Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
03/2008
03/27/2008WO2008034891A2 Novel genes related to glutaminyl cyclase
03/27/2008WO2008034863A2 Sulfonylpyrazoline carboxamidine derivatives as 5-ht6 antagonists
03/27/2008WO2008034534A1 3-cyano-5-thiazaheteroaryl-dihydropyridine and the use thereof for the treatment of cardiovascular diseases
03/27/2008WO2008009405A3 Novel pyridazine derivatives
03/27/2008WO2008008431A3 Heteroaryl sulfonamides and ccr2/ccr9
03/27/2008WO2008005651A3 Cyclic carboxylic acid rhodanine derivatives for the treatment and prevention of tuberculosis
03/27/2008WO2008002674A3 Bicyclic compositions and methods for modulating a kinase cascade
03/27/2008WO2007136668A9 N-benzoyl-and n-benzylpyrrolidin-3-ylamines as histamine-3 antagonists
03/27/2008WO2007136573A3 Antidiabetic bicyclic compounds
03/27/2008WO2007117381A9 2 -aminopyridine analogs as glucokinase activators
03/27/2008WO2007109334B1 Sip receptor modulating compounds and use thereof
03/27/2008WO2007094513A3 Cyclic amine compound and use thereof for the prophylaxis or treatment of hypertension
03/27/2008WO2007020411A8 Amide derivatives
03/27/2008US20080076920 Preparation of thiazoles
03/27/2008US20080076817 Neurotrophic N-glyoxyl-prolyl ester compounds e.g. 3-phenyl-1-propyl (2S)-1-(3,3-dimethyl-1,2-dioxopentyl)-2-pyrrolidinecarboxylate; non-immunosuppressive; side effect reduction; neurodegenerative diseases
03/27/2008US20080076810 Benzoureas Having Anti-Diabetic Activity
03/27/2008US20080076809 Heterocyclic compound for stimulating or inducing the growth of the hair or eyelashes and/or slowing down their loss composition comprising it and its uses
03/27/2008US20080076795 1H-benzo[F]indazol-5-YL derivatives as selective glucocorticoid receptor modulators
03/27/2008US20080076771 Thrombopoietin Receptor Agonists
03/27/2008US20080076759 Therapeutic Heterocyclic Compounds 507
03/27/2008US20080076752 substituted structure of 3-amino-2-(2,5-difluorophenyl)-2,3-dihydro-1,5-benzothiazepin-4(5H)-one; 6-amino-7-phenyl-1,4-thiazepan-5-one; -amino-2-phenyl-2,3-dihydro-1,5-benzoxazepin-4(5H)-one for treating neurological disorders such as Alzheimer's; inhibit the production of amyloid beta protein
03/27/2008DE102006044696A1 3-Cyano-5-thiazaheteroaryl-dihydropyridine und ihre Verwendung 3-cyano-5-thiazaheteroaryl-dihydropyridines and their use
03/27/2008DE102006042143A1 Neue substituierte Bipyridin-Derivate und ihre Verwendung New substituted bipyridine derivatives and their use
03/27/2008CA2664411A1 Platelet adp receptor inhibitors
03/27/2008CA2663901A1 Pyridine derivatives for the treatment of metabolic disorders related to insulin resistance or hyperglycemia
03/27/2008CA2663635A1 Novel genes related to glutaminyl cyclase
03/27/2008CA2663057A1 N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
03/27/2008CA2662574A1 Heterocyclic organic compounds
03/27/2008CA2662484A1 Sulfonylpyrazole and sulfonylpyrazoline carboxamidine derivatives as 5-ht6 antagonists
03/26/2008EP1903043A1 Novel pharmaceutical
03/26/2008EP1903042A2 An improved process for hydrogenation of 5-(substituted Benzylidene) 2,4- Thiazolidine Dione compounds to give corresponding ( +/- ) 5- (substituted Benzyl ) 2,4-Thiazolidine Dione
03/26/2008EP1902713A1 Pharmaceutical composition containing thiazolidinedione compound
03/26/2008EP1902052A1 Heteroaryl benzamide derivatives for use as glk activators in the treatment of diabetes
03/26/2008EP1902051A1 Azacyclohexane derivatives as inhibitors of stearoyl-coenzyme a delta-9 desaturase
03/26/2008EP1902050A1 Oxazolidinone derivatives and use thereof as antibiotics
03/26/2008EP1902026A2 Tetrahydrocarbazole derivatives useful as androgen receptor modulators (sarm)
03/26/2008EP1902025A1 Kinase inhibitors
03/26/2008EP1901752A2 Compositions and methods for viral inhibition
03/26/2008EP1901731A1 Niacin receptor agonists, compositions containing such compounds and methods of treatment
03/26/2008EP1696924B1 Acidic quinoline derivatives and their use for the prevention and/or treatment of hyperglycaemia-related pathologies
03/26/2008EP1583763B1 Benzoazolylpiperazine derivatives having vr1-antagonist activity
03/26/2008CN101151259A Heteroaryl urea derivatives useful for inhibiting CHKI
03/26/2008CN101151249A Cyclopentapyridine and tetrahydroquinoline derivatives
03/26/2008CN101151019A Pharmaceutical preparation of n -[5-(aminosulfonyl)-4-methyl-1,3-thiazol-2-yl]-n-methyl-2-[4-(2-pyridinyl)phenyl] acetamide
03/26/2008CN100377005C Organophotoreceptor with charge transport compound with an azine group
03/26/2008CN100376572C Anti-infective agents
03/26/2008CN100376569C Inhibitors of farnesyl protein transferase
03/26/2008CN100376560C New tricyclic compounds and their use as medicine, process for their preparation and pharmaceutical compositions containing them
03/25/2008US7348440 Mitotic kinesin inhibitors
03/25/2008US7348427 Substituted with an amido heterocylic groups; infection by Gram-positive bacteria.
