Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397) |
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03/18/2010 | CA2736970A1 Pyrimidinone derivatives for use as medicaments |
03/18/2010 | CA2736530A1 Piperazine derivatives for binding and imaging amyloid plaques and their use |
03/18/2010 | CA2736039A1 Novel prostaglandin i2 derivative |
03/18/2010 | CA2735184A1 Heteroaryls amide derivatives and their use as glucokinase activators |
03/18/2010 | CA2734454A1 A process for preparing [1s-[1-alpha,2-alpha,3-beta(1s*, 2r*)5-beta]]-3-[7-[2-(3,4-difluorophenyl)-cyclopropylamino]-5-(propylthio)-3h-1,2,3-triazolo [4,5-d]pyrimidin-3-yl]-5-(2-hydroxyethoxy)cyclopentane-1,2-diol and to its intermediates |
03/17/2010 | EP2163553A1 Arene connected polyamine macroring derivatives, preparation methods and pharmaceutical uses thereof |
03/17/2010 | EP2163543A1 Nitrogen-containing heterocyclic derivative having 11 beta-hydroxysteroid dehydrogenase type i inhibitory activity |
03/17/2010 | EP2163541A1 Piperazine derivatives for binding and imaging amyloid plaques and their use |
03/17/2010 | EP2162453A1 Crystalline form b of olmesartan medoxomil |
03/17/2010 | EP2162450A1 ((bicylicheteroaryl) imidazolyl) methylheteroaryl compounds as adrenergic receptor agonists |
03/17/2010 | EP2162442A1 Dual-acting benzoimidazole antihypertensive agents |
03/17/2010 | EP2162436A1 Novel case of renin inhibitors |
03/17/2010 | EP2162433A2 4' substituted compounds having 5-ht6 receptor affinity |
03/17/2010 | EP1713822B1 Hcv ns-3 serine protease inhibitors |
03/17/2010 | EP1689742B1 Quinolonecarboxylic acid compounds having 5-ht4 receptor agonistic activity |
03/17/2010 | EP1620411B1 Inhibitors of akt activity |
03/17/2010 | EP1513814B1 Novel piperidine compound |
03/17/2010 | EP1284966B1 Process for the synthesis of amine ethers from secondary amino oxides |
03/17/2010 | CN101675042A Novel 2-heteroaryl substituted benzothiophenes and benzofuranes 709 |
03/17/2010 | CN101675036A dual-acting benzoimidazole antihypertensive agents |
03/17/2010 | CN101671335A Cytotoxins, prodrugs, linkers and stabilizers useful therefor |
03/17/2010 | CN101671310A Compounds and compositions useful as cathepsin s inhibitors |
03/17/2010 | CN101671307A 杂环天冬氨酰蛋白酶抑制剂 Heterocyclic aspartyl protease inhibitors |
03/16/2010 | US7678904 or to treat autoimmune and inflammatory disorders; improved water solubility characteristics |
03/16/2010 | US7678813 8a-Benzyl-2-(4-methoxyphenyl)-1,3,4,7,8,8a-hexahydro-2H-isoquinolin-6-one; psychotic major depression, schizoaffective disorder, Alzheimer's Disease and cocaine addiction |
03/16/2010 | US7678812 Aminotetralin-derived urea modulators of vanilloid VR1 receptor |
03/16/2010 | US7678804 Pyrimidine derivatives for treatment of hyperproliferative disorders |
03/16/2010 | US7678802 Voltage gated sodium and calcium channel inhibitors |
03/16/2010 | US7678798 5-({4-[(3S)-4-(5-bromo-2,3-dihydro-1H-inden-1-yl)-3-methylpiperazin-1-yl]-4-methylpiperidin-1-yl}carbonyl)-4,6-dimethylpyrimidine; inflammatory diseases, immune diseases and viral infections; HIV |
03/16/2010 | US7678790 sulfonylurea derivatives, sulfonylthiourea derivatives, sulfonylguanidine derivatives, sulfonylcyanoguanidine derivatives, thioacylsulfonamide derivatives, and acylsulfonamide derivatives; effective for prevention and treatment of cardiovascular diseases, antithrombotic agents |
03/16/2010 | CA2493966C Benzopyran derivatives substituted with secondary amines including imidazole, their preparation and pharmaceutical compositions containing them |
03/16/2010 | CA2386980C Benzodiazepine derivatives for use in acute or chronic neurological disorders |
