Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
09/2001
09/19/2001CN1313854A Antiviral pyrimidinedione derivatives and process for the preparation thereof
09/19/2001CN1313853A Oxindole derivatives as growth hormone releasers
09/19/2001CN1313280A Benzheterocyclic derivatives
09/19/2001CN1071333C Quinoline derivative
09/19/2001CN1071322C Process for producing 5,6-dihydro-1,3-oxazines
09/18/2001US6291685 Reacting 1-(2-thienyl)allyl derivative in solvent medium containing base and carboxylic acid anhydride with carbon monoxide in presence of carbonylation catalyst to form ester compound; saponification to form 4-hydroxybenzothiophene
09/18/2001US6291672 Human NK3 receptor-selective antagonist compounds, method for obtaining them and pharmaceutical compositions containing them
09/18/2001US6291514 Heteroaryl amidines, methylamidines and guanidines, preparation thereof, and use thereof as protease inhibitors
09/18/2001US6291505 Pyrazole estrogen receptor agonist and antagonist
09/18/2001US6291492 3-aryl alkenyl-1,2,4-oxadiazole derivatives and their use as parasiticides for animals
09/18/2001US6291480 Diaryl piperidyl pyrrole derivatives as antiprotozoal agents
09/18/2001US6291474 Bicyclic amine derivatives
09/18/2001US6291458 Morpholinobenzamide salts
09/18/2001US6289745 High temperature insertion type flow element and mounting extension
09/13/2001WO2001066534A2 Cyclic and bicyclic diamino histamine-3 receptor antagonists
09/13/2001WO2001066531A1 Substituted 3-phenyl-5-alkoxi-1,3,4-oxdiazol-2-one and use thereof for inhibiting hormone-sensitive lipase
09/13/2001WO2001066522A1 Acylated phenyl or pyridine herbicides
09/13/2001WO2001066520A1 Indole derivatives, process for preparation of the same and use thereof
09/13/2001US20010021782 Production of amide derivatives and intermediates therefor
09/13/2001US20010021775 Benzimidazolinones, benzoxazolinones, benzopiperazinones, indanones, and derivatives thereof as inhibitors of factor Xa
09/13/2001US20010021714 Compounds such as n-(4-bromo-3-methyl-5-isoxazolyl)-2-n-benzylbenzo(b)thiophene-3-sufonamide administered as endothelin peptide receptor antagonists
09/13/2001US20010021709 Integrin inhibitors used to treat circulatory disorders, for thrombosis, myocardial infarct, coronary heart disease, arteriosclerosis, osteoporosis, pathological processes maintained or propagated by angiogenesis and tumor therapy
09/13/2001DE19954228A1 New epothilone derivatives used for treating e.g. malignant melanoma, breast carcinoma, psoriasis, multiple sclerosis and arthritis
09/13/2001DE10010968A1 New 5-alkoxy-3-phenyl-3H-1,3,4-oxadiazol-2-one derivatives, are hormone-sensitive lipase inhibitors useful for treating metabolic disorders such as non-insulin dependent diabetes mellitus
09/13/2001CA2402174A1 Indole derivatives, process for preparation of the same and use thereof
09/13/2001CA2401953A1 Substituted 3-phenyl-5-alkoxi-1,3,4-oxdiazol-2-one and use thereof for inhibiting hormone-sensitive lipase
09/12/2001EP1132368A2 Process for the preparation of 2-fluoro-1,1-dichloro-acrylyl chloride
09/12/2001EP1131320A1 Isoxazoline fibrinogen receptor antagonists
09/12/2001EP1131319A2 3- benz(ox/thi)azol-7-yl -1h-pyrimidine-2,4-diones
09/12/2001EP1131318A1 Process for making 5-substituted pyrazoles using dithietanes
09/12/2001EP1131309A2 Thiophendioximether
09/12/2001EP1131308A1 New piperazine and piperidine compounds
09/12/2001EP1131306A2 Isoxazoline fibrinogen receptor antagonists
09/12/2001EP1131295A1 Quinoline-4-carboxamide derivatives as nk-3 and nk-2 receptor antagonists
09/12/2001EP0888317B1 Substituted 4-hydroxy-phenylalcanoic acid derivatives with agonist activity to ppar-gamma
09/12/2001EP0832066B1 Substituted n-(indole-2-carbonyl-) amides and derivatives as glycogen phosphorylase inhibitors
09/12/2001EP0820450B1 N-substituted azaheterocyclic carboxylic acids and alkylesters thereof
09/12/2001EP0817775B1 Quinazoline derivatives
09/12/2001EP0794945B1 Iminooxybenzylcrotonic acid esters, process for their preparation and use thereof
09/12/2001CN1312807A Inhibitors of glycogen synthase kinase 3
09/12/2001CN1312803A Novel benzopykan or thiobenzopyran derivatives
09/12/2001CN1312799A Bispiperidines as antithrombotic agents
09/12/2001CN1070701C Pyrimidine ortriazine carboxylic acid derivatives to be used as medicaments
09/11/2001US6288236 Benzimidazole compounds containing a benzoxazole or benzothiazole ring, and compositions and methods of use containing the same
09/11/2001US6288234 Fluorinated heterocyclic amido amine compounds as drugs
09/11/2001US6288231 Peptide-containing α-ketoamide cysteine and serine protease inhibitors
09/11/2001US6288228 Triazine angiogenesis inhibitors
09/11/2001US6288225 Substituted benzolactam compounds as substance P antagonists