03/25/2008US7348426 Substituted bicyclic heterocycles, process for their preparation and their use as antiobesity and hypocholesterolemic agents
03/25/2008US7348357 bactericide; derivatives of pseudopeptide Andrimid in which beta-phenylalanine amide is replaced by heteroaromatic or substituted aromatic amide; N-{(1S)-3-[((1S)-1-{[(3R,4S)-1,4-Dimethyl-2,5-dioxo-3-pyrrolidinyl]carbonyl}-2-methylpropyl)amino]-3-oxo-1-phenylpropyl}-2-pyridinecarboxamide; antibiotics
03/25/2008US7348348 Aryl-link-aryl substituted thiazolidine-dione and oxazolidine-dione as sodium channel blockers
03/25/2008US7348347 Serotonin reuptake inhibitors; for depression and pain; 2-cyclohexyl-N-{4-[4-(2-dimethylaminoethyl)piperazin-1-carbonyl]-4,5,6,7-tetrahydrobenzthiazol-2-yl)-acetamide
03/25/2008US7348346 Use as antidiabetic agents, treating hyperglycemia, syndrome X, hyperinsulinemia, obesity, atherosclerosis; (3S, 5S)-4-([5-(Thiazolidine-3-carbonyl)-pyrrolidin-3-ylmethyl]-sulfamoyl)-benzoic acid for example
03/25/2008US7348343 N-(N-heteroaryl)1-pyridyl- or -pyrimidyl-hydropyridine-4-carboxamides; e.g., 3'-Chloro-3,6-dihydro-2H-[1,2']bipyridinyl-4-carboxylic acid (6-trifluoromethyl-pyridin-3-yl)-amide and 1-pyrimidin-2-yl-1,2,3,6-tetrahydro-pyridine-4-carboxylic acid (6-trifluoromethyl-pyridin-3-yl)-amide
03/25/2008US7348341 Chemical compounds
03/25/2008US7348340 "caused" by the stimulation of nociceptive receptors and transmitted over intact neural pathways; 2-(4-Chlorophenyl)-quinoline-4,6-diamine; acute, persistent and neuropathic pain
03/25/2008US7348327 (2S)-4,4-difluoro-1-(2-{[1-(2-pyrazinyl)piperidin-4-yl]amino}acetyl)-2-pyrrolidine carbonitrile; enzyme inhibitors; diabetes
03/25/2008US7348326 in brain; (2,5-difluorodifluorophenyl)-N-methyl-N-((1-propylbenzimidazol-2-yl)methyl)carboxamide; anxiolitic and antidepressant; finding and altering the signal-transducing activity of gamma aminobutyric acid (GABA) receptors; detectably-labeled antagonist/agonist of GABAR
03/25/2008US7348324 Cyclic amine compounds as CCR5 antagonists
03/25/2008US7348017 such as 2-[Benzyl[(4-methoxyphenyl)sulfonyl]amino]-N-(3-thioxo-3H-1,2,4-dithiazol-5-yl)acetoamide; cosmetics; antiaging agents
03/25/2008CA2268709C Hiv protease inhibitors
03/25/2008CA2268394C New heterocyclylmethyl-substituted pyrazol derivates
03/20/2008WO2008033934A1 Substituted heteroaryl carboxylic acid derivatives as ptb-1b inhibitors
03/20/2008WO2008033931A1 Para-xylylene carboxylic acids and isothiazolones useful as protein tyrosine phosphatases (ptps) in particular ptp-ib
03/20/2008WO2008033854A1 Certain substituted amides, method of making, and method of use thereof
03/20/2008WO2008032858A2 Thiadiazole compound and use thereof
03/20/2008WO2008032191A2 Spiro-oxazolidinone compounds and their use as metabotropic glutamate receptor potentiators
03/20/2008WO2008031734A1 5-phenyl-nicotinamide derivatives
03/20/2008WO2008016692A3 Chemical compounds
03/20/2008WO2008015189A3 Fungicidal n-cycloalkyl-carboxamide derivatives
03/20/2008WO2008005910A3 Pyridone/hydroxypyridine 11-beta hydroxysteroid dehydrogenase type i inhibitors
