Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773) |
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04/14/2009 | US7517894 Endothelial growth factor; angiogenesis inhibitor; antitumor agents; skin disorders; endometriosis; Crohn's disease; leukemia; antiarthritic agents |
04/14/2009 | US7517879 Pyrrolidine derivatives as factor Xa inhibitors |
04/14/2009 | US7517877 5-substituted-alkylaminopyrazole derivatives as pesticides |
04/14/2009 | US7517875 Piperidine derivatives having CCR3 antagonism |
04/14/2009 | US7517535 Agonists and antagonists of nicotinergic acetylcholine receptors of insects like fleas, lice and flies, on humans or animals; chloronicotinyl insecticides such as imidaclopridas veterinary medicine; collars; tags |
04/14/2009 | US7517517 Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands |
04/14/2009 | CA2409841C Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists |
04/14/2009 | CA2408934C Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists |
04/14/2009 | CA2256007C Substituted heterocyclic benzocycloalkenes and their use as analgesic |
04/09/2009 | WO2009046416A1 Anilinopyrimidines as jak kinase inhibitors |
04/09/2009 | WO2009045313A2 Oxypiperidine derivatives as histamine receptor antagonists |
04/09/2009 | WO2009044788A1 Benzoxazinone derivative |
04/09/2009 | WO2009044250A1 New compounds as adenosine a1 receptor antagonists |
04/09/2009 | WO2009044162A1 Pyrazin-2-yl-pyridin-2-yl-amine and pyrazin-2-yl-pyrimidin-4-yl-amine compounds and their use |
04/09/2009 | WO2009043884A1 Azabicyclo [3. 1. 0] hexyl derivatives as modulators of dopamine d3 receptors |
04/09/2009 | WO2009043883A1 Azabicyclo [3. 1. o] hexyl derivatives as modulators of dopamine d3 receptors |
04/09/2009 | WO2009026227A3 Highly selective sigma receptor ligands |
04/09/2009 | WO2009022311A3 1,2-diamido-ethylene derivatives as orexin antagonists |
04/09/2009 | WO2008155666A3 Heteroarylamide-substituted pyrimidone derivatives for the treatment of neurodegenerative diseases |
04/09/2009 | WO2008152093A3 Diaminopyrimidines as modulators of the ep2 receptor |
04/09/2009 | WO2008121592A3 Acetyl coenzyme a carboxylase inhibitors |
04/09/2009 | WO2005054429A3 Synthesis of the c1-c6 keto-acid synthon of the epothilones |
04/09/2009 | US20090093527 [3-(2-{(3S)-3-[2-(Trifluoromethyl)phenoxy]pyrrolidin-1-yl}-1,3-thiazol-5-yl)-1,2,4-oxadiazol-5-yl]methanol, useful for the prevention and treatment of conditions related to abnormal lipid synthesis and metabolism, including cardiovascular disorders, atherosclerosis, obesity, diabetes and fatty liver |
04/09/2009 | US20090093507 Cdk inhibitors containing a zinc binding moiety |
04/09/2009 | US20090093478 N-aroyl cyclic amines |
04/09/2009 | US20090093455 Quinolone analogs and methods related thereto |
04/09/2009 | US20090093452 Pyrrole, Thiophene, Furan, Imidazole, Oxazole, and Thiazole Derivatives |
04/09/2009 | US20090093416 Caspase inhibitors and uses thereof |
04/09/2009 | DE4448032B4 Zusammensetzung enthaltend organische Materialien und 3-Aryl-benzofuranone als Stabilisatoren A composition comprising organic materials and 3-aryl-benzofuranones as stabilizers |
04/09/2009 | DE102007047735A1 Thiazolderivate Thiazole derivatives |
04/09/2009 | CA2738980A1 Pyrazin-2-yl-pyridin-2-yl-amine and pyrazin-2-yl-pyrimidin-4-yl-amine compounds and their use |
04/09/2009 | CA2701406A1 Benzoxazinone derivative |
04/09/2009 | CA2701124A1 C-met protein kinase inhibitors |
