Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226) |
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11/21/2002 | WO2002092076A1 Substituted coumarins and quinolines as caspases activators |
11/21/2002 | WO2002070507A3 Glycorticoid receptor antagonists for treatment of diabetes |
11/21/2002 | WO2002057246A3 Inhibitors of cruzipain and other cysteine proteases |
11/21/2002 | WO2002055514A3 Substituted benzimidazol-2-ones as vasopressin receptor antagonists and neuropeptide y modulators |
11/21/2002 | WO2002022598A8 Quinolinone derivatives as tyrosine kinase inhibitors |
11/21/2002 | US20020173667 Use in photochromic articles such as lenses; 2H-naphtho(1,2-b)pyran structure characterized by having an aromatic substituent in the 5 position |
11/21/2002 | US20020173645 Acylating a 2-aryl-6-alkoxy-benzo(b)thiophene with a p-(tertiaryaminoethoxy)benzoic acid hydrohalide salt or the corresponding benzoyl halide in presence of a boron trihalide |
11/21/2002 | US20020173631 4-((5,5-dimethyl-5,6,7,8-tetrahydro-8-hydroxynaphthalen-2 -yl)carbonyloxy)benzoic acid, benzyl ester for example; receptor subtype selectivity for side effect reduction |
11/21/2002 | US20020173536 Enantiomerically pure basic arylcycloalkylhydroxycarboxylic esters, processes for their preparation and their use in medicaments |
11/21/2002 | US20020173527 Tumor necrosis factor antagonist; antiinflammatory agents |
11/21/2002 | US20020173518 Anticoagulant in mammls |
11/21/2002 | US20020173515 Antiproliferative agents |
11/21/2002 | US20020170125 Bridged diaminopyrazole compounds and dye compositions containing same |
11/21/2002 | DE10125294A1 New heterocyclylmethyl-substituted anthranilamide derivatives and analogs as KDR/FLT tyrosine kinase inhibitors, used for treating e.g. psoriasis, restenosis, leukemia, arthritis, eye or kidney disease or arteriosclerosis |
11/21/2002 | CA2447184A1 5-cyano-1h-indole derivatives as antagonists of the interleukine-8 receptors |
11/21/2002 | CA2446879A1 2,5-disubstituted pyridine, pyrimidine, pyridazine and 1, 2, 4-triazine derivatives for use as p38 inhibitors |
11/21/2002 | CA2446797A1 Furan and thiophene derivatives that activate human peroxisome proliferator activated receptors |
11/21/2002 | CA2446717A1 Novel 4-anilinoquinoline-3-carboxamides |
11/21/2002 | CA2446586A1 Aromatic sulfone hydroxamates and their use as protease inhibitors |
11/20/2002 | EP1258252A1 Integrin expression inhibitors |
11/20/2002 | EP1258244A1 High affinity ligands for nociceptin receptor ORL-1 |
11/20/2002 | EP1257550A1 Platelet adp receptor inhibitors |
11/20/2002 | EP1257544A2 Piperazine and piperidine derivatives for treatment or prevention of neuronal damage |
11/20/2002 | EP1257543A1 Pyridinylimidazoles |
11/20/2002 | EP1150969B1 Alpha-azacyclomethyl quinoline derivatives for treating urinary incontinence |
11/20/2002 | CN1380882A C10 ester substituted taxanes as antitumor agents |
11/20/2002 | CN1380289A Amide capable of inhibiting ApoB-secretion/MTP |
11/19/2002 | US6482963 C9 hydrido, hydroxy and acyloxy taxane derivatives and pharmaceutical compositions containing them |
11/19/2002 | US6482956 Endothelin receptor antagonists |
11/19/2002 | US6482955 Organometallic reagent reacted with an activated carboxylic acid to produce a ketone reacted with carbon disulfide and dihalomethane, further reacting the dithietane product with a secondary amine, and condensing the thioamide with hydrazine |
11/19/2002 | US6482832 Heterocyclically substituted amides, their production and their use |
11/19/2002 | US6482822 N-(iminomethyl)amines derivatives, their preparation, their use as medicines and compositions containing them |
11/18/2002 | WO2001087878A1 Novel benzothiophene derivatives |
11/18/2002 | WO2001087855A1 Triazole derivatives |
11/18/2002 | CA2409821A1 Novel benzothiophene derivatives |
11/15/2002 | WO2001087875A1 Novel benzofuran derivatives |
11/15/2002 | CA2409096A1 Novel benzofuran derivatives |
11/14/2002 | WO2002090355A1 N-aroyl cyclic amines |
11/14/2002 | WO2002090353A1 Sulfonamides |
11/14/2002 | WO2002090352A2 Selective anthranilamide pyridine amides as inhibitors of vegfr-2 and vegfr-3 |
11/14/2002 | WO2002090348A1 Sulfonamides |
11/14/2002 | WO2002090347A1 Amide compounds |
11/14/2002 | WO2002090346A1 Phthalazine derivatives with angiogenesis inhibiting activity |
11/14/2002 | WO2002090342A1 Chromene compound |
11/14/2002 | WO2002090336A1 Substituted arylketones |
11/14/2002 | WO2002090334A1 Isoquinolinone derivatives as parp inhibitors |
11/14/2002 | WO2002090332A2 Novel aeylheteroalkylaminε derivatives |
11/14/2002 | WO2002090330A1 Substituted 2-pyridine-cyclohexane-1,4-diamine derivatives |
11/14/2002 | WO2002090317A1 Substituted cyclohexane-1,4-diamine derivatives |
11/14/2002 | WO2002089793A1 Sulfonamides |
11/14/2002 | WO2002089792A1 Sulfonamides |
