Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
10/2009
10/08/2009WO2009121507A2 Substituted enaminothiocarbonyl compounds
10/08/2009WO2009121247A1 Luminescence quenchers and fluorogenic probes for detection of reactive species
10/08/2009US20090253908 Novel m3 muscarinic acetylchoine receptor antagonists
10/08/2009US20090253762 Preparation and use of aryl alkyl acid derivatives for the treatment of obesity
10/08/2009US20090253749 Substituted enaminocarbonyl compounds
10/08/2009US20090253736 Azaindole derivatives as cftr modulators
10/08/2009US20090253700 N-'4-4(4-morpholinyl) phenyl!- '(4-piperidinyl) methyl! carboxamide derivatives and their use as glycine transporter inhibitors
10/08/2009US20090253697 Novel Indole Derivatives, Preparation Thereof as Medicinal Products and Pharmaceutical Compositions, and Especially as KDR Inhibitors
10/08/2009US20090253694 Fused hetrocyclic compounds
10/08/2009US20090253684 Leukotriene b4 inhibitors
10/08/2009US20090253682 Heterocyclic derivatives for modulation of calcium channels
10/08/2009US20090253656 Bcrp/abcg2 inhibitor
10/08/2009US20090253645 Methods and materials for treating and preventing inflammation of mucosal tissue
10/08/2009CA2720275A1 Indolinone compound
10/08/2009CA2719907A1 Hydroxymethyl pyrrolidines as beta 3 adrenergic receptor agonists
10/08/2009CA2718488A1 Novel dhsp90 inhibitory carbazole derivatives, compositions containing same, and use thereof
10/08/2009CA2718310A1 Pyridyl derivatives as cftr modulators
10/08/2009CA2685716A1 Compounds for treating muscular dystrophy
10/07/2009EP2107058A1 Substituted enaminothiocarbonyl compounds
10/07/2009EP2107052A1 Novel n-(2-aminophenyl)benzamide derivative having an urea structure
10/07/2009EP2106400A2 Benzoquinazole derivatives
10/07/2009EP2106398A2 Isoquinolinecarboxamides as inhibitors of stearoyl-coa desaturase (scd)
10/07/2009EP1756087B1 Amino-5,5-diphenylimidazolone derivatives for the inhibition of beta-secretase
10/07/2009EP1709027B1 Hydrazide type compounds and the use thereof in pharmaceutical compositions for the treatment of cardiovascular diseases
10/07/2009EP1309566B1 Dihydroxypyrimidine carboxylic acids as viral polymerase inhibitors
10/07/2009EP1308441B1 2-aminopyridine compounds and use thereof as drugs
10/07/2009EP1248774B1 Polyhydroxystilbenes and stilbene oxides as antipsoriatic agents and protein kinase inhibitors
10/07/2009EP0861247B1 Novel imidazole n-benzyldioxol derivatives, method for preparing same, resulting intermediates, pharmaceutical compositions and use of said derivatives as endothelin antagonists
10/07/2009CN101553484A Thrombin receptor antagonists based on the modified tricyclic unit of himbacine
10/07/2009CN101553468A Organic compounds
10/07/2009CN101550132A Arylvinylazacycloalkane compounds and methods of preparation and use thereof
10/07/2009CN101550119A Aryl (ethanoic) propanoic acid ascorbyl ester, preparation method thereof and medicament containing same
10/06/2009US7598377 (+-)-7-Methyl-2-morpholin-4-yl-9-(1-phenylaminoethyl)-pyrido[1,2-a]pyrimidin-4-one, for example; selective inhibitors of phosphoinositide (PI) 3-kinase beta for use in anti-thrombotic therapy
10/06/2009US7598288 Inhibitors of glycogen synthase kinase-3 (GSK-3) for treating glaucoma
10/06/2009US7598285 N-[4-((1S)-1-{3-(3,5-Dichlorophenyl)-5-[6-(trifluoromethoxy)-2-naphthyl]-1H-pyrazol-1-yl}ethyl)benzoyl]- beta -alanine; type 2 diabetes, hyperglycemia, or insulin resistance
