Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
07/2002
07/25/2002WO2002057246A2 Inhibitors of cruzipain and other cysteine proteases
07/25/2002WO2002057240A1 Substituted triazole diamine derivatives as kinase inhibitors
07/25/2002WO2002057224A2 Synthesis and antimicrobial activityof novel dicationic 'reversed amidines'
07/25/2002WO2002050061A8 Piperazine derivatives for treatment of bacterial infections
07/25/2002WO2002042268A3 Ep4 receptor selective agonists in the treatment of osteoporosis
07/25/2002WO2002008177A3 N-substituted-1-amino-1,1-dialkylcarboxylic acid derivatives
07/25/2002WO2002006229A3 Heterocyclic beta-3 adrenergic receptor agonists
07/25/2002WO2001068096A3 Combination therapy for the prophylaxis and treatment of hyperlipidemic conditions and disorders
07/25/2002US20020099212 Sulfonamide compounds and pharmaceutical use thereof
07/25/2002US20020099071 Protein tyrosine kinase and protein serin/threonine kinase inhibitory activity; anticancer agents; treating chemotherapy induced alopecia
07/25/2002US20020099038 O- or S- substituted tetrahydronaphthalene derivatives having retinoid and/or retinoid antagonist-like biological activity
07/25/2002US20020099035 Method for preparing alpha-sulfonyl hydroxamic acid derivatives
07/25/2002DE10158803A1 Production of difluoromethoxy-bridged compounds, involves addition of acid to ketene dithioketal, reaction of the carbenium salt with hydroxy compound and fluorodesulfurisation of the dithio-ortho-ester
07/25/2002CA2435117A1 Cyclic 2-carbonylaminoketones as inhibitors of cruzipain and other cysteine proteases
07/25/2002CA2434068A1 Inhibitors of cruzipain and other cysteine proteases
07/25/2002CA2432870A1 Substituted triazole diamine derivatives as kinase inhibitors
07/25/2002CA2425135A1 Synthesis and antimicrobial activity of novel dicationic "reversed amidines"
07/24/2002EP1225169A1 Radiation-activated cytotoxin therapy
07/24/2002EP1224197A1 Hygromycin derivatives
07/24/2002EP1224183A2 Heterocyclic sodium/proton exchange inhibitors and method
07/24/2002EP1224182A1 N-substituted 1-(lactone) isoquinolones for treating nervous disorders
07/24/2002EP1224180A2 Substituted azoles
07/24/2002EP1224175A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
07/24/2002EP1224174A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
07/24/2002EP1223933A2 5-membered heterocycle derivatives, production thereof and use thereof as medicaments
07/24/2002EP1223932A1 Compounds and methods
07/24/2002EP1223809A1 Methods of treating hair loss comprising administering indoline compound
07/24/2002EP0889041B1 Novel iridoid derivatives and neovascularization inhibitors containing the same as active ingredient
07/24/2002CN1360583A Novel compounds, their use and preparation
07/24/2002CN1360577A Hydroxamic acid derivs. as matrix metalloprotease inhibitors
07/24/2002CN1088063C Sulfmidyl (thio) carbonyl-1,2,4-triazolineone deriv. and preparation method and application as weed killer
07/23/2002US6423840 Forming n-acylamino compound
07/23/2002US6423729 Therapeutic or prophylactic agent for glomerulopathy
07/23/2002US6423725 Analgesics
07/23/2002US6423717 Nervous system disorders
07/23/2002US6423713 Substituted pyrazoles as p38 kinase inhibitors
07/23/2002US6423710 Cyclic AMP-specific phosphodiesterase inhibitors
07/23/2002US6423707 Nitroimidazole ester analogues and therapeutic applications
07/23/2002US6423704 Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic diseases
07/23/2002CA2102180C Novel immunosuppressive pyrrolidine/piperidine/azepane-2-carboxylic acid derivatives
07/18/2002WO2002055514A2 Substituted benzimidazol-2-ones as vasopressin receptor antagonists and neuropeptide y modulators
07/18/2002WO2002055501A2 N-pyridyl carboxamide derivatives and pharmaceutical compositions containing them
07/18/2002WO2002055496A1 Aryl piperidine and piperazine derivatives as inducers of ldl-receptor expression
07/18/2002WO2002055484A1 Biaryl compound, process for producing the same, and agent
07/18/2002WO2002040455A8 Substituted amidoalkyl uracils and their use as inhibitors of the poly(adp-ribose) synthetase (pars)
07/18/2002WO2001096299A3 Indole derivatives and their use as 15-lipoxygenase inhibitors
07/18/2002WO2001072685A3 Polyamine analogues as cytotoxic agents
07/18/2002WO2001056974A3 Inha inhibitors and their use as antibacterials
07/18/2002US20020094994 Pyrrolidine carboxylic Acid or ester derivatives are useful for treating alpha 4 beta 1 mediated cell adhesion
07/18/2002US20020094989 Pyrrolidine modulators of CCR5 chemokine receptor activity
07/18/2002CA2434274A1 N-pyridyl carboxamide derivatives and pharmaceutical compositions containing them
07/17/2002EP1223169A1 Agent for potentiating nerve growth factor activity containg 1,2-ethanediol derivate or salt thereof
07/17/2002EP1223166A1 Linked cyclic polyamines with activity against hiv.
