 05/06/2009 | CN101423518A Imidazole derivates and medical use thereof |
| 05/06/2009 | CN101423517A Gamma-carbolines derivates as well as preparation method and application thereof |
| 05/06/2009 | CN101423489A Indoline-2-one derivates and uses thereof |
| 05/06/2009 | CN100484935C Benzimidazole-derivatives as factor Xa inhibitors |
| 05/05/2009 | US7528252 Derivatives of triazoly-imidazopyridine useful as ligands of the adenosine A2a receptor and their use as medicaments |
| 05/05/2009 | US7528251 Oxidizing a (pyridinylmethyl]thioimidazo[4,5-b]pyridine derivative using titanium(IV)-based catalyst and a cyclic beta- or gamma-amino-alcohol chiral ligand (1-amino-2-indanol) in a polar aprotic solvent to form a (pyridinylmethyl]sulfinylimidazo[4,5-b]pyridine derative such as tenatoprazole |
| 05/05/2009 | US7528160 {6-[5-Methyl-2-(4-trifluoromethyl-phenyl)-oxazol-4-ylmethoxy]-benzo[b]thiophen-3-yl}-acetic acid; antidiabetic agent; metabolic Syndrome, hyperglycemia, hyperlipidemia, obesity, coagaulopathy, hypertension, atherosclerosis; lowering fibrinogen, increasing HDL levels |
| 05/05/2009 | US7528149 e.g. N-[1-(2-aminoethyl)-4-piperidinyl]-7-methyl-3-(8-quinolinylmethyl)-3H-imidazo[4,5-b]pyridin-2-amine tetrahydrochloride trihydrate; immunostimulant; lower respiratory tract illness during infancy and childhood, asthma, pneumonia |
| 05/05/2009 | US7528148 Pyrazolo[3,4-B]pyridine compounds, and their use as phosphodiesterase inhibitors |
| 05/05/2009 | US7528147 e.g. 2 {5,6-dimethoxy-1-[2-(4-methylpiperazin- 1 -yl)ethyl]-1H-indol-3 -yl}-1H-pyrrolo[2,3- b]pyridine; Insulin Growth Factor-1 (somatomedin) antagonist; antiproliferative, antitumor agent; solid tumor; prostate, lung and breast cancer |
| 05/05/2009 | US7528146 Substituted 1H-pyrrolo[2,3-b]pyridines and preparation thereof |
| 05/05/2009 | US7528139 Sulfonamides |
| 05/05/2009 | CA2204747C New azo derivatives of 5-aminosalicylic acid |
| 04/30/2009 | WO2009055828A1 New tetracyclic compounds |
| 04/30/2009 | WO2009055696A1 CARBACEPHEM β-LACTAM ANTIBIOTICS |
| 04/30/2009 | WO2009055331A2 Bicyclic heterocycle derivatives and their use as modulators of the activity of gpr119 |
| 04/30/2009 | WO2009055033A1 Pyrazolo-pyridinone derivatives and methods of use |
| 04/30/2009 | WO2009054970A1 Mesylate salt of an ikk inhibitor |