Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
02/2006
02/01/2006EP1620410A1 Use of derivatives of 2, 4-dihydro- 1,2,4 triazole-3-thione as inhibitors of the enzyme myeloperoxidase (mpo)
02/01/2006EP1620091A2 Inhibitors of glutaminyl cyclase
02/01/2006EP1620088A2 Indole acetic acid derivatives and their use as pharmaceutical agents
02/01/2006EP1620086A1 Compounds that modulate ppar activity and methods of preparation
02/01/2006EP1500654B1 Benzoxazinone derivatives, the preparation and use thereof as medicaments
02/01/2006EP1119563B1 Tetrahydrobenzazepine derivatives useful as modulators of dopamine d3 receptors (antipsychotic agents)
02/01/2006CN1729178A N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines
02/01/2006CN1729177A New uracils having a herbicidal activity
02/01/2006CN1729173A N-(indolethyl-) cacloamine compounds
02/01/2006CN1728999A Substituted 1-piperidin-3-yl-4-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists
02/01/2006CN1239501C A thiazolidniedione derivative and its use as antidiabetic
02/01/2006CN1239497C Intermediate product for preparing aralkyl and aryl alkylene heterocyclic lactam and imide
02/01/2006CN1239496C Respiratory syncytial virus replication inhibitors
01/2006
01/31/2006US6992191 Hydrogenation of precursors to thiazolidinedione antihyperglycemics
01/31/2006US6992097 such as methyl-1-{2-[4-((2R)-2-{2-[(tert-butoxy)carbonylamino]-2-methylpropanoylamino}-3-indol-3-ylpropanoylamino)imidazolyl]-2-phenylacetyl}pyrrolidine-2-carboxylate
01/31/2006US6992082 for treatment of cellular proliferative diseases such as cancer, hyperplasias, restenosis, cardiac hypertrophy, immune disorders and inflammation
01/31/2006CA2224635C Pyridine derivatives, process for preparing the same, and intermediate therefor
01/31/2006CA2119261C Novel sidechain-bearing taxanes and intermediates thereof
01/26/2006WO2006008260A1 Dimeric piperidine derivatives
01/26/2006WO2006008259A1 Dimeric compounds of piperidine, piperazine or morpholine or their 7-membered analogs suitabale for the treatment of neurodegenerative disorders
01/26/2006WO2005118579A3 Thiazole derivatives as chemokine receptor antagonists
01/26/2006WO2005116009B1 Substituted 2-quinolyl-oxazoles useful as pde4 inhibitors
01/26/2006WO2005097787A3 Novel benzothiazoles and the use thereof as medicaments
01/26/2006WO2005097134A3 Quinazoline based protein kinase inhibitors
01/26/2006WO2005092304A3 Antifungal agents
01/26/2006WO2005085234A3 Bycyclic anthranilamide derivatives useful as insecticides
01/26/2006WO2005077922A3 Process for the preparation of substituted triazole compounds
01/26/2006WO2004096798A3 Derivatives of 2-acylamino-4-phenylthiazole, preparation method thereof and use of same as chemokine antagonists
01/26/2006US20060020138 E.g., 3-arylmethyl-7-hydroxy-coumarins as intermediates; affects both the Tumor Necrosis Factor alpha level and transcription activity of NuclearFactor kappa Beta; antiimmunoinflammatory agents and autoimmune properties; antiarthritis agents; rheummatic diseases; osteoporosis; leukemia
01/26/2006US20060020132 high binding efficiencies between D3 and D2 dopaminergic receptor subtypes; drug abuse, drug dependence
01/26/2006US20060020008 Compounds, compositions and methods
01/26/2006US20060020000 N,N-Dibutyl-2-[3-(2,2-dimethylpropanoyl)-6-methoxy-1H-indazol-1-yl]acetamide; potassium channel blocker; eye neuroprotectant; hypotensive agent; glaucoma, intraoccular pressure in the eye
01/26/2006US20060019994 I-sulphonlyl piperidine derivatives
01/26/2006US20060019970 Methods and compositions for the treatment of neuroleptic and related disorders using ziprasidone metabolites
01/26/2006US20060019950 Benzathiazol-acetamides
01/26/2006US20060019947 Therapeutic chromone compounds
01/26/2006US20060018846 Animo substituted hydroxyphenyl benzophenone derivatives
01/26/2006US20060018825 Probe for diseases with amyloid accumulation, amyloid-staining agent, remedy and preventive for diseases with amyloid accumulation and diagnostic probe and staining agent for neurofibrillary change
01/26/2006DE102004033312A1 Kontinuierliches Metatheseverfahren mit Ruthenium-Katalysatoren Continuous metathesis with ruthenium catalysts
01/26/2006CA2574193A1 Benzothiazole derivatives as adenosine receptor ligands
01/26/2006CA2573210A1 Viral polymerase inhibitors
01/26/2006CA2572822A1 Dimeric piperidine derivatives
01/26/2006CA2572821A1 Dimeric compounds of piperidine, piperazine or morpholine or their 7-membered analogs suitable for the treatment of neurodegenerative disorders
01/26/2006CA2570968A1 Gonadotropin releasing hormone receptor antagonists
01/26/2006CA2567569A1 Selective inhibitors against cdk4 and cdk6 having aminothiazole skeleton
01/25/2006EP1618099A2 Biaryl substituted thiazoles, oxazoles and imidazoles as sodium channel blockers
01/25/2006EP1618094A1 Substituted heteroaryls as inhibitors of protein tyrosine phosphatases
01/25/2006EP1618093A2 Indazole derivatives as jnk inhibitors
01/25/2006EP1506179B1 Benzoxazine derivatives as 5-ht6 modulators and uses thereof
01/25/2006EP1235825B1 Novel benzoimidazole derivatives useful as antiproliferative agents
