Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
02/2008
02/27/2008CN101133054A 1,3-thiazole-5-carboxamides useful as cancer chemotherapeutic agents
02/27/2008CN101133036A Novel benzimidazole derivatives useful as selective androgen receptor modulators (SARMS)
02/27/2008CN101133027A Pyridine-2-carboxamide derivatives as mglur5 antagonists
02/27/2008CN101130526A Aryl carbonyl derivatives as therapeutic agents
02/27/2008CA2660758A1 Morpholino pyrimidine derivatives useful in the treatment of proliferative disorders
02/26/2008US7335775 Effector conjugates, process for their production and their pharmaceutical use
02/26/2008US7335774 Quinolinone derivatives
02/26/2008US7335753 Bifunctional heterocyclic compounds and methods of making and using same
02/26/2008US7335677 Inhibitors of dipeptidyl peptidase IV
02/26/2008US7335674 Benzothiazole-4,7-diones and benzoxazole-4,7-diones with substituents in position 5 or 6 and method for production thereof
02/26/2008US7335670 Specific inhibitors of the glycine transporters glyt1 and/or glyt2; psychoses, contracture, pain, Parkinson's disease, epilepsy, and sleep apnea
02/26/2008US7335660 Using a 2-benzopyran-6-carboxamide compound
02/26/2008US7335657 Cytokine inhibitors
02/26/2008US7335656 Medical devices employing triazine compounds and compositions thereof
02/26/2008US7335652 Introducing into the subject a ligand capable of labelling aggregated paired helical filament (PHF) tau protein, determining the presence and\or amount of ligand bound to extracellular aggregated PHF tau in the medial temporal lobe of the brain, correlating the result of the determination
02/26/2008US7335649 3-{N'-[1-(3,4-dimethylphenyl)-3-methyl-5-oxo-1,5-dihydropyrazol-4-ylidene]hydrazino}-2-hydroxy-3'-(tetrazol-5-yl)biphenyl for treatment of thrombocytopenia; colony stimulating factors
02/21/2008WO2008022002A2 2-amido-4-isoxazolyl thiazole compounds exhibiting atp-utilizing enzyme inhibitory activity, and compositions, and uses thereof
02/21/2008WO2008021338A2 Tricyclic oxazolidone derivatives useful as pr modulators
02/21/2008WO2008021337A1 Oxazinan-2-one derivatives useful as pr modulators
02/21/2008WO2008021309A1 Imidazolidin-2-one derivatives useful as pr modulators
02/21/2008WO2008020902A1 Substituted spirocyclic cgrp receptor antagonists
02/21/2008WO2008020229A2 Antibacterial pyrrolecarboxamides
02/21/2008WO2008020227A2 Antibacterial pyrrolecarboxamides
02/21/2008WO2008020222A1 Pyrrole derivatives with antibacterial activity
02/21/2008WO2008019477A1 Viral polymerase inhibitors
02/21/2008WO2007146981A3 2-anilino-4-(heterocyclic)amino-pyrimidines as inhibitors of protein kinase c-alpha
02/21/2008WO2007130064A8 2-n-(5-[[4-(2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2,4-thiazolidinedione) butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
02/21/2008WO2007121389A3 4,4-disubstituted piperidine derivatives as nk-i and serotonin transporter inhibitors
02/21/2008WO2007101213A3 Novel 2-oxo-1,2,3,4-tetrahydropyrimidines, bicyclic pyrimidine diones and imidazolidine-2,4-diones useful as inducible nitric oxide synthase inhibitors
02/21/2008WO2006130493A8 Heterocycles useful as modulators of ion channels
02/21/2008US20080045578 2-(4,4-Dimethyl-2-oxo-1,3-oxazolidin-3-yl)-4,5-dihydronaphtho[1,2-d] [1,3]thiazole-7-carbonitrile; progesterone receptor (PR); contraception, fibroids, endometriosis, dysfunctional bleeding, uterine leiomyomata, polycystic ovary syndrome, or hormone-dependent carcinomas, hormone replacement therapy
