Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
12/2000
12/14/2000WO2000075136A1 Aminoalkyl substituted (benzodioxan, benzofuran or benzopyran) derivatives
12/14/2000WO2000075120A1 Diaminothiazoles and their use for inhibiting protein kinases
12/14/2000WO2000075119A2 Substituted 2-aryl-1,2,4-triazine-3,5-di(thi)ones used as herbicides
12/14/2000WO2000075111A1 Formazan metal complex
12/14/2000WO2000074681A1 Metalloprotease inhibitors
12/14/2000WO2000074679A1 Substituted piperidines as melanocortin-4 receptor agonists
12/14/2000WO2000047568A3 1,2-benzothiazepines for the treatment of hyperlipidemic diseases
12/14/2000WO2000046187A3 Antizyme modulators and their use
12/14/2000WO2000029378A3 Acyclic and cyclic guanidine- and acetamidine derivatives, their preparation and their use as pesticides, esp. as parasiticides
12/14/2000DE19926620A1 Neue Cycloiminodepsipeptide, Verfahren zu ihrer Herstellung und ihre Verwendung zur Bekämpfung von Endoparasiten New Cycloiminodepsipeptide, processes for their preparation and their use for controlling endoparasites
12/14/2000CA2377369A1 Substituted piperidines as melanocortin-4 receptor agonists
12/14/2000CA2375942A1 Substituted 2-aryl-1,2,4-triazine-3,5-di(thi)ones
12/14/2000CA2375882A1 Metalloprotease inhibitors
12/14/2000CA2375740A1 Ph sensitive cyanine dyes as reactive fluorescent reagents
12/14/2000CA2375734A1 Benzothiazinone and benzoxazinone compounds
12/14/2000CA2371158A1 Diaminothiazoles and their use for inhibiting protein kinases
12/13/2000EP1058690A1 Thiadiazole compounds useful as inhibitors of cysteine activity dependent enzymes
12/13/2000EP1058684A1 Glycine transport inhibitors
12/13/2000EP1058683A1 Farnesyl transferase inhibitors having a piperidine structure and process for preparation thereof
12/13/2000EP1058679A1 Synthesis of epothilones, intermediates thereto and analogues therof
12/13/2000EP1058549A1 THROMBIN OR FACTOR Xa INHIBITORS
12/13/2000EP0874834B1 Processes and intermediates for preparing 3-(1-piperazinyl)-1,2-benzisothiazole
12/13/2000CN1276790A Carboxamidothiazole derivs., preparation, pharmaceutical composition contg. them
12/13/2000CN1276789A 4-aminothiazole derivs, their preparation and their use as inhibitors of cyclin-dependent kinases
12/13/2000CN1276373A Oxa(thia)diazolylpyridazinone derivative and its preparing process and application
12/13/2000CN1276370A Process for preparing anticancer compound, and intermediate
12/13/2000CN1276211A Use of non-peptides NK3-antagonist
12/13/2000CN1059442C Use of 1,2-bridged 1,4-dihydropyridines as medicaments
12/13/2000CN1059439C Arylthiadiazolones with herbicidal activity
12/12/2000US6160121 Pyridyl-thiazoles and their use to protect plants against infections by micro-organisms
12/12/2000US6160024 Photoactivated antiviral and antitumor compositions
12/12/2000US6160001 Halobenzimidazoles and their use as microbicides
12/12/2000US6159998 Administered as vasodilators, analgesics, anesthetics, sedatives, and anitspasmodic agents
12/12/2000US6159996 Polycyclic thiazolidin-2-ylidene amines, process for their preparation, and their use as pharmaceuticals
12/12/2000US6159994 Imidazole derivatives; antiallergens, antihistamines, antiasthmatic agents
12/12/2000US6159983 Method and composition for treatment of inflammatory bowel disease
12/12/2000US6159976 Polymorph of zopolrestat monohydrate
12/12/2000US6159967 such as 1-(2-((2R)-(3,4-dichlorophenyl)-4-(3,4,5-trimethoxybenzoyl) morpholin-2-yl)ethyl)spiro(benzo(c)thiophene-1-(3H), 4'-piperidine)-(2S)-oxide; respiratory disease such as asthma
12/12/2000US6159966 Azolidinediones useful for the treatment of diabetes, dyslipidemia and hypertension: process for their preparation and pharmaceutical compositions containing them
12/12/2000US6159938 Serine protease inhibitors comprising α-keto heterocycles
12/07/2000WO2000073290A1 Isothiazolecarboxamides and their use as microbicides
12/07/2000WO2000073284A2 1,4-benzodiazepin-2-ones useful as hiv reverse transcriptase inhibitors
12/07/2000WO2000072815A1 Indole derivatives
12/07/2000WO2000031247A3 Recombinant methods and materials for producing epothilone and epothilone derivatives
12/07/2000WO2000009104A3 Use of sulfonamides for treating vision and memory disorders
12/07/2000DE19925593A1 Substituierte 2-Aryl-1,2,4-triazin-3,5-di(thi)one Substituted 2-aryl-1,2,4-triazine-3,5-di (thi) ones
12/07/2000CA2370141A1 1,4-benzodiazepin-2-ones useful as hiv reverse transcriptase inhibitors
12/06/2000EP1057819A1 Phthalazine derivatives and remedies for erectile dysfunction
