Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
06/2001
06/05/2001US6242612 Multistage reaction of forming pyrazoles as kinase and cox-2 enzyme inhibitors
06/05/2001US6242601 Heterocyclic sulfamides
06/05/2001US6242596 Preparation of betamethyl carbapenem intermediates
06/05/2001US6242475 Pesticidal 1-polyarylpyrazoles
06/05/2001US6242458 Tricyclic amide and urea compounds useful for inhibition of G-protein function and for treatment of proliferative diseases
06/05/2001US6242450 Substituted piperidines
06/05/2001US6242439 Azetidinone derivatives for the treatment of HCMV infections
06/05/2001US6242422 (Substituted)Acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
06/05/2001CA2216291C Tricyclic compounds useful for inhibition of g-protein function and for treatment of proliferative diseases
06/03/2001CA2327385A1 Sulfamoylheteroaryl pyrazole compounds as anti-inflammatory/analgesic agents
06/03/2001CA2327256A1 Heteroaryl phenyl pyrazole compounds as anti-inflammatory/analgesic agents
05/2001
05/31/2001WO2001038332A1 Gamma-hydroxy-2-(fluoroalkylaminocarbonyl)-1-piperazinepentanamides as hiv protease inhibitors
05/31/2001WO2001038325A1 5-membered n-heterocyclic compounds with hypoglycemic and hypolipidemic activity
05/31/2001WO2001038324A2 Imidazole derivatives and their use as raf kinase inhibitors
05/31/2001WO2001037835A1 Novel compounds
05/31/2001WO2000005214A3 Isoquinolines as urokinase inhibitors
05/31/2001US20010002400 Administering an antifungal agent
05/31/2001DE19957156A1 New amino and fluoro substituted 1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocine derivatives useful in treatment of e.g. arrythmias, spasms, ischaemia, pain and neurodegenerative disorders
05/31/2001CA2395564A1 Novel compounds
05/31/2001CA2390923A1 5-membered n-heterocyclic compounds with hypoglycemic and hypolipidemic activity
05/30/2001EP1103549A1 Photoprotective cosmetic compositions containing aminoamidine derivatives and uses thereof
05/30/2001EP1103547A1 Formazan metal complex
05/30/2001EP1102764A1 Paroxetine salts
05/30/2001EP1102763A2 Fsh mimetics for the treatment of infertility
05/30/2001EP1102761A2 Cyclopentabenzofuran derivatives and their use
05/30/2001EP1102754A1 Imidazoles and related compounds as alpha-1a agonists
05/30/2001EP1102752A1 Succinoylamino lactams as inhibitors of a beta protein production
05/30/2001EP1102587A2 Vitronectin receptor antagonists
05/30/2001EP1102535A2 Compounds and methods
05/30/2001EP0861242B1 Heterocyclic fungicides
05/30/2001EP0750616B1 Acid addition salts of 2,3,4,5-tetrahydro-1h-3-benzazepine compounds
05/30/2001EP0665834B1 Quinolone and acridinone derivatives for the treatment of urinary incontinence
05/30/2001EP0656778B1 Enantiomerically pure beta-d-dioxolane-nucleosides
05/30/2001EP0641320B1 Substituted (s)-3-phenylpiperidine derivatives, their preparation and their use as dopamine autoreceptor antagonists
05/30/2001CN1297448A Paroxetine ascorbate
05/30/2001CN1297442A 5-aminoindeno [1,2-c] pyrazol-4-ones as anti-cancer and anti-proliferative agents
05/30/2001CN1297441A Heterocyclically substd. amides used as calpain inhibitors
05/30/2001CN1297436A Substd. pyrrolidine hydroxamate metalloprotease inhibitors
05/30/2001CN1066438C Preparation of beta-methyl carbapenem intermediates
05/29/2001US6239173 Antiinflammatory, antipyretic, analgesic, and antiarthritic agents
05/29/2001US6239151 Compounds as inhibitor of tumor necrosis factor alpha release
05/29/2001US6239147 To treat cns, gastrointestinal and other disorders. substance p antagonists having improved activity and fewer side effects, treatment of emesis induced by antineoplastic agents, isochroman ring
05/29/2001US6239143 5-HT7 receptor antagonists
05/29/2001US6239131 1,5 Benzodiazepine derivatives
05/29/2001US6239074 Substituted 3-phenyluracils
05/29/2001US6239071 2,4-diamino-1,3,5-triazines, processes for their preparation and their use as herbicides and plant growth regulators
05/29/2001CA2325783A1 Ultraviolet-protecting cosmetic compounds containing amino- amidine derivatives and uses
05/25/2001WO2001036408A1 Compounds with antibacterial and antiparasitic properties
05/25/2001WO2001036403A1 Urea derivatives as anti-inflammatory agents
05/25/2001WO2001036395A1 Triazoles as farnesyl transferase inhibitors
