Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
05/2001
05/09/2001EP1097147A1 Novel angiogenesis inhibitors
05/09/2001EP1097142A1 Phthalazine derivatives phosphodiesterase 4 inhibitors
05/09/2001EP1097137A1 N-substituted naphthalene carboxamides as neurokinin-receptor antagonists
05/09/2001EP1096925A2 Use of inhibitors of prenyltransferases for for inhibiting fungal growth
05/09/2001CN1294580A Indole derivatives with antiviral activity
05/09/2001CN1065532C Thiazolidine and oxaxoliding derivatives, their prepn. and their medical use
05/08/2001US6228942 Dehydration to esterify or amidate surface of oxidized or aminated carbon powder or fiber suspended in solution containing a monomer or polymer having amine, hydroxy, and/or viny ether groups
05/08/2001US6228808 Carbamoylphenylsulfonylureas, processes for their preparation and their use as herbicides and plant growth regulators
05/08/2001CA2032330C Benzyl-substituted rhodanine derivatives for treating inflammatory bowel disease
05/03/2001WO2001030778A1 Thiazole and imidazo [4,5-b] pyridine compounds and their pharmaceutical use
05/03/2001WO2001030766A1 Phthalazinone derivatives as pde 4 inhibitors
05/03/2001WO2001030762A1 Imidazol-4-ylmethanols use as inhibitors of steroid c17-20 lyase
05/03/2001WO2001030749A1 Novel compounds
05/03/2001WO2001030387A1 Preventives or remedies for arrhythmia
05/03/2001WO2001007439A3 Process for the production of epothiolone b and derivatives as well as intermediate products for this process
05/03/2001CA2388479A1 Preventives or remedies for arrhythmia
05/03/2001CA2388121A1 Phthalazinone derivatives as pde 4 inhibitors
05/03/2001CA2387869A1 Imidazol-4-ylmethanols use as inhibitors of steroid c17-20 lyase
05/02/2001EP1095936A1 Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses, and methods and intermediates useful for their preparation
05/02/2001EP1095935A1 6-Hydroxy-5,6-dihydrouracils as herbicides
05/02/2001EP1094826A1 Novel therapeutic agents that modulate alpha-1a adrenergic receptors
05/02/2001EP1094816A1 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
05/02/2001EP1078926A9 Pyran derivatives
05/02/2001EP0984959A4 Aromatic sulfonyl alpha-hydroxy hydroxamic acid compounds
05/02/2001EP0983257A4 Aromatic sulfonyl alpha-cycloamino hydroxamic acid compounds
05/02/2001EP0973392A4 Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds
05/02/2001EP0885218B1 Oxa- and thia-diazole muscarinic receptor antagonists
05/02/2001EP0769947B1 Indolinone compounds for the treatment of disease
05/02/2001CN1293673A 1-(3-heteroarylpropyl-or-prop-2-enyl)-4-benzylpiperidines used as NMDA receptor antagonists
05/02/2001CN1293669A Benzylpiperazingl-and benzylipeeridinyl ethanone derivatives, their preparation method and their use as dopamine D receptor antagonists
05/02/2001CN1293665A New compounds and their use as positive AMPA receptor modulators
05/02/2001CN1065242C Byridyl-thiazoles
05/01/2001US6225478 Iridoid derivatives and neovascularization inhibitors containing the same as active ingredient
05/01/2001US6225335 3-(4′-bromobenzylindenyl)-2-indolinone and analogues thereof for the treatment of disease
05/01/2001US6225330 For treatment of abnormal conditions such as feeding disorders (obesity and bulimia nervosa), sexual/reproductive disorders, depression, epileptic seizure, hypertension, cerebral hemorrhage, congestive heart failure, sleep disturbances
05/01/2001US6225324 Antidepressant heterocyclic compounds
04/2001
04/26/2001WO2001029029A1 Tetrahydrobenzindolone derivatives, their preparation and their use as 5-ht7 receptor antagonists
04/26/2001WO2001029028A1 9- (piperazinylalkyl) carbazoles as bax-modulators
04/26/2001WO2001029025A2 Tyrosine kinase inhibitors
04/26/2001WO2001029021A1 Neuraminidase inhibitors
04/26/2001WO2001029012A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
04/26/2001WO2001029011A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
04/26/2001WO2001028996A2 Pyrrolidine derivatives, their preparation and their use as inhibitors of neuraminidases
04/26/2001WO2001028987A1 Benzylcycloalkyl amines as modulators of chemokine receptor activity
04/26/2001WO2001028561A1 Gram-positive selective antibacterial compounds, compositions containing such compounds and methods of treatment
04/26/2001WO2001028537A2 Bissulfonamide derivatives as enzyme inhibitors
04/26/2001WO2000059902A3 Aryl sulfonyls as factor xa inhibitors
04/26/2001WO2000055125A3 N-cyanomethyl amides as protease inhibitors
04/26/2001DE19932621A1 Neue substituerte alpha, beta-anellierte Butyrolactone New substituerte alpha, beta-fused butyrolactones
04/26/2001CA2388859A1 Inhibitors of neuraminidases
04/26/2001CA2387593A1 Enzyme inhibitors
04/26/2001CA2384240A1 Benzylcycloalkyl amines as modulators of chemokine receptor activity
04/25/2001EP1094063A1 9-(Piperazinylalkyl)carbazoles as Bax-modulators
04/25/2001EP1093372A1 CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING $g(b)-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS
04/25/2001EP1093367A1 Protease inhibitors
04/25/2001CN1292788A Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors
04/25/2001CN1064962C Arylalkyl-thiadiazinones
04/24/2001US6222048 Diaryl-2-(5H)-furanones as Cox-2 inhibitors
04/24/2001US6222040 Selective NPY (Y5) antagonists (tricyclics)
04/24/2001US6221865 Inhibitors of protein farnesyltransferase and protein geranylgeranyltransferase.
