Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
08/2009
08/13/2009CA2713519A1 Amide derivatives as positive allosteric modulators and methods of use thereof
08/13/2009CA2713347A1 Mesoionic pesticides
08/13/2009CA2713173A1 (dihydro)pyrrolo[2,1-.alpha.]isoquinolines
08/13/2009CA2712574A1 Polymorphic form of a [1,2,4]triazolo[4,3-a]pyridine derivative for treating inflammatory diseases
08/13/2009CA2711937A1 Pyrido[4,3-d]pyrimidinone derivatives as kinase inhibitors
08/12/2009EP2088149A1 Pharmacologically active n,n'-substituted 3,7-diazabicyclo ý3.3.1¨nonanes, pharmaceutical compositions based thereon and a method for the use thereof
08/12/2009EP2086999A1 Inhibitors for disrupting the interaction of ubiquitination related enzymes and uses thereof
08/12/2009EP2086977A2 Polymorphs of nicotinic intermediates
08/12/2009EP2086976A1 Method for producing pradofloxacin
08/12/2009EP2086975A2 7,8-dihydro-1,6-naphthyridin-5(6h)-ones and related bicyclic compounds as inhibitors of dipeptidyl peptidase iv and methods
08/12/2009EP2086973A2 Imidazo- and triazolo-pyridine compounds and methods of use therof
08/12/2009EP2086972A2 Compounds modulating c-fms and/or c-kit activity and uses therefor
08/12/2009EP2086968A1 5-hydroxymethyl-oxazolidin-2-one derivatives
08/12/2009EP2086965A1 Aminopyridines and aminopyrimidines useful as inhibitors of protein kinases
08/12/2009EP2086958A2 Substituted-quinoxaline-type-piperidine compounds and the uses thereof
08/12/2009EP2086643A1 Compounds which potentiate ampa receptor and uses thereof in medicine
08/12/2009EP2086542A1 Topical formulations
08/12/2009EP2086540A1 Triazolopyridine compounds useful for the treatment of degenerative & inflammatory diseases
08/12/2009EP2086539A1 Selective glycosidase inhibitors
08/12/2009EP1981886B1 7h-pyrido[3,4-d]pyrimidin-8-ones, their manufacture and use as protein kinase inhibitors
08/12/2009EP1904461B1 Cyclic anilino-pyridinotriazines as gsk-3 inhibitors
08/12/2009EP1899337B1 Process for the preparation of 3,7-diazabicyclo[3.3.1]nonane compounds
08/12/2009EP1778686B9 Triazolopyridinylsulfanyl derivatives as p38 map kinase inhibitors
08/12/2009EP1663238B1 HEXA- AND OCTAHYDRO-PYRIDO[1,2-a] PYRAZINE DERIVATIVES WITH NK1 ANTAGONISTIC ACTIVITY
08/12/2009EP1427415B1 Lactam-containing compounds and derivatives thereof as factor xa inhibitors
08/12/2009EP1385514B9 Spiroindene and spiroindane compounds
08/12/2009EP1089988B1 Fluorophenyl resin compounds
08/12/2009EP0788360B3 Boronic ester and acid compounds, synthesis and uses
08/12/2009CN101506210A 2-phenoxy pyrimidinone analogues
08/12/2009CN101506208A Pyrrolo isoquinolines as kinase inhibitors
08/12/2009CN101506207A Compound having pyridoindole ring structure having substituted pyridyl group attached thereto, and organic electroluminescence element
08/12/2009CN101506206A Inhibitors of Akt activity
08/12/2009CN101506165A Phenyl, pyridine and quinoline derivatives
08/12/2009CN101503407A Imidazopyridine compound
08/12/2009CN100526314C Production of high-purity corydalis
08/12/2009CN100526313C Imidazopyridine substituted tropane derivatives with CCR5 receptor antagonist activity for the treatment of HIV and inflammation
08/12/2009CN100526312C Benzimidazole quinolinones and uses thereof
08/12/2009CN100526307C Metalloproteinase inhibitors
08/12/2009CN100525768C Novel compounds
