Patents
Patents for C07D 419 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms (1,431)
07/2001
07/17/2001US6262089 Using these compounds to treat diseases associated with amyloidosis, such as alzheimer's disease, maturity onset diabetes mellitus, familial amyloid polyneuropathy, scrapie, and kreuzfeld-jacob disease.
06/2001
06/27/2001EP1110954A1 Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics
06/26/2001US6251907 1-(aryloxyalkyl)-4-(heteroaryl) piperazines and related compounds useful as antipsychotics and analgesics
06/20/2001EP1108426A2 Use of prostaglandin agonists to treat erectile dysfunction or impotence
06/13/2001CN1299360A Pesticidal methoximinomethyloxathiazines
06/02/2001CA2327164A1 Use of prostaglandin agonists to treat erectile dysfunction or impotence
05/2001
05/15/2001US6232309 2-chloropyridine or 2-chlorothiazole derivatives of heterocyclic compounds used as pesticides
05/09/2001CN1065532C Thiazolidine and oxaxoliding derivatives, their prepn. and their medical use
04/2001
04/19/2001WO2000018767A9 2-piperazino alkylamino benzoazole derivatives: dopamine receptor subtype specific ligands
04/17/2001US6218431 Substituted biphenyls
04/17/2001CA2080475C Neuroprotective indolone and related derivatives
04/10/2001US6214825 Aza-heterocycloakenes, pesticidal compositions containing them, pesticidal methods of using them, and processes for preparing them
04/05/2001WO2001022919A2 Spiro[bicyclic -azacycloalkyl and -cycloalkyl] derivatives and uses thereof
03/2001
03/27/2001US6207680 Heteroarylpiperidines and their use as antipsychotics and analgesics
02/2001
02/21/2001EP0835248B1 1-amino-3-benzyluracils
02/15/2001DE19936520A1 New benzoylpyrazolyl derivatives useful as pre- and post-emergent herbicides for protection of crops and application to non-agricultural surfaces
02/14/2001EP0714897B1 Fused heteroaromatic cyclopentene derivative having endothelin-antagonist activity
01/2001
01/31/2001CN1061339C Novel sulfonamide inhibitors of aspartyl protease
01/23/2001USRE37029 Antipsychotic and analgesic agents
01/16/2001US6175012 Processes and intermediates for the preparation of piperazine derivatives
01/10/2001CN1279674A 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analoguse), their preparation and their use in the treatment of neurological disorders
01/10/2001CN1279673A ((Cyclo) alkyl substituted-.gamma.-aminobutyric acid derivatives (=GABA analogurs), their preparation and their use in the treatment of neurolog disorders
01/10/2001CN1279667A 4(3)-substituted-4(3)-aminonethyl-(thioxo)pyran(thiapyran)or-piperidine derivatives(=gabapendin analogues), their preparation and their use in treatment of neurological disorders
12/2000
12/26/2000US6165944 4-(3-heterocyclyl-1-benzoyl) pyrazoles and their use as herbicides
12/13/2000CN1276370A Process for preparing anticancer compound, and intermediate
12/13/2000CN1059440C Wood preservative oxathiazines
11/2000
11/15/2000EP1052255A1 Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics.
11/02/2000EP1047678A1 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
10/2000
10/31/2000US6140345 For treating psychoses and pain
10/25/2000EP1045839A2 Novel amines as pharmaceutical agents
10/25/2000EP1045834A1 4(3)substituted-4(3)-aminomethyl-(thio)pyran or -piperidine derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
10/18/2000EP1044969A2 Processes and intermediates for preparing anti-cancer compounds
10/17/2000US6133449 Processes and intermediates for the preparation of piperazine derivatives
09/2000
09/20/2000EP0705816B1 Benzene derivative useful for ischemic diseases
09/06/2000CN1056144C New use of 6-heterocyclic-4-amino-3,4,5-tetrahydrobenz (CD) indoles compound
08/2000
08/29/2000US6110938 1-(arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-4-(heteroaryl)piperidines and related compounds useful as antipsychotics and analgesics
08/23/2000CN1055686C Substituted benzisoxazole and benzisothaazole herbicidal agents
08/15/2000US6103910 D-proline derivatives
08/08/2000US6100252 Specified compounds including methyl 2-butyl-1-((2'-(2-oxo-3h-1,2,3,5-oxathiadiazol-4-yl)biphenyl) methyl)-benzimidazole-7-carboxylate; use to treat circulatory diseases such as hypertensive diseases and heart diseases
07/2000
07/27/2000WO2000018767A3 2-piperazino alkylamino benzoazole derivatives: dopamine receptor subtype specific ligands
06/2000
06/08/2000WO2000032371A1 Wood preservative formulations
06/08/2000CA2352052A1 Wood preservative formulations
06/07/2000CN1255496A Application of heterobicyclic alcohol antimer for preparing piperazine derivative
05/2000
05/30/2000US6069160 Heteroatom-containing benzocyclopentane-oxazolidinones
05/23/2000US6066650 Inhibitors of microsomal triglyceride transfer protein and method
05/17/2000EP1000621A2 Use of 6-heterocyclic-4-amino-1,3,4,5-tetrahydrobenz (CD) indoles for treating motion sickness and vomiting
05/10/2000CN1052231C 2-oxo-5-oxazolidone methyl compound their preparing method and medicinal composition containing them
04/2000
04/26/2000EP0554247B1 Neuroprotective indolone and related derivatives
04/12/2000CN1250447A 4-(3-heterocyclyl-1-benzoyl) pyrazoles and their use as herbicides
04/06/2000WO2000018767A2 2-piperazino alkylamino benzoazole derivatives: dopamine receptor subtype specific ligands
04/06/2000CA2345944A1 2-piperazino alkylamino benzoazole derivatives: dopamine receptor subtype specific ligands
