| Patents for C07D 419 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms (1,431) |
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| 11/09/2010 | US7829563 sleep disorders; (R)-2-[(S)1-(5-chloro-2-methoxy-phenyl)-3-(6-trifluoromethyl-pyridin-3-yl)-propylamino]-2-(4-fluoro-phenyl)-N-methyl-acetamide |
| 10/26/2010 | US7820682 3-{[(3R)-1-(3,5-dimethoxy-4-methylbenzoyl)-5-(2-phenylethyl)-3-pyrrolidinyl]oxy}benzoic acid methyl ester; treatment of urinary system disease; anticarcinogenic agent, antiarthritic agent, treats proliferative disease, inflammation/immune system disease, Sjogren*s syndrome, brain-related disease |
| 10/20/2010 | EP0959075B1 Heteroarylpiperidines and piperazines and their use as antipsychotics and analgetics |
| 10/19/2010 | US7816380 1-hydroxycycloalkanecarboxamide derivatives |
| 10/19/2010 | CA2362715C Quinazoline derivatives as angiogenesis inhibitors |
| 10/06/2010 | EP1268446B1 Method for producing asymmetrical 4,6-bis(aryloxy)pyrimidine derivatives |
| 09/21/2010 | US7799915 Several exemplified (pyrimidin-2-ylamino)benzenesulfonamide compounds such as N-phenyl-4-[(4-thien-2-ylpyrimidin-2-yl)amino]benzenesulfonamide; I kappa B kinase inhibitors (IKK inhibitors); anticancer agents, autoimmune diseases, osteoporosis |
| 09/21/2010 | CA2499429C Novel oxazole and thiazole compounds as transforming growth factor (tgf) inhibitors |
| 09/16/2010 | WO2010105048A1 Thiazolidinedione analogues |
| 09/15/2010 | CN101835377A Pyrazole compounds for controlling invertebrate pests |
| 09/14/2010 | US7795179 Substituted azole compounds and its preparation and use thereof |
| 09/10/2010 | WO2010100144A1 Fused bicyclic compounds as inhibitors for pi3 kinase |
| 09/08/2010 | EP1931659B1 Derivatives of 2 -aminthiazoles and 2-aminooxazoles, processes for their preparation and their use as pharmaceuticals |
| 09/07/2010 | US7790710 Imidazopyridine derivatives useful as iNOS inhibitors |
| 09/01/2010 | CN101821241A Gamma secretase modulators |
| 08/31/2010 | US7786141 Treating neurodegenerative diseases, psychological disorders, pain, glaucoma, dru eye, dry mouth, Sjogren's syndrome, asthma, bradycardia, wound healing, gastrointestinal disorders; amide- or urea-functional C5.C5N.C6 SPIRO(INDENE-2,4'-PIPERIDINE) RING structures; selective as to subtypes M1-M5 |
| 08/31/2010 | US7786125 Neuroprotective small organic molecules, compositions and uses of related thereto |
| 08/24/2010 | US7781456 The desired characteristics of chiral compounds helps reduce the toxicity of compound; to treat mood disorders, depression; pain, neurodegenerative disorders, sexual disorders, drug abuse etc. |
| 08/19/2010 | US20100210603 Novel sulfonamide inhibitors of aspartyl protease |
| 08/17/2010 | US7777036 1'-(2-Trifluoromethylbenzoyl)-1',2',3',6'-tetrahydro-[2,4']bipyridinyl-5-carboxylic acid (2-cyclopropylethyl)amide; for diseases mediated by stearoyl-CoA desaturase enzymes, preferably SCD1, especially those related to elevated lipid levels, cardiovascular disease, diabetes, obesity, metabolic syndrome |
| 08/17/2010 | US7776876 administering cyclic Glycyl-2-Allyl Proline as as neuroprotectants, for the prophylaxis of nervous system disorders |
| 08/12/2010 | WO2010090716A1 Heteroaryls and their use as pi3k inhibitors |
| 08/12/2010 | CA2750935A1 Heteroaryls and their use as pi3k inhibitors |
| 08/11/2010 | EP1881979B1 Novel oxadiazole derivatives and their medical use |
| 08/03/2010 | US7767812 Crystals of pyrimidine compound and process for producing the same |
| 08/03/2010 | US7767706 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication |
| 07/28/2010 | EP2029546B1 Aryl-substituted heterocycles, and use thereof |
| 07/21/2010 | EP1844044B1 Thiazole-4-carboxamide derivatives as mglur5 antagonists |
| 07/14/2010 | EP2206709A2 Thiophene derivatives as antiviral agents for flavivirus infection |
| 07/14/2010 | EP1778236B1 Modified pyrimidine glucocorticoid receptor modulators |
