Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
04/2001
04/17/2001US6218412 Therapy and prophylaxis of diseases where an increased concentration of interleukin-1.beta. participates in their course, for example septic shock, leukemia, hepatitis, muscular degeneration, degenerative joint diseases
04/17/2001US6218408 Selective NPY (Y5) antagonists (bicyclics)
04/17/2001US6218376 For treating inflammatory diseases
04/17/2001US6218365 Serine protease inhibitors
04/17/2001US6217845 Protein labelling
04/17/2001CA2080475C Neuroprotective indolone and related derivatives
04/12/2001WO2001025229A1 Amide compounds
04/12/2001WO2001025227A2 Quinolyl propyl piperidine derivatives and their use as antibacterial agents
04/12/2001WO2001025220A1 Triazine kinase inhibitors
04/12/2001WO2001025210A2 Substituted 2-thio-3,5-dicyano-4-aryl-6-aminopyridines and the use thereof as adenosine receptor ligands
04/12/2001WO2001025209A1 Pyridinium derivatives for the treatment of diabetic and aging-related vascular complications
04/12/2001WO2001025200A1 Cyclic amine compounds as ccr5 antagonists
04/12/2001WO2001025181A1 Carboxylic acid derivatives and drugs containing the same
04/12/2001WO2001024828A2 MODULATORS OF CYTOKINE MEDIATED SIGNALLING PATHWAYS AND INTEGRIN αVβ3 RECEPTOR ANTAGONISTS FOR COMBINATION THERAPY
04/12/2001WO2001024827A2 INHIBITORS OF THE ENDOTHELIN SIGNALLING PATHWAY AND αVβ3 INTEGRIN RECEPTOR ANTAGONISTS FOR COMBINATION THERAPY
04/12/2001WO2001024796A1 1,2,4-triazole derivatives, composition, process of making and methods of use
04/12/2001DE19948269A1 New compounds as integrin antagonists useful for treating e.g. cardiovascular disorders, rheumatoid arthritis, kidney failure, stroke, cancer, osteoporosis, psoriasis or infection
04/12/2001CA2608807A1 Cyclic amine compounds as ccr5 antagonists
04/12/2001CA2386457A1 Inhibitors of the endothelin signalling pathway and .alpha.v.beta.3 integrin receptor antagonists for combination therapy
04/12/2001CA2386218A1 Triazine kinase inhibitors
04/12/2001CA2386157A1 Amide compounds
04/12/2001CA2386147A1 Substituted 2-thio-3,5-dicyano-4-aryl-6-aminopyridines and the use thereof
04/12/2001CA2383836A1 Quinolyl propyl piperidine derivatives and their use as antibacterial agents
04/12/2001CA2351075A1 Pyridinium derivatives for the treatment of diabetic and aging-related vascular complications
04/11/2001EP1090914A2 Processes and intermediates for manufacturing retroviral protease inhibiting compounds
04/11/2001EP1090912A1 Amino acid derivatives and drugs containing the same as the active ingredient
04/11/2001EP1089998A2 Epothilone derivatives and their synthesis and use
04/11/2001EP1089993A1 5-ht 1f? agonists
04/11/2001EP1089989A1 Inhibitors of alpha4beta1 mediated cell adhesion
04/11/2001EP1089981A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis.
04/11/2001EP1089980A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
04/11/2001EP1089977A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
04/11/2001EP1089964A1 Hydrazine derivatives
04/11/2001EP1089752A1 Alpha-keto oxadiazoles as serine protease inhibitors
04/11/2001EP1089735A1 4-benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective nmda receptor antagonists
04/11/2001EP0984963B1 Novel compounds
04/11/2001CN1291190A 5-substituted pyrimidine-2-yloxy carboxylic acid derivatives, the production of the same and their utilization as endothelin antagonist
04/11/2001CN1064359C Diindole heterocyclic compounds, preparing method and its use
04/11/2001CN1064358C Benyl piperidine derivatives
04/11/2001CN1064350C Aryl and heteroaryl alkoxynaphtalene derivatives
04/10/2001US6215016 Hematopoietic agents; preventing cytopenia
04/10/2001US6214996 Naphthalene derivates, process for the preparation thereof, and intermediates therefor
04/10/2001US6214991 3-(4,5,7-trifluorobenzothiazol-2-yl)methyl-indole-n-acetic acid, ethyl ester for example; treating complications of diabetes mellitus, such as cataracts, retinopathy, nephropathy, and neuropathy
04/10/2001US6214870 Antiarthritic agents; anticancer agents
04/10/2001US6214853 Selective NPY (Y5) antagonists (bicyclics)
04/10/2001US6214852 N-[5-[[[5-alkyl-2-oxazolyl]methyl]thio]-2-thiazolyl]-carboxamide inhibitors of cyclin dependent kinases
04/10/2001US6214845 Insecticidal N-(substituted arylmethyl)-4[bis(substituted phenyl or pyridyl)methyl] piperidines
