Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773) |
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10/25/2005 | US6958339 Pyrazole derivative |
10/25/2005 | US6958336 Anticancer agents; immunosuppressants; antiallergens; antiinflammatory agents |
10/25/2005 | US6958333 N'-(isoindolino[3,2-b]perhydro-1,3-oxazin-5-on-9-yl)-N-(pyridin-2-yl) urea, for example; cyclin-dependent kinase inhibitors; colon cancer treatment |
10/25/2005 | CA2332461C New benzenesulfonamide derivatives, their method of preparation and the pharmaceutical compositions containing them |
10/25/2005 | CA2304974C 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders |
10/20/2005 | WO2005097791A1 Inhibitors of iap |
10/20/2005 | WO2005097787A2 Novel benzothiazoles and the use thereof as medicaments |
10/20/2005 | WO2005097786A1 Oxadiazolone derivatives as ppar delta agonists |
10/20/2005 | WO2005097784A1 Phenylthioacetic acid derivatives and use thereof |
10/20/2005 | WO2005097782A1 Piperidine derivative |
10/20/2005 | WO2005097776A1 Composition comprising an optically-active monomeric compound, method implementing said composition, monomeric compound, polymer comprising same, and use thereof |
10/20/2005 | WO2005097774A1 Substituted 4-alkyl- and 4-alkanoyl-piperidine derivatives and their use as neurokinin antagonists |
10/20/2005 | WO2005097767A1 2-aminothiazole compounds useful as aspartyl protease inhibitors |
10/20/2005 | WO2005097766A1 2-aminomethylthiazole-5-carboxamides as protein kinase modulators |
10/20/2005 | WO2005097765A1 Anaplastic lymphoma kinase modulators and methods of use |
10/20/2005 | WO2005097764A1 Thiazole derivative |
10/20/2005 | WO2005097763A2 1,3,4-oxadiazol-2-ones as ppar delta |
10/20/2005 | WO2005097762A2 1,3,4-oxadiazol-2-ones as ppar delta modulators |
10/20/2005 | WO2005097758A1 Certain triazole-based compounds, compositions, and uses thereof |
10/20/2005 | WO2005097750A1 Substituted pyridones as inhibitors of poly(adp-ribose) polymerase (parp) |
10/20/2005 | WO2005097746A2 2-propene-1-ones as hsp 70 inducers |
10/20/2005 | WO2005097738A1 Novel sulfonamide derivative |
10/20/2005 | WO2005097137A2 Advanced quinazoline based protein kinase inhibitors |
10/20/2005 | WO2005097136A1 Biaryl substituted pyrazinones as sodium channel blockers |
10/20/2005 | WO2005097134A2 Quinazoline based protein kinase inhibitors |
10/20/2005 | WO2005097117A1 Thiadiazolidinones as gsk-3 inhibitors |
10/20/2005 | WO2005097116A1 Composition comprising a jnk inhibitor and cyclosporin |
10/20/2005 | WO2005097114A2 Thiazole sulfonamide compounds for the treatment of neurodegenerative disorders |
10/20/2005 | WO2005097112A2 Ion channel modulators |
10/20/2005 | WO2005085236A3 Caspase inhibitors and uses thereof |
10/20/2005 | WO2005070891A3 Compounds and methods of use |
10/20/2005 | WO2005061450A3 Hiv protease inhibiting sulfonamides |
10/20/2005 | WO2005055715A3 Insecticidal n-(heteroarylalkyl) alkanediamine derivatives |
10/20/2005 | WO2005051931A3 Phosphodiesterase inhibitors |
10/20/2005 | WO2004071460A3 Cyclic derivatives as modulators of chemokine receptor activity |
10/20/2005 | WO2003106413A3 Process for the preparation of oxazolidinones and method of use thereof |
10/20/2005 | US20050234247 New effector conjugates, process for their production and their pharmaceutical use |
10/20/2005 | US20050234242 Coupling of a 2-haloindole with an (hetero)aryl zinc intermediate in the presence of a palladium or nickel-containing catalyst, phosphine ligand and a solvent selected from tetrahydrofuran, dimethylformamide and N-methylpyrrolidone; by-product inhibition; hepatitis C virus polymerase inhibitors |
