Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
03/2010
03/18/2010CA2736970A1 Pyrimidinone derivatives for use as medicaments
03/18/2010CA2736530A1 Piperazine derivatives for binding and imaging amyloid plaques and their use
03/18/2010CA2736039A1 Novel prostaglandin i2 derivative
03/18/2010CA2735184A1 Heteroaryls amide derivatives and their use as glucokinase activators
03/18/2010CA2734454A1 A process for preparing [1s-[1-alpha,2-alpha,3-beta(1s*, 2r*)5-beta]]-3-[7-[2-(3,4-difluorophenyl)-cyclopropylamino]-5-(propylthio)-3h-1,2,3-triazolo [4,5-d]pyrimidin-3-yl]-5-(2-hydroxyethoxy)cyclopentane-1,2-diol and to its intermediates
03/17/2010EP2163553A1 Arene connected polyamine macroring derivatives, preparation methods and pharmaceutical uses thereof
03/17/2010EP2163543A1 Nitrogen-containing heterocyclic derivative having 11 beta-hydroxysteroid dehydrogenase type i inhibitory activity
03/17/2010EP2163541A1 Piperazine derivatives for binding and imaging amyloid plaques and their use
03/17/2010EP2162453A1 Crystalline form b of olmesartan medoxomil
03/17/2010EP2162450A1 ((bicylicheteroaryl) imidazolyl) methylheteroaryl compounds as adrenergic receptor agonists
03/17/2010EP2162442A1 Dual-acting benzoimidazole antihypertensive agents
03/17/2010EP2162436A1 Novel case of renin inhibitors
03/17/2010EP2162433A2 4' substituted compounds having 5-ht6 receptor affinity
03/17/2010EP1713822B1 Hcv ns-3 serine protease inhibitors
03/17/2010EP1689742B1 Quinolonecarboxylic acid compounds having 5-ht4 receptor agonistic activity
03/17/2010EP1620411B1 Inhibitors of akt activity
03/17/2010EP1513814B1 Novel piperidine compound
03/17/2010EP1284966B1 Process for the synthesis of amine ethers from secondary amino oxides
03/17/2010CN101675042A Novel 2-heteroaryl substituted benzothiophenes and benzofuranes 709
03/17/2010CN101675036A dual-acting benzoimidazole antihypertensive agents
03/17/2010CN101671335A Cytotoxins, prodrugs, linkers and stabilizers useful therefor
03/17/2010CN101671310A Compounds and compositions useful as cathepsin s inhibitors
03/17/2010CN101671307A 杂环天冬氨酰蛋白酶抑制剂 Heterocyclic aspartyl protease inhibitors
03/16/2010US7678904 or to treat autoimmune and inflammatory disorders; improved water solubility characteristics
03/16/2010US7678813 8a-Benzyl-2-(4-methoxyphenyl)-1,3,4,7,8,8a-hexahydro-2H-isoquinolin-6-one; psychotic major depression, schizoaffective disorder, Alzheimer's Disease and cocaine addiction
03/16/2010US7678812 Aminotetralin-derived urea modulators of vanilloid VR1 receptor
03/16/2010US7678804 Pyrimidine derivatives for treatment of hyperproliferative disorders
03/16/2010US7678802 Voltage gated sodium and calcium channel inhibitors
03/16/2010US7678798 5-({4-[(3S)-4-(5-bromo-2,3-dihydro-1H-inden-1-yl)-3-methylpiperazin-1-yl]-4-methylpiperidin-1-yl}carbonyl)-4,6-dimethylpyrimidine; inflammatory diseases, immune diseases and viral infections; HIV
03/16/2010US7678790 sulfonylurea derivatives, sulfonylthiourea derivatives, sulfonylguanidine derivatives, sulfonylcyanoguanidine derivatives, thioacylsulfonamide derivatives, and acylsulfonamide derivatives; effective for prevention and treatment of cardiovascular diseases, antithrombotic agents
03/16/2010CA2493966C Benzopyran derivatives substituted with secondary amines including imidazole, their preparation and pharmaceutical compositions containing them
03/16/2010CA2386980C Benzodiazepine derivatives for use in acute or chronic neurological disorders
