Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
03/2003
03/18/2003CA2217351C Carbonyl-piperazinyl and piperidinyl compounds which inhibit farnesyl protein transferase
03/13/2003WO2004043335A2 Methods of treating infection by drug resistant bacteria
03/13/2003WO2003020718A1 Photochromic bis-naphthopyran compounds and methods for their manufacture
03/13/2003WO2003020248A1 Plaster for the treatment of dysfunctions and disorders of nails, comprising sertaconazole
03/13/2003WO2003020217A2 Novel pyrazole analogs acting on cannabinoid receptors
03/13/2003WO2002076950A3 Imidiazole derivatives and their use as agonists selective at alpha 2b or 2b/2c adrenergic receptors
03/13/2003WO2002066469A3 Novel heterocyclic amide derivatives and their use as dopamine d3 receptor ligands
03/13/2003US20030050330 And inflammation-associated disorders, such as arthritis
03/13/2003US20030050320 A therapeutic agent for treating hepatitis C, based on polymerase inhibitory activity
03/13/2003US20030050315 An inhibitors of trypsin-like serine protease enzymes, as anticoagulant agents for treatment and prevention of thromboembolic disorders
03/13/2003US20030050288 Substituted indoline derivative compounds which are antagonists of the progesterone receptor; oral contraception using multiphase progestotational agents, antiprogestins, indole or thiophene derivatives and placebo
03/13/2003US20030050251 A polypeptide which inhibits or reduces tumor progression and/or metastasis
03/13/2003CA2459866A1 Photochromic bis-naphthopyran compounds and methods for their manufacture
03/13/2003CA2458926A1 Methods of treating infection by drug resistant bacteria
03/13/2003CA2458399A1 Cyclic indole and heteroindole derivatives, the production and use thereof as medicaments
03/13/2003CA2457922A1 Novel pyrazole analogs acting on cannabinoid receptors
03/12/2003EP1291345A1 Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
03/12/2003EP1290000A1 Novel chromophores for polymeric thin films and optical waveguides and devices comprising the same
03/12/2003EP1289980A1 Bicyclyl or heterobicyclylmethanesulfonylamino-substituted n-hydroxyformamides
03/12/2003EP1289972A1 Serine protease inhibitors
03/12/2003EP1289965A1 Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists
03/12/2003EP1289964A1 Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists
03/12/2003EP1289963A1 Fungicidal 5-phenyl substituted 2-(cyanoamino) pyrimidines
03/12/2003EP1289957A1 Pharmaceutically active piperidine derivatives, in particular as modulators of chemokine receptor activity
03/12/2003EP1289956A1 Chemical compounds
03/12/2003EP1289955A1 Piperidines for use as orexin receptor antagonists
03/12/2003EP1289954A1 Serine protease inhibitors
03/12/2003EP1289525A2 Tricyclic pyrazole derivatives as protein kinase inhibitors
03/12/2003CN1402712A Novel heterocyclic compounds and salts thereof and medicinal use of same
03/12/2003CN1402710A Antipicornaviral compound and compositions, their pharmaceutical uses, and material for their synthesis
03/12/2003CN1402708A Process for production of pyridine derivs.
03/11/2003US6531599 Compounds having activity as inhibitors of cytochrome P450RAI
03/11/2003US6531502 3-Methylidenyl-2-indolinone modulators of protein kinase
03/11/2003US6531497 Epothilone derivatives and their synthesis and use
03/11/2003US6531479 Anti-cancer compounds
03/11/2003CA2254117C 2,4-diaminopyrimidine derivatives
03/10/2003CA2401358A1 Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
03/06/2003WO2003018575A1 5-substituted-3(2h)-furanones useful for inhibition of farnesyl-protein transferase
03/06/2003WO2003018556A1 Piperidine derivatives useful as modulators of chemokine receptor activity
03/06/2003WO2003018547A2 An improved process for the preparation of amorphous atorvastatin calcium salt (2:1)
03/06/2003WO2003018538A1 Novel diarylalkene derivatives and novel diarylalkane derivatives
03/06/2003WO2003018008A1 Apo ai expression accelerating agent
03/06/2003WO2003017764A1 Substituted propargylamines
03/06/2003WO2002100844A3 Hiv protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
03/06/2003WO2002072570A3 Non-imidazole compounds as histamine h3 antagonists
03/06/2003WO2002066443A3 2-thioxo-1,2,3,4-tetrahydropyrimidine derivatives
03/06/2003WO2002057224A3 Synthesis and antimicrobial activityof novel dicationic 'reversed amidines'
03/06/2003WO2002000650A9 Novel compounds possessing antibacterial, antifungal or antitumor activity
03/06/2003US20030045755 Polyamine analogues as cytotoxic agents
03/06/2003US20030045728 Indol-3-yl derivatives
03/06/2003US20030045726 Novel immunotherapeutic agents
