Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
01/2003
01/23/2003US20030018025 Psychological disorders, antidepressants, Parkinson's disease
01/23/2003US20030018012 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
01/23/2003CA2453503A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003CA2453175A1 Interaction inhibitors of tcf-4 with beta-catenin
01/23/2003CA2451566A1 Use of nk-1 receptor antagonists for the treatment of brain, spinal or nerve injury
01/23/2003CA2446726A1 Piperazine oxime derivatives having nk-1 receptor antagonistic activity
01/23/2003CA2418173A1 N-substituted-1-amino-1,1-dialkylcarboxylic acid derivatives
01/23/2003CA2417156A1 3,4-dihydroisoquinoline derivative compound and a pharmaceutical agent comprising it as active ingredient
01/22/2003EP1277751A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277749A1 2- and 2,5-substituted phenylketo enols
01/22/2003EP1277744A1 Oxadiazole derivatives having anticancer effects
01/22/2003EP1277743A1 Oxa(thia)zolidine derivative and anti-inflammatory drug
01/22/2003EP1277738A1 Condensed heteroaryl derivatives
01/22/2003EP1277735A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277734A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277733A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1276741A1 Phenyl substituted 4-hydroxy tetrahydropyridone
01/22/2003EP1276738A1 2-amino-3-(alkyl)-pyrimidone derivatives as gsk3.beta. inhibitors
01/22/2003EP1276726A2 Substituted phenyl farnesyltransferase inhibitors
01/22/2003EP1276725A2 5-substituted tetralones as inhibitors of ras farnesyl transferase
01/22/2003EP1276723A2 Pyrazole compounds having anti proliferative activity
01/22/2003EP1276720A2 2-acyl indol derivatives and their use as anti-tumour agents
01/22/2003EP1030835B1 Urea derivatives and their use as integrin inhibitors
01/22/2003EP0909174A4 Treatment of cystic disease with tnf-alpha
01/22/2003EP0898562B1 Hydroxamic acid derivatives for use with the treatment of diseases related to connective tissue degradation
01/22/2003EP0782575B1 Substituted pyrazolyl-pyrazole derivatives, processes for their preparation and their use as agents with herbicidal action
01/22/2003EP0646115B1 Heterocyclic-cyclic amine derivatives
01/22/2003CN1392874A Cyclic amidine compounds
01/22/2003CN1099413C Certain fused N-pyrrolylaniline: new class of GABA brain receptor ligand
01/21/2003US6509469 Process for the production of pyridine derivatives
01/21/2003US6509369 Triphenylpropanamide compounds; useful in treating inflammations but which do not demonstrate side effects associated with other anti-inflammatory treatments such as glucocorticoids
01/21/2003US6509362 Cholesteryl acyl transferase (ACAT) inhibitors; treatment of hyperlipidaemia and atherosclerosis.
01/21/2003US6509357 1-aryl or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands
01/21/2003US6509346 Chemokine receptor antagonists and methods of use therefor
01/21/2003US6509331 Deoxyamino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting β-amyloid peptide release and/or its synthesis by use of such compounds
01/21/2003US6509328 Glutamate receptor antagonists
01/21/2003US6508957 Fluorescent maleimides and uses thereof
01/16/2003WO2003004493A1 Novel compounds, their preparation and use
01/16/2003WO2003004486A2 Process for preparing isocoumarins
01/16/2003WO2003004485A1 Benzo-fused 5-membered hetrocycle compounds, process for preparation of the same, and use thereof
01/16/2003WO2003004480A2 Substituted piperazine and diazepanes as histamine h3 receptor agonists
01/16/2003WO2003004475A1 Heterocyclic amines for the treatment of conditions associated with gsk-3
01/16/2003WO2003004028A1 Tetrahydroquinoline derivatives
01/16/2003WO2003004027A1 Substituted anilinic piperidines as mch selective antagonists
01/16/2003WO2003004023A1 1-alkyl-2-aryl-benzimidazole derivatives, their use for producing medicaments and pharmaceutical preparations containing said derivatives
01/16/2003WO2003004022A1 Aryl (or heteroaryl) azolylcarbynol derivatives for the treatment of urinary incontinence
01/16/2003WO2002051837A3 Heterocyclindazole and azaindazole compounds as 5-hydroxytryptamine-6 ligands
01/16/2003WO2002050062A3 Benzimidazole and pyridylimidazole derivatives as ligands for gaba receptors
01/16/2003WO2002012196A3 Lactam compounds and their use as inhibitors of serine proteases and method
01/16/2003US20030013894 Comprises conversion of oxalamide to dithiooxalamide, followed by conversion of the dithiooxalamide to either a 4,5-bisimino-(1,3)dithiolane or 2,3-bisimino-(1,4)dithiane
01/16/2003US20030013892 Production of chirally pure alpha-amino acids and N-sulfonyl alpha-amino acids
