Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
09/2001
09/04/2001CA2224062C Substituted n-(indole-2-carbonyl)-glycinamides and derivatives as glycogen phosphorylase inhibitors
08/2001
08/30/2001WO2001062765A2 Small molecule modulators of g protein-coupled receptor six
08/30/2001WO2001062756A1 Pyridinylimidazoles
08/30/2001WO2001062736A1 Aryl fused azapolycyclic compounds
08/30/2001WO2001062726A2 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
08/30/2001WO2001062245A2 Bilirubin or biliverdin degradation fragments
08/30/2001WO2001062233A2 Adenosine receptor modulators
08/30/2001WO2001016131A3 Five membered-ring compounds and utilization thereof in liquid crystal mixtures
08/30/2001WO2001014576A3 Process and intermediates for the preparation of isoxazolecaroxamides and analogues
08/30/2001WO2000075119A3 Substituted 2-aryl-1,2,4-triazine-3,5-di(thi)ones used as herbicides
08/30/2001US20010018525 Modulating blood glucose concentration
08/30/2001US20010018438 Nervous system disorders; psychological disorders
08/30/2001CA2401036A1 Pyridinylimidazoles
08/30/2001CA2368447A1 Small molecule modulators of g protein-coupled receptor six
08/29/2001EP1127883A2 Oxamides as IMPDH inhibitors
08/29/2001EP1127055A2 Stereoselective process for producing cryptophycins
08/29/2001EP1127054A1 Novel inhibitors of impdh enzyme
08/29/2001EP1127053A1 Novel 1-aryl-4-thiouracils
08/29/2001EP1127051A2 Tricyclic pyrazole derivatives
08/29/2001EP1126843A1 Compounds derived from an amine nucleus that are inhibitors of impdh enzyme
08/29/2001EP0889043B1 5,11-DIHYDRODIBENZ b,e] 1,4]OXAZEPINE DERIVATIVES AND DRUG COMPOSITIONS CONTAING THE DERIVATIVES
08/29/2001CN1310718A Heterocyclic compound as inhibitors of rotamase enzymes
08/29/2001CN1310706A Inhibitors of phospholipase enzymes
08/29/2001CN1310179A Oxamide being as IMPDH inhibitor
08/28/2001US6281356 Substituted pyrroles
08/28/2001US6281352 Antiinflammatory agents
08/28/2001US6281209 Fungicidal alkoximinomethyldioxazine derivatives
08/28/2001CA2101572C Benzoxazinones as inhibitors of hiv reverse transcriptase
08/28/2001CA2017252C Retroviral protease inhibiting compounds
08/24/2001CA2337588A1 Oxamides as impdh inhibitors
08/23/2001WO2001060820A2 Matrix metalloproteinase inhibitors and uses thereof
08/23/2001WO2001060819A1 Novel isoxazole and thiazole compounds and use thereof as drugs
08/23/2001WO2001060816A1 Kinase inhibitors
08/23/2001WO2001060813A1 Beta-alanine derivatives and their use as receptor antagonists
08/23/2001WO2001060802A1 4-imidazole derivatives of benzyl and restricted benzyl sulfonamides, sulfamides, ureas, carbamates, and amides and their use as alpha-1a agonists
08/23/2001WO2001060797A1 Phenyl-substituted heterocyclic enaminones
08/23/2001WO2001060362A1 TNF-α INHIBITORS
08/23/2001WO2001016111A3 Hypoglycemic sulfonyl pyrazolones and pyrazolines
08/23/2001WO2001012625A3 Substituted benzoxazoles
08/23/2001WO2001007436A3 Substituted oxoazaheterocyclyl compounds
08/23/2001WO2001004116A3 Neurotrophic pyrrolidines and piperidines, and related compositions containing them
08/23/2001US20010016657 Substituted isoquinoline derivatives and their use as anticonvulsants
08/23/2001US20010016583 Therapeutic application of pro-apoptotic benzodiazepines
08/23/2001US20010016579 Serotonin 5-HT, receptor partial activator
08/23/2001DE19960683A1 Substituierte 2,4-Diamino-1,3,5-triazine, Verfahren zur Herstellung und Verwendung als Herbizide und Pflanzenwachstumsregulatoren Substituted 2,4-diamino-1,3,5-triazines, to processes for preparation and use as herbicides and plant growth regulators
08/23/2001DE10007286A1 New phenyl-substituted heterocyclic enaminone and enaminethione derivatives useful as herbicides and pesticides, especially insecticides, acaricides, nematocides and fungicides
08/23/2001CA2651825A1 Substituted arylpyrazines
08/23/2001CA2400631A1 Beta-alanine derivatives and their use as receptor antagonists
08/23/2001CA2399147A1 4-imidazole derivatives of benzyl and restricted benzyl sulfonamides, sulfamides, ureas, carbamates, and amides and their use as alpha-1a agonists
08/23/2001CA2395841A1 Matrix metalloproteinase inhibitors and uses thereof
08/22/2001EP1124827A1 3-(substituted phenyl)-5-(substituted heterocyclyl)-1,2,4-triazole compounds
08/22/2001EP1124826A1 Process for the preparation of 2-(r)-(1- (r)-(3,5-bis (trifluoromethyl) phenyl)ethoxy) -4-((5-dimethylaminomethyl) -1,2,3-triazol -4-yl)methyl) -3-(s)-(4- fluorophenyl) morpholine
08/22/2001EP1124823A1 Thrombin inhibitors
08/22/2001EP1124822A1 Thrombin inhibitors
08/22/2001EP1124821A1 Compounds
08/22/2001EP1124804A1 Prostaglandin endoperoxide h synthase biosynthesis inhibitors
08/22/2001EP1124797A1 N-arylsulfonyl amino acid omega amides
08/22/2001EP1124528A1 Multivalent macrolide antibiotics
08/22/2001EP0752854B1 Pyrimidine or triazine carboxylic acid derivatives to be used as medicaments
08/22/2001CN1309656A Thioalkyl alpha-substd. pyrimidine compounds
08/22/2001CN1309654A Biphenyl derivs.
