Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
04/2003
04/03/2003WO2003027074A1 Pyrazole derivatives useful in the treatment of hyper-proliferative disorders
04/03/2003WO2003027061A2 Muscarinic agonists
04/03/2003WO2003026666A1 2-phenylamino-4- (5-pyrazolylamino)-pyrimidine derivatives as kinase inhibitors, in particular, as src kinase inhibitors
04/03/2003WO2003026665A1 2-phenylamino-4-(5-pyrazolylamino)-pyrimidine derivatives as kinase inhibitors, in particular, src kinase inhibitors
04/03/2003WO2003026664A1 2-phenylamino-4- (5-pyrazolylamino) -pyramidine derivatives as kinase inhibitors, in particular, src kinase inhibitors
04/03/2003WO2003026660A1 An enantiomerically pure diarylmethylpiperazine and methods of using same
04/03/2003WO2003026648A1 4,5-dihydro-1h-pyrazole derivatives having potent cb1-antagonistic activity
04/03/2003WO2003026647A1 Novel 4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic activity
04/03/2003WO2003026587A2 Compounds useful for treating hepatitus c virus
04/03/2003WO2003002531A3 Fluoropyrrolidines as dipeptidyl peptidase inhibitors
04/03/2003WO2003002530A3 Pyrrolidines as dipeptidyl peptidase inhibitors
04/03/2003WO2002100974A3 Core guest host system comprising a chromophore in a polycarbonate matrix
04/03/2003WO2002092563A3 Protease inhibitors
04/03/2003WO2002074738A3 Spiro-cyclic beta-amino acid derivatives as inhibitors of matrix metalloproteinases and tnf-alpha converting enzyme (tage)
04/03/2003WO2002039954A3 Novel compounds
04/03/2003WO2002013808A3 Treatment of tumors with acetylenes distributed with a phenyl or heteroaromatic group and a substituted chromanyl, thiochromanyl or tetrahydroquinolinyl group in combination with other anti-tumor agents
04/03/2003US20030065200 Taxanes having T-butoxycarbonyl substituted side-chains and pharmaceutical compositions containing them
04/03/2003US20030065187 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
04/03/2003US20030065179 Diabetic therapy
04/03/2003US20030065176 Anticoagulant; cardiovascular disorders
04/03/2003US20030065034 Antiinflammatory agents; coupling sulfonyl halide with aromatic amine compound
04/03/2003US20030065012 Estrogen receptor modulators
04/03/2003US20030065007 Analgesics; psychological disorders; antidepressants
04/03/2003US20030065004 Androgen receptor modulators and methods for use thereof
04/03/2003US20030064997 Novel compounds
04/03/2003US20030064992 N-aryl (thio) anthranilic acid amide derivatives, their preparation and their use as VEGF receptor tyrosine kinase inhibitors
04/03/2003US20030064982 Pyrazole compounds useful as protein kinase inhibitors
04/03/2003US20030064981 Anticancer agents; antidiabetic agents; Alzheimer's disease
04/03/2003US20030064980 Respiratory system disorders; antiinflammatory agents
04/03/2003US20030064977 Viricides
04/03/2003US20030062509 Field effect transistor, OLED, electroluminescent device, RFID tag, backlight, photovoltaic or sensor device, or electrophotographic recording device; security marking; charge injection layer, planarising layer, antistatic film
04/03/2003CA2461709A1 Small organic molecule regulators of cell proliferation
04/03/2003CA2461363A1 Substituted 3-pyridyl indoles and indazoles as c17,20 lyase inhibitors
04/03/2003CA2461360A1 3-pyridyl or 4-isoquinolinyl thiazoles as c17,20 lyase inhibitors
04/03/2003CA2461128A1 Pyrazole derivatives useful in the treatment of hyper-proliferative disorders
04/03/2003CA2460000A1 Inhibitors of glycogen synthase kinase-3 (gsk-3) for treating glaucoma
04/02/2003WO2002030891A1 Aliphatic nitrogenous five-membered ring compounds
04/02/2003EP1298496A2 Electrophotographic organophotoreceptors
04/02/2003EP1298125A1 Substituted benzimidazole compounds and their use for the treatment of cancer
04/02/2003EP1296978A2 N-ureidoheterocycloaklyl-piperidines as modulators of chemokine receptor activity
04/02/2003EP1296975A1 4-heteroaryl-3-heteroarylidenyl-2-indolinones and their use as protein kinase inhibitors
04/02/2003EP1296974A2 2-cyanopyrrolidine derivatives and their use as medicaments
04/02/2003EP1296973A1 Guanidine derivatives of quinazoline and quinoline for use in the treatment of autoimmune diseases
04/02/2003EP1296972A1 Arylmethylamine derivatives for use as tryptase inhibitors
04/02/2003EP1296961A1 1,4-diazepan-2,5-dione derivatives and their use as nk-1 receptor antagonists
04/02/2003EP1296950A2 Aminopiperidines for use as glyt-1 inhibitors
04/02/2003EP1296931A2 Polyamine analogues as cytotoxic agents
04/02/2003EP1204668B1 Bisimidino compounds and the transitional metal complexes thereof as well as the use thereof as catalysts
04/02/2003EP1135386B1 Method for producing pyrazolylbenzoyl derivatives and novel pyrazolylbenzoyl derivatives
04/02/2003EP1015446B1 (4-piperidinyl)-1h-2-benzopyran derivatives useful as antipsychotic agents
04/02/2003EP0991643B1 Novel aminooxyamide tricyclic inhibitors of farnesylprotein transferase
04/02/2003EP0951467B1 SUBSTITUTED NITROGEN CONTAINING HETEROCYCLES AS INHIBITORS OF p38 PROTEIN KINASE
04/02/2003EP0912512B1 Sulphonamide derivatives and their use in the treatment of cns disorders
04/02/2003EP0880504B1 Heterocyclo-substituted imidazoles for the treatment of inflammation
04/02/2003EP0681574B1 C7 Taxane derivatives and pharmaceutical compositions containing them
04/02/2003CN1407971A Substituted 2-thio-3,5-dicyano-4-aryl-6-aminopyridines and the use thereof
04/02/2003CN1407970A Urea compounds having muscarinic receptor antagonist activity
04/02/2003CN1406937A 1-[1-(hetero) aryl-1-perhydroxyalkylmethyl]-piperazine compound, preparation thereof and pharmaceutics containing it
04/02/2003CN1104429C 4-(3-heterocycly-1-benzoyl) pyrazoles and their use as herbicides
04/02/2003CN1104418C Benzoheterocyclic derivatives
04/01/2003US6541638 (2S,4S)-1-(4-Mercapto-1-(naphthalene-2-sulfonyl)-pyrrolidine-2 -carbonyl)-piperidine-4-carboxylic acid ethyl ester for example; zinc protease inhibitors; for treating diseases associated with vasoconstriction
04/01/2003US6541505 Inhibiting the activity of Factor Xa; treating a disease state associated with a physiologically detrimental excess amount of thrombin.