01/16/2003US20030013886 Such as (E)-1-(2-Pyridyl)-2-styryl-1H-benzimidazole; antiinflammatory and analgesic agents; prostaglandin inhibitors
01/16/2003US20030013875 3-azabicyclo[3.1.0]hexane derivatives useful in therapy
01/16/2003US20030013757 Aromatic dicarboxylic acid derivatives
01/16/2003US20030013744 3,4-diaryl thiophenes and analogs thereof having use as anti-inflammatory agents
01/16/2003US20030013742 Antiinflammatory agents; skin disorders
01/16/2003US20030013724 Novel prolines as antimicrobial agents
01/16/2003US20030013712 Antiinflammatory agents
01/16/2003US20030013706 Autoimmune disease; antiinflammatory agents
01/16/2003US20030013041 Write-once optical data carrier
01/16/2003CA2454613A1 Substituted anilinic piperidines as mch selective antagonists
01/16/2003CA2452646A1 Derivatives of aryl(or heteroaryl) azolylcarbinols for the treatement ofurinary incontinence
01/16/2003CA2448913A1 Sulfone containing bicyclic aromatic ring compounds, their preparation and use as nicotinic acetyl-chloine receptors
01/15/2003EP1275644A1 Benzenesulfonamide derivatives, process for their preparation and pharmaceutical compositions containing them
01/15/2003EP1275389A1 Compositions containing C7 Taxanes
01/15/2003EP1274706A1 Pyrazoles for inhibiting protein kinases
01/15/2003EP1274705A1 2-substituted 4-heteroaryl-pyrimidines and their use in the treatment of proliferative disorders
01/15/2003EP1274701A1 Chemical compounds
01/15/2003EP1274683A2 Heterocyclic acylsulfimides, a method for their production, agents containing the same and their use as pesticides
01/15/2003EP1274424A1 Compounds and methods
01/15/2003EP0974584B1 Fused ring compounds, process for producing the same and use thereof
01/15/2003EP0925287B1 Heterocyclic metalloprotease inhibitors
01/15/2003EP0907643B1 Compounds with growth hormone releasing properties
01/15/2003EP0729468B1 Non-peptide tachykinin receptor antagonists
01/15/2003EP0722442B1 Polyazacycloalkanes as dichelants
01/15/2003EP0713483B1 Amidine derivatives with nitric oxide synthetase activities
01/15/2003EP0649412B1 Pharmaceutical pyridine compounds
01/15/2003CN1391571A Heterocyclic compounds and their use as medicines
01/15/2003CN1391565A Benzophenones as inhibitors of reverse transcriptase
01/15/2003CN1391563A Therapeutic quinazoline derivatives
01/15/2003CN1391562A Quinazoline derivatives as pharmaceuticals
01/15/2003CN1391560A 喹唑啉衍生物 Quinazoline derivatives
01/15/2003CN1391558A Substituted 1,3-diaryl-2-pyridine-2-yl-3-(pyridine-2-ylamino)-propanol derivatives, methods for their production, pharmaceutical compositions containing the same and their use
01/15/2003CN1391556A IL-8 receptor antagonists
01/15/2003CN1391555A Benzamides and related inhibitors of factor Xa
01/15/2003CN1391475A Optically active isomers of ketotifen and therapeutically active metabolites thereof
01/15/2003CN1391474A 5-membered heterocycle derivatives, production thereof and use as medicaments
01/15/2003CN1390834A Indenoindolone compounds, their preparation and medicinal compositions containing them
01/15/2003CN1098838C Substituted N-(indole-2-carbonyl)-beta-alanimamides and derivatives as antidiabetic agents
01/14/2003US6506936 N-substituted arylsulfonylamino hydroxamic acids useful as inhibitors of c-proteinase and for treating or preventing disorders related to unregulated collagen production
01/14/2003US6506901 1-(9H-Carbazol-4-yloxy)-3-((1-(7-trifluoromethyl-quinolin-4-yl) -piperidin-4-lmethyl)-amino)-propan-2-ol, for example; treating diabetes, urinary continence, atherosclerosis, gastrointestinal disorders, glaucoma
01/14/2003US6506876 LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use
01/14/2003US6506777 Method for modulation of CCR-3 or CCR-5 chemokine receptor activity in a mammal in need thereof to treat asthma, allergic rhinitis, dermatitis, conjunctivitis, atherosclerosis or rheumatoid arthritis, which comprises the administration of an
01/14/2003US6506770 Antiviral compounds
01/14/2003US6506747 Method of treating an inflammatory disease which comprises administering to a patient in need of such treatment-a N-(4-(5-Ethyl-3-pyridin-3-yl-pyrazol-1-yl)phenyl)pyridine-3-carboxamide;
01/14/2003US6506538 Ophthalmic lenses, contact lenses, solar protection glasses, filters, camera optics or photographic apparatus optics or other optical devices
01/14/2003US6506517 Surface modified carbonaceous materials
01/14/2003US6506507 Methine compound, material for organic luminescence element, and organic luminescence element using the same
01/14/2003CA2217516C Triazole antifungal agent
01/14/2003CA2217477C Tricyclic compounds useful for inhibition of farnesyl protein transferase