| 07/13/2010 | US7754727 Hypotensive agents; atherosclerosis; congestive heart failure; hypertrophy; cardiomyopathy; diabetic nephropathy; restenosis; cognition activator; Alzheimer's disease; anxiolytic agents |
| 07/13/2010 | US7754723 Therapeutic agents useful for treating pain |
| 07/01/2010 | WO2010072310A1 4-amino-1,2,3- benzoxathiazine derivatives as pesticides |
| 07/01/2010 | US20100168189 Therapeutic substituted lactams |
| 06/30/2010 | EP2201009A2 Monomethine dyes |
| 06/30/2010 | CN101765591A Pyrimidine derivatives useful for the treatment of inflammatory or allergic conditions |
| 06/29/2010 | US7745453 Hydroxypyrimidinone derivatives having inhibitory activity against HIV integrase |
| 06/29/2010 | US7745442 Methods of reducing risk of infection from pathogens |
| 06/16/2010 | EP2196461A1 4-Amino-1,2,3-benzoxathiazine-derivatives as pesticides |
| 06/15/2010 | US7737275 simple and low cost chemical process of 2-chloro-5-[3,6-dihydro-2,6-dioxo-4-(trifluoromethyl)-1(2H)-pyrimidinyl]-4-fluoro-N-[[methyl(1-methylethyl)amino]sulfonyl]benzamide |
| 06/15/2010 | US7737153 Heteroaryloxy-substituted phenylaminopyrimidines as rho-kinase inhibitors |
| 06/09/2010 | EP2192839A1 Synergistic pesticidal mixtures |
| 06/09/2010 | CN1852712B Dual NK1/NK3 antagonists for treating schizophrenia |
| 06/01/2010 | US7728136 Such as 5-(2-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)ethyl)-6-chloro-1,3-dihydro-2H-indol-2-one via coupling piperazine derivative with alkyl halide by heating in solvent free conditions |
| 05/19/2010 | EP2186811A1 Synthesis of epothilones, intermediates thereto, analogues and uses thereof |
| 05/19/2010 | EP2185550A1 Substituted aryloxazoles and the use thereof |
| 05/11/2010 | US7714130 To a suspension of 2-(4-t-butylphenyl)-4-piperazin-1-yl-1H-benzimidazole and potassium carbonate in acetone was added 6-bromomethylquinoxaline to produce 2-(4-tert-butylphenyl)4-{[4-(6-quinoxalyl)methyl]piperazin-1-yl}benzimidazole Dihydrochloride Dihydrate |
| 04/29/2010 | US20100105894 Cyclopropane compounds and pharmaceutical use thereof |
| 04/27/2010 | US7704995 Protein kinase modulators and methods of use |
| 04/21/2010 | EP2176233A1 Gamma secretase modulators |
| 04/20/2010 | US7700631 Use of pyridine N-oxide analogs at doses which do not induce emesis |
| 04/20/2010 | US7700552 Macrocyclic inhibitors of hepatitis C virus |
| 04/14/2010 | EP2173722A2 Pyrimidine derivatives useful for the treatment of inflammatory or allergic conditions |
| 04/14/2010 | EP1694410B1 Cyclopropane derivatives and pharmaceutical use thereof |
| 03/30/2010 | US7687508 Cyclic derivatives as modulators of chemokine receptor activity |
| 03/30/2010 | US7687502 Substituted quinazoline or pyridopyrimidine derivative |
| 03/30/2010 | CA2418084C Substituted and unsubstituted benzooxathiazoles and compounds derived therefrom |
| 03/24/2010 | CN101677570A synergistic pesticidal mixtures |
| 03/23/2010 | US7683050 Anticancer agents; parasiticides, viricides, fungicides, bactericides; sealed container consisting of an aqueous solution of homoharringtonine (4-methyl-2-hydroxy-2-(4-hydroxy-4-methylpentyl) (HHT), wherein solution is free of pharmaceutical excipients and said sealed container is an ampule or vial |
| 03/16/2010 | US7678798 5-({4-[(3S)-4-(5-bromo-2,3-dihydro-1H-inden-1-yl)-3-methylpiperazin-1-yl]-4-methylpiperidin-1-yl}carbonyl)-4,6-dimethylpyrimidine; inflammatory diseases, immune diseases and viral infections; HIV |
| 03/09/2010 | US7674901 Process for preparation of imatinib base |
| 03/02/2010 | US7671077 Kits for neurodegenerative diseases such as Parkinson's disease and amyotrophic lateral sclerosis (ALS) |
| 02/16/2010 | US7662811 1,2,3,4-tetrahydropyrazin-2-yl acetamides and methods of use |
| 02/10/2010 | EP1747196B1 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication |
| 01/14/2010 | US20100010045 PYRAZOLE-DERIVATIVES AS FACTOR Xa INHIBITORS |
| 01/13/2010 | CN101624391A Thiophene derivatives as antiviral agents for flavivirus infection |
| 01/05/2010 | US7642354 Polycyclic pyrazines as potassium ion channel modulators |