04/01/2003US6541491 4-mercaptopyrrolidine derivatives as farnesyl transferase inhibitors
04/01/2003US6541489 Excellent inhibitory activity of one or more matrix metalloprotease (MMP) enzymes, such as MMP-2, MMP-9, and MMP-13, while exhibiting substantially less inhibition at least of MMP- 1
04/01/2003US6541477 Inhibitors of p38-a kinase
04/01/2003US6541476 Piperazine derivatives and their use as anti-inflammatory agents
04/01/2003US6541474 Administering a pharmaceutically effective dose of the heterocycle-containing carboxylic acid derivative or salt to a patient suffering form acute promyelocytic leukemia
04/01/2003US6541470 Have a potent antiviral activity against picornaviruses and rotaviruses.
04/01/2003US6541209 Bioassay; identification of compounds as agonists; use in treatment of diseases and disorders that are related to 5-HT2A and or 5-HT2C serotonin receptors
03/2003
03/27/2003WO2003024961A1 Insecticidal 3-(2,6-disubstituted phenyl)-5-[4- or 5-arylthien-2- or -3-yl]-1,2,4-triazoles
03/27/2003WO2003024955A2 Small molecule inhibitors of caspases
03/27/2003WO2003024954A1 Novel terthiophene-3-carboxylic acid compound and fabricating method thereof, functionalized conductive terthiophene polymer with the compound as a monomer, process for dna hybridizatioon detection using the polymer, and fabricating method of probe dna
03/27/2003WO2003024950A1 Coumarin derivative
03/27/2003WO2003024949A1 Dna-pk inhibitors
03/27/2003WO2003024948A1 Benzofuran and dihydrobenzofuran derivatives useful as beta-3 adrenoreceptor agonists
03/27/2003WO2003024935A2 Substituted pyrazolyl compounds for the treatment of inflammation
03/27/2003WO2003024933A1 2-phenyl-3-heteroarylpropionic acid derivative or salt thereof and medicine containing the same
03/27/2003WO2003024929A1 Substituted piperidines with selective binding to histamine h3-receptor
03/27/2003WO2003024926A2 Methods and compositions of novel triazine compounds
03/27/2003WO2003024453A1 Excitatory amino acid receptor antagonists
03/27/2003WO2003024451A1 2-(2-phenylethyl)-benzimidazole-5-carboxamide derivatives and their use as tryptase inhibitors
03/27/2003WO2003024448A2 Inhibitors of histone deacetylase
03/27/2003WO2003024441A1 Novel use of tricyclic compound
03/27/2003WO2003024220A1 Delta 1-pyrrolines used as pesticides
03/27/2003WO2002101007A3 Antipathogenic benzamide compounds
03/27/2003WO2002078628A3 Cyanamide, alkoxyamino, and urea derivatives of 1,3-benzodiazapines as hiv reverse transcriptase inhibitors
03/27/2003WO2002060879A3 Bacterial gyrase inhibitors and uses thereof
03/27/2003WO2001092218A3 Polyamine analogues as therapeutic and diagnostic agents
03/27/2003US20030060638 C7 carbamate substituted taxanes
03/27/2003US20030060626 Fungicides
03/27/2003US20030060474 A piperazine compound as antithrombotic agent
03/27/2003US20030060473 Piperazine compounds as inhibitors of MMP or TNF
03/27/2003US20030060461 Cyclic diamine compound with condensed-ring groups
03/27/2003US20030060453 Such as 4-((4-fluorophenyl)hydrazono)-4H-pyrazole- 3,5-diamine for antiproliferative activity, and promoting apoptosis in cells lacking normal regulation of cell cycle and death
03/27/2003US20030060452 N-heterocyclic derivatives as NOS inhibitors
03/27/2003DE10207217C1 Production of 1,2-dichloroethane, used as intermediate for vinyl chloride, involves dissolving chlorine in circulating liquid medium containing catalyst and removing undissolved gas before contact with ethylene solution
03/27/2003CA2465978A1 Inhibitors of histone deacetylase
03/27/2003CA2461074A1 Methods and compositions of novel triazine compounds
03/27/2003CA2460942A1 Substituted pyrazolyl compounds for the treatment of inflammation
03/27/2003CA2460149A1 2-phenyl-3-heteroarylpropionic acid derivative or salt thereof and medicine containing the same