Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
06/2000
06/13/2000CA2014062C Pyridine derivatives
06/08/2000WO2000032606A1 IMIDAZO[4,5-b]PYRIDINIUMMETHYL-CONTAINING CEPHEM COMPOUNDS HAVING BROAD ANTIBACTERIAL SPECTRUM
06/08/2000WO2000032599A1 Oxazolidinone antibacterial agents having a thiocarbonyl functionality
06/08/2000WO2000032598A1 Methods and compositions for treating inflammatory diseases utilizing inhibitors of tumor necrosis factor activity
06/08/2000WO2000032588A2 Carboxylic acids and carboxylic acid isosteres of n-heterocyclic compounds
06/08/2000WO2000032586A1 Method for preparing 3-chromene derivatives, use of said derivatives for preparing thiazolidinones
06/08/2000WO2000032577A2 Substituted benzo[de]isoquinoline-1,3-diones
06/08/2000WO2000032575A1 β-ALANINE DERIVATIVES AS α4 INTEGRIN INHIBITORS
06/08/2000WO2000032216A1 Peptoid and nonpeptoid containing alpha-keto oxadiazoles as serine protease inhibitors
06/08/2000WO2000032190A1 Compositions and methods for the treatment of alzheimer's disease, central nervous system injury, and inflammatory diseases
06/08/2000WO2000032180A2 Antihypertriglyceridemic, antihyperglycemic, anti-angiogenic and wound healing substituted indolealkanoic acids
06/08/2000WO2000032175A2 METHODS AND COMPOSITIONS FOR RESTORING CONFORMATIONAL STABILITY OF A PROTEIN OF THE p53 FAMILY
06/08/2000WO2000009103A9 N-linked sulfonamides of n-heterocyclic carboxylic acids or isosteres for vision and memory disorders
06/08/2000CA2385845A1 Methods of reducing serum glucose and triglyceride levels and for inhibiting angiogenesis using substituted indolealkanoic acids
06/08/2000CA2352045A1 Substituted benzo[de]isoquinoline-1,3-diones
06/08/2000CA2351062A1 Oxazolidinone antibacterial agents having a thiocarbonyl functionality
06/08/2000CA2350597A1 Methods and compositions for restoring conformational stability of a protein of the p53 family
06/08/2000CA2347701A1 .beta.-alanine derivatives as .alpha.4 integrin inhibitors
06/08/2000CA2291506A1 Process for the preparation of dithiazolyl disulfides
06/07/2000EP1006114A1 Pyrazole derivatives and cox inhibitors containing them
06/07/2000EP1005465A2 New epothilone derivatives, method for producing same and their pharmaceutical use
06/07/2000EP1005456A1 Method for producing organic compounds
06/07/2000EP1005455A1 Method for producing substituted-2-nitroguanidine derivatives
06/07/2000EP1005454A1 2-acylaminopropanamines as tachykinin receptor antagonists
06/07/2000EP0855909A4 Radiosensitizing taxanes and their pharmaceutical preparations
06/06/2000US6071948 Treatment of diseases caused by excessive blood vessel growth
06/06/2000US6071921 4-phenyl-7-arylquinoazolines; angiogenisis inhibitors and/or vascular permeability reducing effects in warm-blooded animals; anticarcinogenic and -arthritic agents; rheumatic diseases; vascular endothelium growth factor inhibitors
06/06/2000US6071908 Radiation-activated cytotoxin therapy of neoplastic disease
06/06/2000US6071860 For selective control of broad-leaved and grass weeds in crops of useful plants
06/02/2000WO2000031247A2 Recombinant methods and materials for producing epothilone and epothilone derivatives
06/02/2000WO2000031074A2 Indole derivatives and their use as serotonin receptor ligands
06/02/2000WO2000031072A1 Process for making 5-substituted pyrazoles using dithietanes
06/02/2000WO2000031063A1 SUBSTITUTED PYRAZOLES AS p38 KINASE INHIBITORS
06/02/2000WO2000031054A1 Il-5 inhibiting 6-azauracil derivatives
06/02/2000WO2000031053A1 Il-5 inhibiting 6-azauracil derivatives
06/02/2000WO2000031037A1 Quinoline-4-carboxamide derivatives as nk-3 and nk-2 receptor antagonists
06/02/2000WO2000030639A1 Use of n-substituted azabicycloalkane derivatives for treating diseases of the central nervous system
06/02/2000CA2352526A1 Use of n-substituted azabicycloalkane derivatives for treating diseases of the central nervous system
06/02/2000CA2351865A1 Quinoline-4-carboxamide derivatives as nk-3 and nk-2 receptor antagonists
06/02/2000CA2351725A1 Substituted pyrazoles as p38 kinase inhibitors
06/02/2000CA2351526A1 Indole derivatives and their use as serotonin receptor ligands
06/02/2000CA2350189A1 Recombinant methods and materials for producing epothilone and epothilone derivatives
06/02/2000CA2350081A1 Process for making 5-substituted pyrazoles using dithietanes
05/2000
05/31/2000EP1003740A2 Pyrrolidine-3-carboxylic acid derivatives and their use as endothelin antagoists
05/31/2000EP1003739A2 2-(4-aryl or heteroaryl-piperazin-1-ylmethyl)-1h-indole derivatives
05/31/2000EP1003737A1 Phenyl urea and phenyl thiourea derivatives as hfgan72 antagonists