03/06/2003US20030045554 Such as 1-(2-thien-2'-yl- 2-oxoethyl)-3-((3-phenylmethyl) pyrazol-5-yl)pyridinium bromide for treating diseases caused by the accumulation of AGE (Advanced Glycation Endproducts); antidiabetic/ antiaging agents
03/06/2003US20030045552 Isoindole-imide compounds, compositions, and uses thereof
03/06/2003US20030045546 Anticancer agents
03/06/2003US20030045531 Antileukemia and antitumor agents
03/06/2003US20030045519 Treating allergy, allergy-induced airway responses, and congestion (e.g., nasal congestion)
03/06/2003US20030045516 Chemokine receptor antagonists and methods of use therefor
03/06/2003US20030044402 Oligo(ethylene glycol)-terminated 1,2-dithiolanes and their conjugates useful for preparing self-assembled monolayers
03/06/2003US20030044399 Method of treatment
03/05/2003EP1288202A1 N-acyltetrahydroisoquinoline derivatives
03/05/2003EP1286986A1 Quinolinyl-piperidin-4-ylidene-methyl-benzamide derivatives for the treatment of pain
03/05/2003EP1286985A1 Substituted pyridine herbicides
03/05/2003EP1286984A2 Method for the preparation of tetrahydrobenzothiepines
03/05/2003EP1286966A1 4-aminopiperidine derivatives and their use as medicine
03/05/2003EP1286955A1 Aryl and heteroarylcyclopropyl oxime ethers and their use as fungicides
03/05/2003EP1286704A2 Ethylenedicysteine (ec)-drug conjugates
03/05/2003EP1286673A2 Ligands of integrin receptors
03/05/2003EP1194427B1 Thiophene-ethyl thiourea compounds and use in the treatment of hiv
03/05/2003EP1169316B1 Novel lipoic acid derivatives, their preparation, and pharmaceutical compositions containing them
03/05/2003EP1119560B1 Naphthopyrans annelated in c5-c6, their preparation and compositions and (co) polymer matrices containing them
03/05/2003EP1115719B1 Novel amidine derivatives, their preparation and application as medicines and pharmaceutical compositions containing same
03/05/2003EP0966447B1 Small molecules useful in the treatment of inflammatory disease
03/05/2003EP0945438B1 Pyrazole derivatives
03/05/2003EP0942901B1 Cyclic imines as pesticides
03/05/2003EP0832069B1 BIPHENYL-2-CARBOXYLIC ACID-TETRAHYDRO-ISOQUINOLIN-6-YL AMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS INHIBITORS OF MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN AND/OR APOLIPOPROTEIN B (Apo B) SECRETION
03/05/2003EP0831830B1 Imidazole compounds
03/05/2003CN1400970A Substituted arylpyrazines
03/05/2003CN1400968A Method for preparing alpha sulfonyl hydroxamic acid derivatives
03/05/2003CN1400210A Oligothiophene derivative, its preparation method and application
03/05/2003CN1102580C Arylethenesulfonamide derivatives and drug composition containing the same
03/05/2003CN1102573C Aryl or heteroaryl substd, 3,4-dihydroanthracene and benzo [1,2-g]-chrom-3-ene, benzo[1,2-g]-thiochrom-3-ene and benzo [1,2-g]-1,2-dihydroquinoline derivs having bioactivity of visual pigmentoid
03/04/2003US6528659 Condensation between protected and unprotected pyrroles to form chemical intermediates; deprotecting; easier purifi-cation, isolation, storage and transportation
03/04/2003US6528655 Aromatic derivatives with HIV integrase inhibitory properties
03/04/2003US6528538 Cyclic compounds useful in the treatment of dyslipidaemia, atherosclerosis and diabetes, pharamaceutical compositions and preparation process
03/04/2003US6528535 Bicyclic inhibitors of protein farnesyl transferase
03/04/2003US6528532 Benzenesulfonamide group
03/04/2003US6528510 HIV protease inhibitors
03/04/2003CA2218913C Substituted oximes, hydrazones and olefins as neurokinin antagonists
03/04/2003CA1341424C Diketohexanoic acids and 2- and 3-diloweralkyl derivatives thereof
02/2003
02/27/2003WO2003016308A1 N-heterocyclyl substituted thienyloxy-pyrimidines used as herbicides
02/27/2003WO2003016306A1 Hiv inhibiting pyrimidines derivatives
02/27/2003WO2003016297A1 Lactone derivative, and plant growth regulator and rooting agent each containing the same as active ingredient
02/27/2003WO2003016286A1 3-phenoxy-4-pyridazinol derivative and herbicide composition containing the same
02/27/2003WO2003016276A2 3-substituted oxindole beta-3 agonists
02/27/2003WO2003016275A1 Antiviral agent
02/27/2003WO2003015790A1 Thiopyrane-4-ones as dna protein kinase inhibitors
02/27/2003WO2003015774A1 Compounds effecting glucokinase
02/27/2003WO2003015769A1 Aminoalkyl-substituted aromatic bicyclic compounds, method for the production thereof and their use as medicaments
02/27/2003WO2003000181A3 Dipeptidyl peptidase inhibitors for the treatment of diabetes
02/27/2003WO2002100851A3 Thiophene derivatives as antiviral agents for flavivirus infection