Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
03/2010
03/04/2010WO2010022412A1 Octahydroquinolizines for antidiabetic treatment
03/04/2010WO2010004215A3 Substituted 1-benzyl-cinnolin-4(1h)-one derivatives, preparation thereof, and therapeutic use thereof
03/04/2010WO2009106471A3 Angiotensin ii receptor blocker derivatives
03/04/2010US20100056796 Compounds Suitable As Precursors to Compounds that are Useful for Imaging Amyloid Deposits
03/04/2010US20100056779 Synthesis of methyl nonactate derivatives
03/04/2010US20100056602 Substituted Pyrrole Derivatives And Their Use As HMG-CO Inhibitors
03/04/2010US20100056582 Modulators of LXR
03/04/2010US20100056571 Novel pyrazole compounds as transforming growth factor (tgf) inhibitors
03/04/2010US20100056528 Sulfonamide derivatives with therapeutic indications
03/04/2010US20100056512 Pyrimidine compounds
03/04/2010US20100056506 Substituted 2-amino-fused heterocyclic compounds
03/04/2010CA2735730A1 2,4-diaminopyrimidine compound
03/04/2010CA2735497A1 New compounds suitable as precursors to compounds that are useful for imaging amyloid deposits
03/04/2010CA2734981A1 Oxotetrahydrofuran-2-yl-benzimidazole derivative
03/04/2010CA2734551A1 Pyridine derivatives as vegfr-2 receptor and protein tyrosine kinase inhibitors
03/04/2010CA2733648A1 Novel pyrrole derivative having, as substituents, ureide group, aminocarbonyl group and bicyclic group which may have substituent
03/03/2010EP2159223A2 6 -acyloxy- 7-meth0xy- 2, 2 -dimethylchromane compounds and their use as pigmentation-regulators
03/03/2010EP2081572B1 Benzimidazole cannabinoid agonists bearing a substituted heterocyclic group
03/03/2010EP2016064B1 Methods for the preparation of pyrazole-containing compounds
03/03/2010EP1753719B1 Substituted pyrrolidine-2-ones
03/03/2010EP1749001B1 3-piperidinylisochroman-5-ols as dopamine agonists
03/03/2010EP1107964B1 Isoquinoline derivatives with angiogenesis inhibiting activity
03/03/2010CN101663296A Twelve-membered cyclomacrolactam derivative
03/03/2010CN101659659A Pyridine derivative and medical application thereof
03/02/2010US7671221 Modulators of ATP-Binding Cassette transporters
03/02/2010US7671088 Water-soluble etoposide analogs and methods of use thereof
03/02/2010US7671076 N-(4-piperidin-1-yl-phenyl)-2-[5-(thiaxolidine-3-carbonyl)-pyrrolidin-3-ylidene]-acetamide;antidiabetic agents; hyperglycemia, syndrome X, hyperinsulinemia, obesity, atherosclerosis
03/02/2010US7671072 benzyl-carbamic acid cis-3-[5-(cyclohexanecarbonyl-amino)-1H-pyrazol-3-yl]-cyclobutyl ester; glycogen synthase kinase-3 (GSK-3) inhibitors; inter alia, Alzheimer's Disease, cancer, dementia, depression, diabetes, hair loss, schizophrenia, and stroke
03/02/2010US7671063 2,4 Di (hetero) -arylamino-pyrimidine derivatives as ZAP-70 and/or syk inhibitors
03/02/2010US7671056 5-fluoro-8-(4-(4-(6-methoxyquinolin-8-yl)piperazin-1-yl)piperidin-1-yl)quinoline; central nervous system disorders, such as cognition disorders, anxiety disorders, depression and sexual dysfunction
03/02/2010US7671053 such as 2-chloro-N-(1-hydroxy-cycloheptylmethyl)-5-[4-(2-hydroxy-3-methoxy-propyl)-3,5-dioxo-4,5-dihydro-3H-[1,2,4]triazin-2-yl]-benzamide for treatment of asthma and COPD; purinergic receptors (P2X7)
03/02/2010US7671049 1-{3-[(6-amino-5-nitropyridin-2-yl)amino]propyl}-4-(2,4-dichlorophenyl)-N-[(1S)-2-hydroxy-1-methylethyl]-1H-pyrrole-3-carboxamide; Antidiabetic, hypotensive, antiischemic, anticarcinogenic agents; Alzheimer*s disease, obesity, polycystic ovary syndrome; brain, neurodegenerative and autoimmune diseases