08/11/2009US7572914 2-hydroxy-1H-indol derivatives enzyme inhibitors for preventing or treating inflammation, inflammatory bowel disease, psoriasis, dementia related diseases Alzheimer's Disease, Cognitive Impairment, arthritis, neurodegenerative diseases, amyotrophic lateral sclerosis, Down syndrome, Huntington's Disease
08/11/2009US7572913 Inhibitors of Rho kinase; N-Benzyloxycarbonyl-4-[N''-(tert-butyloxycarbonyl)hydrazino]piperidine; 4-{[N''-(tert-butyloxycarbonyl)-N'-(1'-propyl)]hydrazino}piperidine
08/11/2009US7572883 Somatostatin-dopamine chimeric analogs
08/11/2009US7572808 2-substituted 7-aryl-[1,2,4]triazolo[4,3-c]pyrimidin-3(2H)-one; mitogen-activated protein kinase inhibitor; physiological and psychotropic effects including regulation of appetite, immunosuppression, analgesia, inflammation, emesis, anti-nocioception, sedation, and intraocular pressure
08/11/2009US7572807 3-Cycloheptyl-8-((2,6-dichlorophenoxy)methyl)H-imidazo[1,5-a]pyridine; N-((3-((2,6-Dichlorophenoxy)methyl)pyridin-2-yl)methyl)cycloheptane-carboxamide; diabetes; cardiovascular diseases, Metabolic Syndrome, inflammatory diseases
08/11/2009US7572806 PPAR active compounds
08/11/2009US7572805 (+-)-cis-6-(Trifluoromethyl)-2,3,3a,4-tetrahydro-1H-pyrrolo[3,4-c]isoquinolin-5(9bH)-one hydrochloride; modulation of serotonin receptors; obesity, diabetes, atherosclerosis, dyslipidemia; anxiety, depression, obsessive compulsive disorder, panic disorder, psychosis, schizophrenia, sleep disorder
08/11/2009US7572802 For central nervous system diseases, in particular Parkinson's disease, Extra Pyramidal Syndrome, restless legs syndrome and attention deficit hyperactivity disorder
08/11/2009US7572801 Pyridopyrimidinone derivatives which are HM74A agonists
08/11/2009US7572796 excitatory amino acid antagonists for treating neurodegenerative diseases as cerebrovascular diseases, epilepsy, schizophrenia, Alzheimer's disease, Parkinson's disease, Huntington's disease, cerebral ischaemia, infarction, psychoses; 6-{3-[4-(4-fluorobenzyl)-1-piperidyl]propyl}-1H-indole-3-carbonitrile
08/11/2009US7572791 Long-term stability, extended delivery using a suitable reservoir; pumped or metered at a controlled rate; implantable or external pump device, pen style injection device; stable at physiologic temperatures for duration of therapeutic exposure; supply of therapeutically active material for up to 2 years
08/11/2009US7572787 Substituted naphthalene sulfonamides
08/11/2009CA2482551C 1-(4-piperidinyl) benzimidazolones as histamine h3 antagonists
08/11/2009CA2395846C Diazepan derivatives or salts thereof
08/11/2009CA2222552C N-oxides as antibacterial agents
08/06/2009WO2009097515A2 [a]-fused indole compounds, their use as mtor kinase and pi3 kinase inhibitors, and their syntheses
08/06/2009WO2009097287A1 Compounds and compositions as kinase inhibitors
08/06/2009WO2009097014A2 Therapeutic kinase modulators
08/06/2009WO2009096549A1 Compound having substituted pyridyl group and pyridoindole ring structure linked through phenylene group, and organic electroluminescent device
08/06/2009WO2009095752A1 Fused pyrazole derivatives as cannabinoid receptor modulators
08/06/2009WO2009095394A1 Diazepanes as histamine h3 receptor antagonists
08/06/2009WO2009095253A1 6-halo-pyrazolo[1, 5-a]pyridines, a process for their preparation and their use as metabotropic glutamate receptor (mglur) modulators
08/06/2009WO2009095162A1 Cyclic azaindole-3-carboxamides, their preparation and their use as pharmaceuticals
08/06/2009WO2009094831A1 Heteroaromatic compounds, the preparation method and the use thereof