03/2000
03/28/2000US6043240 Useful as antipsychotic and analgesic agents
03/22/2000CN1248255A 3-heterocyclyl-substituted benzoyl derivatives
03/22/2000CN1050603C Prepn. of intermediate product used in process for diastereoselective synthesis of nucleosides
03/07/2000US6034098 Inhibitors of microsomal triglyceride transfer protein and method
03/01/2000EP0981521A2 Novel macrocyclic compounds as metalloprotease inhibitors
02/2000
02/09/2000CN1049219C Fused heteroaromatic cyclopentene derivative having endothelin-antagonist activity
02/08/2000US6022967 Heterocyclic compounds
01/2000
01/06/2000WO1999057116A3 Pesticidal methoximinomethyloxathiazines
12/1999
12/28/1999US6008245 Treatment of prophylaxis and cardiovascular disorders, in particular arrhythmias, for the treatment of ulcers of the gastrointestinal disorders, diarrheal diseases
12/22/1999CN1239474A Substituted pyridines and biphenyls as anti-hypercholesterinemic, anti-hyperlipoproteinemic and anti-hyperglycemic agents
12/15/1999EP0963984A1 Heteroarylpiperidines and piperazines and their use as antipsychotics and analgetics
12/14/1999US6001834 [(4-heteroaryl-1-piperazinyl)alkoxy]-3,4-dihydro-1(2h)-naphthalenones and related compounds and their therapeutic utility
12/07/1999US5998452 Benzene derivatives, compositions and methods for treating ischemic diseases
12/07/1999US5998417 N-[(4-heteroaryl-1-piperazinyl) alkyl]phthalimides and related compounds and their therapeutic utility
11/1999
11/24/1999EP0959076A1 Heteroarylperidines and piperazines and their use as antipsychotics and analgetics
11/24/1999EP0959075A1 Heteroarylpiperidines and piperazines and their use as antipsychotics and analgetics
11/24/1999EP0958292A1 4-(3-heterocyclyl-1-benzoyl)pyrazoles and their use as herbicides
11/24/1999EP0958291A1 3-heterocyclyl-substituted benzoyl derivatives
11/17/1999EP0957102A1 Heteroarylpiperidines and piperazines and their use as antipsychotics and analgetics
11/11/1999WO1999057116A2 Pesticidal methoximinomethyloxathiazines
11/11/1999WO1998004528A3 Substituted pyridines and biphenyls as anti-hypercholesterinemic, anti-hyperlipoproteinemic and anti-hyperglycemic agents
11/11/1999DE19819828A1 Methoximinomethyloxathiazine Methoximinomethyloxathiazine
11/04/1999WO1999031074A3 ((cyclo)alkyl substituted)-.gamma.-aminobutyric acid derivatives (=gaba analogues), their preparation and their use in the treatment of neurological disorders
11/02/1999US5977140 N-[(4-Heteroaryl-1-Piperidinyl)Alkly] Phthalimides and related compounds and their therapeutic utility
11/02/1999US5977113 4-heteroaryl-1-piperazine alkylamines and their therapeutic utility
10/1999
10/13/1999CN1231664A Sulfonamicles and derivatives thereof that moulate the activity of endothelin
10/12/1999US5965546 1-[(2-pyrimidinyloxy)alkyl]4-(heteroaryl)piperazines and related compounds and their therapeutic utility
10/06/1999EP0946552A1 Sulfonamides and derivatives thereof that modulate the activity of endothelin
10/05/1999US5962490 Thienyl-, furyl- and pyrrolyl-sulfonamides and derivatives thereof that modulate the activity of endothelin
09/1999
09/29/1999CN1230196A Modified aminoacids, pharmaceuticals containing these compounds and method for their prodn.
09/22/1999CN1229080A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/22/1999CN1229079A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/22/1999CN1229078A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/01/1999EP0939135A1 Substantially pure hetero-bicyclic alcohol enantiomers
08/1999
08/11/1999EP0934274A1 Substituted pyridines and biphenyls as anti-hypercholesterinemic, anti-hyperlipoproteinemic and anti-hyperglycemic agents
07/1999
07/13/1999US5922113 Antibacterial and antifouling oxathiazines and their oxides
07/07/1999EP0927192A1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production
07/06/1999US5919798 4-heteroaryl-1-piperidinealkanols and derivatives thereof and their therapeutic utility
06/1999
06/24/1999WO1999031075A1 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
06/24/1999WO1999031074A2 ((cyclo)alkyl substituted)-.gamma.-aminobutyric acid derivatives (=gaba analogues), their preparation and their use in the treatment of neurological disorders
06/24/1999WO1999031057A1 4(3)substituted-4(3)-aminomethyl-(thio)pyran or -piperidine derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
06/23/1999CN1043786C Method for preparing antibiotic compound
06/22/1999US5914263 Enzymatic process for the stereoselective preparation of a hetero-bicyclic alcohol enantiomer
06/09/1999CN1219172A Novel benzo-1,3-dioxolyl- and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists
06/02/1999CN1218050A Sulfonamide-substituted benzopyran derivates processes for their preparation, their use as medicament, and pharmaceutical preparations comprising them
05/1999
05/26/1999CN1217327A D-proline derivative
05/12/1999EP0915088A1 D-Proline derivatives
05/06/1999EP0913396A2 Sulphonamide substituted benzopyran derivatives, process of preparation, their use as medicines and pharmaceutical compositions containing them
05/03/1999CA2252733A1 Sulfonamide-substituted benzopyran derivatives, processes for their preparation, their use as a medicament, and pharmaceutical preparations comprising them
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15