Patents
Patents for C07D 419 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms (1,431)
08/2008
08/05/2008US7407950 N-(heteroaryl)-1H-indole-2-carboxamide derivatives and their use as vanilloid TRPV1 receptor ligands
07/2008
07/30/2008CN101233128A Heteroaryl benzamide derivatives for use as glk activators in the treatment of diabetes
07/24/2008WO2008073956A3 Cyclic sulfonamide derivatives and methods of their use
07/17/2008WO2008050101A3 Benzoyl amino heterocyclyl compounds useful in the treatment of a disease mediated through glk
07/15/2008US7399767 Heterocyclic benzo[c]chromene derivatives useful as modulators of the estrogen receptors
07/02/2008EP1937677A1 Cb-1 modulating compounds and their use
07/02/2008EP1937676A1 Biocompatible fluorescent imaging agents
07/02/2008CN100398537C Cycloalkyl derivatives having bioisosteric carboxylic acid groups, processes for their preparation and their use as pharmaceuticals
07/02/2008CN100398105C 1,3-substitued cycloalkyl derivatives having acidic, mostly heterocyclic groups, processes for their preparation and their use as pharmaceuticals
06/2008
06/25/2008EP1934211A1 Biocompatible n, n-disubstituted sulfonamide-containing fluorescent dye labels
06/25/2008EP1606266A4 Chemical compounds
06/25/2008CN101208094A Pharmacokinetically improved compounds
06/19/2008WO2008073956A2 Cyclic sulfonamide derivatives and methods of their use
06/19/2008WO2008044027A3 Pharmaceutical compounds having hsp90 inhibitory or modulating activity
06/19/2008US20080146569 Nicotinamide Derivatives
06/18/2008EP1931662A1 Pyrimidine derivatives for the inhibition of igf-ir tyrosine kinase activity
06/18/2008EP1931659A1 Derivatives of 2 -aminthiazoles and 2-aminooxazoles, processes for their preparation and their use as pharmaceuticals
06/05/2008US20080132500 Antibiotic compounds
06/04/2008EP1927594A1 1,2,3-Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia
06/03/2008US7381723 Antiserotonine agents; stroke, brain disorders;trauma; Alzheimer's disease; neurodegenerative disease; schizophrenia; psychological disorders; anxiolytic agents; controlling stresses; eating disorders; sleep disorders; sexual disorders
06/03/2008US7381719 To treat obesity and Related Diseases; oral bioavailablility, oral administration; inhibition of orexigenic effects; side effects reduction; weight loss while maintaining or minimizing the loss of lean muscle mass; 6-[4-(2-Benzylamino-ethyl)-phenoxy]-nicotinamide
05/2008
05/29/2008WO2008064218A2 Amido anti-viral compounds
05/20/2008US7375229 Dihydro-dibenzo[B,E]oxepine based selective estrogen receptor modulators, compositions and methods
05/20/2008CA2191874C Novel processes and intermediates for the preparation of piperazine derivatives
05/08/2008US20080108668 compounds with biological activity against all sorts of plant diseases and insects at very low dosage, to control plant diseases like cucumber downy mildew, cucumber grey mold, cucumber powdery mildew, tomato early blight, tomato late blight, phytophthora blight of pepper, grape downy mildew and etc
05/06/2008US7368451 N-(3,5-diamino-6-chloropyrazine-2-carbonyl)-N'-(4-{4-[3-(1H-tetrazol-5-yl)propoxy]phenyl}butyl)guanidine hydrochloride; hydrates mucosal surfaces; are absorbed less rapidly, thus have a prolonged pharmacodynamic half-life; skin and respiratory disorders, vision deffects
05/02/2008CA2667435A1 Chemical compounds
04/2008
04/29/2008US7365068 Hepatitis C virus infections; -(3-cyclopropyl-4-(pentyloxy)phenyl)-3-nicotinoylthiourea;methyl 2-oxo-2-(5-((3-(4-(pentyloxy)-3-(trifluoromethyl)phenyl)thioureido)carbonyl)pyridin-2-ylamino)acetate
04/23/2008CN101166735A Novel oxadiazole derivatives and their medical use
04/17/2008WO2008044045A1 Pharmaceutical combinations
04/03/2008WO2008039023A1 Heteroaryl-pyrazole derivatives as cannabinoid cb1 receptor antagonists
