Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
04/2010
04/07/2010EP2170866A1 Phthalazine compounds, compositions and methods of use
04/07/2010EP2170861A2 Derivatives of 4-(n-azacycloalkyl) anilides as potassium channel modulators
04/07/2010EP2170857A2 3',4',5-trimethoxy flavone derivatives as stimulant of mucus secretion, method of the same, and pharmaceutical composition comprising the same
04/07/2010EP2170843A1 Hetero bicyclic carboxamide derivatives and their pharmaceutical use and compositions
04/07/2010EP2170831A1 Benzazepine derivatives useful as vasopressin antagonists
04/07/2010EP2170329A2 Crystalline polymorph of 7-ethyl-10-hydroxycamptothecin
04/07/2010EP2170328A2 Crystalline polymorph of exemestane
04/07/2010EP1673368B1 Azole derivative useful as antifungal agents with reduced interaction with metabolic cytochromes
04/07/2010EP1551829B1 Novel compounds with antibacterial activity
04/07/2010EP1527050B1 Quinoline derivatives and their use as mycobacterial inhibitors
04/07/2010CN101691360A Preparation method of carbamyl benzotriazole
04/07/2010CN101691353A N-Boc-3,5-(E)-diarylidene-4-piperidone and application thereof in preparation of anti-tumor drugs
04/06/2010US7692028 for treating neurological disorders such as epilepsy, neuropathic pain, bipolar disorder or migraine; 2-(2-oxo-4-propyl-1-pyrrolidinyl)butanamide; neuroprotective agent
04/06/2010US7692009 Reference standard for characterization of rosuvastatin
04/06/2010US7691883 decreases expression of a Type I collage gene in a tissue to induce a reduction in accumulation of collagen and thereby improves tissue fibrosis
04/06/2010US7691881 1-isopropyl-2-oxo-1,2-dihydropyridine-3-carboxamide derivatives having 5-HT4 receptor agonistic activity
04/06/2010US7691854 Diethyl 2-amino-4-(4-cyanophenyl)-6-methyl-1-(3-methylphenyl)-1,4-dihydro-3,5-pyridine-dicarboxylate; chronic obstructive pulmonary disease, acute coronary syndrome, acute myocardial infarction or development of heart failure
04/06/2010US7691853 Pyrazole compounds useful as protein kinase inhibitors
04/06/2010US7691843 Inhibitors of UPD-3-O (R-3-hydroxymyristoyl)-N-acetylglucosamine deacetylase, an enzyme present in gram negative bacteria; azetidine, pyrrolidine, or 3-pyrroline 2-carboxylic acid hydroxyamides; 1-(3,4-dimethoxy-5-propylbenzoyl)pyrrolidine-2R-carboxylic acid hydroxyamide for example
04/06/2010US7691837 e.g. 1-{[1,5-bis(4-cholorophenyl)-2-methylpyrrol-3-yl]methyl}-4-(4-fluoro-phenyl)piperazine; Mycobacterium tuberculosis, drug resistant Mycobacterium tuberculosis, Mycobacterium avium-intracellulare complex, Mycobacterium fortuitum or Mycobacterium kansasi
04/06/2010US7691785 Pyridine-3-ketone compound; plant growth controllers
04/06/2010CA2496712C New process for synthesizing derivatives of 1,3,4,5-tetrahydro-2h-3-benzazepin-2-one and its application to the synthesis of ivabradine and its pharmaceutically acceptable acid addition salts
04/06/2010CA2449899C Piperazinylpyrazines compounds as antagonists of serotonin 5-ht2 receptor
04/06/2010CA2397636C Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses
04/06/2010CA2319807C Novel antifungal compound and process for producing the same
04/01/2010WO2010037129A1 Quinazolinone, quinolone and related analogs as sirtuin modulators
04/01/2010WO2010037066A2 Dosage units of 3-(6-(1-(2,2-difluorobenzo [d] [1,3] dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic acid