04/09/2009 | CA2700963A1 Oxypiperidine derivatives and methods of use thereof |
04/09/2009 | CA2700526A1 New compounds as adenosine a1 receptor antagonists |
04/08/2009 | EP2045242A1 Heterocyclic compounds having inhibitory activity against HIV integrase |
04/08/2009 | EP2045238A1 Bridged cyanine compounds and optical recording materials containing the same |
04/08/2009 | EP2045237A1 Pyrrole compounds as inhibitors of mycrobacteria, synthesis thereof and intermediates thereto |
04/08/2009 | EP2044939A1 Therapeutic agent for liver fibrosis |
04/08/2009 | EP2044066A2 Crystalline forms of n-[5-[[[5-(1,1-dimethylethyl)-2-oxazolyl]methyl] thio]-2-thiazolyl]-4-piperidinecarboxamide |
04/08/2009 | EP2044062A1 Indole compounds |
04/08/2009 | EP2044060A1 Fungicide hydroximoyl-tetrazole derivatives |
04/08/2009 | EP2044057A2 Derivatives of ureas of piperidine or pyrrolidine, their preparation and their therapeutical use |
04/08/2009 | EP2044052A1 Fungicide hydroximoyl-tetrazole derivatives |
04/08/2009 | EP2044041A2 Isothiazolidines useful in the treatment of ocular hypertensive conditions |
04/08/2009 | EP2044038A2 Novel piperazines, pharmaceutical compositions and methods of use thereof |
04/08/2009 | EP2044031A1 2-(heteroaryl) alkyl indazole 6-phenyl and thienyl methyl amide as thrombin inhibitors |
04/08/2009 | EP2044028A2 Cyanoisoquinoline compounds that stabilize hypoxia inducible factor (hif) |
04/08/2009 | EP2043993A2 Cyclopentane derivatives as antiglaucoma agents |
04/08/2009 | EP2043744A2 Chemical compounds |
04/08/2009 | EP2043441A1 Fungicide hydroximoyl-tetrazole derivatives |
04/08/2009 | EP1718667A4 Heterocyclic self-immolative linkers and conjugates |
04/08/2009 | EP1668162B1 Detection of immobilized nucleic acid |
04/08/2009 | EP1442026B1 Triazole derivatives as cyclooxygenase (cox) inhibitors |
04/08/2009 | EP1212299B1 Substituted piperidine compounds useful as modulators of chemokine receptor activity |
04/08/2009 | CN101405283A HIV inhibiting 5-amido substituted pyrimidines |
04/08/2009 | CN101405282A Aurora kinase modulators and method of use |
04/08/2009 | CN101405278A Novel heterocyclic NF-kB inhibitors |
04/08/2009 | CN101405275A Triazolone derivative |
04/08/2009 | CN101405270A Pyrazoles as 11-beta-HSD-1 |
04/08/2009 | CN101402554A 2- and 2,5-substituted phenylketo-enols |
04/08/2009 | CN100475810C Novel 2-arylthiazole compounds as pparalpha and ppargamma agonists |
04/08/2009 | CN100475796C Thiazole derivatives as cannabinoid receptor modulators |
04/08/2009 | CN100475792C Novel gamma-secretase inhibitors |
04/08/2009 | CN100475778C Diketohydrazine derivative compounds and drugs containing the compounds as the active ingredient |
04/07/2009 | US7514570 Derivatives of 3-hydroxy-4-(cyclyl-alkylaminoalkyl)-5-phenyl-1h-pyrazole as antagonists of the gonadotropin releasing hormone (GnRH) for use in the treatment of sex hormone related conditions, such as prostatic of uterine cancer |
04/07/2009 | US7514565 3,5-Difluoropyridines |
04/07/2009 | US7514564 Substituted amine derivatives and methods of use |
04/07/2009 | US7514557 Hepatitis C; preparing 8-bromo-7-alkoxyquinolines 2-substituted with a hetercyclic ring having an amine, carbamate, amine or urea group an 4-substituted with a 3-prolineoxy- group or derivative; intermediates |
04/07/2009 | US7514461 Chroman derivatives |
04/07/2009 | US7514460 Benzazole analogues and uses thereof |
04/07/2009 | US7514459 Gamma-secretase inhibitors |
