Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
02/2003
02/13/2003US20030032654 Useful for the treatment or prevention of asthma and other allergic diseases.
02/13/2003US20030032623 E.g., 1-(2-(1-adamantyl)ethyl)-1-pentyl-3-(3-(4-pyridyl)propyl)urea; useful as therapeutic agents for autoimmune diseases such as rheumatoid arthritis.
02/13/2003CA2468925A1 Platelet adp receptor inhibitors
02/13/2003CA2456096A1 Novel amine derivative having human .beta.-tryptase inhibitory activity and medecine containing the same
02/13/2003CA2455833A1 1,3,5-triazine-2,4,6-triones, preparation and use as gonadotropin-releasing hormone receptor antagonists
02/13/2003CA2455772A1 Substituted isoindoles and their use
02/13/2003CA2455235A1 1,2,4-triazin-3,5-diones as gonadotropin-releasing hormone receptor (gnrh) antagonists
02/13/2003CA2455179A1 Androgen receptor modulators and methods of use thereof
02/13/2003CA2449804A1 Aromatic hydroxamic acid derivatives useful as hdac inhibitors
02/12/2003EP1283448A2 Electrophotographic organophotoreceptors with charge transport compounds
02/12/2003EP1283210A1 Process for preparation of sulfonamide derivatives and crystals thereof
02/12/2003EP1283209A1 Novel benzothiophene derivatives
02/12/2003EP1283208A1 Novel benzofuran derivatives
02/12/2003EP1283055A1 Soluble beta amyloid precursor protein secretion promoters
02/12/2003EP1282617A1 Hydantoin derivatives with affinity for somatostatin receptors
02/12/2003EP1282616A1 Hydroxyphenyl-piperidin-4-ylidene-methyl-benzamide derivatives for the treatement of pain
02/12/2003EP1282614A1 Hydroxamic acid derivatives
02/12/2003EP1282609A2 Piperazinedione compounds
02/12/2003EP1282600A1 Inhibitors of dipeptidyl peptidase iv
02/12/2003EP1282445A2 N-substituted dithiocarbamates for the treatment of biological disorders
02/12/2003EP1282418A2 Use of pyrazole derivatives for treating infertility
02/12/2003EP1064262B1 Substituted isoindolones and their use as cyclic gmp modulators in medicaments
02/12/2003EP0988292B1 Piperazine derivatives and their use as anti-inflammatory agents
02/12/2003EP0926146B1 Chromene compounds
02/12/2003CN1397148A Luminescent element material and luminescent element comprising the same
02/12/2003CN1396833A Integrin expression inhibitors
02/12/2003CN1396827A Remedies or preventives for pulmonary insufficiency containing diaminotrifluoromethylpyridine derivatives
02/12/2003CN1396807A 除草组合物 Herbicidal compositions
02/12/2003CN1396163A Thiophen sulfuryl compound
02/12/2003CN1101384C Process for preparing 1-biphenylmethylmidazole derivatives
02/12/2003CN1101380C 4-mercaptopyrrolidine derivatives as farnesyl transferase inhibitors
02/11/2003US6518429 Anticancer agents, treating restenosis, atherosclerosis and hepatitis virus
02/11/2003US6518303 Selectively inhibit COX-2 in preference to COX-1 and are useful in the treatment of COX-2 mediated diseases, such as inflammation, pain, fever and asthma with fewer side effects
02/11/2003US6518301 Better selectivity than estrogen for the estrogen receptor-beta over receptor-alpha; treatment of Alzheimer's disease, anxiety, depression, osteoporosis, cardiovascular disease, rheumatoid arthritis, or prostate cancer
02/11/2003US6518295 Utilization of aryl(or heteroaryl)azolylcarbinol derivatives in the preparation of a medicament for the treatment of troubles mediated by an excess of substance P
02/11/2003US6518292 Heterocyclic aromatic compounds usefuls as growth hormone secretagogues
02/11/2003US6518289 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
02/11/2003US6518286 Compounds
02/11/2003US6518279 Cyclopentanone dihydropyridine compounds useful as potassium channel openers
02/11/2003US6518267 Protease inhibitors
02/11/2003US6518266 1- Aryl-3-thioalkyl pyrazoles, the synthesis thereof and the use thereof as insecticides
02/11/2003US6518264 For treatment/prevention of psychoses, other brain disorders, and cardiovascular disorders
02/11/2003CA2047237C Chroman derivatives
02/11/2003CA2041135C Method for the photochemical isomerisation of organic compounds under the influence of a photosensitizer
02/06/2003WO2003010361A2 Nitrogen atom transfer
02/06/2003WO2003010164A1 Arylsulfonamide derivatives as c-jun-n-terminal kinases (jnk's) inhibitors
02/06/2003WO2003010163A1 Novel compounds
02/06/2003WO2003010160A2 1-glycinyl-4 (methylpiperidin-4-yl) piperazines and -piperridines as factor xa antagonists
02/06/2003WO2003010158A1 Novel compounds
02/06/2003WO2003010141A2 Hepatitis c virus polymerase inhibitors with a heterobicyclic structure
02/06/2003WO2003010140A2 Hepatitis c virus polymerase inhibitors with heterobicyclic structure
02/06/2003WO2003009847A1 Substituted piperidines as modulators of the melanocortin receptor
02/06/2003WO2003009845A1 Substituted urea neuropeptide y y5 receptor antagonists