03/11/2010 | WO2010027848A2 Forms of lapatinib compounds and processes for the preparation thereof |
03/11/2010 | WO2010026771A1 Nitrogenated heterocyclic compound and salt thereof, and bactericidal agent for agricultural or horticultural applications |
03/11/2010 | WO2010026388A1 Isatin derivatives for use as in vivo imaging agents |
03/11/2010 | WO2010026255A1 Process for preparing olmesartan medoxomil intermediate |
03/11/2010 | WO2010026212A1 Novel inhibitors |
03/11/2010 | WO2010026096A1 7-(piperazine-1-ymethyl)-1h-indole-2-carboxylic acid (phenyl)-amide derivatives and allied compounds as p38 map kinase inhibitors for the treatment of respiratory diseases |
03/11/2010 | WO2010026095A1 Novel benzamides, production thereof, and use thereof as medicaments |
03/11/2010 | WO2010025850A1 Heterocyclically substituted anilinopyrimidines as fungicides |
03/11/2010 | WO2010025831A1 Heterocyclically substituted anilinopyrimidines as fungicides |
03/11/2010 | WO2010006755A3 Cyclic polyamines for binding phosphatidylserine |
03/11/2010 | WO2009156099A8 6-substituted isoquinolines and isoquinolinones |
03/11/2010 | WO2008094909A3 Quinazolinone and fused pyrimidinone compounds and their use in treating sodium channel-mediated diseases or conditions |
03/11/2010 | US20100063129 4-Diallylaminomethylene-6-hydroxy-1- alpha -methoxymethyl-10 beta ,13 beta -dimethyl-3,7,17-trioxo-1,3,4,7,10,11 beta ,12,13,14 alpha ,15,16,17-dodecahydro-2-oxa-cyclopenta[ alpha ] phenanthren-11-ol or its acetate in a carrier; PI-3 kinase inhibitor; treating color cancer |
03/11/2010 | US20100063119 Substituted carbinol compound |
03/11/2010 | US20100063105 Pharmaceutical uses and synthesis of nicotinanilide-n-oxides |
03/11/2010 | US20100063100 Modulators of aldehyde dehydrogenase activity and methods of use thereof |
03/11/2010 | US20100063087 5-Amino-4-Hydroxy-7-(Imidazo [1,2-A] Pyridin-6-Ylmethyl)-8-Methyl-Nonamide Derivatives and Related Compounds as Renin Inhibitors for the Treatment of Hypertension |
03/11/2010 | US20100063079 Pyrimidyl Sulphone Amide Derivatives as Chemokine Receptor Modulators |
03/11/2010 | US20100063075 Aryl-quinazoline/aryl-2amino-phenyl methanone derivatives |
03/11/2010 | US20100063062 Novel use of 1-[4-(5-cyanoindol-3-yl)butyl]-4-(2-carbamoyl-benzofuran-5-yl)-piperazine and its physiologically acceptable salts |
03/11/2010 | US20100063056 Bipyridine carboxamide orexin receptor antagonists |
03/11/2010 | US20100063040 Sulfonamide Derivative Having PGD2 Receptor Antagonistic Activity |
03/11/2010 | US20100062996 Dioxolane derivates for the treatment of cancer |
03/11/2010 | US20100062972 Triazole compounds and uses related thereto |
03/11/2010 | US20100062942 Pyrazolyl-substituted heterocycles and their use as phytosanitary products |
03/11/2010 | US20100062937 Benzanilides with insecticidal activity |
03/11/2010 | US20100062065 Pharmaceutical composition containing naphthoquinone-based compound for intestine delivery system |
03/11/2010 | US20100061982 3-substituted-1h-indole, 3-substituted-1h-pyrrolo[2,3-b]pyridine and 3-substituted-1h-pyrrolo[3,2-b]pyridine compounds, their use as mtor kinase and pi3 kinase inhibitors, and their syntheses |
03/11/2010 | CA2735970A1 Isatin derivatives for use as in vivo imaging agents |
03/11/2010 | CA2735795A1 Novel inhibitors |
03/11/2010 | CA2735770A1 7-(piperazine-1-ymethyl)-1h-indole-2-carboxylic acid (phenyl)-amide derivatives and allied compounds as p38 map kinase inhibitors for the treatment of respiratory diseases |
03/11/2010 | CA2735208A1 Novel benzamides, production thereof, and use thereof as medicaments |