09/11/2001US6288092 Triaryl compounds
09/11/2001US6288088 Such as 1-(2,6-dichloro-4-trifluoromethylphenyl)-3-(4-( n,n-dimethylcarbamoyl)-.delta..sup.2-1,2,4-oxadiazolin-3-yl)-5 -isopropoxymethyleneamino-4-trifluoromethylsulfinylpyrazole
09/11/2001US6288062 Interleukin and tumor necrosis factor inhibitors; antiinflammatory agents; rheumatic diseases; antiarthritic agents; respiratory system disorders
09/11/2001US6288059 Acylated hetero-alicyclic derivatives
09/11/2001US6288055 Analgesic agents
09/11/2001CA2200742C Quinoxaline derivatives useful in therapy
09/07/2001WO2001064755A2 Isoxazole gegen virale erkrankungen
09/07/2001WO2001064673A1 Flavone derivatives, preparation method and use as medicines
09/07/2001WO2001064670A1 Novel cyclic amide derivatives
09/07/2001WO2001064656A1 2,4,di(hetero-)arylamino(-oxy)-5-substituted pyrimidines as antineoplastic agents
09/07/2001WO2001064654A1 Pyrimidine compounds
09/07/2001WO2001064652A1 Substituted 5-methyldihydropyridazinones and their use in the prophylaxis and/or treatment of anemias
09/07/2001WO2001064637A1 2-oxo-1-pyrrolidine derivatives, process for preparing them and their uses
09/07/2001WO2001064632A1 Azetidine derivatives, preparation thereof and pharmaceutical compositions containing same
09/07/2001WO2001064216A1 4-alkyl piperidinyl pyrrolidine modulators of chemokine receptor activity
09/07/2001CA2401405A1 Medicament for viral diseases
09/07/2001CA2400116A1 Azetidine derivatives, preparation thereof and pharmaceutical compositions containing same
09/07/2001CA2339676A1 Use of heteroaryl substituted n-(indole-2-carbonyl-) amides for treatment of infection
09/06/2001US20010020033 Selective factor xa inhibitors
09/06/2001US20010020021 Metalloprotease inhibitor
09/06/2001DE10010429A1 New 6-(4-sulfonamido-phenyl)-5-methyl-dihydropyridazinones, having erythropoietin sensitizing and erythropoiesis stimulating activity, useful for treating anemia
09/06/2001DE10010426A1 Medicaments, especially for treating anemia, containing 6-(4-(acylamino)-phenyl)-dihydropyridazinones having erythropoietin sensitizing and erythropoiesis stimulating activity
09/06/2001DE10010425A1 Medicaments for treating anemia, containing new or known 6-(4-(acylamino)-phenyl)-5-methyl-dihydropyridazinones having erythropoietin sensitizing and erythropoiesis stimulating activity
09/05/2001EP1130017A2 Azole derivatives and their use as superoxide radical inhibitors
09/05/2001EP1130016A1 Thiocarbamic acid derivatives
09/05/2001EP1129082A1 Method and novel intermediate products for producing isoxazolin-3-yl-acylbenzenes
09/05/2001EP1129075A1 N-aryl(thio)anthranilic acid amide derivatives, their preparation and their use as vegf receptor tyrosine kinase inhibitors
09/05/2001EP1129074A2 Antrhranilic acid amides and the use thereof as medicaments
09/05/2001EP0946545B1 Novel carboxy substituted cyclic carboxamide derivatives
09/05/2001EP0807112B1 Hetero-aromatic ring substituted phenyloxazolidinone antimicrobials
09/05/2001EP0699185B1 GUANIDINE DERIVATIVES AS INHIBITORS OF Na+ /H+ EXCHANGE IN CELLS
09/05/2001CN1311793A Antipicornaviral compounds, their prepn. and use
09/05/2001CN1311787A Oxazolidinone derivatives, process for their prepn. and pharmaceutical compositions contg. same
09/05/2001CN1311786A Oxadiazoline derivatives and their use as insecticides
09/05/2001CN1311783A Sulfonyl amino (thio) carbonyl triazoline (thi) one having alkenyl substitutents
09/05/2001CN1311692A Farnesyl protein transferase inhibitors with i(IN VIVO) Radiosensitizing
09/05/2001CN1311679A Benzimidazole derivatives as modulators of IgE
09/05/2001CN1311676A Compound that inhibit the binding of integrins to their receptors
09/05/2001CN1311675A Compounds having IgE affecting properties
09/05/2001CN1070490C 吲哚衍生物 Indole derivatives
09/05/2001CN1070488C Substituted arylalkylthioalkylthiopyridines for use in the control of helicobacter bacteria
09/05/2001CN1070481C Use of dioxomorpholines to combact endopharasites, movel dioxomopholines and process for their prodn.
09/05/2001CN1070480C 2-amino-benzoxanones for treatment of viral infections
09/04/2001USH1992 Metalloproteinase inhibitors, pharmaceutical compositions containing them, and their pharmaceutical uses
09/04/2001US6284781 Anticancer agent
09/04/2001US6284779 Nervous system disorders
09/04/2001US6284774 4-Benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective NMDA receptor antagonists
09/04/2001US6284768 Src family SH2 domain inhibitors
09/04/2001US6284767 Retroviral protease inhibiting compounds
09/04/2001US6284764 Antiproliferative agent
09/04/2001US6284759 2-piperazinoalkylaminobenzo-azole derivatives: dopamine receptor subtype specific ligands
09/04/2001US6284755 Inhibitors of prenyl-protein transferase