02/06/2003WO2003009841A1 Novel pyrroles having hypolipidemic hypocholesteremic activities, process for their preparation and pharmaceutical compositions containing them and their use in medicine
02/06/2003WO2002079146A3 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same
02/06/2003WO2002070516A3 Cyclopropaheterocycles as non-nucleoside reverse transcriptase inhibitors
02/06/2003WO2002059112A3 Pyrazole compounds useful as protein kinase inhibitors
02/06/2003WO2002048134A3 Di-substituted aminomethyl chroman derivative beta-3 adrenoreceptor agonists
02/06/2003WO2002046172A3 Substituted 1, 3, 5-triazines and pyrimidines as abca-1 elevating compounds against coronary artery disease or atherosclerosis
02/06/2003WO2002046141A3 Coumpounds of the formula r1-x-y-z-nr2r3 as abca-1 elevating agents against coronary artery disease or atherosclerosis
02/06/2003WO2002010137A9 Indazole derivatives as jnk inhibitors
02/06/2003US20030028034 Nematicidal pyrazoles
02/06/2003US20030028026 Nitrate salts of Salbutamol, Cetirizine, Loratadine, Terfenadine, Emedastine, Ketotifen, Nedocromil, Ambroxol, Dextromethorphan, Dextorphan, Isoniazide, Erythromycin, and Pyrazinamide; respiratory system pathology treatment
02/06/2003US20030028022 Preferably tertiary amines comprising tetrahydroquinoline and benzimidazole; use treating human immunodeficiency virus (HIV) and Feline Immunodeficiency Virus (FIV)
02/06/2003US20030028018 Treating diseases characterized by activity of vascular endothelial growth factor receptor tyrosine kinases such as cancer
02/06/2003US20030027855 Preparation of a derivative or analog of baccatin III or 10-desacetyl baccatin III having a C9 hydroxy substituent by selective reduction of the C9 keto compound
02/06/2003US20030027842 Halogenobenzimidazoles
02/06/2003US20030027836 Arylalkoxy-substituted tetrahydroisoquinoline-3-carboxylic acids or esters
02/06/2003US20030027829 Potassium channel inhibitors
02/06/2003US20030027814 Bis(5-aryl-2-pyridyl) compound having excellent immunoglobulin (IgE) antibody production inhibiting activity, useful for the prevention or treatment of allergic immune diseases
02/06/2003US20030027810 Nicotine receptor ligands
02/06/2003US20030027794 N-heterocyclic derivatives as NOS inhibitors
02/06/2003CA2454903A1 Substituted piperazines as modulators of the melanocortin receptor
02/06/2003CA2454702A1 Novel compounds
02/06/2003CA2452328A1 Substituted piperidines as modulators of the melanocortin receptor
02/06/2003CA2452259A1 Arylsulfonamide derivatives as c-jun-n-terminal kinases (jnk's) inhibitors
02/05/2003EP1280800A1 N-sulfonyl hydroxamic acid derivatives as inhibitors of cd 23
02/05/2003EP1280793A2 Cyclic amidine compounds and their use as alpha4beta2 nicotinic acetylcholine receptor ligands
02/05/2003EP1280781A1 5-ht 7 receptor antagonists
02/05/2003EP1280777A1 Tetrahydroisoquinoline analogs useful as growth hormone secretagogues
02/05/2003EP1280773A1 5-aryl-1.3.3.-trimethyl-2-methylene-indoline derivatives and salts thereof, methods for the production and use of said compounds for the temporary coloration of fibres
02/05/2003EP1117653B1 Quinoline and quinazoline derivatives and their use as inhibitors of cytokine mediated diseases
02/05/2003CN1395575A Novel piperidine compounds and drugs containing the same
02/05/2003CN1395568A 1,2-diaryl benzimidazole derivative for treating illnesses associated with microglia activation
02/05/2003CN1395567A New imidazole derivatives
02/05/2003CN1395566A Corticotropin releasing factor antagonists
02/05/2003CN1395563A Isatine derivatives with neurotrophic activity
02/05/2003CN1395562A Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
02/05/2003CN1394859A Intermediate for preparing cyclopentane formamide compound and its preparation method
02/05/2003CN1100777C N-heterocyclic derivatives as NOS inhibitor
02/05/2003CN1100771C Phosphononooxymethyl ethers for taxame derivatives
02/05/2003CN1100762C Substituted pyrazolyl-pyrazole derivatives and their use as herbicides
02/05/2003CN1100761C Benzyloxy substituted aryl copounds and their use as fungicides and insecticides
02/05/2003CN1100759C Xanthene and arcridine derivative and its use
02/05/2003CN1100540C Protein tyrosine kinase aryl and heteroaryl quinazoline compounds having selective inhibition of HER-2 autophosphorylation properties
02/04/2003US6515151 Method for the preparation of novel sidechain-bearing taxanes and intermediates thereof
02/04/2003US6515133 Certain diaryl imidazoles act as partial agonists or antagonists for NPY receptors, in particular NPY 5 receptors. They are of use, for example in treating loss of appetite. Such compounds bear aryl groups in the 2 position.
02/04/2003US6515124 Dehydroamino acids
02/04/2003US6515013 For diseases or conditions caused by or exacerbated by histamine-3 receptor activity
02/04/2003US6515002 Compounds and compositions for treating C1s-mediated diseases and conditions