10/06/2009US7598284 Indazole compounds as B3 adrenoceptor agonist
10/06/2009US7598271 Crystalline paroxetine methane sulfonate
10/06/2009US7598268 Vascular endothelial growth factor; tyrosine kinase inhibitor;angiogenesis inhibitor; anticarcinogenic agents
10/06/2009US7598260 CDK-inhibitory pyrimidines, their production and use as pharmaceutical agents
10/06/2009US7598251 aminopyrazine derivatives; ROCK inhibitors; 3-(1-ethyl-1H-imidazo[4,5-c]pyridin-2-yl)pyrazin-2-amine; antiinflammatory, antidiabetic, antiproliferative agents
10/06/2009US7598250 for treating neurodegenerative disease such as Alzheimer's disease
10/01/2009WO2009119880A1 Substituted pyrazole derivatives and use thereof
10/01/2009WO2009119785A1 Method for purifying ethynylthymidine compound
10/01/2009WO2009119528A1 Heterocyclic compound
10/01/2009WO2009119167A1 Aniline derivative having anti-rna viral activity
10/01/2009WO2009119088A1 Heterocyclic compound
10/01/2009WO2009118765A2 Novel monoamine re-uptake inhibitor
10/01/2009WO2009118473A2 Azetidine-derived compounds, preparation method therefor and therapeutic use of same
10/01/2009WO2009118411A2 3,4-dihydro-2h-pyrazino[1,2-a]indol-1-one derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
10/01/2009WO2009118305A1 Hydroxamate-based inhibitors of deacetylases b
10/01/2009WO2009118254A1 Aminopiperidinyl derivatives and uses thereof
10/01/2009WO2009074300A3 Hedgehog pathway antagonists and therapeutic applications thereof
10/01/2009WO2009060835A8 Novel ubiquilin-binding small molecule
10/01/2009US20090247745 adenosine A3 receptor antagonists; improved bioavailability; treatment of diseases such as asthma, COPD and ARDS, glaucoma, tumor, allergic and inflammatory diseases, ischemia, hypoxia, arrythmia and renal diseases; e.g. 4-Methoxy-N-[6-(morpholin-4-yl)-4-benzylamino-3-cyanoquinolin-2-yl]-benzamide
10/01/2009US20090247617 Process for the preparation of benzo-fused heteroaryl sulfamates
10/01/2009US20090247587 1,3-dihydroisobenzofuran derivatives
10/01/2009US20090247509 for treating central nervous system disorders such as psychological disorders, drug dependence and abuse, dyskinesia, dementia, anxiety disorders, sleep disorders and mood disorders
10/01/2009US20090247503 5-demethoxyfumagillol and derivatives thereof
10/01/2009US20090247489 Dihydroxyl compounds and compositions for cholesterol management and related uses
10/01/2009US20090247474 3-Aminopyrrolidine Derivatives As Modulators Of Chemokine Receptors
10/01/2009US20090246390 Aziridine crosslinking agents having water solubilizing groups are more environmentally friendly, do not require VOCs, lower cost
10/01/2009US20090246137 Pyridyl derivatives as cftr modulators
10/01/2009CA2719477A1 Hydroxamate-based inhibitors of deacetylases b
10/01/2009CA2718727A1 Heterocyclic compound
10/01/2009CA2716961A1 Azetidine-derived compounds, preparation method therefor and therapeutic use of same
10/01/2009CA2716932A1 Aza-bicyclohexyl substituted indolyl alkyl amino derivatives as novel inhibitors of histone deacetylase
10/01/2009CA2712468A1 Aminopiperidinyl derivatives and uses thereof
09/2009
09/30/2009EP2105441A1 Alanyl aminopeptidase and dipeptidylpeptidase IV dual inhibitors for the treatment of immunological, inflammatory, neuronal and other illnesses
09/30/2009EP2104673A2 New 2, 4-dianilinopyrimidines, preparation thereof as drugs, pharmaceutical compositions and use thereof essentially as ikk inhibitors