03/02/2010US7671032 19-(7-Methoxy-2-phenyl-quinolin-4-yloxy)-2, 16-dioxo-3,15,17-triaza-tricyclo[15.3.0.0*4,6*]icos-7-ene-4,14-dicarboxylic acid 4-ethyl ester 14-methyl ester, for example; inhibits the NS3 protease of flavivirus such as hepatitis C virus (HCV)
03/02/2010CA2445207C Process for the preparation of 2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]chroman
02/2010
02/25/2010WO2010022125A1 Ethynyl-substituted pyridine and pyrimidine derivatives and their use in treating viral infections
02/25/2010WO2010022121A1 Substituted pyridine and pyrimidine derivatives and their use in treating viral infections
02/25/2010WO2010021878A1 Cold menthol receptor antagonists
02/25/2010WO2010020548A1 Glyt1 receptor antagonists
02/25/2010WO2009091433A3 Spiro and dispiro 1,2,4-trioxolane antimalarials
02/25/2010US20100048893 Substituted arylalkanoic acid derivatives and use thereof
02/25/2010US20100048636 Aspartic Protease Inhibitors
02/25/2010US20100048618 Derivatives of 8-epiblechnic Acid and their Effects on Down-Regulation of Endothelin (ETA) receptor mRNA
02/25/2010US20100048600 such as trans-2-[3'-oxospiro [cyclohexane- 1,1'(3'H)-isobenzofuran]-4yl]-5-(2-pyridyl) imidazo[4,5-b]pyridine, exhibiting neuropeptide Y antagonistic effects, used for the treatment of cardiovascular, nervous system, metabolic, gastrointestinal, sexual and respiratory system disorders; pharmacokinetics
02/25/2010US20100048590 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
02/25/2010US20100048588 Aminocarbonyl-derivatives as novel inhibitors of histone deacetylase
02/25/2010US20100048585 Quinoline derivatives as antibacterial agents
02/25/2010US20100048565 Benzimidazole derivatives
02/25/2010US20100048539 Compounds and compositions as protein kinase inhibitors
02/25/2010US20100048531 GlyT1 RECEPTOR ANTAGONISTS
02/25/2010US20100048529 New 2-Azetidinone Derivatives Useful In The Treatment Of Hyperlipidaemic Conditions
02/25/2010US20100048500 Anti-viral nucleoside analogs and methods for treating viral infections, especially HIV infections
02/25/2010CA2734487A1 Ethynyl-substituted pyridine and pyrimidine derivatives and their use in treating viral infections
02/25/2010CA2734486A1 Substituted pyridine and pyrimidine derivatives and their use in treating viral infections
02/24/2010EP2157084A1 5-phenyl-3-pyridazinone derivative
02/24/2010EP2157081A1 Indolinones substituted in six locations, their manufacture and their application as medicine
02/24/2010EP2155732A1 Amorphous olmesartan medoxomil
02/24/2010EP2155731A1 1, 3-dihydroimidazole- 2 -thione derivatives as inhibitors of dopamine-beta-hydroxylase
02/24/2010EP2155717A1 2-[4-(pyrazol-4-ylalkyl)piperazin-1-yl]-3-phenyl pyrazines and pyridines and 3-[4-(pyrazol-4-ylalkyl)piperazin-1-yl]-2-phenyl pyridines as 5-ht7 receptor antagonists
02/24/2010EP2155716A2 Substituted heterocyclic derivatives and compositions and their pharmaceutical use as antibacterials
02/24/2010EP2155714A2 Substituted aromatic heterocyclic compounds as fungicides
02/24/2010EP2155693A1 Novel 4-phenyl-imidazole-2-thiones used as tyrosinase inhibitors, method for preparing same and use thereof in human medicine and cosmetology
02/24/2010EP2155666A1 Azetidine derivatives and their use as prostaglandin e2 antagonists
02/24/2010EP2154966A1 Benzimidazoles and pharmaceutical compositions thereof
02/24/2010EP2001873B1 Active ingredient combinations with insecticidal properties
02/24/2010EP1981880B1 Use of 4-imidazole derivatives for cns disorders
02/24/2010EP1848705B1 Exo- and diastereo- selective syntheses of himbacine analogs
