Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
09/2005
09/15/2005WO2005085238A1 2-pyridinylethylcarboxamide derivatives and their use as fungicides
09/15/2005WO2005085236A2 Caspase inhibitors and uses thereof
09/15/2005WO2005085234A2 Bycyclic anthranilamide derivatives useful as insecticides
09/15/2005WO2005085230A1 4-benzimidazol-2-yl-pyridazine-3-one-derivatives, production and use thereof in medicaments
09/15/2005WO2005085226A1 Mtp inhibiting aryl piperidines or piperazines substituted with 5-membered heterocycles
09/15/2005WO2005085225A1 Novel hydroxy-6-heteroarylphenanthridines and their use as pde4 inhibitors
09/15/2005WO2005085220A1 Use of thiadiazole urea derivatives
09/15/2005WO2005085216A1 Isoxazoline-substituted benzamide compound and noxious organism control agent
09/15/2005WO2005085214A1 Diaryl-substituted five-membered heterocycle derivative
09/15/2005WO2005085209A1 Basic amine compound and use thereof
09/15/2005WO2005085201A1 Novel cyclic compound having 4-pyridylalkylthio group having (un)substituted amino introduced therein
09/15/2005WO2005085198A2 Amino cyclopropane carboxamide derivatives as bradykinin antagonists
09/15/2005WO2005085194A2 Indole-2-carboxylic acid hydrazides as glycogen phosphorylase inhibitors
09/15/2005WO2005085177A2 Biaryl amino acids and their use in dna binding oligomers
09/15/2005WO2005084222A2 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
09/15/2005WO2005068433A9 Benzimidazole derivatives
09/15/2005WO2005065050A3 Bicyclic compound
09/15/2005WO2005055940A3 Novel m3 muscarinic acetylcholine receptor antagonists
09/15/2005WO2005054430A3 Hepatitis c virus inhibitors
09/15/2005WO2005051300A3 Bicyclic inhibitors of mek and methods of use thereof
09/15/2005WO2005049604A3 Antithrombotic aromatic ethers
09/15/2005WO2005039496A3 Inhibitors of cathepsin s
09/15/2005WO2005037258A3 Cyanoguanidine-based azole compounds useful as malonyl-coa decarboxylase inhibitors
09/15/2005WO2005026111A3 Heteroaromatic selective inhibitors of neuronal nitric oxide synthase
09/15/2005US20050203159 Calcium channel modulators 2-(alkyl or (hetero)arylalkylthio)-imidazoles and S-oxides thereof; angina, hypertension, congestive heart failure, myocardial ischemia, arrhythmia, diabetes, urinary incontinence, stroke, pain, brain injury, or neuronal disorders
09/15/2005US20050203152 Polymorph of a pharmaceutical
09/15/2005US20050203151 carboxy- or tetrazole functional thiazole and oxazole compounds; peroxisome proliferator-activated receptor (PPAR) modulators; Type 2 diabetes, syndrome X, dyslipidemia, and atherosclerotic diseases
09/15/2005US20050203149 Alkanamide alpha-monohydrazone derivatives, e.g., N-(4-chlorobenzyl)-2-(4-trifluoromethylphenylhydrazono)propionamide, for agricultural and horticultural use, clothing, food and housing-related use, or livestock and pet use
09/15/2005US20050203147 Biaryl heterocyclic compounds and methods of making and using the same
09/15/2005US20050203146 P2Y1 Purinoreceptor; thromboembolic disorders; compounds are 2-((hetero)arylamino) benzimidazoles, benzoxazoles or benzothiazoles such as [2-(2-tert-butyl-phenoxy)-pyridin-3-yl]-(6-methyl-1H-benzoimidazol-2-yl)-amine
09/15/2005US20050203127 2-(Phenyl)-2h-pyrazole-3-carboxylic acid-n-4-(thioxo-heterocyclyl)-phenyl-amide derivatives and corresponding imino-heterocyclyl derivatives and relates compounds for use as inhibitors of the coagulation factors xa and/or viia for treating thromboses
