Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397) |
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01/19/2010 | CA2472115C Colorant compounds |
01/19/2010 | CA2402751C Decahydro-isoquinolines |
01/19/2010 | CA2368097C Amide derivatives of 3,4-dihydroquinazolinone compounds useful as cytokine inhibitors |
01/19/2010 | CA2239904C Inhibitors of interleukin-1.beta. converting enzyme |
01/14/2010 | WO2010006191A1 4-phenoxymethylpiperidines as modulators of gpr119 activity |
01/14/2010 | WO2010005783A1 Pyrrolidinyl and piperidinyl compounds useful as nhe-1 inhibitors |
01/14/2010 | WO2010004782A1 Prolineamide derivative, salt thereof with acid, organic catalyst consisting of the same and method of producing β-hydroxycarbonyl compound using the organic catalyst |
01/14/2010 | WO2010004215A2 Substituted 1-benzyl-cinnolin-4(1h)-one derivatives, preparation thereof, and therapeutic use thereof |
01/14/2010 | WO2010003624A2 Heterocyclic compounds, processes for their preparation, medicaments comprising these compounds, and the use thereof |
01/14/2010 | WO2009132453A8 Cyclylamine derivatives as calcium channel blockers |
01/14/2010 | US20100010241 Cosmetics |
01/14/2010 | US20100010042 Arylvinylazacycloalkane compounds and methods of preparation and use thereof |
01/14/2010 | US20100010023 Quinazoline derivatives and pharmaceutical compositions containing them |
01/14/2010 | US20100010007 Piperidine derivatives as modulators of chemokine receptor ccr5 |
01/14/2010 | US20100010004 Inhibitors of histone deacetylase |
01/14/2010 | US20100010003 Pyrimidine Derivatives And Their Use As Pesticides |
01/14/2010 | US20100009988 Piperazinyl-, piperidinyl- and morpholinyl-derivatives as novel inhibitors of histone deacetylase |
01/14/2010 | US20100009973 Integrase Inhibitors 3 |
01/14/2010 | US20100009972 Pyridyl Non-Aromatic Nitrogen-Containing Heterocyclic-1-Carboxylate Compound |
01/14/2010 | US20100009971 Pyridyl Non-Aromatic Nitrogen-Containing Heterocyclic-1-Carboxylate Compound |
01/14/2010 | CA2730511A1 4-phenoxymethylpiperidines as modulators of gpr119 activity |
01/14/2010 | CA2730280A1 5-quinolinone and imidazopyridine compounds and use thereof |
01/14/2010 | CA2730116A1 Pyrrolidinyl and piperidinyl compounds useful as nhe-1 inhibitors |
01/14/2010 | CA2729896A1 Substituted 1-benzyl-cinnolin-4(1h)-one derivatives, preparation thereof, and therapeutic use thereof |
01/13/2010 | EP2143714A1 Tetrahydroisoquinoline compound |
01/13/2010 | EP2143713A1 Novel pyrrolinone derivative and medicinal composition containing the same |
01/13/2010 | EP2142538A1 Derivatives and analogs of chroman as functionally selective alpha2c adrenoreceptor agonists |
01/13/2010 | EP2142528A1 1-(1-benzylpiperidin-4-yl)benzimidaz0le -5-carboxylic acid derivatives for the treatment of diabetes mellitus |
01/13/2010 | EP2142524A1 Novel 5-cyano-prostacyclin derivatives and their use as agents for the treatment of influenza a viral infection |
01/13/2010 | EP2142515A1 Novel inhibitors |
01/13/2010 | EP2142514A1 Thiourea derivatives as glutaminyl cyclase inhibitors |
01/13/2010 | EP2142513A1 Nitrovinyl-diamine derivatives as glutaminyl cyclase inhibitors |
01/13/2010 | EP2142509A2 Quinolones and azaquinolones that inhibit prolyl hydroxylase |
01/13/2010 | EP2142503A2 Process for the manufacture for non-steroidal anti-inflammatory agents and intermediates thereof |