04/07/2009 | US7514458 Heterocyclic-substituted benzamide derivatives, e.g., benzyl [2-(4-{1-[5-(5-tert-Butyl-3-methanesulfonylamino-2-methoxy-phenylcarbamoyl)-2-methyl-phenyl]-1H-1,2,3-triazol-4-yl}-2-phenyl-2H-pyrazol-3-yl)-ethyl]-carbamate; inhibit production of cytokines; useful for treating chronic inflammatory disease |
04/07/2009 | US7514456 Nicotinamide derivatives useful as p38 inhibitors |
04/07/2009 | US7514445 Heteroaryl amines as glycogen synthase kinase 3β inhibitors (GSK3 inhibitors) |
04/07/2009 | US7514439 Oxime derivative and preparations thereof |
04/07/2009 | US7514437 2-(2,4-difluorophenyl)-2-[(3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-isobutyl-2,5-dioxopiperazin-1-yl]-N,N-dimethylethanamide; to suppress uterine contractions; cyclization of leucine analogs |
04/07/2009 | US7514431 Piperidinyl cyclopentyl aryl benzylamide modulators of chemokine receptor activity |
04/07/2009 | US7514430 Nitrogen compounds such as N-phenyl-N'-{(1R,2S)-2-[(2S)-2-benzyl-6-oxo-morpholin-4-yl-methyl]-cyclohexyl }-urea, used to control chemotactic cytokines, and administered for the prevention of asthma or allergies; inhibition of the migration of eosinophils |
04/07/2009 | US7514429 Benzoxazinone-derived compounds, their preparation and use as medicaments |
04/07/2009 | US7514428 Pesticidal 1-aryl-3-amidoxime-pyrazole derivatives |
04/07/2009 | US7514225 detecting drugs that inhibits the binding of macrophage migration inhibitory factor (MIF) to an antimacrophage migration inhibitor factor monoclonal or polyclonal antibody; drug screening |
04/07/2009 | CA2415890C N-oxides as nk1 receptor antagonist prodrugs of 4-phenyl-pyridine derivatives |
04/07/2009 | CA2393757C Cycloamine ccr5 receptor antagonists |
04/07/2009 | CA2381243C 1-cycloalkylpyrazoyl-benzoyl derivatives |
04/07/2009 | CA2373880C Isoquinoline derivatives or salts thereof |
04/07/2009 | CA2352505C Epothilone derivatives and their use as antitumor agents |
04/07/2009 | CA2352503C Il-5 inhibiting 6-azauracil derivatives |
04/07/2009 | CA2281133C Multiple-agents-binding compound and use thereof |
04/07/2009 | CA2217737C Thf-containing sulfonamide inhibitors of aspartyl protease |
04/02/2009 | WO2009042694A1 (3-hydroxy-4-amino-butan-2-yl) -3- (2-thiazol-2-yl-pyrrolidine-1-carbonyl) benzamide derivatives and related compounds as beta-secretase inhibitors for treating |
04/02/2009 | WO2009042485A1 Indole compounds bearing aryl or heteroaryl groups having sphingosine-1-phosphate (s1p) receptor biological activity |
04/02/2009 | WO2009042435A1 Pyridin-2 -yl-amino-i, 2, 4 -thiadiazole derivatives as glucokinase activators for the treatment of diabetes mellitus |
04/02/2009 | WO2009041559A1 Indazole acrylic acid amide compound |
04/02/2009 | WO2009040755A2 Pyrrole compounds as inhibitors of mycobacteria, synthesis thereof ans intermediates thereto |
04/02/2009 | WO2009039944A1 Phenothiazine derivative having a double bond, method for the production thereof, and use thereof as a pharmaceutical |
04/02/2009 | WO2009039553A1 Benzothiazole compounds |
04/02/2009 | WO2009014910A3 N-azacyclic substituted pyrrole, pyrazole, imidazole, triazole and tetrazole derivatives as agonists of the rup3 or gpr119 receptor for the treatment of diabetes and metabolic disorders |
04/02/2009 | WO2009011880A3 Heterocyclic modulators of pkb |
04/02/2009 | WO2009010299A8 Substituted heteroarylpiperidine derivatives as melanocortin-4 receptor modulators |