Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
04/2009
04/15/2009CN101410397A Organic compounds
04/15/2009CN101410396A Chromane derivatives
04/15/2009CN101410390A Hydantoin compounds for the treatment of inflammatory disorders
04/15/2009CN101410388A Compounds for the treatment of inflammatory disorders
04/15/2009CN101410385A Benzothiazoles having histamine H3 receptor activity
04/15/2009CN101410377A Process for preparing 6,7-dihydro-5h-imidazo[1,5-A]pyridin-8-one
04/15/2009CN101410114A A3 adenosine receptor allosteric modulators
04/15/2009CN101407516A Camptothecine derivative having anticancer activity
04/15/2009CN101407515A Chinoline polycyclic compounds as CDK inhibitors
04/15/2009CN101407492A New nitrogen-containing heterocyclic derivative and organic electroluminescent element using the same
04/15/2009CN101407489A 2-alkyl acrylate compounds and uses thereof
04/15/2009CN101406471A Novel heterocyclic compounds which are active as inhibitors of beta-lactamases
04/15/2009CN100478031C The use of substituted tetracyclic imidazole derivatives as anti-histaminics
04/14/2009US7517994 Heterocyclic inhibitors of MEK and methods of use thereof
04/14/2009US7517990 Method for deuteration of a heterocyclic ring
04/14/2009US7517987 Interleukin converting enzyme inhibitors such as 5-Fluoro-4-oxo-3-(2-(6-oxo-6H-pyrimidin-1-yl)-butyrylamino)-pentanoic acid, administered as modulators of cell apoptosis and inflammation
04/14/2009US7517986 Such as N-(6-ethoxycarbonyl-3-cyano-4,5,6,7-tetrahydrothieno[2,3-c]pyridin-2-yl)nicotinamide; cell-cycle specific inducers of apoptosis specific to cells with aberrant cell growth
04/14/2009US7517904 Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
04/14/2009US7517899 Phenylaminopropanol derivatives and methods of their use
04/14/2009US7517887 Reversible inhibitors of S-adenosyl-L-homocysteine hydrolase and uses thereof
04/14/2009US7517532 Dihydroxypyridopyrazine-1,6-dione compounds useful as HIV integrase inhibitors
04/14/2009US7517517 Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands
04/14/2009CA2468658C [1,2,4]-triazole bicyclic adenosine a2a receptor antagonists
04/09/2009WO2009045753A1 Triazolopyridine 11-beta hydroxysteroid dehydrogenase type i inhibitors
04/09/2009WO2009045489A2 Process for the synthesis of cmhtp, a paliperidone intermediate
04/09/2009WO2009044777A1 Oxazolidinone derivative having 7-membered hetero ring
04/09/2009WO2009044413A2 Improved process for preparing paliperidone, novel polymorphic forms of the same and process thereof
04/09/2009WO2009044147A1 Indolizine derivatives with crth2 receptor affinity for the treatment of inflammatory diseases
04/09/2009WO2009044134A1 Indolizine derivatives with crth2 receptor affinity for the treatment of inflammatory diseases
04/09/2009WO2009023253A3 IMIDAZO[L,2-α]PYRIDINE DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO
04/09/2009WO2009007535A3 Derivatives of 7-alkynyl-1,8-naphthyridones, preparation method thereof and use of same in therapeutics
04/09/2009WO2008155666A3 Heteroarylamide-substituted pyrimidone derivatives for the treatment of neurodegenerative diseases
04/09/2009WO2008151927A3 6-n-substituted benz imidazole derivatives as acid pump antagonists
04/09/2009WO2008149163A3 Potassium ion channel modulators and uses thereof
04/09/2009WO2008021342A3 Amorphous and crystalline forms of 9-hydroxy-risperidone ( paliperidone )
04/09/2009WO2007123732A3 Antifungal and antiparasitic indoloquinoline derivatives
04/09/2009WO2007089336A3 Certain chemical entities, compositions and methods
04/09/2009US20090093634 For therapy and prophylaxis of cardiovascular diseases, diabetes, diabetes- associated disorders, inflammatory diseases, immunological disorders, dermatological disorders, oncological disorders and central nervous system disorders
04/09/2009US20090093516 Triazolopyridine 11-beta hydroxysteroid dehydrogenase type i inhibitors
04/09/2009US20090093515 Substituted pyrroline kinase inhibitors
04/09/2009US20090093512 1, 2, 3, 3a, 8, 8a-hexahydro-2, 7a-diada-cyclopenta[a]inden-7-one derivatives which bind to neuronal nicotinic acetylcholine specific receptor sites and are useful in modulating cholinergic function and in the treatment of addictive disorders
04/09/2009US20090093501 Heterocyclic antiviral compounds
04/09/2009US20090093478 N-aroyl cyclic amines
04/09/2009US20090093473 Spiro-benzimidazoles as inhibitors of gastric acid secretion
04/09/2009US20090093469 Phenylaminopropanol Derivatives and Methods of Their Use
04/09/2009US20090093465 Therapeutic kinase modulators
04/09/2009US20090093455 Quinolone analogs and methods related thereto
04/09/2009US20090091252 Binaphthyl compound and organic light emitting element using the same
04/09/2009US20090091240 Compound containing fused ring and organic electroluminescent element employing the same
04/09/2009CA2701630A1 Quinolone analogs and methods related thereto
04/09/2009CA2701355A1 Triazolopyridine 11-beta hydroxysteroid dehydrogenase type i inhibitors
04/08/2009EP2045252A2 Derivatives of 1,2-dihydro-7-hydroxyquinolines containing fused rings