01/13/2010 | EP1451160B1 Pyrazole-amides for use in the treatment of pain |
01/13/2010 | EP1144388B1 Acyl derivatives which treat vla-4 related disorders |
01/13/2010 | CN101627032A Process for the preparation of (r) -5- (2-aminoethyl) -1- (6, 8-difluorochroman-3-yl) -1, 3-dihydroimidazole-2-thione |
01/13/2010 | CN100579976C P38 inhibitors and methods of use thereof |
01/12/2010 | US7645891 E.g., 4-(2-methyl-3-oxo-hept-6-en-2-yl)-2,2-dimethyl-[1,3]-dioxane chemical intermediate; chemical/metabolic stabilization of microtubuli; antitumor, -carcinogenic agents; malignant melanoma, acute lymphocytic/myelocytic leukemia; angiogenesis inhibitors; antiinflammatory/-arthritic agents; psoriasis |
01/12/2010 | US7645878 Reacting an aniline derivative with an acylchloride to form an intermeidate, cyclizing the intermediate, replacing hydroxy group with a leaving group (chloride), racting the product with an amino-heterocyclic compound |
01/12/2010 | US7645789 Modulators of ATP-Binding Cassette transporters; Cystic Fibrosis Transmembrane Conductance Regulator; N-(5-hydroxy-2,4-ditert-butyl-phenyl)-4-oxo-1H-quinoline-3-carboxamide |
01/12/2010 | US7645784 Benzimidazole derivatives |
01/12/2010 | US7645774 Sulfonamide-containing benzene derivatives; cancer and inflammatory, immunomodulatory or respiratory diseases; allergy, seasonal allergic rhinitis, reversible airway obstruction, adult respiratory distress syndrome, asthma, or bronchitis |
01/12/2010 | US7645770 Phenylalanine enamide derivatives |
01/12/2010 | US7645761 Indoline derivatives |
01/12/2010 | US7645759 (4-(S)-amino-5-(4-{4-[2,4-dichloro-3-(2,4-dimethyl-quinolin8yloxy-methyl) benzenesulfonylamino] tetrahydropyran-4carbonyl}-piperazin-1-yl)-5-oxo-pentyl] trimethyl-ammonium chloride, dihydrochloride; asthma or chronic bronchitis |
01/12/2010 | US7645757 Derivatives of heteroaryl-alkylcarbamates, methods for their preparation and use thereof as fatty acid amido hydrolase enzyme inhibitors |
01/12/2010 | CA2560489C Pyranone compounds useful to treat retroviral infections |
01/12/2010 | CA2511242C Inhibitors of human tumor-expressed ccxckr2 |
01/12/2010 | CA2411418C Hydroxyformamidine derivatives and medicines containing the same |
01/12/2010 | CA2407463C N-substituted peptidyl nitriles as cysteine cathepsin inhibitors |
01/12/2010 | CA2399062C Stereoselective synthesis of nucleoside analogues |
01/12/2010 | CA2391643C Gamma-hydroxy-2-(fluoroalkylaminocarbonyl)-1-piperazinepentanamides as hiv protease inhibitors |
01/12/2010 | CA2384018C Muscarinic antagonists |
01/12/2010 | CA2306428C 3-oxo-2(h)-1,2,4 - triazine derivatives as ligands of 5ht1a receptors |
01/07/2010 | WO2010003048A1 Benzimidazoles and related analogs as sirtuin modulators |
01/07/2010 | WO2010003025A1 Bicyclic heterocycles as mek kinase inhibitors |
01/07/2010 | WO2010002483A1 Optionally condensed dihydro pyridine, dihydropyrimidine and dihydro pyrane derivatives acting as late sodium channel blockers |
01/07/2010 | WO2010002075A1 Methods for preparing amide derivatives |
01/07/2010 | WO2010001946A1 Triazole derivative or salt thereof |
01/07/2010 | WO2010000773A1 5-heterocyclylalkyl-3-hydroxy-2-phenylcyclopent-2-enones as herbicides |
01/07/2010 | WO2010000668A1 A crystalline form of posaconazole |
