Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773) |
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08/17/2005 | CN1215069C Sulfonamicles and derivatives thereof that moulate the activity of endothelin |
08/17/2005 | CN1215061C Process for preparing anticancer compound, and intermediate |
08/16/2005 | US6930185 Anorectic agents; obesity; such as 4'-chloro-N-(6-((N,N-dimethylamino)methyl)-2-naphthyl)(1,1'-biphenyl)-4 -carbox-amide |
08/16/2005 | US6930131 Hetero or aromatic-alkyloxyalkylphenylsulfonamide or analogs or derivatives useful in treating metabolic disorders mediated by insulin resistance or hyperglycemia |
08/16/2005 | US6930117 N-alkyl-4-methyleneamino-3-hydroxy-2-pyridones |
08/16/2005 | US6930116 Such as 4-chloro-5-(2-phenyl-thiazol-5-yl)-2H-pyrazole-3-carboxylic acid ethyl amide; for inhibiting topoisomerases; treating bacterial infections in mammals |
08/16/2005 | US6930111 Substituted heterocyclic compounds |
08/16/2005 | US6930107 treating obesity, overweight condition, hyperlipidemia, thyroid disease, hypothyroidism, thyroid cancer and related disorders |
08/16/2005 | US6930104 beta -amyloid precursor protein secretory stimulators; treating neurodegenerative disorders; n-carbamoyl- quinoxaline or quinoline derivatives |
08/16/2005 | US6930102 16-halogen-epothilone derivatives, process for their production, and their pharmaceutical use |
08/16/2005 | CA2342974C Methods and compositions for inhibition of angiogenesis |
08/16/2005 | CA2323703C New cyano-indole serotonin reuptake inhibitors, the procedure for preparing them and the pharmaceutical formulations that contain them |
08/16/2005 | CA2220438C (n-(pyridinylmethyl)-heterocyclic)ylideneamine compounds as nicotinic acetylcholine receptor binding agents |
08/11/2005 | WO2005073230A1 Heterocyclically substituted 7-amino-4-quinolone-3-carboxylic acid derivatives, method for the production thereof and their use as medicaments |
08/11/2005 | WO2005073227A2 A process for the preparation of 5-[4-[2-[n-methyl-n-(2-pyridyl) amino] ethoxy] phenyl methyl] thiazolidine-2, 4-dione maleate |
08/11/2005 | WO2005073226A1 Acylaminothiazole derivatives, preparation method thereof and use of same in therapeutics |
08/11/2005 | WO2005073225A1 2-(3-substituted-aryl)amino-4-aryl-thiazoles as tyrosine kinase inhibitors |
08/11/2005 | WO2005073224A2 Quinoline quinazoline pyridine and pyrimidine counds and their use in the treatment of inflammation angiogenesis and cancer |
08/11/2005 | WO2005073216A2 Hcv ns-3 serine protease inhibitors |
08/11/2005 | WO2005073203A1 MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1, AND/OR NF-κB ACTIVITY AND USE THEREOF |
08/11/2005 | WO2005073202A1 Acylaminothiazole derivatives and use thereof as beta-amyloid inhibitors |
08/11/2005 | WO2005073195A2 Hcv ns-3 serine protease inhibitors |
08/11/2005 | WO2005073192A1 Novel piperidines as chemokine modulators (ccr) |
08/11/2005 | WO2005072732A1 Modulators of the glucocorticoid receptor, ap-1, and/or nf-kb activity and use thereof |
08/11/2005 | WO2005072729A1 Modulators of glucocorticoid receptor, ap-1, and/or nf-kb activity and use thereof |
08/11/2005 | WO2005072376A2 Anionic-sweetener-based ionic liquids and methods of use thereof |
08/11/2005 | WO2005072308A2 Cgrp receptor antagonists |
08/11/2005 | WO2005072132A2 TRICYCLIC MODULATORS OF THE GLUCOCORTICOID RECEPTOR, AP-1, AND/OR NF-κB ACTIVITY AND USE THEREOF |
08/11/2005 | WO2005051302A3 Bicyclic inhibitors of mek and methods of use thereof |
08/11/2005 | WO2005034856A3 Targeted drug-formaldehyde conjugates and methods of making and using the same |
08/11/2005 | WO2005020897A3 Compositions and methods for the treatment of disease associated with trp-p8 expression |
08/11/2005 | US20050176965 Process for preparing 2-aminothiazole-5-carboxamides useful as kinase inhibitors |