02/21/2008US20080045577 4-[2-(3,5,5-Trimethyl-2-oxoimidazolidin-1-yl)-1,3-thiazol-4-yl]benzonitrile; 1-[4-(4-Bromophenyl)-1,3-thiazol-2-yl]-3-methylimidazolidin-2-one; contraception, fibroids, endometriosis, dysfunctional bleeding, uterine leiomyomata, polycystic ovary syndrome, or hormone-dependent carcinomas
02/21/2008US20080045576 Therapeutic n-aryl or n-heteroaryl pyrazolidine and pyrazolidinone derivatives
02/21/2008US20080045560 Pyrrolidine and related derivatives useful as PR modulators
02/21/2008US20080045528 6-o-substituted benzoxazole and benzothiazole compounds and methods of inhibiting csf-1r signaling
02/21/2008US20080045524 Selective NPY (Y5) antagonists
02/21/2008US20080045516 Viral Polymerase Inhibitors
02/21/2008US20080045505 1-(isopropyl)-4-{[4-(tetrahydro-2H-pyran4-yloxy)phenyl]carbonyl}hexahydro-1H-1,4-diazepine, used in the treatment of nervous system and psychological disorders such as Alzheimer's disease or as cognition activators
02/21/2008US20080045503 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
02/21/2008US20080045493 such as Parkinson's disease, schizophrenia, cognitive disorders, depression, anxiety, drug addiction, eating disorders and urogenital disorders; 4-(2,2-Difluoro-cyclopropyl)-N-[4-(1-propyl-piperidin-3-yl)-phenyl]-benzenesulfonamide
02/21/2008CA2660555A1 Viral polymerase inhibitors
02/21/2008CA2660318A1 Modulators of glucocorticoid receptor, ap-1, and/or nf-kb activit y and use thereof
02/21/2008CA2659299A1 Azetidine compounds
02/21/2008CA2659276A1 2-amido-4-isoxazolyl thiazole compounds exhibiting atp-utilizing enzyme inhibitory activity, and compositions, and uses thereof
02/21/2008CA2659208A1 Oxazolidone derivatives as pr modulators
02/21/2008CA2650932A1 Substituted spirocyclic cgrp receptor antagonists
02/20/2008EP1889844A2 Polymorphic forms of ziprasidone sulphates
02/20/2008EP1889843A1 Bisheterocycle tandem compounds useful as antiviral agents, the uses thereof and the compositions comprising such compounds
02/20/2008EP1889842A1 Heterocyclic compound
02/20/2008EP1889838A1 Thrombopoietin mimetics
02/20/2008EP1889619A1 Use of thiadiazolidine-derived compounds as neurogenic agents
02/20/2008EP1888576A1 Process for making aztreonam
02/20/2008EP1888575A2 Compounds for modulating trpv3 function
02/20/2008EP1888574A2 New antibiotic derivatives
02/20/2008EP1888573A1 Thiazole derivatives and use thereof
02/20/2008EP1888567A1 Heteroaryl-carboxylic acid (sulfamoyl alkyl) amide - derivatives as factor xa inhibitors
02/20/2008EP1888565A2 2, 6-di (hetero) aryl -4-amido-pyrimidines as adenosine receptor antagonists
02/20/2008EP1888558A1 Bicyclic derivatives as modulators of ion channels
02/20/2008EP1888547A1 Indane derivatives as modulators of ion channels
02/20/2008EP1888546A1 Thiazole derivatives and use thereof
02/20/2008EP1888542A1 Substituted spiro-compounds and the use thereof for producing medicaments
02/20/2008EP1888531A2 (5z)-5-(6-quinoxalinylmethylidene)-2-ý(2,6-dichlorophenyl)amino¨-1,3-thiazol-4(5h)-one
02/20/2008EP1888530A2 Quinoline derivatives as neurokinin receptor antagonists
02/20/2008EP1888528A2 Phosphodiesterase 4 inhibitors
02/20/2008EP1740569B1 Imidazole derivatives used as tafia inhibitors
02/20/2008EP1556381B1 Pyrazole amides for treating hiv infections
02/20/2008EP1305310B1 Tartrate salts of thiazolidinedione derivative
02/20/2008CN101128460A Tricyclic delta-opioid modulators
02/20/2008CN101128457A 凝血酶受体拮抗剂 Thrombin receptor antagonists
02/20/2008CN101128445A 4-cyclopropyl-1,2,3-thiadiazole derivative, agrohorticultural plant disease controlling agent, and method for using the same