04/01/2008US7351825 4-[5-((1S,2R)-1-Carboxy-2-phenyl-cyclopropylsulfamoyl)-thiophen-2-yl]-3,6-dihydro-2H-pyridine-1-carboxylic acid tert-butyl ester; aggrecanase and matrix metalloproteinase (with zinc in the catalytic active center) (MMP) inhibitor; antiarthritic agent: osteoarthritis, rheumatoid arthritis
03/2008
03/18/2008CA2277893C 4-(3-heterocyclyl-1-benzoyl)pyrazoles and their use as herbicides
03/12/2008CN100374434C Microbiocidal N-Phenyl-N-[4-pyridyl-pyrimidin-2-yl]-amine derivatives
03/11/2008US7341700 Method for recovery of metals from metal-containing materials using medium temperature pressure leaching
03/05/2008CN101137653A Thiazole-4-carboxamide derivatives as MGLUR5 antagonists
02/2008
02/27/2008EP1891058A1 Heteroaryl benzamide derivatives for use as glk activators in the treatment of diabetes
02/20/2008EP1888567A1 Heteroaryl-carboxylic acid (sulfamoyl alkyl) amide - derivatives as factor xa inhibitors
02/20/2008CN100369905C Antibiotic & antifouling oxathiazine and its oxide
02/14/2008US20080039327 3-heterocyclyl-substituted benzoyl derivatives
02/13/2008EP1480973B1 1,4-disubstituted benzofused cycloalkyl urea compounds useful in treating cytokine mediated diseases
02/06/2008EP1884511A1 Aromatic ether compounds,preparation and usage thereof
02/06/2008EP1135239B1 Wood preservative formulations
01/2008
01/31/2008WO2008013414A1 Novel compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist; and pharmaceutical compositions containing the same
01/31/2008CA2658925A1 Novel sulfonylamino acrylamide derivatives, isomer thereof,or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist; and pharmaceutical compositions containing the same
01/30/2008EP1881979A1 Novel oxadiazole derivatives and their medical use
01/23/2008EP1879886A1 Mitotic kinesin inhibitors and methods of use thereof
01/17/2008WO2007068374A3 Thienylpyridyl carboxamides
01/10/2008WO2008005338A1 Modulators of the histamine h3-receptor useful for the treatment of disorders related thereto
01/10/2008WO2007123853A3 Five-membered heterocyclic invertebrate pest control agents
01/10/2008US20080008655 Cyanine dye bioconjugates useful for diagnostic imaging and therapy; for photoacoustic imaging and detection of tumors; do not aggregate in solution, form starburst dendrimers, are capable of absorbing or omitting light in the near infrared region; Bis(ethylcarboxymethyl)indocyanine Dye
12/2007
12/26/2007CN100357270C D-proline derivative
12/21/2007WO2007059359A3 Substituted pyrazalones
12/20/2007US20070293509 treating eating disorders, obesity, type II diabetes, and substance abuse and/or addiction (including alcohol dependency and nicotine dependency); 6-(4-chloro-phenyl)-5-[methyl-(3-methyl-butyl)-amino]-pyrazine-2-carboxylic acid ((R)-2-cyclopropyl-2-hydroxy-propyl)-amide
12/19/2007EP1865775A1 Diarylamine-containing compounds and compositions, and their use as modulators of steroid hormone nuclear receptors
12/19/2007CN101090894A Macrocyclic compounds and compositions useful as BACE inhibitors
12/12/2007CN101087755A Substituted aryl acylthioureas and related compounds; inhibitors of viral replication
12/06/2007WO2007137800A1 Isoindolin-1-one-, isoindolin-3-one- and isoindolin-1,3-dione-derivatives and use thereof
12/06/2007WO2007137791A1 Aryl-substituted heterocycles, and use thereof
12/06/2007CA2653673A1 Isoindolin-1-one, isoindolin-3-one and isoindoline-1,3-dione derivatives and their use
12/04/2007US7304160 intermediates for enantiomerically pure analogs having silyl or alkyl groups at C4 position; organometallic nucleophile or Grignard and an silyl or alkyl acyl halide reacted with nicotine; oxidation and deacylation to 4-hydroxy; modulate nicotinic acetylcholine receptors; Alzheimer's, Parkinson's
11/2007
11/29/2007WO2007060541A3 Piperazine derivatives and their use as insecticides, acaricides, molluscicides, and nematicides
11/29/2007WO2007057407A3 Insecticidal methods using 3-amino-1,2-benzisothiazole derivatives
11/28/2007CN100351242C Processes and intermediates for preparing anti-cancer compounds