04/10/2001US6214842 Treating metabolic disorders related to insulin resistance or hyperglycemia typically associated with obesity or glucose intolerance; treating diabetes types i and ii
04/10/2001US6214841 Anticoagulants
04/10/2001US6214834 Angiogenesis inhibitors; antiinflammatory agents; anticancer agents
04/10/2001US6214825 Aza-heterocycloakenes, pesticidal compositions containing them, pesticidal methods of using them, and processes for preparing them
04/10/2001US6214822 Substituted aza and diazacycloheptane and cyclooctane compounds and their use
04/10/2001US6214813 Azopyrazoles
04/05/2001WO2001023382A1 Pharmaceutically active sulfonyl hydrazide derivatives
04/05/2001WO2001023378A1 Pharmaceutically active sulfonamide derivatives
04/05/2001WO2001023376A1 Isonipecotamides for the treatment of integrin-mediated disorders
04/05/2001WO2001023375A2 Substituted pyridines and pyridazines with angiogenesis inhibiting activity
04/05/2001WO2001023357A2 Fused cycloheptane and fused azacycloheptane compounds and their use as integrin receptor antagonists
04/05/2001WO2001022966A1 Caspases and apoptosis
04/05/2001WO2000073284A3 1,4-benzodiazepin-2-ones useful as hiv reverse transcriptase inhibitors
04/05/2001WO2000068198A3 Heterosubstituted pyridine derivatives as pde 4 inhibitors
04/05/2001CA2385001A1 Pharmaceutically active sulfonyl hydrazide derivatives
04/05/2001CA2352957A1 Isonipecotamides for the treatment of integrin-mediated disorders
04/04/2001EP1088822A1 Pharmaceutically active sulfonyl hydrazide derivatives
04/04/2001EP1088821A1 Pharmaceutically active sulfonamide derivatives
04/04/2001EP1088819A2 6-azauracil derivatives as thyroid receptor ligands
04/04/2001EP1087981A2 Prenyl transferase inhibitors
04/04/2001EP1087975A2 Epothilone minor constituents
04/04/2001EP1087967A1 1,3-oxazoline and 1,3-thiazoline derivatives, method for producing the same and their use as pesticides
04/04/2001EP1087963A1 Inhibitors of glycogen synthase kinase 3
04/04/2001EP1087962A1 Preparation of heteroaryl compounds
04/04/2001EP1087959A1 Novel benzopyran or thiobenzopyran derivatives
04/04/2001EP1087951A1 Carbon substituted aminothiazole inhibitors of cyclin dependent kinases
04/04/2001EP1087948A1 2,4-diamino-1,3,5-triazine, method for the production and use of the same as herbicides and plant growth regulators
04/04/2001EP1087941A2 Thiolesters and uses thereof
04/04/2001EP1087937A1 Cyclic hydroxamic acids as metalloproteinase inhibitors
04/04/2001EP0805805B1 Substituted arylazadioxacyclo alkene fungicides
04/04/2001CN1290266A Benzofuran-4-carboxamides and their therapeutical use
04/04/2001CN1290265A Thrombin receptor antagonists
04/04/2001CN1290264A Triazine angiogenesis inhibitors
04/04/2001CN1290263A Arylpiperidine derivatives and use thereof
04/04/2001CN1290262A Heteroaromatic derivatives
04/04/2001CN1290250A Sulfonylamino derivatives which inhibit matrix-degrading metallopr teinases
04/04/2001CN1290249A Aminoguanidine hydrazone derivatives, process for producing the same and drugs thereof
04/04/2001CN1290165A Benzothiazole Protein tyrosine kinase inhibitors
04/04/2001CN1290164A Inhibition of RAF kinase using substituted heterocyclic ureas
04/04/2001CN1289773A Preparation of intermediate for thiazolylisopseudoindole dyes
04/04/2001CN1064044C Heterocyclic compounds, their production and use
04/04/2001CN1063942C Use of thiazolidine derivative for making medicaments
04/03/2001US6211412 Reacting beta-keto ester with hydrogenating agent in presence of asymmetric organometallic molecular catalyst comprising metal atom having one or more chiral ligands coupled thereto, converting hydroxyester formed to epothilone precursor
04/03/2001US6211381 Chemical intermediates
04/03/2001US6211379 Process for preparing heterocyclic compounds
04/03/2001US6211376 8-hydroxy-7-substituted quinolines as anti-viral agents
04/03/2001US6211240 O-benzyl oxime ether derivatives and their use as pesticides
04/03/2001US6211234 Substituted phenyl compounds
04/03/2001US6211214 Pesticides, insecticides or miticides
04/03/2001US6211204 Thiadiazole, hydrogenated pyridine derivatives
04/03/2001US6211183 Selective factor Xa inhibitors
04/03/2001US6211178 Antiprotozoa agents for coccidioides; cyclization
04/03/2001US6211170 Azetidinone derivatives for the treatment of HCMV infections