Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
01/2001
01/03/2001CN1278818A Process for preparation of thiazolidinedione derivatives
01/03/2001CN1278806A Aminothiazole inhibitors of cyclin dependent protein kinasses of cells
01/03/2001CN1278805A Novel heterocyclioally substituted and a-hydroxycarboxlic acid derivatives, method for producing the same and their use as endothelin receptor antagonists
01/03/2001CN1278804A Isothiazolcarboxylic acid derivatives
01/03/2001CN1278794A Substituted di-hydroxyl-indol derivatives as protein tyrosine kinase and as protein serine/threenine kinase inhibitors
01/03/2001CN1278790A Chemical compound
01/03/2001CN1278726A IL-8 receptor antagonists
01/03/2001CN1060173C Heterocyclic compound with activity against diabetes and preparation nad application of same
01/03/2001CN1060171C Substituted biphenyl isoxazole sulfonamides
01/02/2001US6169188 Treating cyclooxygenase-2 mediated diseases
01/02/2001US6169181 Compounds useful to treat retroviral infections
01/02/2001US6169097 1-(1,2-Disubstituted piperidinyl)-4-substituted piperidine derivatives
01/02/2001US6169088 1,3 diazines with platelet-derived growth factor receptor inhibitory activity
01/02/2001US6169086 Pyrazole derivatives
01/02/2001CA2161662C Process for preparing intermediates for the synthesis of antifungal agent
01/02/2001CA2068064C Fibrinogen receptor antagonists
01/02/2001CA1341162C Sbustituted aminomethyltetralins and their heterocyclic analogues
12/2000
12/28/2000WO2000078758A1 Novel imidazole derivatives
12/28/2000WO2000078757A1 Inhibitors of il-12 production
12/28/2000WO2000078756A1 Thiophene-ethyl thiourea compounds and their use in the treatment of hiv
12/28/2000WO2000078755A1 Thiophene-ethyl thiourea compounds and use in the treatment of hiv
12/28/2000WO2000078747A1 Acylhydrazine derivatives, process for preparing the same and use thereof
12/28/2000WO2000078746A1 Antiviral agents
12/28/2000WO2000078312A1 Arylthiazolidinedione and aryloxazolidinedione derivatives
12/28/2000WO2000061551A3 Pyrimidine-2-one derivatives as integrin receptor ligands
12/28/2000WO2000049021A3 16-halogen-epothilone derivatives, method for producing them and their pharmaceutical use
12/28/2000WO2000049020A3 Novel epothilon derivatives, method for the production thereof and their pharmaceutical application
12/28/2000WO2000047584A3 Epothilon derivatives, method for the production and the use thereof as pharmaceuticals
12/28/2000WO2000043373A3 Kinase inhibitors
12/28/2000WO1999052493A3 Compounds that inhibit the binding of integrins to their receptors
12/28/2000CA2383492A1 Acylhydrazine derivatives, their production and use
12/28/2000CA2375261A1 Thiophene-ethyl thiourea compounds and use in the treatment of hiv
12/28/2000CA2375211A1 Antiviral agents
12/27/2000EP1063235A1 Benzofurylpyrone derivatives
12/27/2000EP1062216A1 Inhibitors of phospholipase a2
12/27/2000EP1062212A1 Heterocyclyl anthracyclinone derivatives
12/27/2000EP1062205A2 Inhibitors of phospholipase enzymes
12/27/2000EP1061921A1 Vitronectin receptor antagonists
12/27/2000EP0821671B1 Arylsulfonyl hydroxamic acid derivatives as mmp and tnf inhibitors
12/27/2000CN1278175A Compositions of lipid lowering agents
12/27/2000CN1277965A Luogelie ketone hydrochloride and its use
12/26/2000US6166222 Reacting a pyrrolecarboxylic acid derivative in ammonia with an alkali metal or alkaline earth metal and then an aqueos salt solution of a alkyl- or silyl-leaving group compound
12/26/2000US6166219 Treatment of diabetes and related disorders
12/26/2000US6166216 Compounds useful as neuro-protective agents
12/26/2000US6166056 Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings
12/26/2000US6166054 A 1,2,3-thiadiazole derivative for treating plant diseases
12/26/2000US6166041 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma
12/26/2000US6166033 Drugs for preventing and treating dopamine d receptor-related morbid states such as schizophrenia and problematic behavior caused by cerebrovascular accidents and senile dementia and do not induce extrapyramidal disorders as side effects
12/26/2000US6166028 Diaminopuridine-containing thiourea inhibitors of herpes viruses
12/26/2000US6166027 Treatment of high blood pressure and cardiac insufficiency, angina pectoris, arrhythmias, thromboembolic diseases, ischaemias, myocardial infarction, cerebral stroke, restenoses, coronary angioplasties, arteriosclerosis