05/31/2000EP1003736A1 Substituted 4-benzoyl-pyrazoles
05/31/2000EP1003729A1 6-azauracil derivatives as il-5 inhibitors
05/31/2000EP1003723A1 2-acylaminopropanamines as tachykinin receptor antagonists
05/31/2000EP1003721A1 Benzylidene-1,3-dihydro-indol-2-one derivatives as receptor tyrosine kinase inhibitors, particularly of raf kinases
05/31/2000EP1003540A1 $g(b)2-ADRENERGIC RECEPTOR AGONISTS
05/31/2000EP1003512A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
05/31/2000EP1003511A1 ALPHA 1aADRENERGIC RECEPTOR ANTAGONISTS
05/31/2000EP1003509A1 Il-8 receptor antagonists
05/31/2000EP0820448B1 Novel taxoids, preparation thereof, and pharmaceutical compositions containing same
05/31/2000CN1255162A Protease inhibitors
05/31/2000CN1255136A Substituted 4-arylmethylene-2-imino-2,3-dihydrothiazoles and derivatives and their pharmaceutical use
05/31/2000CN1255124A Substituted isoquinoline derivatives and their use as anticonulsants
05/31/2000CN1255119A Protease inhibitors
05/31/2000CN1255042A Diaryl ethers and processes for their preparation and herbicidal and desiccant compositions containing them
05/31/2000CN1254596A Process for preparing composition to kill internal parasites
05/31/2000CN1052984C New erythromycin derivative and its preparing process and application in medicine
05/30/2000US6069162 Indolyl and benzofuranyl carboxamides as inhibitors of nitric oxide production
05/30/2000US6069160 Heteroatom-containing benzocyclopentane-oxazolidinones
05/30/2000US6069157 Parasiticidal compounds
05/30/2000US6069156 Indole derivatives as cGMP-PDE inhibitors
05/30/2000US6069141 Substituted aminophenyl isoxazoline derivatives useful as antimicrobials
05/25/2000WO2000029410A1 Thiazolone derivatives having fused polycyclic heterocycle at the 2-position and pesticides containing the same as the active ingredient
05/25/2000WO2000029409A1 Novel heterocyclyl-substituted oxazolidone derivatives
05/25/2000WO2000029406A2 Novel isoxazoline fibrinogen receptor antagonists
05/25/2000WO2000029399A1 Antiherpes compounds
05/25/2000WO2000029398A1 Isothiazolecarboxylic acid derivatives
05/25/2000WO2000029397A1 New piperazine and piperidine compounds
05/25/2000WO2000029396A1 Novel substituted phenyloxazolidone derivatives
05/25/2000WO2000029378A2 Acyclic and cyclic guanidine- and acetamidine derivatives, their preparation and their use as pesticides, esp. as parasiticides
05/25/2000WO2000028822A2 Herbicidal 3-(benzo(ox/thi)azol-7-yl)-1h-pyrimidine-2,4-diones
05/25/2000DE19854147A1 Control of cocaine addiction comprises administration of N-substituted azabicycloalkane derivative
05/25/2000CA2351564A1 Herbicidal 3-(benzo(ox/thi)azol-7-yl)-1h-pyrimidine-2,4-diones
05/25/2000CA2350742A1 Acyclic and cyclic guanidine- and acetamidine derivatives, their preparation and their use as pesticides, esp. as parasiticides
05/25/2000CA2345210A1 Novel isoxazoline fibrinogen receptor antagonists
05/24/2000EP1001973A1 Compounds which inhibit leukocyte adhesion mediated by vla-4
05/24/2000EP1001951A1 Thiazole derivatives, method for their production and use
05/24/2000EP1001939A1 Heterocyclic substituted 4-benzoyl-pyrazole as herbicides
05/24/2000EP1001934A1 Indole compounds as cox-2 inhibitors
05/24/2000EP1001933A1 Caspases and apoptosis
05/24/2000EP1001927A2 Novel polyamine analogues as therapeutic and diagnostic agents
05/24/2000EP0793674B1 Human neutrophil elastase inhibitors
05/24/2000CN1254337A N-hydroxy 4-sulfonyl butyramide compounds
05/24/2000CN1254335A Nicotinamide derivatives
05/23/2000US6066740 From thiourea intermediate; for treatment of respiratory disorders, ocular disorders, gastrointestinal disorders, nasal decongestion, hypertension, migraine, disorders associated with sympathetic nervous system activity, and substance abuse
05/23/2000US6066657 For the treatment of disease states associated with proteins which mediate cellular activity, for example by inhibiting tumor necrosis factor or phosphodiesterase iv
05/23/2000US6066650 Inhibitors of microsomal triglyceride transfer protein and method
05/23/2000US6066443 Provides good speed and improved color reproduction; maximum blue sensitivity at less than 485 nm.
05/23/2000CA2010578C Piperidine compounds and their preparation and use
05/18/2000WO2000027842A1 Compounds
05/18/2000WO2000027832A2 Thiazole derivatives as ppar gamma ligands
05/18/2000WO2000027830A1 Thiocarbamic acid derivatives
05/18/2000WO2000027822A2 Tricyclic pyrazole derivatives
05/18/2000WO2000027819A2 Antrhranilic acid amides and the use thereof as medicaments
05/18/2000WO2000027812A1 Phenyl-substituted cyclic enaminones