04/01/2010WO2010036631A2 Compounds which selectively modulate the cb2 receptor
04/01/2010WO2010036630A2 Compounds which selectively modulate the cb2 receptor
04/01/2010WO2010036613A1 Novel cyclic benzimidazole derivatives useful anti-diabetic agents
04/01/2010WO2010035766A1 Method for producing triazole derivative
04/01/2010WO2010035745A1 Heterocyclic biaryl derivative, and pde inhibitor comprising same as active ingredient
04/01/2010WO2010035727A1 Novel pyrrolinone derivative and medicinal composition containing same
04/01/2010WO2010034797A1 1h-benzimidazole-5-carboxamides as anti-inflammatory agents
04/01/2010WO2010034796A1 1h-benz imidazole-5-carboxamides as anti-inflammatory agents
04/01/2010WO2010034671A1 Pyrine or pyrazine derivatives for treating hcv
04/01/2010WO2010017545A3 Triazole compounds that modulate hsp90 activity
04/01/2010US20100081686 Pyridone derivatives having a binding activity to the cannabinoid type 2 recepter
04/01/2010US20100081670 N-pyrazinyl-phenylsulphonamides and their use in the treatment of chemokine mediated diseases
04/01/2010US20100081658 Heterocyclic antiviral compounds
04/01/2010US20100081203 Fluorescent isotope tags and their method of use
04/01/2010CA2738809A1 Quinazolinone, quinolone and related analogs as sirtuin modulators
04/01/2010CA2738083A1 1h-benzimidazole-5-carboxamides as anti-inflammatory agents
04/01/2010CA2737694A1 Novel cyclic benzimidazole derivatives useful anti-diabetic agents
04/01/2010CA2737645A1 Compounds which selectively modulate the cb2 receptor
04/01/2010CA2737639A1 Compounds which selectively modulate the cb2 receptor
04/01/2010CA2737384A1 1h-benzimidazole-5-carboxamides as anti-inflammatory agents
04/01/2010CA2736545A1 Dosage units of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic acid
04/01/2010CA2736472A1 Pyrine or pyrazine derivatives for treating hcv
03/2010
03/31/2010EP2168962A2 Phenylacetamides and their use as glucokinase modulators
03/31/2010EP2168958A1 Isoindole-Imide Compounds, Compositions And Uses Thereof
03/31/2010EP2168951A1 Azolylmethylenehydrazine derivative and use thereof
03/31/2010EP2168947A1 Novel compound having secretase inhibitory activity
03/31/2010EP2168576A2 New utilities of tricyclic compounds
03/31/2010EP2167494A1 3-amino-6-(1-amino-ethyl)-tetrahydropyran derivatives
03/31/2010EP2167487A1 Pyrrole derivatives as p2y12 antagonists
03/31/2010EP2167485A2 2-acylaminopropoanol-type glucosylceramide synthase inhibitors
03/31/2010EP2167484A2 Condensed anthranilamide insecticides
03/31/2010EP2167472A2 1-benzylpyrazole derivatives, preparation thereof and therapeutic use thereof
03/31/2010EP2167466A1 N-phenyl hydrazides as modulators of the ghrelin receptor
03/31/2010EP2167083A2 Novel 1- heteroaryl-3-azabicycloý3.1.0¨hexanes, methods for their preparation and their use as medicaments
03/31/2010EP2166854A1 Triazole derivatives for treating alzheimer's disease and related conditions
03/31/2010EP2166850A1 New heteocyclic h3 antagonists
03/31/2010EP2166849A1 Substituted pyrazole compounds
03/31/2010EP1904465B1 Method of synthesis of imidazole-amino acid derivatives and related compounds
03/31/2010EP1546107B1 Cox-2 inhibiting pyridine derivatives
03/31/2010EP1252139B1 Trifluoromethylpyrrole carboxamides and trifluoromethylpyrrolethioamides as fungicides
03/31/2010CN101687913A kallikrein 7 modulators