12/26/2000US6166023 1,5- and 3-O-substituted 1H-indazoles having anti-asthmatic, anti-allergic, anti-inflammatory, immunomodulating and neuroprotective action, process for their preparation and their use as medicaments
12/26/2000US6166020 Aryl and heteroaryl alkoxynaphthalene derivatives
12/26/2000US6166005 Heterocyclic metalloprotease inhibitors
12/26/2000US6165944 4-(3-heterocyclyl-1-benzoyl) pyrazoles and their use as herbicides
12/26/2000US6165943 Herbicides
12/26/2000US6165941 Substituted 2-phenylpyridines
12/21/2000WO2000077027A2 Serine protease inhibitors
12/21/2000WO2000076995A1 Process for the preparation of (-)-1,4-benzothiazine-2-acetic acid derivatives
12/21/2000WO2000076988A1 Rhodanine derivatives and their use in inhibiting and imaging amyloids
12/21/2000WO2000076987A1 Rhodanine derivatives for use in a method of inhibiting amyloid protein aggregation and imaging amyloid deposits
12/21/2000WO2000076985A1 Cyclo-imino depsipeptides and their utilization in controlling endoparasites
12/21/2000WO2000076984A2 Novel compounds, their use and preparation
12/21/2000WO2000076972A1 N-cyclopentyl modulators of chemokine receptor activity
12/21/2000WO2000076971A2 Serine protease inhibitors
12/21/2000WO2000076970A2 Serine protease inhibitors
12/21/2000WO2000076521A1 Antiviral indoleoxoacetyl piperazine derivatives
12/21/2000WO2000076514A1 Cyclopentyl modulators of chemokine receptor activity
12/21/2000WO2000076489A2 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits
12/21/2000CA2383008A1 Compounds
12/21/2000CA2375920A1 Compounds
12/21/2000CA2375551A1 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits
12/21/2000CA2374632A1 Cyclo-imino depsipeptides and their utilization in controlling endoparasites
12/21/2000CA2374616A1 Rhodanine derivatives for use in a method of inhibiting amyloid protein aggregation and imaging amyloid deposits
12/21/2000CA2370316A1 Rhodanine derivatives and their use in inhibiting and imaging amyloids
12/21/2000CA2340663A1 Antiviral indoleoxoacetyl piperazine derivatives
12/20/2000EP1061074A1 Novel process and intermediates
12/20/2000EP1061072A1 Pyrrolic compounds with a high herbicidal activity and their agronomic use
12/20/2000EP1060178A1 Heterocyclic compounds as inhibitors of rotamase enzymes
12/20/2000EP1060166A1 Five-membered, benzo-condensed heterocycles used as antithrombotic agents
12/20/2000EP1060163A1 New piperazinyl-substituted pyridylalkane, alkene and alkine carboxamides
12/20/2000EP0751944B1 Thiazolidines and oxazolidines substituted by a pyridine ring and their use as hypoglycemic agents
12/20/2000CN1277610A Process for preparation of 2-aminothiazolecarboxamide derivatives
12/20/2000CN1277607A 2-substituted 1,2-benzisothiazole derivatives and their use as serotonin antagonists (5-HT1A, 5-HT1b and 5-HT1D)
12/20/2000CN1277605A Arylpyridazinones as prostaglandin endoperoxide H synthase biosynthesis inhibitors
12/20/2000CN1277604A Heteraryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors
12/20/2000CN1059674C Hypolipidemic benzothiazepines
12/20/2000CN1059673C Hypolipidemic 1,4-benzothiazepine-1,1-dioxides
12/19/2000US6162927 (2s,3r,4s)-2-(2,2-dimethylpentyl)-4-(7-methoxy-1,3-benzodioxol-5-yl)-1-(n,n-di(n-butyl)aminocarbonylmethyl)-pyrrolidine-3-carboxylic acid, or salt or ester thereof, in pure form; adminstering to treat hypertension, other diseases
12/19/2000US6162819 Pyrazole derivatives, their preparation and their use in pharmaceuticals
12/19/2000US6162812 Pharmaceutical compositions containing HIV protease inhibitors and methods of their use
12/19/2000US6162809 Pyridylthio compounds for controlling helicobacter bacteria
12/19/2000US6162808 Compounds
12/19/2000US6162804 Tyrosine kinase inhibitors
12/19/2000US6162791 Thiadiazole compounds useful as inhibitors of cysteine activity dependent enzymes
12/19/2000CA2001225C Antimicrobial lactam-quinolones
12/18/2000CA2311872A1 Processes and intermediates for preparing (indole-2-carbonyl)-amides
12/14/2000WO2000075237A2 pH SENSITIVE CYANINE DYES AS REACTIVE FLUORESCENT REAGENTS
12/14/2000WO2000075140A1 7-oxo-2-azabicyclo[2.2.1]heptanes as selective muscarinic receptor antagonist
12/14/2000WO2000075139A2 Benzothiazinone and benzoxazinone compounds
12/14/2000WO2000075138A1 Oxime derivatives, process for the preparation thereof and pesticides