10/20/2005 | US20050234238 8-(Biaryl)quinoline pde4 inhibitors |
10/20/2005 | US20050234098 antitumor, anticarcinogenic agents; cytotoxic activity and angiogensis inhibitors; leukemia, colorectal cancer; orally |
10/20/2005 | US20050234082 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto |
10/20/2005 | US20050234081 for inhibiting the enzyme C1s, a protease in the classical pathway of the complement system; and the use of this inhibition to treat or ameliorate acute or chronic disorders in mammals |
10/20/2005 | US20050234080 Mitotic kinesin inhibitors |
10/20/2005 | US20050234079 Novel crystalline form of 5-[4-[[3-methyl-4-oxo-3,4-dihydroquinazolin-2-yl]methoxy] benzyl]thiazolidine-2,4-dione potassium salt |
10/20/2005 | US20050234065 Dipeptidyl peptidase-IV inhibitors |
10/20/2005 | US20050234064 2-(4-Methoxyphenyl)-amino-),3-(aminocarbonyl-)quinoxaline; janus(JAK) kinase inhibitors;spleen tyrosine kinase(SYK) inhibitors; glycogen synthase-3(GSK-3) kinase inhibitors; immunocompetance; antiinflammatory agents; antiallergens; autoimmune diseases; antiproliferative agents; respiratory disorders |
10/20/2005 | US20050234062 Such as 2-{4-[(4aS,8aR)-4-(3,4-dimethoxyphenyl)-1-oxo-4a,5,8,8a-tetrahydro-1H-phthalazin-2-yl]-piperidin-1-yl}-2H-acetamide; phosphodiesterase inhibitors; for treatment of respiratory disorders |
10/20/2005 | US20050234059 4-(5-Methyl-2-phenyl-pyrimidin-4-yl)-1H-pyrrole-2 carboxylic acid (2-hydroxy-1-(S)-phenyl-ethyl)-amide; Mitogen-activated protein kinase inhibitor; anticarcinogenic, antiinflammatory agent,neurodegenerative disorders, restenosis, antidiabetic, antiallergen, and cardiovascular disease |
10/20/2005 | US20050234057 1-Phenylpiperidin-3-one derivatives and processes for the preparation thereof |
10/20/2005 | US20050234055 Pyrazole derivative |
10/20/2005 | US20050234049 Methods of treating or preventing autoimmune diseases with 2, 4-pyrimidinediamine compounds |
10/20/2005 | US20050234048 substituted 4,5-dihydro-1H-benzo[b][1,4]-diazepin-2-one; amidation of a substituted monoprotected 1,2-diaminobenzene with an ester, deprotecting, cyclization; chronic neurological disorders, psychosis, schizophrenia, Alzheimer's disease |
10/20/2005 | US20050234047 Respiratory syncytial virus replication inhibitors |
10/20/2005 | US20050234046 Aryl sulfonamide and sulfonyl compounds as modulators of PPAR and methods of treating metabolic disorders |
10/20/2005 | US20050234045 N-alkyl-4-methyleneamino-3-hydroxy-2-pyridones |
10/20/2005 | US20050234044 Cyclic amine derivatives and methods of use |
10/20/2005 | US20050234042 Organic compounds |
10/20/2005 | US20050234041 Substituted 1-benzazepines and derivatives thereof |
10/20/2005 | US20050234038 Protease inhibitors |
10/20/2005 | US20050234033 1-(2-naphthylsulfonyl)-4-(5-hydroxyaminocarbonylthiazol-2-yl)piperazine;antiprolifrative agent; cell cycle arrest, cellular differentiation, apoptosis and reversal of the transformed phenotype; |
10/20/2005 | US20050234030 Modulators of CRTH2, COX-2 and FAAH |
10/20/2005 | US20050234020 e.g. 3'-(1-Cyclohexyl-5-hydroxy-3-methyl-1H-pyrazol-4-ylazo)-2'-hydroxy-biphenyl-3- carboxylic acid; agonists of TPO receptor; non-peptide; thrombocytopenia is due to bone marrow, stem cell, or liver transplant, idiopathic thrombocytopenia purpura, myelodysplastic syndromes, aplastic anemia or leukemia |
