Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
07/2001
07/17/2001US6262272 Reacting furan carboxylic acid derivative with acid chloride or acid anhydride in inert solvent containing acid receptor; adding aromatic amine compound to form pyrrole carboxamide compound
07/17/2001US6262089 Using these compounds to treat diseases associated with amyloidosis, such as alzheimer's disease, maturity onset diabetes mellitus, familial amyloid polyneuropathy, scrapie, and kreuzfeld-jacob disease.
07/17/2001US6262088 Polyhydroxylated monocyclic N-heterocyclic derivatives as anti-coagulants
07/17/2001US6262084 Compounds that inhibit the binding of integrins to their receptors
07/17/2001US6262082 Diaminopyridine-containing thiourea inhibitors of herpes viruses
07/17/2001US6262073 Pharmaceutical methods of use of 5-substituted and 5,5 disubstituted-3,4-dihydroxy-2(5H)-furanones
07/17/2001US6262069 1-amino-7-isoquinoline derivatives as serine protease inhibitors
07/17/2001US6262060 Treatment of hyperglycaemia, diabetes, obesity or inflammation
07/17/2001US6262052 Amino acid ester containing azole antifungals
07/12/2001WO2001049684A1 Novel tetrahydropyridines, preparation method and pharmaceutical compositions containing same
07/12/2001WO2001049681A1 A method for the preparation of substituted benzene derivatives
07/12/2001WO2001049678A1 Substituted phenyl-piperazine derivatives, their preparation and use
07/12/2001WO2001049677A1 Phenylpiperazinyl derivatives
07/12/2001WO2001049676A1 Substituted piperidines, medicaments containing these compounds, and methods for the production thereof
07/12/2001WO2001049674A2 Glycosidase inhibitors and preparation thereof
07/12/2001WO2001049673A2 Compounds and methods for modulation of estrogen receptors
07/12/2001WO2001049667A1 Method for preparing hydroxypicolinic acid derivatives
07/12/2001WO2001049666A1 Picolinic acid derivatives and their use as fungicides
07/12/2001WO2001049664A1 Trifluoromethylpyrrole carboxamides and trifluoromethylpyrrolethioamides as fungicides
07/12/2001WO2001044207A8 Novel branched substituted amino derivatives of 3-amino-1-phenyl-1h[1,2,4]triazol, methods for producing them and pharmaceutical compositions containing them
07/12/2001WO2001004113A3 Process for the preparation of paroxetine and synthetic intermeditates thereof
07/12/2001WO2001004093A3 Process for producing paroxetine derivatives by mitsunobu reaction
07/12/2001WO2001002391A3 Bicyclic aromatic compounds for treating drug addiction
07/12/2001WO2000005223A3 Heterocyclic derivatives and their use as integrin inhibitors
07/12/2001US20010007877 Novel anti-infectives
07/12/2001US20010007870 Compounds useful for inhibition of farnesyl protein transferase
07/12/2001DE19963868A1 Neue substituierte Piperidine, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung New substituted piperidines, pharmaceutical compositions containing them and methods for their preparation
07/12/2001DE19963174A1 Substituierte Pyrrol-Mannichbasen Substituted pyrrole Mannich bases
07/12/2001DE19962998A1 New integrin receptor ligands, especially integrin-alphavbeta3 ligands, useful for treating e.g. atherosclerosis, rheumatoid arthritis, restenosis, angioplasty and acute kidney failure
07/12/2001CA2396688A1 Glycosidase inhibitors and methods of synthesizing same
07/12/2001CA2396306A1 Method for preparing hydroxypicolinic acid derivatives
07/12/2001CA2396299A1 Picolinic acid derivatives and their use as fungicides
07/12/2001CA2396059A1 Compounds and methods for modulation of estrogen receptors
07/12/2001CA2395867A1 Phenylpiperazinyl derivatives
07/12/2001CA2395267A1 Trifluoromethylpyrrole carboxamides and trifluoromethylpyrrolethioamides as fungicides
07/11/2001EP1114821A1 Benzopyrans and their use as therapeutic agents
07/11/2001EP1114817A1 Substituted benzylamino piperidine compounds
07/11/2001EP1114522A1 Rf receiver having cascaded filters and an intermediate amplifier stage
07/11/2001EP1114040A1 PROCESS FOR OBTAINING HMG-CoA REDUCTASE INHIBITORS OF HIGH PURITY
07/11/2001EP1114030A1 Pyridine ketones useful as herbicides
07/11/2001EP1114028A1 Aza-bicycles which modulate the inhibition of cell adhesion
07/11/2001EP1114022A1 Process for producing stereoselective nitro compounds
07/11/2001EP0823896B1 Substituted oximes, hydrazones and olefins as neurokinin antagonists
07/11/2001EP0725779B1 Novel (r)-5-carbamoyl-8-fluoro-3-n,n-disubstituted-amino-3,4-dihydro-2h-1-benzopyranes
07/11/2001CN1303378A 3-(Amino-or aminoalkyl) pyridinone derivatives and their use for treatment of HIV related diseases
07/11/2001CN1303373A N-Aryloxyethylamine derivatives for treatment of depression
07/11/2001CN1303371A Indole derivatives
07/11/2001CN1302801A Substituted aminoquinazolone (thio-ketone) derivative or its salt, its intermediate and pest controlling agent and its application method