03/31/2010CN101687860A Novel n- (8-heteroaryltetrahydronaphtalene-2yl) or n- (5- heteroarylchromane-3-yl) carboxamide derivatives for the treatment of pain
03/31/2010CN101687859A Process for the preparation of alfuzosin and salts thereof
03/31/2010CN101687858A 1, 3-dihydroimidazole- 2 -thione derivatives as inhibitors of dopamine-beta-hydroxylase
03/31/2010CN101687853A Pyrimidine derivatives and compositions as C-KIT and PDGFR kinase inhibitors
03/31/2010CN101687850A Substituted pyrimidines as adenosine receptor antagonists
03/31/2010CN101687844A Imidazole derivatives as CCR2 receptor antagonists
03/31/2010CN101687843A Substituted aromatic heterocyclic compounds as fungicides
03/31/2010CN101687842A modulators of cftr
03/31/2010CN101687841A Benzimidazole derivatives
03/31/2010CN101687817A Tri-amino-pyrimidine cyclobutenedione derivatives used as phosphatase cdc25 inhibitors
03/31/2010CN101687816A Triaminopyrimidine derivatives as inhibitors of cdc25 phosphatase
03/31/2010CN101687812A 2 -imidazolines having a good affinity to the trace amine associated receptors (TAAR)
03/31/2010CN101687807A 1-benzylpyrazole derivatives, preparation thereof and therapeutic use thereof
03/31/2010CN101687805A Benzazepine derivatives useful as vasopressin antagonists
03/31/2010CN101687786A Hydroxylamine compounds and methods of their use
03/31/2010CN101686969A crystalline polymorph of exemestane
03/31/2010CN101686968A crystalline polymorph of 7-ethyl-10-hydroxycamptothecin
03/31/2010CN101684115A 4-(5-((2-(4-morpholinyl-6-phenylamino group-1,3,5-triazine-2-base) hydrazono) methyl) furan-2-base) benzoic acid, preparing method and application thereof
03/31/2010CN101684097A Phenylpyrimidine amines as ige inhibitors
03/31/2010CN101684095A Novel organic electroluminescent compounds and organic electroluminescent device using the same
03/31/2010CN101684091A cannabinoid receptor ligands
03/31/2010CN101684089A bicycloester derivative
03/30/2010US7687643 For angiogenesis mediated diseases; cancer; acylation, cyclization and Heck-type reduction
03/30/2010US7687640 3-methoxy-4-(4-methyl-1H-imidazol-1-yl)benzaldehyde; inhibits production of A beta 40 and A beta 42 from amyloid precursor protein ; Alzheimer's disease and Down syndrome
03/30/2010US7687639 Useful as adjuvants to chemotherapy or radiation therapy to treat cancer; as inhibitors of checkpoint kinase Cds1 (in man also known as Chk2); 2-[4-(3,4-dichloro-phenoxy)-phenyl]-1H-imidazo[4,5-b]pyridine-5-carboxylic acid amide
03/30/2010US7687631 Synthesis of diethyl{[5-(3-fluorophenyl)-pyridine-2yl]methyl}phosphonate
03/30/2010US7687535 Substituted 3-sulfur indoles
03/30/2010US7687532 Fused heteroaryl derivatives for use as p38 kinase inhibitors in the treatment of I.A. rheumatoid arthritis
03/30/2010US7687525 e.g. N-(2-aminophenyl)-4-(N-benzoylaminomethyl)benzamide hydrochloride; anticarcinogenic, antitumor agents; hematologic malignancy and a solid carcinoma; autoimmune disease, skin disorders;
03/30/2010US7687514 Benzimidazole derivatives
03/30/2010US7687510 Pyrimidinone derivatives as therapeutic agents against acute and chronic inflammatory, ischaemic and remodelling processes
03/30/2010US7687503 2-(methylamino)-2-oxoethyl 4-{5-[3-(trifluoromethyl)-phenyl]-2-pyridyl}-1-piperazinecarboxylate, for example; enzyme inhibitors of fatty acid amide hydrolases; treatment of pain, eating disorders, neurological and psychiatric pathologies, among other disorders