03/11/2010WO2010027848A2 Forms of lapatinib compounds and processes for the preparation thereof
03/11/2010WO2010026771A1 Nitrogenated heterocyclic compound and salt thereof, and bactericidal agent for agricultural or horticultural applications
03/11/2010WO2010026388A1 Isatin derivatives for use as in vivo imaging agents
03/11/2010WO2010026255A1 Process for preparing olmesartan medoxomil intermediate
03/11/2010WO2010026212A1 Novel inhibitors
03/11/2010WO2010026096A1 7-(piperazine-1-ymethyl)-1h-indole-2-carboxylic acid (phenyl)-amide derivatives and allied compounds as p38 map kinase inhibitors for the treatment of respiratory diseases
03/11/2010WO2010026095A1 Novel benzamides, production thereof, and use thereof as medicaments
03/11/2010WO2010025850A1 Heterocyclically substituted anilinopyrimidines as fungicides
03/11/2010WO2010025831A1 Heterocyclically substituted anilinopyrimidines as fungicides
03/11/2010WO2010006755A3 Cyclic polyamines for binding phosphatidylserine
03/11/2010WO2009156099A8 6-substituted isoquinolines and isoquinolinones
03/11/2010WO2008094909A3 Quinazolinone and fused pyrimidinone compounds and their use in treating sodium channel-mediated diseases or conditions
03/11/2010US20100063129 4-Diallylaminomethylene-6-hydroxy-1- alpha -methoxymethyl-10 beta ,13 beta -dimethyl-3,7,17-trioxo-1,3,4,7,10,11 beta ,12,13,14 alpha ,15,16,17-dodecahydro-2-oxa-cyclopenta[ alpha ] phenanthren-11-ol or its acetate in a carrier; PI-3 kinase inhibitor; treating color cancer
03/11/2010US20100063119 Substituted carbinol compound
03/11/2010US20100063105 Pharmaceutical uses and synthesis of nicotinanilide-n-oxides
03/11/2010US20100063100 Modulators of aldehyde dehydrogenase activity and methods of use thereof
03/11/2010US20100063087 5-Amino-4-Hydroxy-7-(Imidazo [1,2-A] Pyridin-6-Ylmethyl)-8-Methyl-Nonamide Derivatives and Related Compounds as Renin Inhibitors for the Treatment of Hypertension
03/11/2010US20100063079 Pyrimidyl Sulphone Amide Derivatives as Chemokine Receptor Modulators
03/11/2010US20100063075 Aryl-quinazoline/aryl-2amino-phenyl methanone derivatives
03/11/2010US20100063062 Novel use of 1-[4-(5-cyanoindol-3-yl)butyl]-4-(2-carbamoyl-benzofuran-5-yl)-piperazine and its physiologically acceptable salts
03/11/2010US20100063056 Bipyridine carboxamide orexin receptor antagonists
03/11/2010US20100063040 Sulfonamide Derivative Having PGD2 Receptor Antagonistic Activity
03/11/2010US20100062996 Dioxolane derivates for the treatment of cancer
03/11/2010US20100062972 Triazole compounds and uses related thereto
03/11/2010US20100062942 Pyrazolyl-substituted heterocycles and their use as phytosanitary products
03/11/2010US20100062937 Benzanilides with insecticidal activity
03/11/2010US20100062065 Pharmaceutical composition containing naphthoquinone-based compound for intestine delivery system
03/11/2010US20100061982 3-substituted-1h-indole, 3-substituted-1h-pyrrolo[2,3-b]pyridine and 3-substituted-1h-pyrrolo[3,2-b]pyridine compounds, their use as mtor kinase and pi3 kinase inhibitors, and their syntheses
03/11/2010CA2735970A1 Isatin derivatives for use as in vivo imaging agents
03/11/2010CA2735795A1 Novel inhibitors
03/11/2010CA2735770A1 7-(piperazine-1-ymethyl)-1h-indole-2-carboxylic acid (phenyl)-amide derivatives and allied compounds as p38 map kinase inhibitors for the treatment of respiratory diseases
03/11/2010CA2735208A1 Novel benzamides, production thereof, and use thereof as medicaments