01/25/2006EP1135127B1 New pharmaceutical composition and the process for its preparation
01/25/2006EP0978392B1 Optical recording media
01/25/2006EP0914158B2 Pharmaceutical combination containing a compound having angiotensin ii antagonistic activity and a compound which increases the insulin-sensitivity
01/25/2006CN1726207A Substituted 1-piperidin-4-yl-4-pyrrolidin-3-yl-piperazine derivatives and their use as neurokinin antagonists
01/25/2006CN1726205A 2-substituted quinazolin-4-ylamine analogues as capsaicin receptor modulators
01/25/2006CN1726197A 5-substituted-pyrazine or -pyridine glucokinase activators
01/25/2006CN1726042A Benzo[d]azepine derivatives for the treatment of neurological disorders
01/25/2006CN1238347C Heterocyclic derivatives
01/25/2006CN1238343C Pyrimidine derivatives and herbicides containing the same
01/24/2006US6989452 Anticancer agents
01/24/2006US6989451 Substituted isothiazole compounds are useful for treating the diseases associated with abnormality in protein kinases(especially MAP kinases)
01/24/2006US6989450 Aldol condensation of a ketonic compound containing free or protected alcohol group with a acid or or metallic salt group containing compound to form intermediate, performing macrolactonizing of the intermediate
01/24/2006US6989398 Benzanilides as potassium channel openers
01/24/2006US6989391 Lactam-containing compounds and derivatives thereof as factor Xa inhibitors
01/24/2006US6989385 Pyrazole compounds useful as protein kinase inhibitors
01/24/2006US6989384 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
01/24/2006US6989379 Selective NPY (Y5) antagonists
01/24/2006CA2166415C Acylated aminophenylsulfonylureas; preparation and use as herbicides and plant growth regulators
01/24/2006CA2123093C Sulfonamide herbicides
01/19/2006WO2006006741A1 Fused benzamide compound and vanilloid receptor 1 (vr1) activity inhibitor
01/19/2006WO2006006573A1 Filter and cyanine compound
01/19/2006WO2006005914A1 2, 4, 6-trisubstituted pyrimidines as phosphotidylinositol (pi) 3-kinase inhibitors and their use in the treatment of cancer
01/19/2006WO2006005444A1 Cationic metal complexes for use as light-absorbing compounds in the information layer of optical data carriers
01/19/2006WO2005097746A3 2-propene-1-ones as hsp 70 inducers
01/19/2006WO2005095357A3 Pyrimidine derivatives and methods of treatment related to the use thereof
01/19/2006US20060014962 Thiadiazole compound and use thereof
01/19/2006US20060014958 4-Aminothiazole derivatives
01/19/2006US20060014948 e.g 1-[3,5-bis(trifluoromethyl)benzoyl]-2-[3-[(2-methoxyethoxy)-methoxy]-4-methylbenzyl]-4-[2-[(3R)-3-methoxymethyl-morpholino]ethyl]piperazine; treating or preventing Tachykinin-mediated diseases in humans or animals
01/19/2006US20060014836 e.g. 1-(Benzofuran-2-carbonyl-3-(3-phenoxy-phenyl)-thiourea;viricides; hepatitis virus
01/19/2006US20060014796 Epothilone derivatives
01/19/2006US20060014794 CXCR1 and CXCR2 chemokine antagonists
01/19/2006US20060014792 Heterocyclo inhibitors of potassium channel function
01/19/2006US20060014783 Sulfonylamino-acetic acid derivatives
01/19/2006US20060014781 Thiazole, imidazole and oxazole compounds and treatments of disorders associated with protein aging
01/19/2006US20060014755 17 Beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
01/19/2006US20060014749 (R)-2-{4-[(1H-Indol-2-ylmethyl)-amino]-piperidin-1-yl}-1-(6-methoxyquinolin-4-yl)-ethanol; effective against both gramnegative and grampositive bacteria
01/19/2006US20060014743 Methods of preventing bacterial infections with florfenicol-type antibiotics
01/19/2006US20060014740 Analogs exhibiting inhibition of cell proliferation, methods of making, and uses thereof
01/19/2006US20060014736 Phenothiazine kinesin inhibitors
01/19/2006US20060013860 Anticancer agents; side effect reduction
01/19/2006DE102004031323A1 Substituierte Pyridazincarboxamide und Derivate hiervon And derivatives thereof substituted Pyridazincarboxamide
01/19/2006DE102004023332A1 Chinoxalin-2-on-derivate, diese enthaltende nutzpflanzenschützende Mittel und Verfahren zu ihrer Herstellung und deren Verwendung Quinoxalin-2-one derivatives, useful-plant-protecting compositions containing them and processes for their preparation and their use
01/19/2006CA2571748A1 2, 4, 6-trisubstituted pyrimidines as phosphotidylinositol (pi) 3-kinase inhibitors and their use in the treatment of cancer
01/18/2006EP1615919A1 7-([1,4]dioxan-2-yl)-benzothiazole derivatives as adenosine receptor ligands
01/18/2006EP1615918A1 Process for preparing a polymorph of rosiglitazone maleate
01/18/2006EP1615909A1 Piperazine derivatives and their use for the treatment of neurological and psychiatric diseases
01/18/2006EP1615907A1 5-amino-2-carbonylthiophene derivatives for use as p38 map kinase inhibitors in the treatment of inflammatory diseases
01/18/2006EP1615906A1 Compositions useful as inhibitors of protein kinases
01/18/2006EP1615900A1 Benzisothiazol-3-one-carboxylic acid amides as phospholipase inhibitors
01/18/2006EP1615899A1 Alpha-substituted carboxylic acids as ppar modulators