08/11/2005 | US20050176964 Nicotinamide derivatives useful as p38 inhibitors |
08/11/2005 | US20050176801 Acyl bicyclic derivatives of pyrrol |
08/11/2005 | US20050176799 drugs such as 1-Benzyl-3-(2-furyl)-5-trifluoromethylpyrazole, capable of modulating biosynthesis of cyclic guanosine monophosphate, used for therapy and prophylaxis of cardiovascular disorders such as hypertension, angina pectoris, cardiac insufficiency, thrombosis or atherosclerosis |
08/11/2005 | US20050176789 Modulators of ATP-Binding Cassette transporters |
08/11/2005 | US20050176787 Thiazolidinediones alone or in combination with other therapeutic agents for inhibiting or reducing tumour growth |
08/11/2005 | US20050176776 Mitotic kinesin inhibitors |
08/11/2005 | US20050176775 Substituted pyridinones |
08/11/2005 | US20050176773 Antimetastasis agents e.g. 6-[4-Amino-5-(2,6-difluoro-benzoyl)-thiazol-2-ylamino]-N-2-dimethylamino-2-methyl-propyl)-nicotinamide; protein kinase inhibitor |
08/11/2005 | US20050176767 Pyridine carboxamide and methods for inhibiting HIV integrase |
08/11/2005 | US20050176765 For therapy of glaucoma, dementia such as Alzheimer's disease and vascular dementia, depression, attention deficit disorder, sleep disorder, schizophrenia, pain, ischemia; -[1-[1-(3-Thienoyl)piperidin-4-yl]piperidin-4-yl]-1,3-dihydro-2H-benzimidazol-2-one |
08/11/2005 | US20050176763 Administering a therapeutically effective amount of 3-thia-4-(2-oxy/hydroxyphenyl)quinolin-2-one derivative to a patient to treat erectile dysfunction or irritable bowel syndrome |
08/11/2005 | US20050176762 Tachykinin receptor subtypes NK3 and NK2 (NK neurokinin); various diseases including respiratory system disorders, autoimmune disorders, psychological disorders, skin disorders |
08/11/2005 | US20050176749 Modulators of glucocorticoid receptor, AP-1, and/or NF-kB activity and use thereof |
08/11/2005 | US20050176727 Male erectile dysfunction; 1-(3-chlorophenyl)-3-(4-pyridin-2-yl-piperazin-1-yl)propan-1-one O-methyloxime |
08/11/2005 | US20050176726 Pyrimidine ether derivatives; antiinflammatory; analgesic; antiarthritis; antirheumatic;diseases involving sensory nerve function; 2-((6-(4-((1S)-1-(4-fluorophenyl)ethyl)-1-piperazinyl)-4-pyrimidinyl)oxy)quinoline |
08/11/2005 | US20050176722 Piperazinylacylpiperidine derivatives, their preparation and therapeutic use thereof |
08/11/2005 | US20050176719 An enzyme inhibitors of cyclin-dependent kinases, antitumor agents; chemical intermediate synthesis |
08/11/2005 | US20050176716 (2,3-5,6 aryl-heteroaryl)-bicyclo(2,2,2,)octane-amide derivatives; antiinflammatory, obesity, antidiabetic agent, autoimmune disease, asthma, arthritis; non-steroidal; side effect reduction; pharmacokinetics |
08/11/2005 | US20050176713 Amide derivatives as glycogen synthase kinase 3-beta inhibitors |
08/11/2005 | US20050176712 Integrin expression inhibitor |
08/11/2005 | US20050176709 Selective NPY (Y5) antagonists |
08/11/2005 | US20050176705 5-Chloro-1-(3,5-dichloro-2-methoxy benzenesulfonyl)-4-piperazin-1-yl-1H-indole trifluoroacetic acid salt; 5-hydroxytryptamine (serotonin) HT6 receptor antagonists; antidepressant, anxiolytic agent, cognition activator; ADHD, Alzheimer's and Parkinson's disease, drug and nicotine abuse |
08/11/2005 | US20050176701 Inhibitors of hepatitis C virus RNA-dependent RNA polymerase, and compositions and treatments using the same |
08/11/2005 | US20050176699 Benzodiazepine derivatives, preparation thereof and use thereof |
08/11/2005 | DE102004003812A1 Arylsubstituierte Heterozyklen, Verfahren ihrer Herstellung und ihre Verwendung als Arzneimittel Aryl substituted heterocycles, processes for their preparation and their use as medicaments |
08/11/2005 | CA2554925A1 2-(3-substituted-aryl)amino-4-aryl-thiazoles as tyrosine kinase inhibitors |