03/20/2008WO2007138110A3 Compounds that interact with ion channels, in particular with ion channels from the kv family
03/20/2008WO2007115058A3 Thiadiazolidinone inhibitors of ptpase
03/20/2008WO2007113327A3 Fungicide n-cyclopropyl-sulfonylamide derivatives
03/20/2008WO2007084391A3 Thiazole compounds as protein kinase b ( pkb) inhibitors
03/20/2008WO2006094187A3 Phthalazine, aza- and diaza-phthalazine compounds and methods of use
03/20/2008US20080071083 Methods for minimizing thioamide impurities
03/20/2008US20080070948 Including indanones, indolinones and benzoxazolinones containing a piperidine ring, e.g., 1-[3-(4-(Hydroxymethyl)piperidin-1-yl)propyl]-1,3-dihydrobenzoimidazol-2-one; particularly for the M1 and/or M4 receptor subtypes; increase acetylcholine signaling or effect in the brain
03/20/2008US20080070929 Thiazoline and oxazoline derivatives and their methods of use
03/20/2008US20080070928 Novel 2-Heteroaryl-Substituted Benzimidazole Derivative
03/20/2008US20080070921 Melanocortin receptor modulators; sexual disorders, obesity, cachexia, eating disorders; for example 1,4-bis(2-amino-3-p-tolyl-propionyl)-2-isobutyl-5-(4-(2-aminoethylamino)butyl)piperazine
03/20/2008US20080070916 Treating disorders such as proliferative diseases, and cancer; compounds can act as probes of biological function; libraries; for example, 2-ethoxy-3-(2-hydroxyethoxyethoxyethyl)-4-(1-acetylindol-3-yl)-6-(morpholinocarbonyl)-2H-3,4-dihydropyran
03/20/2008US20080070915 Poly(ADP-ribose)polymerase (PARP); ischemia, reperfusion injuries, neurological disorders, neuroprotectants, sensitizer for chemotherapy or radiotherapy, anticancer
03/20/2008US20080070906 Quinolinone derivatives
03/20/2008US20080070905 An enzyme in the tryptophan degradation pathway, used to treat neurodegenerative disorders, certain cancers, drug addiction; 2-sulfonamido-substituted oxazole, imidazole or thiazole compounds such as 3,4-dimethoxy-N-[4-(3-nitrophenyl)-5-dimethylaminomethyl-1,3-thiazole-2-yl]benzenesulfonamide
03/20/2008US20080070903 New pyrimidine derivatives and new pyridine derivatives
03/20/2008US20080070902 Cinnamide Compound
03/20/2008US20080070895 Heteroaryl substituted spirocyclic sulfamides for inhibition of gamma secretase
03/20/2008US20080070869 Malonyl-CoA Decarboxylase Inhibitors Useful as Metabolic Modulators
03/20/2008CA2663113A1 Nicotinic acid derivatives as modulators of metabotropic glutanate receptors
03/20/2008CA2662409A1 5-phenyl-nicotinamide derivatives
03/20/2008CA2661951A1 Substituted amides, method of making, and method of use thereof
03/20/2008CA2661654A1 Certain substituted amides, method of making, and method of use thereof
03/20/2008CA2660611A1 Thiadiazole compound and use thereof
03/19/2008EP1900736A1 5-[4-[2-(n-methyl-n-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione and pharmaceutical compositions comprising the same
03/19/2008EP1899330A1 Substituted glycinamides having an antithrombotic and factor xa-inhibiting effect
03/19/2008EP1899296A1 Histamine-3 receptor antagonists
03/19/2008EP1660487B1 Pyrrole compositions useful as inhibitors of c-met