10/20/2005 | US20050233979 Use in controlling apoptosis, as antiinflammatory agents, in treating autoimmune disease, as antiischemic agents, in treating cardiovascular disorders; for example, (S,S)-3-[2-(3-Acetylamino-2-oxo-2H-pyridin-1-yl)-butyrylamino]-4-oxo-5-(2,3,5,6-tetrafluoro-phenoxy)-pentanoic acid |
10/20/2005 | US20050233909 such as 6-(5-chlorobenzoxazol-2-yl)-2-(3-trifluoromethylphenoxy)pyridine, used on monocotyledonus or dicotyledonus weeds |
10/20/2005 | CA2562780A1 Nucleic acid melting analysis with saturation dyes |
10/20/2005 | CA2562140A1 Phenylthioacetic acid derivatives and use thereof |
10/20/2005 | CA2561967A1 Substituted 4-alkyl- and 4-alkanoyl-piperidine derivatives and their use as neurokinin antagonists |
10/20/2005 | CA2561928A1 Thiazole sulfonamide compounds for the treatment of neurodegenerative disorders |
10/20/2005 | CA2561907A1 Composition comprising a jnk inhibitor and cyclosporin |
10/20/2005 | CA2561738A1 1,3,4-oxadiazol-2-ones as ppar delta modulators_and their use thereof |
10/20/2005 | CA2561627A1 Oxadiazolone derivatives as ppar delta agonists |
10/20/2005 | CA2561280A1 Substituted pyridones as inhibitors of poly(adp-ribose) polymerase (parp) |
10/20/2005 | CA2561267A1 2-aminothiazole compounds useful as aspartyl protease inhibitors |
10/20/2005 | CA2561249A1 2-aminomethylthiazole-5-carboxamides as protein kinase modulators |
10/20/2005 | CA2561230A1 1,3,4-oxadiazol-2-ones as ppar delta modulators and their use thereof |
10/20/2005 | CA2560954A1 Certain triazole-based compounds, compositions, and uses thereof |
10/20/2005 | CA2560796A1 Biaryl substituted pyrazinones as sodium channel blockers |
10/20/2005 | CA2560683A1 Novel benzothiazoles and the use thereof as medicaments |
10/20/2005 | CA2560162A1 Inhibitors of iap |
10/20/2005 | CA2559866A1 Anaplastic lymphoma kinase modulators and methods of use |
10/20/2005 | CA2559740A1 Thiadiazolidinones as gsk-3 inhibitors |
10/20/2005 | CA2557721A1 Ion channel modulators |
10/19/2005 | EP1586573A1 Oxadiazolones, processes for their preparation and their use as pharmaceuticals |
10/19/2005 | EP1586567A1 Compounds useful in the treatment of inflammatory diseases |
10/19/2005 | EP1586565A1 Substituted polycyclic aryl and heteroaryl pyrazinones useful for selective inhibition of the coagulation cascade |
10/19/2005 | EP1586564A1 8-azaprostaglandin derivatives and medicinal uses thereof |
10/19/2005 | EP1586558A2 Bis-sulfonamide hydroxyethylamino retroviral protease inhinitors |
10/19/2005 | EP1586319A1 Thiadiazolidinones as GSK-3 inhibitors |
10/19/2005 | EP1586318A1 Thiadiazolidinones as GSK-3 inhibitors |
10/19/2005 | EP1585827A2 Modulation of protein functionalities |
10/19/2005 | EP1585739A1 Substituted arylcyclopropylacetamides as glucokinase activators |
10/19/2005 | EP1585737A2 Uracils having a herbicidal activity |
10/19/2005 | EP1585734A2 Anti-inflammatory medicaments |
10/19/2005 | EP1585728A1 Imino acid derivatives for use as inhibitors of matrix metalloproteinases |
10/19/2005 | EP1585727A1 Indoles useful in the treatment of androgen-receptor related diseases |
10/19/2005 | EP1585726A1 Fused heterocyclic derivatives as ppar modulators |
10/19/2005 | EP1585725A2 Compounds which mimic the chemical and biological properties of discodermolide |
10/19/2005 | EP1585720A1 Process for converting a cis-trans mixture of substituted benzylidene amines into the pure cis isomer |
10/19/2005 | EP1585541A2 Pharmaceutical compositions comprising insulin and legends of insulin hexamer |
10/19/2005 | EP1585521A2 Derivatives of aryl-quinazoline/aryl-2amino-phenyl methanone which promote the release of parathyroid hormone |