Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773) |
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11/02/2005 | EP1591443A1 Pyrazole derivative |
11/02/2005 | EP1590358A1 9-ketospinosyn derivatives |
11/02/2005 | EP1590347A1 Isothiazole derivatives |
11/02/2005 | EP1590346A1 4- {'3-(sulfonylamino) phenyl! '1-(cyclymethyl) piperidin-4-ylidene! methyl} benazmide derivatives as delta opioid receptor ligands for the treatment of pain, anxiety and functional gastrointestinal disorder |
11/02/2005 | EP1590344A2 Anti-cancer medicaments |
11/02/2005 | EP1590337A1 Acylaminothiazole derivatives, preparation method thereof and use of same as beta-amyloid peptide production inhibitors |
11/02/2005 | EP1590329A1 N-aryl heteroaromatic products, compositions containing same and use thereof |
11/02/2005 | EP1590326A2 Substituted alkyl amido piperidines |
11/02/2005 | EP1507530B1 Diaminothiazoles and use thereof as cdk4 inhibitors |
11/02/2005 | EP1446402B1 2-amino-4-heteroarylethyl thiazoline derivatives and their use an inhibitors of inducible no-synthase |
11/02/2005 | EP1383749B1 Arylsulfonamides as antiviral agents |
11/02/2005 | EP1377569B1 Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines with adenosine receptor-binding activity and their use as cardiovascular preparations |
11/02/2005 | EP1246807B1 Novel hydantoin, thiohydantoin, pyrimidinedione and thioxopyrimidinone derivatives, preparation method and use as medicines |
11/02/2005 | EP1159261B1 Antizyme modulators and their use |
11/02/2005 | EP1045833B1 2,3-substituted indole compounds as cox-2 inhibitors |
11/02/2005 | EP0946531B1 Process for the preparation of thiazole derivatives |
11/02/2005 | CN1692108A Pesticidal heterocycles |
11/02/2005 | CN1692100A 4[piperidin-4-yliden-(3-carbamoylphenyl)methyl]benzamide derivatives and their use for the treatment of pain spinal injuries or gastrointestinal disorders |
11/02/2005 | CN1690051A Novel azoles having an insecticidal action |
11/02/2005 | CN1225471C Compounds with growth hormone releasing properties |
11/02/2005 | CN1225462C New piperazine and piperidine compounds |
11/01/2005 | US6960606 Adamantyl Thiazole Thioureas |
11/01/2005 | US6960605 Thiazole, imidazole and oxazole compounds and treatments of disorders associated with protein aging |
11/01/2005 | US6960601 Imidazole derivatives; appetite suppressants |
11/01/2005 | US6960599 Dopamine D2 receptor and 5-HT1A antagonists; schizophrenia; cognitive activators; Alzheimer's disease; brain disorders; strokes; antiischemic agents; anxiolytic agents; obsessive compulsive disorder; eating, sleeping and sexual disorders |
11/01/2005 | US6960591 Propane-1,3-dione derivative |
11/01/2005 | US6960578 Glutamate receptor antagonists |
11/01/2005 | US6960575 Thiazine derivatives |
10/27/2005 | WO2005101838A2 Piperazinylpiperidine derivatives as chemokine receptor antagonists |
10/27/2005 | WO2005100349A2 Polycyclic pyridines as potassium ion channel modulators |
10/27/2005 | WO2005100348A1 Amorphous ziprasidone hydrochloride |
10/27/2005 | WO2005100344A1 Inhibitors of akt activity |
10/27/2005 | WO2005100338A1 5-morpholinylmethylthiophenyl pharmaceutial compounds as p38 map kinase modulators |
10/27/2005 | WO2005100334A1 Dipeptidyl peptidase-iv inhibitors |
10/27/2005 | WO2005100331A2 Antidiabetic agents |
10/27/2005 | WO2005100303A1 Indene derivatives and process for the preparation thereof |
10/27/2005 | WO2005099709A2 Bicyclic heterocycles useful as serine protease inhibitors |
10/27/2005 | WO2005099673A1 Polycylic thiazoles as potassium ion channel modulators |
10/27/2005 | WO2005099353A2 A novel process for the preparation of linezolid and related compounds |
10/27/2005 | WO2005087725A3 Novel compounds as inhibitors of hepatitis c virus ns3 serine protease |
10/27/2005 | WO2005074642A3 Chemical compounds |
10/27/2005 | WO2005034848A3 Inhibitors of cathepsin s |
10/27/2005 | US20050240035 polymerase inhibitors such as -1-(5-Cyano-pyridin-2-yl)-3-(1,1a,2,7b-tetrahydro-cyclopropa[c]chromene-1-yl)-urea, used as antiviral agents |
10/27/2005 | US20050240023 Cathepsin cysteine protease inhibitors |
10/27/2005 | US20050239865 3-Cyano-2-amide-5,6-dihydrothieno[2,3-b]pyridine derivatives, e.g., tert-butyl 3-cyano-2-[(2-ethylbutanoyl)amino]-5,6-dihydrothieno[2,3-b]pyridine-7(4H) carboxylate; the compounds block the action of glucagon at its receptor and decrease the levels of plasma glucose to treat diabetes |
10/27/2005 | US20050239853 New compounds |
10/27/2005 | US20050239852 2-(3-aminoaryl)amino-4-aryl-thiazoles and their use as c-kit inhibitors |
10/27/2005 | US20050239851 Substituted benzoxazoles as estrogenic agents |
10/27/2005 | US20050239843 Diaminothiazoles |
10/27/2005 | US20050239841 New compounds |
10/27/2005 | US20050239835 controlling weight gain; 1-(1-amino-2-phenylethylcarbonyl)-4-cyclohexylpiperidine compounds |
10/27/2005 | US20050239829 Novel piperidine compound |