03/11/2010CA2733533A1 Hedgehog pathway modulators
03/10/2010EP2161266A1 Benzofuran derivatives as orexin receptor antagonists
03/10/2010EP2160387A2 Heteroarylamide pyrimidone compounds
03/10/2010EP2160380A1 Cyano-guanidine derivatives as glutaminyl cyclase inhibitors
03/10/2010EP1896456B1 Novel tetracyclic tetrahydrofuran derivatives containing a cyclic amine side chain
03/10/2010EP1841737B1 N-(heteroaryl)-1h-indole-2-carboxamide derivatives and their use as vanilloid trpv1 receptor ligands
03/10/2010EP1786801B1 2-arylcarbamoyl-indoles as cytokine inhibitors
03/10/2010EP1780209B1 Oxime ester compound and photopolymerization initiator containing such compound
03/10/2010EP1751113B1 Urea antagonists of p2y1 receptor useful in the treatment of thrombotic conditions
03/10/2010EP1423376B1 Bicyclic compound, production and use thereof
03/10/2010EP1377293B1 Aryl and biaryl piperidines used as mch antagonists
03/10/2010CN101665488A New production technique of hydrobromic acid darifenacin
03/10/2010CN101665487A Method for preparing Flavopiridol
03/09/2010US7674903 Dehydrophenylahistins and analogs thereof and the synthesis of dehydrophenylahistins and analogs thereof
03/09/2010US7674887 3'-{N'-[1-(3,4-Dimethylphenyl)-3-methyl-5-oxo-1,5-dihydropyrazol-4-ylidene]hydrazino}-2'-hydroxybiphenyl-3-carboxylic acid; thrombocytopenia and megakaryocytopoiesis treatment
03/09/2010US7674828 Urea antagonists of P2Y1receptor useful in the treatment of thrombotic conditions
03/09/2010US7674823 DNA-PK inhibitors
03/09/2010US7674818 Aryl, aryloxy, alkyloxy substituted 1H-indol-3-yl glyoxylic acid derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1)
03/09/2010US7674809 Anti-inflammatory and analgesic heterocyclic amidines that inhibit nitrogen oxide (NO) production
03/09/2010US7674796 Inhibitors of the FAK (focal adhesion kinase) protein tyrosine kinases, antiproliferative, antitumor; for example 5-{4-[(1-Hydroxy-cyclopentylmethyl)-amino]-5-trifluoromethyl-pyrimidin-2-ylamino}-1,3-dihydro-indol-2-one
03/09/2010CA2493313C Novel benzodioxoles
03/09/2010CA2482346C Substituted phenylacetamides and their use as glucokinase activators
03/09/2010CA2431952C Muscarinic antagonists
03/09/2010CA2379282C Amido spiropiperidines promote the release of growth hormone
03/09/2010CA2329292C A process for the manufacture of sulfonylaminocarbonyl triazolinones and salts thereof under ph controlled conditions
03/09/2010CA2306313C Dipeptide nitriles
03/09/2010CA2140598C Prolineamide derivatives
03/04/2010WO2010024769A1 New benzofurans suitable as precursors to compounds that are useful for imaging amyloid deposits
03/04/2010WO2010024430A1 2,4-diaminopyrimidine compound
03/04/2010WO2010024227A1 Novel pyrrole derivative having, as substituents, ureide group, aminocarbonyl group and bicyclic group which may have substituent
03/04/2010WO2010024110A1 Oxotetrahydrofuran-2-yl-benzimidazole derivative
03/04/2010WO2010023946A1 Novel uracil compound having nitrogenated heterocyclic ring or salt thereof
03/04/2010WO2010023931A1 1-adamantylazetidin-2-one derivative and pharmaceutical preparation comprising same
03/04/2010WO2010023678A1 A process for preparation of rosuvastatin intermediate
03/04/2010WO2010023512A1 Novel vanilloid receptor modulators, process for their preparation and pharmaceutical compositions containing them
03/04/2010WO2010022725A1 Pyridine derivatives as vegfr-2 receptor and protein tyrosine kinase inhibitors