07/11/2001CN1302612A Preparation method of medicinal composition containing 1,3-oxathin cyclopentane nucleoside analogues
07/10/2001US6258948 An n-acylamino compound; antiinflammatory agents, autoimmune diseases
07/10/2001US6258843 4-oxy-3-(aryl)phenyl-arylcarbonyloxy compounds useful as phosphodiesterase inhibitors
07/10/2001US6258833 Enzyme inhibitors and antiinflammatory agents
07/10/2001US6258817 Substituted pyrazin-2-yl-sulphonamide (-3-pyridyl) compounds and uses thereof
07/10/2001US6258813 D4 receptor selectivity piperazine derivatives
07/10/2001US6258812 Phthalazines with angiogenesis inhibiting activity
07/10/2001US6258811 Methods for preventing, inhibiting or treating graft rejection reactions in graft-versus-host disease (GVHD) and organ transplantation
07/10/2001US6258800 Prodrugs of benzofuranylethyl carbamate NK1 antagonists
07/10/2001CA2175502C Cyclic amide derivatives
07/05/2001WO2001047921A1 Pyrimidine and triazine kinase inhibitors
07/05/2001WO2001047916A1 2-(1h-indol-3-yl)-2-oxo-acetamides with antitumor activity
07/05/2001WO2001047905A1 Pyrrolidine derivatives as cyclic amp-specific phosphodiesterase inhibitors
07/05/2001WO2001047897A1 Cytokine, especially tnf-alpha, inhibitors
07/05/2001WO2001047893A1 New azabicyclooctane derivatives useful in the treatment of cardiac arrhythmias
07/05/2001WO2001047891A1 Heterocyclic compounds having sulfonamide groups
07/05/2001WO2001047890A1 Quinoline and quinazoline derivatives and drugs containing the same
07/05/2001WO2001047889A1 Tricyclic compounds
07/05/2001WO2001047887A1 β-AMINO ACID COMPOUNDS AS INTEGRIN ANTAGONISTS
07/05/2001WO2001047886A1 Nitrile derivatives as cathepsin k inhibitors
07/05/2001WO2001047885A1 Substituted indole mannich bases
07/05/2001WO2001047883A1 Fused-ring compounds and use thereof as drugs
07/05/2001WO2001047878A1 Substituted pyrrole mannich bases to combat pain and allergic reactions
07/05/2001WO2001047875A1 Substituted aminoalkylamide derivatives as antagonists of follicle stimulating hormone
07/05/2001WO2001009094A3 Chemokine receptor antagonists and methods of use therefor
07/05/2001WO2001000584A3 Pyrazolyl derivatives of bicyclic benzoic acids for use as herbicides
07/05/2001WO2000055137A8 Compounds and methods for modulation of estrogen receptors
07/05/2001US20010006969 Pyrimidine nucleus-containing compound and a medicament containing the same for a blood oxygen partial pressure amelioration, and a method for preparing the same
07/05/2001US20010006944 Treating noninvasive fungus-induced rhinosinusitis by mucoadministering an antifungal agent; culturing noninvasive fungus from a mammalian mucus sample for antigen/antibody production; apparatus for collecting nasal mucus
07/05/2001DE19963178A1 Substituierte Indol-Mannichbasen Substituted indole Mannich bases
07/05/2001CA2396693A1 Cytokine, especially tnf-alpha, inhibitors
07/05/2001CA2396502A1 Substituted pyrrole mannich bases
07/05/2001CA2395834A1 Tricyclic compounds
07/05/2001CA2395716A1 Substituted aminoalkylamide derivatives as antagonists of follicle stimulating hormone
07/05/2001CA2395205A1 2-(1h-indol-3-yl)-2-oxo-acetamides with antitumor activity
07/05/2001CA2395179A1 Nitrile derivatives as cathepsin k inhibitors
07/05/2001CA2394727A1 Pyrimidine and triazine kinase inhibitors
07/05/2001CA2394097A1 New azabicyclooctane derivatives useful in the treatment of cardiac arrhythmias
07/05/2001CA2392866A1 Substituted indole mannich bases
07/05/2001CA2363274A1 Fused-ring compounds and use thereof as drugs for hepatitis c
07/04/2001EP1113014A1 Linear or cyclic ureas, a process for their preparation and pharmaceutical compositions containing them
07/04/2001EP1113007A1 Tetrahydroisoquinoline compounds as estrogen agonists/antagonists
07/04/2001EP1112284A1 Piperazine-4-phenyl derivatives as inhibitors of the interaction between mdm2 and p53
07/04/2001EP1112270A1 Dihydrobenzodioxine carboxamide and ketone derivatives as 5-ht4 receptor antagonists
07/04/2001EP1112269A2 Hiv protease inhibitors
07/04/2001EP1112268A1 Condensed heterocyclic compounds and herbicides containing them
07/04/2001EP1112261A1 2-ethyl-2,3-dihydrobenzofuran-carboxylic acid ester derivative, preparation method and use for preparing efaroxan derivatives
07/04/2001EP1112256A1 Cyclohexenonquinolinoyl-derivatives as herbicidal agents
07/04/2001EP1112252A1 Kappa agonist compounds and pharmaceutical formulations thereof
07/04/2001EP1112251A1 Azetidine derivatives, preparation and medicines containing them
07/04/2001EP0850236B1 Piperazino derivatives as neurokinin antagonists
07/04/2001CN1302297A Pyrimidin-aminomethyl-pyridine derivatives, their preparation and their use in control of helicobacter bacteria