02/24/2010EP1748995B1 Arylsulfonyl benzodioxanes useful for modulation the 5-ht6 receptor, the 5-ht2areceptor or both
02/24/2010EP1742935B1 Polycyclic pyrazines as potassium ion channel modulators
02/24/2010EP1729775B1 Process and intermediate compounds useful in the preparation of statins, particularly rosuvastatin
02/24/2010EP1682539B1 Process for preparing thiazolidinediones
02/24/2010EP1625121B1 Pyrimidine derivatives for the treatment of abnormal cell growth
02/24/2010EP1585728B1 Imino acid derivatives for use as inhibitors of matrix metalloproteinases
02/24/2010EP1465631B1 Pyrimidine a2b selective antagonist compounds, their synthesis and use
02/24/2010CN101657444A Derivatives and analogs of chroman as functionally selective alpha2C adrenoreceptor agonists
02/24/2010CN101657443A [1,2,3] triazolyl substituted quinolines and coumarins as inhibitors of leukotriene biosynthesis
02/24/2010CN101654453A Process for the manufacture of the calcium salt of rosuvatatin and crystalline intermediates thereof
02/24/2010CN100591676C 2- and 2,5-substituted phenylketo-enols
02/23/2010USRE41149 Optically active pyridonecarboxylic acid derivatives
02/23/2010US7667053 Cannabinoid-1 (CB1) receptor antagonists and/or inverse agonists; e.g. N-(2,3-bis(4-chlorophenyl)-1-methylpropyl)-1,4-benzodioxane-2-carboxamide; psychological disorders, eating disorders
02/23/2010US7667052 Bioactive substance
02/23/2010US7667041 Cinnamide compound
02/23/2010US7666904 3-aryl-4-hydroxyfuranone compounds and the human and animal health use thereof
02/23/2010US7666892 N-{[(4S)-2,5-dioxoimidazolidinyl]methyl}-4-(4-fluorophenoxy)benzenesulfonamide and N-{[(4S)-2,5-dioxoimidazolidinyl]methyl}[1,1'-biphenyl]-4-sulfonamide; chemical intermediates for enzyme inhibitors; especially as inhibitors of MMP12
02/23/2010US7666869 Nitrogen-containing 5-membered ring compound
02/23/2010US7666863 Benzofuran compounds, compositions and methods for treatment and prophylaxis of hepatitis C viral infections and associated diseases
02/23/2010CA2462289C Heteroaryl substituted tetrazole modulators of metabotropic glutamate receptor-5
02/23/2010CA2433021C Isoindole-imide compounds, compositions, and uses thereof
02/23/2010CA2374905C Pyrrolidinyl, piperidinyl or homopiperidinyl-substituted benzopyran derivatives for treating impaired fundic relaxation
02/23/2010CA2345146C Cyanophenyl derivative
02/18/2010WO2010019930A1 Urea derivatives as inhibitors of map kinases
02/18/2010WO2010018874A1 Amide compound
02/18/2010WO2010018777A1 Odor-controlling method
02/18/2010WO2010018231A2 Salt of, and processes for the preparation of, 1-isopropyl-4-{[4-(tetrahydro-2h-pyran- 4-yloxy)phenyl]carbonyl}hexahydro-1h-1,4-diazepine
02/18/2010WO2010017827A1 6-substituted 1-sulfonyl-2, 3-dihydro-indole derivatives for the treatment of proliferative diseases
02/18/2010WO2009084773A3 Preparation process useful in synthesis of atorvastatin
02/18/2010US20100041708 N-phenylarylsulfonamide compound, pharmaceutical composition comprising the compound as active ingredient, synthetic intermediate for the compound and process for it's preparation
02/18/2010US20100041656 Novel amide derivatives and medicinal use thereof
02/18/2010US20100041654 Pyrimidine Derivatives And Their Use As CB2 Modulators
02/18/2010US20100041652 Tyrosine kinase inhibitors
02/18/2010US20100041649 viricides used for for treating a human papillomavirus (HPV) viral infections, for inhibiting HPV DNA replication or for preventing prenatal transmission of HPV from mother to baby by administering to the mother prior to giving birth