08/11/2005 | CA2554525A1 Heterocyclically substituted 7-amino-4-quinolone-3-carboxylic acid derivatives, method for the production thereof and their use as medicaments |
08/11/2005 | CA2554389A1 Anionic-sweetener-based ionic liquids and methods of use thereof |
08/11/2005 | CA2554351A1 Cgrp receptor antagonists |
08/11/2005 | CA2553433A1 Quinoline quinazoline pyridine and pyrimidine compounds and their use in the treatment of inflammation angiogenesis and cancer |
08/11/2005 | CA2553089A1 Novel piperidines as chemokine modulators (ccr) |
08/11/2005 | CA2552317A1 Hcv ns-3 serine protease inhibitors |
08/11/2005 | CA2551142A1 Acylaminothiazole derivatives, preparation method thereof and use of same in therapeutics |
08/10/2005 | EP1561749A1 TNF-Alpha production inhibitors for the treatment of autoimmune diseases |
08/10/2005 | EP1560827A1 Anti-infective agents |
08/10/2005 | EP1560822A1 4-imidazol-1-ylmethyl-pyrimidine derivatives as ligands for gabaa receptors |
08/10/2005 | EP1560817A1 Methods and compositions of novel triazine compounds |
08/10/2005 | EP1560811A2 Pharmaceutical compositions as inhibitors of dipeptidyl peptidase-iv (dpp-iv) |
08/10/2005 | EP1560580A1 Sulfonamides, sulfamates and sulfamides as gamma-secretase inhibitors |
08/10/2005 | EP1560576A2 Synthesis of oligomeric epicatechin and catechin-derived procyanidins |
08/10/2005 | EP1368340B1 Piperazine derivatives as melanocortin receptor agonists |
08/10/2005 | EP1098891B1 Polycyclic thiazolidin-2-ylidene amines, method for the production and use thereof as medicaments |
08/10/2005 | CN1653054A Benzoxazine derivatives as 5-HT6 modulators and uses thereof |
08/10/2005 | CN1653053A Broadspectrum substituted benzimidazole sulfonamide HIV protease inhibitors |
08/10/2005 | CN1653051A Substituted anthranilamides for controlling invertebrate pests |
08/10/2005 | CN1653049A Pesticidal pyridinecarboxamide derivatives |
08/10/2005 | CN1653048A Pyridine carboxamide derivatives and their use as pesticides |
08/10/2005 | CN1653046A 8-azaprostaglandin derivative compounds and drugs containing the compounds as the active ingredient |
08/10/2005 | CN1652788A Method of treating diabetes |
08/10/2005 | CN1652787A Compositions and methods for combating lower urinary tract dysfunctions with delta opioid receptor agonists |
08/10/2005 | CN1652780A Diaminothiazoles used as CDK4 inhibitors |
08/10/2005 | CN1652776A N3 alkylated benzimidazole derivatives as MEK inhibitors |
08/10/2005 | CN1651392A 2-and 2, 5-substituted phenylketoenols |
08/10/2005 | CN1214040C Peptide derivatives having thiazolyl-alanine residue |
08/10/2005 | CN1214026C Indol-3-yl derivatives |
08/10/2005 | CN1213658C Picolinamide derivatives and pest controllers containing same as active ingredient |
08/09/2005 | US6927230 Triazole derivatives |
08/09/2005 | US6927229 Difluorothioacetamides of oxazolidinones as antibacterial agents |
08/09/2005 | US6927228 Biphenyl compounds usefuf in treatment of human and veterinary medicines such as dermatology, cardivovascular diseases, immune diseases or diseases associated with lipid metabolisms, or in cosmetic formulation |
08/09/2005 | US6927225 Fungicidal 2-pyridyl alkyl amides and their compositions, methods of use and preparation |
08/09/2005 | US6927216 Treatment of inflammatory disorders |
08/09/2005 | US6927214 Non-peptide GLP-1 agonists |
08/09/2005 | CA2231700C Prodrugs of aspartyl protease inhibitors |
08/09/2005 | CA2188164C Benzamide compounds and pharmaceutical use thereof |
08/04/2005 | WO2005070934A1 Substituted diazabicycloheptanes and their use as protein kinase inhibitors |
08/04/2005 | WO2005070929A1 Vanilloid receptor ligands and their use in treatments |
08/04/2005 | WO2005070926A1 Thiazole derivatives as a2b antagonists |
08/04/2005 | WO2005070925A1 Aryl substituted heterocycles, method for production and use thereof as medicaments |