08/22/2001CN1309638A N-substd. naphthalene carboxamides as neurokinin-receptor antagonists
08/21/2001US6277985 As antibiotics; water solubility; in prodrugs
08/21/2001US6277877 Substituted n-(indole-2-carbonyl)glycinamides and derivates as glycogen phosphorylase inhibitors
08/21/2001US6277872 Antiischemic agents; brain disorders
08/21/2001US6277868 Bactericides; skin disorders
08/21/2001US6277859 Highly selective kappa-opioid agonists useful as analgesics and diuretics with reduced physiological side effects
08/21/2001US6277855 Method of treating dry eye disease with nicotinic acetylcholine receptor agonists
08/21/2001US6277853 Indole derivatives as 5-HT1B and 5-HT1D agonists
08/21/2001US6277848 Systemic pesticides for controlling arthropod, nematode, helminth or protozoan pests in agriculture
08/21/2001US6277839 Antiinflammatory agents, antipyretics, analgesics; side effect reduction
08/21/2001CA2094012C 1,2,4-oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents
08/21/2001CA2060652C N-substituted cycloalkyl and polycycloalkyl alpha-substituted trp-phe- and phenethylamine derivatives
08/16/2001WO2001058896A1 Benzoxazole derivatives as tnf and pde iv inhibitors
08/16/2001WO2001058895A1 Benzofuran carboxamides and their therapeutic use
08/16/2001WO2001058890A1 Heteroaromatic carboxamide derivatives and their use as inhibitors of the enzyme ikk-2
08/16/2001WO2001058881A1 Pyrimidine derivatives as selective inhibitors of cox-2
08/16/2001WO2001058871A1 Piperidyl carboxylic acids as integrin antagonists
08/16/2001WO2001058869A2 Cannabinoid receptor modulators, their processes of preparation, and use of cannabinoid receptor modulators in treating respiratory and non-respiratory diseases
08/16/2001WO2001058491A1 Drug comprising combination
08/16/2001WO2001010842A3 Melanocortin-4 receptor binding compounds and methods of use thereof
08/16/2001WO2001010380A3 Benzanilides as potassium channel openers
08/16/2001WO2001009119A3 Chemokine receptor antagonists
08/16/2001WO2000066106A3 Use of benzodiazepines for treating autoimmune diseases induced by apoptosis
08/16/2001US20010014677 Restenosis, kidney diseases, lung diseases
08/16/2001EP1143946A3 Use of benzodiazepines for treating autoimmune diseases induced by apoptosis
08/16/2001EP1123934A1 Benzoxazole derivatives useful as UV filters
08/16/2001EP1123285A1 Substituted benzopyran analogs for the treatment of inflammation
08/16/2001EP1123284A1 Method for the preparation of citalopram
08/16/2001EP0944388A4 Inhibitors of farnesyl-protein transferase
08/16/2001EP0885208B1 Taxoids, their preparation and pharmaceutical compositions containing them
08/16/2001EP0788498B1 Phenyloxazolidinone antimicrobials
08/16/2001DE10006453A1 New piperidylcarboxylic acid derivatives, are integrin antagonists useful for treating inflammatory, autoimmune or immunological diseases, e.g. atherosclerosis, asthma, diabetes, rheumatoid arthritis or transplant rejection
08/16/2001CA2399791A1 Cannabinoid receptor modulators, their processes of preparation, and use of cannabinoid receptor modulators in treating respiratory and non-respiratory diseases
08/16/2001CA2399463A1 Combination drug
08/15/2001CN1308631A Heterocyclic derivatives which inhibit factor xa
08/15/2001CN1308626A Benzothiophenes, benzofurans, and indoles useful in the treatment of insulin resistance and hyperglycemia
08/15/2001CN1308618A Oxazole-aryl-carboxylic acids useful in the treatment of insulin resistance and hyperglycemia
08/15/2001CN1308616A Non-peptidyl inhibitors and VLA-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory disease
08/15/2001CN1308614A Benzimidazoles, production thereof and use thereof medicaments