07/17/2002EP1222308A1 Antiprotozoal histone acetyl transferase inhibitors
07/17/2002EP1222305A2 Enzymatic process for the resolution of enantiomeric mixtures of beta-lactams
07/17/2002EP1222182A2 Substituted (aminoiminomethyl or aminomethyl) dihydrobenzofurans and benozopyrans
07/17/2002EP1222176A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF A$g(b) PROTEIN PRODUCTION
07/17/2002EP1222174A1 Imidazol-4-ylmethanols used as inhibitors of steroid c17-20 lyase
07/17/2002EP1222171A1 Pyridinium derivatives for the management of aging-related and diabetic vascular complications, process for their preparation and therapeutic uses thereof
07/17/2002EP0939629A4 Thiol sulfonamide metalloprotease inhibitors
07/17/2002EP0888340B1 4-(benzo-1,3-dioxolyl)-pyrrolidine-3-carboxylic acid derivatives as endothelin antagonists
07/17/2002EP0882044B1 1,4-dihydropyridine compounds as bradykinin antagonists
07/17/2002CN1359377A Dihydrobenzodiazepins and their use for treating dyslipidemia
07/17/2002CN1358719A Process for synthesizing sertaconazole
07/17/2002CN1087737C Dihygropyridine derivatives as bradykinin ant agonists
07/17/2002CN1087736C Novel amidinonaphthyl derivative or salt thereof
07/16/2002US6420567 Prodrugs
07/16/2002US6420563 Inverse antagonist
07/16/2002US6420541 Non-endogenous, constitutively activated human serotonin receptors and small molecule modulators thereof
07/16/2002US6420438 1-amino-7-isoquinoline derivatives as serine protease inhibitors
07/16/2002US6420417 Combination therapy employing ileal bile acid transport inhibiting benzothiepines and HMG Co-A reductase inhibitors
07/16/2002US6420415 Thiol compounds, their production and use
07/16/2002US6420412 Eprosartan dihydate and a process for its production and formulation
07/16/2002US6420409 Benzimidazole derivatives
07/16/2002US6420396 Biphenyl and biphenyl-analogous compounds as integrin antagonists
07/16/2002US6420393 Nuclear factor .kappa.b-dependent disease selected from the group consisting of inflammatory diseases, immunological disorders, septic shock, transplant rejection, radiation damage, reperfusion injuries after ischemia, stroke or
07/16/2002US6420392 Paf receptor antagonists and/or by inhibiting the enzyme 5-lipoxygenase.
07/16/2002US6420391 Fused thiophone derivatives and drugs containing the same as the active ingredient
07/16/2002US6420385 Substituted pyrimidinone and pyridone compounds and methods of use
07/16/2002US6420375 Fused ring compounds, process for producing the same and use thereof
07/16/2002US6420316 Substituted aromatic thiocarboxylic acid amides and their use as herbicides
07/16/2002US6420315 5-thien-3-yl-2-oxy- or -2-thio-pyridines; high selectivity for broadleaf and grassy weeds in crops, such as maize and rice; pre- and post-emergence
07/16/2002US6420313 Defoliants, desiccants; controlling weeds, such as monocotyledons and dicotyledons in crop fields; pre- and post-emergence; cyclization and alkylation of a biguanide and an alkoxycarbonyl compound
07/11/2002WO2002053558A1 Quinazolone derivatives as alpha 1a/b adrenergic receptor antagonists
07/11/2002WO2002053557A1 Novel sulfamides and their use as endothelin receptor antagonists
07/11/2002WO2002053155A1 Telomerase inhibitor
07/11/2002WO2002028353A3 Phosphate transport inhibitors
07/11/2002WO2001040187A3 Compound having effect of promoting neuron differentiation
07/11/2002US20020091274 Taxane derivatives having an amino substituted C13 side chain useful as antileukemia and antitumor agents
07/11/2002US20020091272 Sulfonamides and derivatives thereof that modulate the activity of endothelin
07/11/2002US20020091270 Sulfonamides containing oxazole and substituted thiophene rings, useful for treating hypertension, cardiovascular disease, asthma, pulmonary hypertension, inflammatory diseases, vision defects, menstrual disorders, renal failure
07/11/2002US20020091210 Group 8-10 transition metal based supported catalyst where the support is treated with a pore-filling agent; improved the catalyst productivity in the presence of hydrogen
07/11/2002US20020091150 Carbamic acid derivatives
07/11/2002US20020091148 3-substituted indole antiproliferative angiogenesis inhibitors
07/11/2002US20020091124 Also used as an antimitotic and for direct and/or indirect inhibition of tubulin polymerization in mammalian
07/11/2002US20020091122 Voltage-dependent
07/11/2002US20020091116 Show selectivity for factor Xa versus other proteases of coagulation or the fibrinolytic cascades
07/11/2002US20020091078 Treating diabetes, especially Type II diabetes
07/10/2002EP1221441A2 LTA4 Hydrolase inhibitors
07/10/2002EP1221440A1 Benzoheterocyclic derivatives useful as vasopressin or oxytocin modulators