09/15/2005US20050203114 Pyrimidine-indole derivatives; cancer, autoimmunological, metabolic, inflammatory, infection (bacterial, viral, yeast, fungal, etc.), diseases of the central nervous system, degenerative neural disease, allergy/asthma, dermatology, angiogenesis, neovascularization, vasculogenesis, and cardiovascular
09/15/2005US20050203108 Glucagon antagonists/inverse agonists
09/15/2005US20050203102 Oxazolidinone derivatives such as (S)-N-[3-[3-fluoro-4-[4-[4-[(3-carboxymethyl-5-oxo-2-thioxo-1,3-thiazolidin-3-yl)methine]phenyl]piperazin-1 -yl]phenyl]-2-oxooxazolidin-5-ylmethyl] acetamide; antibiotics; use against Vancomycin resistant organisms, methicillin resistant organisms
09/15/2005US20050203093 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4
09/15/2005US20050203090 Methods of using N-alkyl-hydroxamic acid-isoindolyl compounds
09/15/2005US20050203078 Inhibitors of factor Xa or related serine proteases; thrombosis; benzamide derivatives with benzimidazole, indole or imidazo(1,2-a)pyridine rings; e.g. 4-(azepan-2-on-1-yl)-N-[(1R)-1-(5-chloro-1H-benzimidazol-2-yl)-2-methoxy-ethyl]-3-methyl-benzamide
09/15/2005US20050203064 Novel oxidized thioether derivatives
09/15/2005US20050203030 Novel effectors of dipeptidyl peptidase IV
09/15/2005DE102004009933A1 Use of 1,3,4-thiadiazole derivatives to prepare medicaments for treating diseases in which the inhibition, regulation or modulation of kinase signal transduction plays a role
09/15/2005DE102004004972B3 Heterocyclisch substituierte 7-Amino-4-chinolon-3-carbonsäure-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel Heterocyclic-substituted 7-amino-4-quinolone-3-carboxylic acid derivatives, to processes for their preparation and their use as medicaments
09/15/2005CA2558848A1 Isoxazoline-substituted benzamide compound and pesticide
09/15/2005CA2558600A1 A substituted-trialkyl amine compound with anti-viral activity based on antagonism against a chemokine receptor cxcr4
09/15/2005CA2558278A1 Diaryl-substituted five-membered heterocycle derivative
09/15/2005CA2557858A1 Amino cyclopropane carboxamide derivatives as bradykinin antagonists
09/15/2005CA2557645A1 Caspase inhibitors and uses thereof
09/15/2005CA2557322A1 Inhibitors of hepatitis c virus ns3 protease
09/15/2005CA2557304A1 Ketoamides with cyclic p4's as inhibitors of ns3 serine protease of hepatitis c virus
09/15/2005CA2557303A1 Use of thiadiazole urea derivatives
09/15/2005CA2556692A1 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
09/15/2005CA2556387A1 Bicyclic anthranilamide derivatives useful as insecticides
09/15/2005CA2555712A1 Novel cyclic compound having 4-pyridylalkylthio group having substituted or unsubstituted amino group introduced therein
09/15/2005CA2553252A1 2-pyridinylethylcarboxamide derivatives and their use as fungicides
09/14/2005EP1574511A1 2-Pyridinylethylcarboxamide derivatives and their use as fungicides
09/14/2005EP1574510A1 Substituted pyridine herbicides
09/14/2005EP1572690A1 Thiazole compounds as integrin receptor antagonists derivatives
09/14/2005EP1572688A1 Oxazolidinone derivatives and their use as antibacterial agents
09/14/2005EP1572687A1 Antibacterial oxazolidinones
09/14/2005EP1572686A1 Anthranilic acid amide derivatives and their pharmaceutical use
09/14/2005EP1572670A1 5-substituted-pyrazine or -pyridine glucokinase activators
09/14/2005EP1572668A2 N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines
09/14/2005EP1572664A1 Pyrazole compounds
09/14/2005EP1572662A1 Pyrazole and imidazole compounds and uses thereof
09/14/2005EP1572655A2 Novel arylheteroalkylamine derivatives
09/14/2005EP1572646A1 N-(indolethyl-)cacloamine compounds
09/14/2005EP1572215A1 Benzo[d]azepine derivatives for the treatment of neurological disorders
09/14/2005EP1572207A1 N-(substituted arylmethyl)-4-(disubstituted methyl) piperidines and pyridines
09/14/2005EP1572072A2 Methods of treating infection by drug resistant bacteria
09/14/2005EP1499609A4 Pesticidal heterocycles
09/14/2005EP1461318B1 Tetrahydroquinoline analogues as muscarinic agonists
09/14/2005EP1289954B1 Serine protease inhibitors
09/14/2005CN1668605A Broadspectrum substituted benzisoxazole sulfonamide HIV protease inhibitors
09/14/2005CN1668585A 3, 6-disubstituted azabicyclo [3.1.0]hexane derivatives useful as muscarinic receptor antagonists
09/14/2005CN1668584A Pyrrole derivatives as antimycobacterial compounds
09/14/2005CN1668297A 丙型肝炎病毒抑制剂 Hepatitis C virus inhibitors
09/14/2005CN1666983A Substituted aminoquinazolinone (thione) derivatives or salts thereof, intermediates thereof, and pest contollers and a method for using the same
09/13/2005US6943187 Shampoos for treating alopecia
09/13/2005US6943184 For therapy of Alzheimer's disease, Parkinson's disease, Pick's disease, Korsakoff s disease cerebral ageing, of mood disorders, of pain and of tobacco withdrawal
09/13/2005US6943183 Antiproliferative agnets; anticancer agents; skin disorders; restenosis
09/13/2005US6943162 Osteoporosis; cardiovascular disorders; anticancer agents;incontinence
09/13/2005US6943160 Morpholine derivatives as antagonists of orexin receptors
09/13/2005US6943159 amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor agonists or antagonists such as 3-Cyclohexyl-7-(1-hydroxyethyl)-1,2,3,4-tetrahydro-1,2,4-benzothiadiazine-1,1-dioxide, used for prophylaxis of nervous system disoders
09/13/2005CA2371587C Piperidine derivatives useful as ccr5 antagonists
09/13/2005CA2358724C New cyclobutene-dione derivatives, their method of preparation and pharmaceutical compositions containing them
09/09/2005WO2005082901A1 Novel chemical compounds
09/09/2005WO2005082900A2 Oxazolidinone amidoximes as antibacterial agents
09/09/2005WO2005082899A1 Oxazolidinone derivatives as antimicrobials
09/09/2005WO2005082897A1 Oxazolidinone antibacterial agents
09/09/2005WO2005082895A1 Novel carboxamides for use as xa inhibitors
09/09/2005WO2005082889A1 Piperidinyl targeting compounds that selectively bind integrins
09/09/2005WO2005082887A1 Pyrimidine derivative
09/09/2005WO2005082884A2 2-pyridin-2yl-pyrimidine derivatives useful in the treatment of gastro-esophagea l reflux disease
09/09/2005WO2005082871A2 Guanidine compounds, and use thereof as binding partners for 5-ht5 receptors
09/09/2005WO2005082865A1 Fused bicyclic pyrimidine derivative
09/09/2005WO2005082864A1 1,4-diaryl-dihydropyrimidin-2-ones and their use as human neutrophil elastase inhibitors
09/09/2005WO2005082859A1 6-substituted 2,3,4,5-tetrahydro-1h-benzo[d]azepines as 5-ht2c receptor agonists
09/09/2005WO2005082858A2 Isoquinoline derivatives
09/09/2005WO2005082856A2 Tetrahydroquinolinones and their use as antagonists of metabotropic glutamate receptors
09/09/2005WO2005082023A2 Heterocyclic self-immolative linkers and conjugates
09/09/2005WO2005068444A3 Thiazole derivatives and use thereof