| 01/05/2010 | US7642274 (+)-3-acetyl-6-chloro-2-[2-(3-(N-(2-hydroxyethyl)-N-isopropylamino)propoxy)-5-methoxyphenyl]benzothiazoline; kappa -opioid receptor agonist |
| 12/24/2009 | US20090318472 Aminopyrazine derivatives and compositions |
| 12/16/2009 | EP2132193A1 Substituted pyrrolidine amides, the production thereof, and the use thereof as medications |
| 12/16/2009 | EP1888567B1 Heteroaryl-carboxylic acid (sulfamoyl alkyl) amide - derivatives as factor xa inhibitors |
| 11/17/2009 | US7618975 4-arylamino-quinazolines and analogs as activators of caspases and inducers of apoptosis; antiproliferative, anticarcinogenic, antimetabolic agents; tubulin and topoisomerase II inhibitors; fungicides; synergistic administration with other anticarcinogenic agents |
| 11/11/2009 | CN100558724C Sulphonic acid amide for regulating bast peptide activity and derivative thereof |
| 11/05/2009 | WO2009134224A1 Synergistic pesticidal mixtures |
| 10/29/2009 | WO2009131977A1 Therapeutic compounds |
| 10/29/2009 | US20090270367 Substituted hydroxyethylamine aspartyl protease inhibitors |
| 10/29/2009 | CA2731279A1 Therapeutic compounds |
| 10/28/2009 | CN101568534A Benzoyl amino heterocyclyl compounds useful in the treatment of a disease mediated through GLK |
| 10/27/2009 | US7608643 Compounds for inhibiting KSP kinesin activity |
| 10/27/2009 | US7608632 Sulfonamide inhibitors of aspartyl protease |
| 10/27/2009 | US7608564 Herbicide; in crops such as wheat, rice, maize, soybeans and cotton they act against broad-leaved weeds and grass weeds without damaging the crop plants; compounds are based on 3-(5,5-disubstituted 2-isoxazolin-3-yl)benzoic acid, esters, thioesters and pyrazolyl ketones thereof |
| 10/22/2009 | WO2009127726A1 Novel microbiocides |
| 10/22/2009 | US20090264401 Substituted pyrimidin-5-carboxamides 281 |
| 10/14/2009 | CN100548987C Pesticidal pyridinecarboxamide derivatives |
| 10/06/2009 | US7598389 Silylated carboxamides |
| 10/06/2009 | US7598255 Pyrimidine compounds as serotonin receptor modulators |
| 10/06/2009 | US7598251 aminopyrazine derivatives; ROCK inhibitors; 3-(1-ethyl-1H-imidazo[4,5-c]pyridin-2-yl)pyrazin-2-amine; antiinflammatory, antidiabetic, antiproliferative agents |
| 09/29/2009 | US7595321 Useful for the prevention and/or treatment of cognitive disorders; 3-Amino-N-(2-cyanoethyl)-6-[4-(pyrrolidin-1-ylsulfonyl)phenyl]pyrazine-2-carboxamide, for example |
| 09/29/2009 | US7595319 Compounds having selective inhibiting effect at GSK3 |
| 09/24/2009 | WO2009027393A3 Pyrazole compounds for controlling invertebrate pests |
| 09/16/2009 | EP2099778A2 Amido anti-viral compounds |
| 09/15/2009 | US7589205 phosphodiesterase inhibitor; antiinflammatory agent; 3-thia-10-aza-phenanthrenes and iintermediates 3-(3,4-dialkoxy-phenyl)-tetrahydro-thiopyran-4-one and 3-(3,4-dialkoxy-phenyl)-1,1-dioxo-hexahydro-1-thiopyran-4-ylamine, useful for its preparation |
| 09/09/2009 | CN101528740A Heteroaryl-pyrazole derivatives as cannabinoid CB1 receptor antagonists |
| 09/08/2009 | US7585853 Compounds having selective inhibiting effect at GSK3 |
| 09/08/2009 | CA2213466C Inhibitors of microsomal triglyceride transfer protein and method |
| 09/02/2009 | CN101522674A Novel compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist |
| 08/18/2009 | US7576209 Breast, prostate and ovarian cancer; such as 1-[4-(9-phenyl-3-pyrimidin-2-yl[1,2,4]triazolo[3,4-f]-1,6-naphthyridin-8-yl)phenyl]cyclobutanamine; serine/threonine kinase (Akt) suppression |
| 08/18/2009 | US7576076 1-Methyl,2,6-dioxo,4-(4-(ethyloxycarbony)piperazin-1-yl-),5-(3-trifluoromethylphenyl)methyl-)-1,2,3,6-tetrahydropyrimidine; antagonist, antagonism; psychoses; antidepressants; schizophrenia; psychological disorders; Alzheimer's disease; neurodegenerative diseases;drug abuse, drug dependence (cocaine) |
| 08/18/2009 | US7576074 Receptor-type kinase modulators and methods of use |
| 08/12/2009 | EP2086964A2 Benzoyl amino heterocyclyl compounds useful in the treatment of a disease mediated through glk |