10/27/2005 | US20050239827 N-(4-(2,2-difluoro-benzo(1,3)dioxol-5-ylcarbamoyl)-3-hydroxy-phenyl)-4,6-Bis-((3R,5S)-3,5-diamino-piperidin-1-yl)-(1,3,5)triazine-2-amine for example; Gram-positive and Gram-negative strains; retains potency against common antibiotic resistant strains |
10/27/2005 | US20050239819 4-Oxoquinoline compounds and utilization thereof as hiv integrase inhibitors |
10/27/2005 | US20050239801 Novel compounds |
10/27/2005 | US20050239800 Polycyclic pyrazines as potassium ion channel modulators |
10/27/2005 | US20050239796 tert-butyl4-{(3,4-dimethoxyphenethyl)[2-(1H-indol-3-yl)acetyl]amino}-1-piperidine carboxylate; somatostatin receptors modulator; anticarcinogenic agent; acromegalia, hypophyseal adenomas, endocrine gastroenteropancreatic tumors including carcinoid syndrome; reducing amination of N-substituted piperidone |
10/27/2005 | US20050239790 Substituted hydroxyethylamine aspartyl protease inhibitors |
10/27/2005 | US20050239786 Triazole derivatives as tachykinin receptor antagonists |
10/27/2005 | US20050239777 Quinazoline derivatives and pharmaceutical compositions containing them |
10/27/2005 | US20050239776 Tachykinin receptor antagonists |
10/27/2005 | US20050239771 Respiratory syncytial virus replication inhibitors |
10/27/2005 | US20050239769 Therapeutic compounds for treating dyslipidemic conditions |
10/27/2005 | US20050239713 Novel tubulysin analogues |
10/27/2005 | US20050239096 via unsymmetrical cyanine dyes that are derivatives of thiazole orange, staining solution and select fluorogenic compounds that are characterized as non-genotoxic; low cost |
10/27/2005 | US20050238614 Polyethylene glycol conjugates of heterocycloalkyl carboxamido propanoic acids |
10/27/2005 | DE102004016845A1 Phenylthioessigsäure-Derivate und ihre Verwendung Phenylthioacetic acid derivatives and their use |
10/27/2005 | CA2562242A1 Polycylic thiazoles as potassium ion channel modulators |
10/27/2005 | CA2562235A1 Piperazinylpiperidine derivatives as chemokine receptor antagonists |
10/27/2005 | CA2561311A1 Inhibitors of akt activity |
10/27/2005 | CA2560346A1 Polycyclic pyridines as potassium ion channel modulators |
10/26/2005 | EP1589017A2 12,13-modified epothilone derivatives |
10/26/2005 | EP1589013A2 Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines with adenosine receptor-binding activity and their use as cardiovascular preparations |
10/26/2005 | EP1589008A1 A crystalline dibenzothiazepine derivative and its use as an antipsychotic agent |
10/26/2005 | EP1589007A2 5-membered heterocycle derivatives, production thereof and their use as medicaments |
10/26/2005 | EP1589006A1 Oxa- and thiazole derivatives useful as antidiabetics and antidiobesity agents |
10/26/2005 | EP1587804A1 Androgen receptor antagonists |
10/26/2005 | EP1587803A1 Pyrimidine-4,6-dicarboxylic acid diamides for use as selective mmp 13 inhibitors |
10/26/2005 | EP1587800A1 Thiazole derivatives and their use as vap-1 inhibitors |
10/26/2005 | EP1587795A1 N- (1-benzyl-2-oxo-2- (1-piperazinyl) ethyl) -1-piperidincarboxamid-derivatives and related compounds use as cgrp-antagonists for treating a headache |
10/26/2005 | EP1587791A1 Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof |
10/26/2005 | EP1587790A2 Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof |
10/26/2005 | EP1587787A1 Viral polymerase inhibitors |
10/26/2005 | EP1587509A2 Androgen receptor antagonists |
10/26/2005 | EP1427408A4 CYCLIC HYDROXAMIC ACIDS AS INHIBITORS OF MATRIX METALLOPROTEINASES AND/OR TNF-$g(a) CONVERTING ENZYME (TACE) |
10/26/2005 | EP1289965B1 Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists |
10/26/2005 | EP1183229B1 Glucagon antagonists/inverse agonists |
10/26/2005 | EP1129071B1 Phenyl-substituted cyclic enaminones |
10/26/2005 | EP0835245B1 Substituted n-methylenethioureas as pesticides |
10/26/2005 | CN1688574A Indole-3-carboxamides as glucokinase(GK) activators |
10/26/2005 | CN1688571A Substituted heterocyclylpyrimidines |
10/26/2005 | CN1688557A Thiazole compounds for treatment of neurodegenerative disorders |
10/26/2005 | CN1688315A Use of selective COX-2 inhibitors for the treatment of urinary incontinence |
10/26/2005 | CN1224623C 1-phenysulfonyl-1, 3-dihydro-2H-indole-2-one derivatives, their preparation and their therapeutic use |
10/26/2005 | CN1224622C Method for preparing 2-alkyl-3-aminothiophene derivative and 3-aminothiophene derivative |
10/25/2005 | US6958401 Method for synthesizing epothilones and epothilone analogs |
10/25/2005 | US6958355 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis |
10/25/2005 | US6958350 Chemical compounds |
10/25/2005 | US6958348 Side effect reduction |
10/25/2005 | US6958340 such as N-[3-methyl-5-(trifluoromethyl)phenyl]-4-(2-phenyl-1H-imidazol-1-yl)pyrimidin-2-amine; treating breast cancer; use in combination with estrogen receptor modulators such as tamoxifen and raloxifene |