03/11/2010 | CA2733533A1 Hedgehog pathway modulators |
03/10/2010 | EP2161266A1 Benzofuran derivatives as orexin receptor antagonists |
03/10/2010 | EP2160387A2 Heteroarylamide pyrimidone compounds |
03/10/2010 | EP2160380A1 Cyano-guanidine derivatives as glutaminyl cyclase inhibitors |
03/10/2010 | EP1896456B1 Novel tetracyclic tetrahydrofuran derivatives containing a cyclic amine side chain |
03/10/2010 | EP1841737B1 N-(heteroaryl)-1h-indole-2-carboxamide derivatives and their use as vanilloid trpv1 receptor ligands |
03/10/2010 | EP1786801B1 2-arylcarbamoyl-indoles as cytokine inhibitors |
03/10/2010 | EP1780209B1 Oxime ester compound and photopolymerization initiator containing such compound |
03/10/2010 | EP1751113B1 Urea antagonists of p2y1 receptor useful in the treatment of thrombotic conditions |
03/10/2010 | EP1423376B1 Bicyclic compound, production and use thereof |
03/10/2010 | EP1377293B1 Aryl and biaryl piperidines used as mch antagonists |
03/10/2010 | CN101665488A New production technique of hydrobromic acid darifenacin |
03/10/2010 | CN101665487A Method for preparing Flavopiridol |
03/09/2010 | US7674903 Dehydrophenylahistins and analogs thereof and the synthesis of dehydrophenylahistins and analogs thereof |
03/09/2010 | US7674887 3'-{N'-[1-(3,4-Dimethylphenyl)-3-methyl-5-oxo-1,5-dihydropyrazol-4-ylidene]hydrazino}-2'-hydroxybiphenyl-3-carboxylic acid; thrombocytopenia and megakaryocytopoiesis treatment |
03/09/2010 | US7674828 Urea antagonists of P2Y1receptor useful in the treatment of thrombotic conditions |
03/09/2010 | US7674823 DNA-PK inhibitors |
03/09/2010 | US7674818 Aryl, aryloxy, alkyloxy substituted 1H-indol-3-yl glyoxylic acid derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1) |
03/09/2010 | US7674809 Anti-inflammatory and analgesic heterocyclic amidines that inhibit nitrogen oxide (NO) production |
03/09/2010 | US7674796 Inhibitors of the FAK (focal adhesion kinase) protein tyrosine kinases, antiproliferative, antitumor; for example 5-{4-[(1-Hydroxy-cyclopentylmethyl)-amino]-5-trifluoromethyl-pyrimidin-2-ylamino}-1,3-dihydro-indol-2-one |
03/09/2010 | CA2493313C Novel benzodioxoles |
03/09/2010 | CA2482346C Substituted phenylacetamides and their use as glucokinase activators |
03/09/2010 | CA2431952C Muscarinic antagonists |
03/09/2010 | CA2379282C Amido spiropiperidines promote the release of growth hormone |
03/09/2010 | CA2329292C A process for the manufacture of sulfonylaminocarbonyl triazolinones and salts thereof under ph controlled conditions |
03/09/2010 | CA2306313C Dipeptide nitriles |
03/09/2010 | CA2140598C Prolineamide derivatives |
03/04/2010 | WO2010024769A1 New benzofurans suitable as precursors to compounds that are useful for imaging amyloid deposits |
03/04/2010 | WO2010024430A1 2,4-diaminopyrimidine compound |
03/04/2010 | WO2010024227A1 Novel pyrrole derivative having, as substituents, ureide group, aminocarbonyl group and bicyclic group which may have substituent |
03/04/2010 | WO2010024110A1 Oxotetrahydrofuran-2-yl-benzimidazole derivative |
03/04/2010 | WO2010023946A1 Novel uracil compound having nitrogenated heterocyclic ring or salt thereof |
03/04/2010 | WO2010023931A1 1-adamantylazetidin-2-one derivative and pharmaceutical preparation comprising same |
03/04/2010 | WO2010023678A1 A process for preparation of rosuvastatin intermediate |
03/04/2010 | WO2010023512A1 Novel vanilloid receptor modulators, process for their preparation and pharmaceutical compositions containing them |
03/04/2010 | WO2010022725A1 Pyridine derivatives as vegfr-2 receptor and protein tyrosine kinase inhibitors |