04/08/2009EP2045243A1 Tetrahydro isoquinoline derivatives, preparation methods and medicinal uses thereof
04/08/2009EP2045242A1 Heterocyclic compounds having inhibitory activity against HIV integrase
04/08/2009EP2044958A2 Pharmaceutical composition for treating arteriosclerosis
04/08/2009EP2044073A1 11beta-hydroxysteroid dehydrogenase type 1 active compounds
04/08/2009EP2044068A1 1-hydroxy naphthyridine compounds as anti-hiv agents
04/08/2009EP2044065A2 Compounds and compositions as hedgehog pathway modulators
04/08/2009EP2044061A2 Benzothiophene inhibitors of rho kinase
04/08/2009EP2044051A1 Pyridine and pyrazine derivatives as mnk kinase inhibitors
04/08/2009EP2044041A2 Isothiazolidines useful in the treatment of ocular hypertensive conditions
04/08/2009EP2044035A1 Process for the covalent coupling of two molecules by means of a diels-alder reaction with inverse electron requirement
04/08/2009EP2044032A2 Novel inhibitors of hepatitis c virus replication
04/08/2009EP2044016A2 4-heteroaryl-substituted 1-aminocyclohexane-1-and cyclohexene-1-derivatives having effects on the opiod receptor system
04/08/2009EP2043655A2 Purine and deazapurine derivatives as pharmaceutical compounds
04/08/2009EP1448566B3 Chemokine receptor antagonists and methods of use thereof
04/08/2009EP1415986B1 Spiro isobenzofuranes as neuropeptide y receptor antagonists
04/08/2009CN101405288A Imidazopyridin-2-one derivatives as inhibitors of endothelial lipase
04/08/2009CN101405282A Aurora kinase modulators and method of use
04/08/2009CN101405281A Inhibitors of the interaction between MDM2 and P53
04/08/2009CN101405277A Dicarbonylic compounds with antibacterial activity
04/08/2009CN101405267A Process for preparing l-halo-2,7-naphthyridinyl derivatives
04/08/2009CN101402636A Propellane compounds, preparation method and application thereof
04/08/2009CN101402635A Process for producing 5-chlorine-7-aza indole
04/08/2009CN100475822C Synthesis method for producing ecteinascidin compound
04/08/2009CN100475814C 7-azaindoles and use thereof as therapeutic agents
04/08/2009CN100475813C 4-oxo-1-3-substituted phenyl-1,4-dihydro-1,8-naphthyridine-3-carboxamide phosphodiesterase-4 inhibitor
04/08/2009CN100475812C Pyrazolopyridines as cyclin dependent kinase inhibitors
04/08/2009CN100475207C 1H-imidazo[4,5-c]quinoline derivatives in the treatment of protein kinase dependent diseases
04/07/2009US7514583 Compounds, compositions and methods for the treatment of amyloid diseases and synucleinopathies such as alzheimer's disease, type 2 diabetes, and parkinson's disease
04/07/2009US7514564 Substituted amine derivatives and methods of use
04/07/2009US7514558 e.g. 3-(4-{[6-({(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)-hexyl]oxy}butyl)benzenesulfonamide; beta 2 adrenergic receptor agonist and muscarinic receptor antagonist activity; bronchodilator agent; pulmonary disorders: chronic obstructive pulmonary disease; asthma
04/07/2009US7514451 1 -cyclopropyl-7- [3-cyclopropylaminomethyl-4-fluoro-1 -pyrrolidinyl]-6-fluoro -1 ,4-dihydro-8-methyl-4-oxo-3-quinolinecarboxylic acid; bactericide; against drug-resistant bacteria and against gram-positive bacteria, such as MRSA, PRSP and VRE
04/07/2009US7514448 Azaindoles useful as inhibitors of rock and other protein kinases
04/07/2009US7514430 Nitrogen compounds such as N-phenyl-N'-{(1R,2S)-2-[(2S)-2-benzyl-6-oxo-morpholin-4-yl-methyl]-cyclohexyl }-urea, used to control chemotactic cytokines, and administered for the prevention of asthma or allergies; inhibition of the migration of eosinophils
04/07/2009US7514420 Steroids having 1,8-unsaturation and formulations comprising same
04/07/2009US7514418 silyl camptothecin derivatives for cancer and/or leukemia; cytotoxic; DNA-topoisomerase I inhibitors; antitumor agents; 7-trimethylsilyl-10-acetoxy camptothecin, 7-trimethylsilyl-11-fluoro camptothecin
04/07/2009CA2341991C Pyrroloindoles, pyridoindoles and azepinoindoles as 5-ht2c agonists
04/07/2009CA2118239C 1h-imidazo{4,5-c}quinolin-4-amines as vaccine adjuvants
04/02/2009WO2009041567A1 Diaryl ketimine derivative having antagonistic activity on melanin-concentrating hormone receptor
04/02/2009WO2009041566A1 Preventive or remedy for posterior eye diseases containing quinazolinone derivative or quinoxaline derivative as the active ingredient
04/02/2009WO2009041565A1 Quinazolinone derivative, and prophylactic or therapeutic agent for corneal/conjunctival disorder comprising quinazolinone derivative as active ingredient
04/02/2009WO2009041559A1 Indazole acrylic acid amide compound
04/02/2009WO2009040399A1 Substituted pyrrolo-pyrimidine derivatives, process for their preparation and their use as kinase inhibitors
04/02/2009WO2009040288A1 1,1,1-trifluoro-2-hydroxy-3-phenylpropane derivatives
04/02/2009WO2009039635A1 Methods of modulating neurotrophin-mediated activity
04/02/2009WO2009019553A3 Imidazopyridinones
04/02/2009US20090088573 Biologically active peptides and compositions, their use
04/02/2009US20090088572 Method for preparing ladderanes
04/02/2009US20090088570 Organic electroluminescent device