12/06/2000EP1057812A1 Aminoguanidine hydrazone derivatives, process for producing the same and drugs thereof
12/06/2000EP1056743A1 Benzamine derivatives
12/06/2000EP1056732A2 4-aminothiazole derivatives, their preparation and their use as inhibitors of cyclin-dependent kinases
12/06/2000EP1056729A1 N-[(substituted five-membered di- or triaza diunsaturated ring)carbonyl]guanidine derivatives for the treatment of ischemia
12/06/2000EP1056724A2 Substituted cycloalkyl-4-oxonicotinic carboxamides; gaba brain receptor ligands
12/06/2000EP1056719A2 Inhibitors of phospholipase enzymes
12/06/2000EP0597088B1 Novel imidazole derivatives, their preparation and therapeutic applications
12/06/2000CN1275982A Novel heterocyclic compounds process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
12/06/2000CN1275912A Novel amide derivatives
12/06/2000CN1059210C Process for preparation of 6-heterocyclic-4-amino-1,3,4,5-tetrahydrbenz [cd] indoles and acid additive salt used as medicine
12/05/2000US6156898 Substituted 1,4-dihydro-4-oxonicotinic carboxamides; GABA brain receptor ligands
12/05/2000US6156787 Substituted thienlycyclohexanone derivatives for enhancing cognition
12/05/2000US6156784 Ester, acid or derivatives of amides, sulfonamides or thioamides
12/05/2000US6156782 Parasiticidal compounds
12/05/2000US6156766 Heterocyclic benzamides as drugs
12/05/2000US6156761 Substituted tetralone derivatives for enhancing cognition
12/05/2000US6156748 Compounds useful as neuro-protective agents
12/05/2000US6156746 1,2,5-benzothiadiazepine-1,1-dioxides with n-2 imidazolylalkyl substituents
12/05/2000US6156702 As herbicides
11/2000
11/30/2000WO2000071572A1 Substituted beta-alanine derivatives as cell adhesion inhibitors
11/30/2000WO2000071540A1 Hydrochloride of fused-heterocycle compound
11/30/2000WO2000071536A1 Heteroaryloxypyrimidine insecticides and acaricides
11/30/2000WO2000071535A1 INDOLE-TYPE DERIVATIVES AS INHIBITORS OF p38 KINASE
11/30/2000WO2000071532A1 Heterocyclic derivatives useful as anticancer agents
11/30/2000WO2000071528A1 4h-1,4-benzothiazine-2-carboxamides and their use as gaba brain receptor ligands
11/30/2000WO2000071521A1 A process for the reduction of oxiranyl epothilones to olefinic epothilones
11/30/2000WO2000071517A1 Phenoxypropylamine compounds
11/30/2000WO2000071132A1 Use of 1,4-benzothiazepine derivatives as drugs overcoming carcinostatic tolerance
11/30/2000WO2000046199A3 Indole derivatives as anti-inflammation agents
11/30/2000WO2000043535A3 Composition and device for detecting leukocytes in urine
11/30/2000WO2000032598A9 Methods and compositions for treating inflammatory diseases utilizing inhibitors of tumor necrosis factor activity
11/30/2000CA2716369A1 Phenoxypropylamine compounds
11/30/2000CA2375029A1 A process for the reduction of oxiranyl epothilones to olefinic epothilones
11/30/2000CA2372567A1 Indole-type derivatives as inhibitors of p38 kinase
11/29/2000EP1054886A1 Heteroaryl amidines, methylamidines and guanidines as protease inhibitors, in particular as urokinase inhibitors
11/29/2000EP1054884A1 Benzofuran-4-carboxamides and their therapeutic use
11/29/2000EP1054882A1 Condensed heterocyclic system derivatives, preparation, pharmaceutical compositions containing them
11/29/2000EP1054877A1 Novel cyclic sulfonamide derivatives as metalloproteinase inhibitors
11/29/2000EP1054876A1 1,3,4-thiadiazoles derivatives as kyn-oh inhibitors
11/29/2000EP1054874A1 Substituted aminophenyl isoxazoline derivatives useful as antimicrobials
11/29/2000EP1054865A1 Farnesyl transferase inhibitors
11/29/2000EP0702727B1 Dyes designed for high sensitivity detection of double-stranded dna
11/29/2000EP0655055B1 Tachykinin antagonists
11/29/2000CN1275124A Phthalazine derivatives and remedies for erectile dysfunction
11/29/2000CN1275123A Prostaglandin agonists and their use to treat bone disorders
11/29/2000CN1058964C Branched-amino-sbustituted thiazoles, process for their preparation and the pharmaceutical compositions which contain them
11/28/2000US6153763 A microbicides comprising an imidazole ring
11/28/2000US6153761 An intermediates for preparing herbicides and/or fungicides
11/28/2000US6153759 Herbicide comprising a 5-membered or 6-membered heterocyclic, saturated or unsaturated radical containing one to three hetero atoms selected from the group consisting of oxygen, sulfur and nitrogen
11/28/2000US6153757 Metalloproteinase inhibitors and intermediates useful for their preparation
11/28/2000US6153642 Useful as antineoplastic and antiviral agents
11/28/2000US6153628 1,3,4-thiadiazoles and 1,3,4-Oxadiazoles as αv β3 antagonists