09/30/2009EP2104671A2 Substituted heterocyclylcarbonylamino-acetic-acid-derivatives as inhibitors of bacterial heptose synthesis, methods for their preparation and biological applications of said inhibitors
09/30/2009EP2104670A2 Novel triazinedione derivatives as gaba-b receptor modulators
09/30/2009EP1962849B1 Quinoline derivatives useful in the treatment of mglur5 receptor-mediated disorders
09/30/2009EP1711181B1 Quinoline derivatives and use thereof as mycobacterial inhibitors
09/30/2009EP1435944B1 4(4-alkoxy-3-hydroxyphenyl)-2-pyrrolidone derivatives as pde-4 inhibitors for the treatment of neurological syndromes
09/29/2009US7595343 Inhibitors of histone deacetylase
09/29/2009US7595339 Such as N-(4-Fluoro-benzyl)-4-(3-phenyl-indole-1-sulfonyl)-benzamide; Cannabinoid-1 (CB1) receptor; dietetics
09/29/2009US7595329 4-{[4-({[(3-isopropyl-2-oxo-2,3-dihydro-1H-benzimidazol-1-yl)carbonyl]amino}methyl)piperidin-1-yl]methyl}tetrahydro-2H-pyran-4-carboxylic acid; serotonin receptor agonist; gastroesophageal reflux disease, analgesic, cognition activator; less toxicity, good absorption, and metabolic stability
09/29/2009US7595321 Useful for the prevention and/or treatment of cognitive disorders; 3-Amino-N-(2-cyanoethyl)-6-[4-(pyrrolidin-1-ylsulfonyl)phenyl]pyrazine-2-carboxamide, for example
09/29/2009US7595319 Compounds having selective inhibiting effect at GSK3
09/29/2009CA2438891C Method for preparing optically active dihydropyrones
09/29/2009CA2368495C Electron-deficient nitrogen heterocycle-substituted fluorescein dyes
09/29/2009CA2348391C Chromenone and chromanone derivatives as integrin inhibitors
09/29/2009CA2315647C Inhibition of p38 kinase activity using aryl and heteroaryl substituted heterocyclic ureas
09/24/2009WO2009117269A1 Substituted 4-hydroxypyrimidine-5-carboxamides
09/24/2009WO2009116055A1 Lamivudine : zidovudine : water 1 : 1 : 1 cocrystal
09/24/2009WO2009115874A2 Novel heterocyclic compounds, pharmaceutical compositions containing them and processes for their preparation
09/24/2009WO2009115547A1 Trisubstituted 1, 2, 4 -triazoiies as nicotinic acetylcholine receptor modulators
09/24/2009WO2009087212A3 Pyridine derivatives
09/24/2009WO2009076142A3 Processes for producing cycloalkylcarboxiamido-pyridine benzoic acids
09/24/2009WO2009067035A3 Method of obtaining of 4-n-furfurylcytosine and/or its derivatives, an anti-aging composition and use of 4-n-furfurylcytosine and/or its derivatives in the manufacture of anti-aging composition
09/24/2009US20090239889 Spiro[2-cyclohexene-1,3'-[3H]indole]-2',4(1'H)-diones and 4-hydroxyspiro[2-cyclohexene-1,3'-[3H]indol]-2'(1'H)-ones; act as antagonists of mdm2 interactions; useful as potent and selective anticancer agents
09/24/2009US20090239883 Treatment of Pulmonary Hypertension
09/24/2009US20090239876 Substituted 4-Hydroxypyrimidine-5-Carboxamides
09/24/2009US20090239866 Peptide deformylase inhibitors
09/24/2009US20090239863 1-aryl-or 1- alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands
09/24/2009US20090239860 Novel benzofuran derivative, medicinal composition containing the same, and uses of these
09/24/2009US20090239845 Pyrazole compounds as prostaglandin receptors ligands
09/24/2009US20090239773 Lubricant additive, lubricant composition and grease composition
09/24/2009US20090238761 Novel Aryl Piperazine Derivatives With Medical Utility
09/24/2009CA2718936A1 Novel heterocyclic compounds and uses therof