08/06/2009WO2009023179A3 Nitrogen containing bicyclic chemical entities for treating viral infections
08/06/2009US20090198063 Novel heterocyclic compound or salt thereof and intermediate thereof
08/06/2009US20090198061 Camptothecin analogs and methods of preparation thereof
08/06/2009US20090198051 Chemical intermediates for sulfiding under mild conditions forming ring compounds for use as marine alkaloids; connecting reaction of 4 components, transforming c22-tert-butyltriphenylsilyl to acety group, cyclization, hydroxy group to methanesulonyl group, reduction of amide, dehydration,Heck reaction
08/06/2009US20090198049 Methods and intermediates for the synthesis of porphyrins
08/06/2009US20090197965 Compounds, compositions and methods for the treatment of amyloid diseases and synucleinopathies such as alzheimer's disease, type 2 diabetes, and parkinson's disease
08/06/2009US20090197910 Novel viral replication inhibitors
08/06/2009US20090197909 Bis-Heterocyclic Imidazolyl Compounds
08/06/2009US20090197906 Reversion of malignant phenotype with 9-hydroxy ellipticine derivatives
08/06/2009US20090197901 Variolin derivatives and their use as antitumor agents
08/06/2009US20090197889 Synthesis and anti-proliferative effect of benzimidazole derivatives
08/06/2009US20090197887 Piperazinylpiperidine derivatives as chemokine receptor antagonists
08/06/2009US20090197881 pyrrolo[2,3-b]pyridine derivatives used as prostaglandin D2 (PGD2) receptor antagonists, for the treatment of allergic diseases such as asthma
08/06/2009US20090197871 Dual Pharmacophores - PDE4-Muscarinic Antagonistics
08/06/2009US20090197862 2-aminopyridine kinase inhibitors
08/06/2009CA2713807A1 Compounds and compositions as kinase inhibitors
08/06/2009CA2712701A1 Cyclic azaindole-3-carboxamides, their preparation and their use as pharmaceuticals
08/06/2009CA2698463A1 Therapeutic kinase modulators
08/05/2009EP2084160A1 Hiv integrase inhibitors
08/05/2009EP2084159A1 Pyrido ý2, 3-d¨pyrimidines and their use as kinase inhibitors
08/05/2009EP2029559B1 Aryl-4-ethynyl-isoxazole derivatives
08/05/2009EP1948132B1 Zolpidem tablets
08/05/2009EP1919474B1 Pyrrolopyridine derivatives and use of same as ppar receptor modulators
08/05/2009EP1805144A4 Heterocyclical chromophore architectures
08/05/2009EP1737459B1 Imidazopyridine and imidazopyrimidine derivatives as antibacterial agents
08/05/2009EP1713803B1 7-phenylamino-4-quinolone-3-carboxylic acid derivatives, methods for production and use thereof as medicaments
08/05/2009EP1699454B1 Pyrazole derivatives and use thereof as orexin receptor antagonists
08/05/2009EP1641457B1 Pyrrolo-dihydroisoquinoline derivatives as pde10 inhibitors
08/05/2009EP1465880B1 5-sulphanyl-4h-1,2,4-triazole derivatives and their use to treat disorders associated with somatostatine
08/05/2009EP1401825B1 Thiophene derivatives as antiviral agents for flavivirus infection
08/05/2009EP1399445B1 Substituted pyrroloquinolines and pyridoquinolines as serotonin agonists and antagonists
08/05/2009EP1357111B1 2-pyridone derivatives having affinity for cannabinoid type 2 receptor
08/05/2009CN101501034A 1, 7-naphthyridine derivatives as p38 map kinase inhibitors
08/05/2009CN101501033A Novel compound having affinity for amyloid
08/05/2009CN101501032A Fused, tricyclic sulfonamide inhibitors of gamma secretase
08/05/2009CN101501024A Muscarinic receptor agonists that are effective in the treatment of pain, alzheimer's disease and schizophrenia
08/05/2009CN101501009A CGRP receptor antagonists