04/24/2001US6221574 Spectral sensitizers
04/24/2001CA2166203C Processes and intermediates for the preparation of 5-[2-(4-(benzoisothiazol-3-yl)-piperazin-1-yl)ethyl]- 6-chloro-1,3-dihydro-indol-2-one
04/19/2001WO2001027308A2 13-alkyl epothilone derivatives
04/19/2001WO2001027145A1 Antibody catalysis of enantio- and diastereo-selective aldol reactions
04/19/2001WO2001027128A1 C-aryl glucoside sglt2 inhibitors
04/19/2001WO2001027108A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF Aβ PROTEIN PRODUCTION
04/19/2001WO2001027107A2 Heterocyclic sodium/proton exchange inhibitors and method
04/19/2001WO2001027096A1 Aminomethyl-(hetero)aryl derivatives and their use as tryptase inhibitors
04/19/2001WO2001027094A1 Hypertriglyceridemia remedies and antiobestics
04/19/2001WO2001027091A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF Aβ PROTEIN PRODUCTION
04/19/2001WO2001027089A1 Pyrimidine derivatives
04/19/2001WO2001027080A2 5-substituted indolinones and use thereof as kinase and cyclin/cdk complex inhibitors
04/19/2001WO2001026656A2 5-membered heterocycle derivatives and use thereof as monoamine oxidase inhibitors
04/19/2001WO2001002558A8 Probe for analysis of nucleic acids
04/19/2001WO2000018767A9 2-piperazino alkylamino benzoazole derivatives: dopamine receptor subtype specific ligands
04/19/2001US20010000344 N-(2-(R)-amino-3-mercaptopropyl)-L-penicillaminyl-1,2,3,4 -tetrahydro-3(S)-isoquinoline carbonyl methionine methylester cyclic disulfide, for example; administering as antitumor agent or to treat restenosis
04/19/2001DE19949209A1 In 5-Stellung substituierte Indolinone, ihre Herstellung und ihre Verwendung als Arzneimittel In the 5-position substituted indolinones, their preparation and their use as medicaments
04/19/2001CA2425620A1 13-alkyl epothilone derivatives
04/19/2001CA2388813A1 Heterocyclic sodium/proton exchange inhibitors and method
04/19/2001CA2388505A1 5-membered heterocycle derivatives, their preparation and application as medicine
04/19/2001CA2387493A1 Amino lactam sulfonamides as inhibitors of a.beta. protein production
04/19/2001CA2384544A1 Amino lactam sulfonamides as inhibitors of a.beta. protein production
04/19/2001CA2382605A1 Pyrimidine derivatives
04/18/2001EP1092715A2 Cyano-indole derivatives as inhibitors of serotonin reuptake, method for their preparation and pharmaceutical compositions containing the same
04/18/2001EP1092711A1 Retinoid-associated receptor regulators
04/18/2001EP1091955A1 Quinolones as serine protease inhibitors
04/18/2001EP1091943A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
04/18/2001EP1091942A1 Potassium channel blocking agents
04/18/2001EP0682663B1 4-hydroxy-benzopyran-2-ones and 4-hydroxy-cycloalkyl b]pyran-2-ones useful to treat retroviral infections
04/18/2001CN1291993A Thiadiazole compounds useful as inhibitors of cysteine activity dependent enzymes
04/18/2001CN1291984A Glycine transport inhibitors
04/18/2001CN1291892A Substituted oxoazaheterocyclyl factor Xa inhibitors
04/18/2001CN1064682C Pyrrolidine derivatives having phospholipase A2 inhibitor activity
04/18/2001CN1064681C Heterocyclic compounds
04/18/2001CN1064679C Herbicidal thiocarbamoyltetrazolinones
04/17/2001US6218544 Heterocyclic esters and amides
04/17/2001US6218431 Substituted biphenyls
04/17/2001US6218423 Administering pyrrolidine derivative for therapy of nerve-related vision disorder, improving vision, treating memory impairment, or enhancing memory performance in animal
04/17/2001US6218418 Therapy of cell proliferative disorders associated with an altered cell dependent kinase activity by administering amino pyrazole derivative to mammal
04/17/2001US6218413 Oxazolidinone antibacterial agents having a thiocarbonyl functionality