11/15/2007WO2007056469A3 Certain chemical entities, compositions, and methods
11/15/2007US20070265308 5-[5-(2-chloro-4-fluorophenyl)-2-piperidin-4-yl-1,3-thiazol-4-yl]-1-(2,6-dichlorophenyl)pyridin-2(1H)-one; p38 MAP kinase inhibitory activity; inflammatory, respiratory , circulatory and central nervous diseases; rheumatoid arthritis
11/14/2007EP1578745B1 BENZOFURAN DERIVATivES, PROCESS FOR THEIR PREPARATION AND INTERMEDIATES THEREOF
10/2007
10/31/2007EP1848435A2 Compounds for inflammation and immune-related uses
10/24/2007CN101061116A Sulfonamide compounds
10/24/2007CN101061096A Cycloalkyl keto piperidine tachykinin receptor antagonists
10/24/2007CN101061095A Cycloalkyl piperidine tachykinin receptor antagonists
10/24/2007CN101058573A 2-hydrazone substituted triazine compound, preparation method thereof, and medicinal composition and use using same as active component
10/23/2007US7285551 For use as therapeutic agent and prophylactic agent for hepatitis C
10/18/2007US20070244103 Novel Compounds Having an Anti-Bacterial Activity
10/18/2007DE69233686T2 Heteoaryl-Piperidine und Piperazine und ihre Anwendung als antipsychotisches und analgetisches Mittel Heteoaryl-piperidines and piperazines and their use as antipsychotic and analgesic agent
10/17/2007EP1844044A1 Thiazole-4-carboxamide derivatives as mglur5 antagonists
10/04/2007US20070232596 10-(o-Hydroxyphenyl)--3a,4,9,10-tetrahydro-2-alkyl-2,9,10a-triazacyclopenty[b]fluorene-1,3-diones or the corresponding 2,10a-diaza-9 oxafluorenediones or 1,10a-diaza-9-thiafluorenediones; antiproliferative, apoptosis-inducing agents; treating color cancer
10/03/2007EP1838680A2 Macrocyclic compounds and compositions useful as bace inhibitors
10/03/2007EP1599468B1 1,2,3-trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia
09/2007
09/26/2007CN101041657A Imines derivative of 4,5-disubstituted-2-aminothiazole having anticancer action and preparation thereof
09/25/2007US7273936 A 2-pyridyl derivatives therapeutic agent for treating cancer, glomerulonephritis, diabetic nephropathy, hepatic fibrosis, pulmonary fibrosis, hyperplasia, restenosis, skin disorders
09/20/2007WO2007105637A1 Nitrogenated heterocyclic derivative, and pharmaceutical agent comprising the derivative as active ingredient
09/20/2007CA2644368A1 Nitrogenated heterocyclic derivative, and pharmaceutical agent comprising the derivative as active ingredient
09/12/2007CN101035785A Novel compounds having an anti-bacterial activity
08/2007
08/29/2007EP1643998B1 Dual nk1/nk3 antagonists for treating schizophrenia
08/23/2007US20070197493 Selenophene anti-tumor agents
08/22/2007EP1819702A1 Thiazepine oxazolidinones as antibacterial agents
08/21/2007CA2304965C ((cyclo)alkyl substituted)-gamma-aminobutyric acid derivatives (=gaba analogues), their preparation and their use in the treatment of neurological disorders
08/16/2007WO2007092638A1 Bicyclic sphingosine 1-phosphate analogs
08/16/2007CA2641718A1 Bicyclic sphingosine 1-phosphate analogs
08/15/2007EP1817285A2 Cycloalkyl keto piperidine tachykinin receptor antagonists
08/08/2007EP1814550A2 N-sulfonylpiperidine cannabinoid receptor 1 antagonists
08/08/2007CN101014591A Novel substituted thiophenecarboxamides, their production and their use as medicaments
08/02/2007WO2006081391A3 Compounds for inflammation and immune-related uses
08/02/2007US20070179122 Beta-Aminoacid-Derivatives As Factor Xa Inhibitors
08/01/2007EP1811844A1 Methods for diagnosis and treatment of cancer
07/2007
07/31/2007US7250421 Diketo acids with nucleobase scaffolds: anti-HIV replication inhibitors targeted at HIV integrase
07/31/2007CA2175212C Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics
07/31/2007CA2121253C Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics
07/12/2007US20070160931 methine dye containing C4O2.C6.C4O2 ring; thermal stability, light fastness; reproduction/playback of the high density information recordings
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