01/07/2010 | WO2009108525A3 Hexahydrocyclopentyl[f]indazole carboxamides and derivatives thereof as selective glucocorticoid receptor modulators |
01/07/2010 | US20100004456 Oxepin derivative |
01/07/2010 | US20100004444 Novel Triazolo pyrimidine compounds |
01/07/2010 | US20100004438 Diarylether derivatives as antitumor agents |
01/07/2010 | US20100004290 Insecticidal n-substituted (heteroaryl)cycloalkyl sulfoximines |
01/07/2010 | US20100004233 Novel coumarin derivative having antitumor activity |
01/07/2010 | US20100004208 Substituted benzofurans, benzothiophenes, benzoselenophenes and indoles and their use as tubulin polymerisation inhibitors |
01/07/2010 | US20100003216 HCV NS-3 Serine Protease Inhibitors |
01/07/2010 | CA2729745A1 Oxindole compounds |
01/07/2010 | CA2729724A1 5-heterocyclylalkyl-3-hydroxy-2-phenylcyclopent-2-enones as herbicides |
01/07/2010 | CA2729408A1 Triazole derivative or salt thereof |
01/07/2010 | CA2729128A1 Benzimidazoles and related analogs as sirtuin modulators |
01/07/2010 | CA2728170A1 A crystalline form of posaconazole |
01/07/2010 | CA2727250A1 Bicyclic heterocycles as mek kinase inhibitors |
01/07/2010 | CA2726999A1 New drugs for inhibiting aggregation of proteins involved in diseases linked to protein aggregation and/or neurodegenerative diseases |
01/06/2010 | EP2141160A1 Ground crystal of olmesartan medoxomil |
01/06/2010 | EP2141159A1 A Crystalline form of posaconazole |
01/06/2010 | EP2140868A1 Use of a cholinesterase inhibitor for the treatment of dementia and cognitive impairments associated with or caused by chemotherapy |
01/06/2010 | EP2140864A2 Use of GAL3 receptor antagonists for the treatment of depression and / or anxiety and compounds useful in such methods |
01/06/2010 | EP2140862A2 Use of GAL 3 receptor antagonists for the treatment of depression and /or anxiety and compounds useful in such methods |
01/06/2010 | EP2139885A1 Co-crystals of propiconazole |
01/06/2010 | EP2139857A1 Sub-type selective azabicycloalkane derivatives |
01/06/2010 | EP1735278B1 Histamine h3 receptor agents, preparation and therapeutic uses |
01/06/2010 | EP1562911B1 Compositions useful as inhibitors of jak and other protein kinases |
01/06/2010 | EP1489078B1 Benzofuran derivative |
01/06/2010 | EP0934281B1 1-phenyl-benzimidazole compounds and their use as baga- a? receptor modulators |
01/06/2010 | CN101622248A N3-heteroaryl substituted triazoles and N5-heteroaryl substituted triazoles useful as AXL inhibitors |
01/06/2010 | CN101619059A Method for preparing osemozotan hydrochloride |
01/06/2010 | CN101619057A N-substituted piperidine derivatives as serotonin receptor agents |
01/06/2010 | CN100577658C 喹唑啉衍生物 Quinazoline derivatives |
01/06/2010 | CN100577643C Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists |
01/06/2010 | CN100577163C Compounds effecting glucokinase |
01/05/2010 | US7642378 Lipid lowering biphenylcarboxamides |
01/05/2010 | US7642359 Pyrazolyl-substituted heterocycles and their use as phytosanitary products |
01/05/2010 | US7642354 Polycyclic pyrazines as potassium ion channel modulators |
01/05/2010 | US7642351 2,4-Pyrimidinediamine compounds and their uses |
01/05/2010 | US7642277 Non-nucleoside reverse transcriptase inhibitors |
01/05/2010 | US7642276 N-[4-methyl-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)phenyl]-2-pyrrolidin-1-ylisonicotinamide; rheumatoid arthritis |