05/25/2001WO2000077027A3 Serine protease inhibitors
05/25/2001WO2000039081A3 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
05/23/2001EP1101761A2 Process for producing 3-phenyluracil compounds
05/23/2001EP1101759A1 Phenylazole compounds, process for producing the same and drugs for hyperlipemia
05/23/2001EP1101755A1 Anthranilic acid derivatives
05/23/2001EP1100805A1 Medicine nitrate salts
05/23/2001EP1100796A1 Process for the preparation of a non-crystalline anhydrate form of paroxetine hydrochloride
05/23/2001EP1100795A1 Disubstituted bicyclic heterocycles having, in particular, a thrombin inhibitive effect
05/23/2001EP1100792A1 Tricyclic sulfonamides and their derivatives as inhibitors of matrix metalloproteinases
05/23/2001EP1100786A1 Antiviral pyrimidinedione derivatives and process for the preparation thereof
05/23/2001EP1100782A1 Amino-aldehyde solid support, linker therefor and methods of preparation and use thereof
05/23/2001EP1100781A1 High affinity ligands for nociceptin receptor orl-1
05/23/2001EP1100506A1 Integrin receptor antagonists
05/23/2001EP1100501A1 Pyrrolidine and pyrroline derivatives having effects on serotonin related systems
05/23/2001EP0788497B1 Bisarylcarbinol derivatives as inhibitors of leukotriene biosynthesis
05/23/2001EP0680950B1 Propenone derivatives
05/23/2001EP0631578B1 Itraconazole and saperconazole stereoisomers
05/23/2001CN1296481A (4-arylsulfonylamino)-tetrahydropyran-4-carboxylic acid hydroxamides
05/23/2001CN1296478A Histamine H3 receptor ligands
05/23/2001CN1296010A Novel cyano-indole thrombotonin reuptaking inhibitor compound, its preparation process and medicinal compositions having the same
05/23/2001CN1066148C Tricyclic benzazepine compounds
05/23/2001CN1066141C 3-(hetero)aryl carboxylic acid derivatives, methods of preparing them and intermediates used in their preparation
05/22/2001US6235907 Intermediates useful in making mappicine and related compounds
05/22/2001US6235768 Osteoporosis; rheumatic disorders; antitumor agents
05/22/2001US6235758 Indole derivatives as 5-HT receptor antagonist
05/22/2001US6235756 Methods and compositions for inhibition of angiogenesis by thalidomide
05/22/2001US6235755 FSH mimetics for the treatment of infertility
05/22/2001US6235750 Nitric oxide synthase inhibitor
05/22/2001US6235747 6-phenyl-pyridin-2-ylamine derivatives
05/17/2001WO2001034632A2 Aliphatic hydroxy substituted piperidyl diaryl pyrrole derivatives as antiprotozoal agents
05/17/2001WO2001034591A2 Substituted 4h-chromene and analogs as activators of caspases and inducers of apoptosis and the use thereof
05/17/2001WO2001034577A1 5-aryl-1h-1,2,4-triazole compounds as inhibitors of cyclooxygenase-2 and pharmaceutical compositions containing them
05/17/2001WO2001034573A1 Compounds
05/17/2001WO2001034566A2 Protease inhibitors
05/17/2001WO2001034158A1 Protease inhibitors
05/17/2001WO2001034157A1 Protease inhibitors
05/17/2001WO2001034155A1 Protease inhibitors
05/17/2001WO2001034149A1 Diaryl piperidyl pyrrole derivatives as antiprotozoal agents
05/17/2001WO2001034146A1 Novel anti-infectives
05/17/2001WO2001024796A8 1,2,4-triazole derivatives, composition, process of making and methods of use
05/17/2001WO2001014358A3 Substituted (aminoiminomethyl or aminomethyl) dihydrobenzofurans and benozopyrans
05/17/2001WO2001007408A3 Novel method for preparing benzoperhydroisoindole compounds
05/16/2001EP1099701A1 7-[(4'-Trifluoromethyl-biphenyl-2-carbonyl)amino]-quinoline-3-carboxylic acid amides, and methods of inhibiting the secretion of apolipoprotein B
05/16/2001EP1099695A1 5-aryl-1H-1,2,4-triazole compounds as inhibitors of cyclooxygenase-2 and pharmaceutical compositions containing them
05/16/2001EP1099690A1 MONOCYCLIC $g(b)-LACTAM COMPOUNDS AND CHYMASE INHIBITORS CONTAINING THE SAME
05/16/2001EP1098893A1 Cyclic compounds useful in the treatment of dyslipidemia, atherosclerosis and diabetes, pharmaceutical compositions and preparation process
05/16/2001EP1098890A1 Dihydrotriazolone derivatives as pesticides
05/16/2001EP1098888A1 Piperazinone derivatives and their uses
05/16/2001EP1098886A1 Phthalazine derivatives as phosphodiesterase 4 inhibitors
05/16/2001EP1098885A1 Imidazole compounds and their use as adenosine deaminase inhibitors