02/20/2008CN101128439A 1,6 - substituted (3r,6r) -3- (2,3-dihydro-1h-inden-2-yl)-2,5-piperazinedione derivatives as oxytocin receptor antagonists for the treatment of pre-term labour, dysmenorrhea and endometriosis
02/20/2008CN101128432A Tetrahydroisoquinoline compounds for treatment of cns disorders
02/20/2008CN101125853A Sodium salts of 5-[4-[2-(n-methyl-n-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione
02/20/2008CN101125852A Sodium salts of 5-[4-[2-(n-methyl-n-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione
02/20/2008CN101125851A Novel pharmaceutical
02/20/2008CN100369904C 2-(replace- amino)-NOBS HIV prolease inhibitor
02/20/2008CN100369903C Five-membered-ring compound
02/20/2008CN100369898C Nicotinamide derivates useful as p38 inhibitors
02/19/2008US7332614 Process for cross coupling indoles
02/19/2008US7332602 Pyridyl substituted heterocycles useful for treating or preventing HCV infection
02/19/2008US7332521 Substituted indoles
02/19/2008US7332520 Fused indoles as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
02/19/2008US7332517 1-(1H-indol-3-ylmethyl)-3-(4-nitrophenyl)-5-[2-(4-phenyl-1H-imidazol-2-yl)ethyl]-2thioxo-4imidazolidinone; somastatin receptor affinity; acromegaly, hypophyseal adenomas, endocrine gastroenteropancreatic tumors, as carcinoid syndrome and gastrointestinal bleeding
02/19/2008US7332513 N-[4-Methyl-5-(2-nitrooxy-ethyl)-thiazol-2-yl]-formamide for example; compound forms a naturally occurring metabolite when NO is released to slow or prevent drug tolerance; treating cardiovascular diseases, inflammation, psychiatric and neurological diseases, respiratory diseases, urogenital disorders
02/19/2008US7332512 Halogenated nitrobutadienes for controlling animal pests
02/19/2008US7332511 Vanilloid receptor ligands and their use in treatments
02/19/2008US7332499 N-[(1R)-1-(2-fluoro-4-{1-[(trifluoromethyl)sulfonyl]-1,2,3,4-tetrahydroquinolin-8-yl}phenyl)ethyl]-1-[(trifluoroacetyl)amino]cyclopropanecarboxamide; bradykinin B1 antagonists or inverse agonists; analgesic and antiinflammatory agent; acute and chronic pain
02/19/2008US7332493 [3-Methyl-4-(pyridin-3-yloxy)-phenyl]-(6-piperidin-3-ylethynyl-quinazolin-4-yl)-amine; selective inhibitors of receptor tyrosine kinases and non-receptor tyrosine kinases (eg: Ick, src, abl) or serine/threonine kinases (e.g.: cyclin dependent kinases); carcinoma
02/19/2008US7332492 Amino substituted dibenzothiophene derivatives for the treatment of disorders mediated by NP Y5 receptor
02/19/2008US7332490 inhibit smooth muscle cell proliferation by modulating Heparan Sulfate Proteoglycans (HSPGs); inhibit or block glycated protein and Advanced Glycation Endproducts (AGE) produced induction of the signaling-associated inflammatory response in endothelial cells; antiproliferative and antiinflammatory agent
02/19/2008US7332489 Methods and compositions of novel triazine compounds
02/19/2008US7332488 Methods and compositions of novel triazine compounds
02/19/2008US7332487 Nitrogen-containing 5-membered ring compound
02/19/2008US7332484 2,4-pyrimidinediamine compounds and their uses
02/19/2008US7332483 3-(5-benzamido-2-chlorophenyl)-7-methoxy-3,4-dihydroquinazolin-4-one;cytokines (tumor necrosis factor and interleukins) inhibitor; antiinflammatory agent, rheumatoid arthritis, osteoarthritis, psoriasis, chronic obstructive pulmonary disease
02/19/2008US7332481 Thrombopoietin mimetics
02/19/2008US7332354 bioconjugation; luciferins; biopolymer labels
02/19/2008CA2207100C Pyrimidine derivatives
02/14/2008WO2008018639A2 Glycine transporter inhibitor
02/14/2008WO2008017852A1 Diamine-containing, tetra- substituted piperazine compounds as melanocortin receptor modulators