11/14/2002 | WO2002089785A1 Sulfonamides |
11/14/2002 | WO2002089783A1 Substituted cyclohexan-1,4-diamine derivatives with constipating and peripheral analgesic properties |
11/14/2002 | WO2002081453A8 Thiohydantoins and use thereof for treating diabetes |
11/14/2002 | WO2002072577A3 Azacycloalkyl substituted acetic acid derivatives for use as mmp inhibitors. |
11/14/2002 | WO2002024650B1 Pyridinone and pyridinethione derivatives having hiv inhibiting properties |
11/14/2002 | US20020169336 Able to inhibit the binding of integrins to their ligands and are of use in the prophylaxis and treatment of immuno or inflammatory disorders |
11/14/2002 | US20020169322 Use of N-alkylamino-heterocylic compounds for the treatment of migraine |
11/14/2002 | US20020169313 Of carbonyl compounds with secondary amines in the presence of a water scavenger, preferably trifluoroacetic acid; preparation of imidazole-containing benzodiazepines, which are inhibitors of farnesyl protein transferase |
11/14/2002 | US20020169203 Modulators of all three classes of calcium channel blocker subtypes (Small, Intermediate and Big conductance K channel (SK, IK and BK)) comprising malonate esters and nitriles; respiratory, brain, cardiovascular, urogenital disorders |
11/14/2002 | US20020169198 Agonists of the progesterone receptor; contraceptives, hormone replacement therapy and treating menopause symptoms |
11/14/2002 | US20020169188 Modulating neurotransmission in the central nervous system |
11/14/2002 | US20020169161 Bicyclic sulfanimde compounds useful for the treatment of cardiac arrhythmias |
11/14/2002 | US20020169155 A nitrogen-ring containing triheterocyclic compound is useful for treating a disease associated with aberrant leukocyte recruitment and/or activation |
11/14/2002 | DE10136449A1 Substituierte Arylketone Substituted aryl ketones |
11/14/2002 | CA2453223A1 Selective anthranilamide pyridinamides as vegfr-2 and vegfr-3 inhibitors |
11/14/2002 | CA2449187A1 Substituted arylketones |
11/14/2002 | CA2446735A1 Substituted cyclohexane-1,4-diamine derivatives with an anti-diarrhoea and peripheral analgesic action |
11/14/2002 | CA2446396A1 N-aroyl cyclic amines |
11/14/2002 | CA2446365A1 Sulfonamides |
11/14/2002 | CA2446120A1 Novel arylheteroalkylamine derivatives |
11/14/2002 | CA2446051A1 Phthalazine derivatives with angiogenesis inhibiting activity |
11/14/2002 | CA2444531A1 Isoquinolinone derivatives as parp inhibitors |
11/13/2002 | EP1255740A2 Substituted arylpyrazines |
11/13/2002 | EP1255739A1 3-aminoquinazolin-2,4-dione antibacterial agents |
11/13/2002 | EP1255738A2 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto |
11/13/2002 | EP1255736A2 Substituted piperazine derivatives and their use as inhibitors of the microsomal triglyceride transfer protein (mtp) |
11/13/2002 | EP1255735A2 Pyridine derivatives as potentiators of glutamate receptors |
11/13/2002 | EP1255734A1 Isatine derivatives with neurotrophic activity |
11/13/2002 | EP1255726A2 (r)-2-aryl-propionamides, useful in the inhibition of il-8 induced chemiotaxis of neutrophils |
11/13/2002 | EP1255536A2 Indolinone derivatives for modulation of c-kit tyrosine protein kinase |
11/13/2002 | EP1140916B1 Heteroaryl-cyclic acetals |
11/13/2002 | EP1012139B1 Azetidinone derivatives as beta-lactamase inhibitors |
11/13/2002 | EP0912515B1 1,4-di-substituted piperidines as muscarinic antagonists |
11/13/2002 | CN1379777A Amino-triazolopyridine derivatives |
11/13/2002 | CN1379774A Compounds |
11/13/2002 | CN1379765A Benzodiazepine derivatives usable as parental metabolic glutamate receptor antagonist |
11/13/2002 | CN1379764A Benzodiazepine derivatives |
11/13/2002 | CN1379763A Pyrazoloanthrone and derivatives thereof as JNK inhibitors and their compositions |
11/13/2002 | CN1379666A Non-peptide GnRH agents, methods and intermediates for their preparation |
11/12/2002 | US6479678 Metal alkoxide taxane and β-lactam compounds |
11/12/2002 | US6479554 Immunotherapeutic agents |
11/12/2002 | US6479536 Benzofuran derivatives, process for the preparation of the same and uses thereof |
11/12/2002 | US6479519 Inhibitors of cell adhesion; treatment of asthma or inflammatory bowel disease |
11/12/2002 | US6479517 Treatment of post-menopausal syndrome: osteoporosis, cardiovascular effects such as hyperlipidemia, and estrogen-dependent cancer, particularly breast and uterine cancer |
11/12/2002 | US6479514 Quinoline-aminomethyl-pyridyl derivatives with anti-helicobacter activity |
11/12/2002 | US6479508 Viral polymerase inhibitors |
11/12/2002 | US6479505 6-arylphenanthridines with PDE-IV inhibiting activity |
11/12/2002 | US6479504 Antagonism of immunostimulatory CpG-oligonucleotides by 4-aminoquinolines and other weak bases |
11/12/2002 | US6479495 Simultaneously treating depression and memory dysfunction in mammals suffering from memory dysfunction and depression |