Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587) |
---|
11/21/2002 | US20020173534 Amorphous form of cell cycle inhibitor having improved solubility and bioavailability |
11/21/2002 | US20020173533 Induce apoptosis; dissolving in critical fluid; separation |
11/21/2002 | US20020173532 Induce apoptosis |
11/21/2002 | US20020173527 Tumor necrosis factor antagonist; antiinflammatory agents |
11/21/2002 | US20020173518 Anticoagulant in mammls |
11/21/2002 | US20020173492 Novel pesticides |
11/21/2002 | US20020173425 Herbicides |
11/21/2002 | CA2447305A1 Novel 5-phenyl-1h-indole derivatives as antagonists of interleukine-8 receptors |
11/21/2002 | CA2446980A1 Substituted pyrazinones, pyridines and pyrimidines as corticotropin releasing factor ligands |
11/21/2002 | CA2445477A1 Antitumor agents |
11/21/2002 | CA2445003A1 Diarylurea derivatives useful as anti-inflammatory agents |
11/20/2002 | EP1258480A1 Pharmaceutical use of N-Carbamoylazole derivatives |
11/20/2002 | EP1258252A1 Integrin expression inhibitors |
11/20/2002 | EP1257547A1 1,3-disubstituted pyrrolidines as alpha-2-adrenoceptor antagonists |
11/20/2002 | EP1257546A1 Kinase inhibitors |
11/20/2002 | EP1257544A2 Piperazine and piperidine derivatives for treatment or prevention of neuronal damage |
11/20/2002 | EP1257543A1 Pyridinylimidazoles |
11/20/2002 | EP1257539A2 Amino pyrazole derivatives useful for the treatment of obesity and other disorders |
11/20/2002 | EP1187832B1 Amino heterocycles useful as pharmaceutical agents |
11/20/2002 | EP1007522B1 2- 4-[4-(4,5-dichloro-2-methylimidazol-1-yl)butyl]piperazin-1-yl -5-fluoropyrimidine, its preparation and therapeutic use |
11/20/2002 | EP0929530B1 Quinazoline derivatives and pharmaceutical compositions containing them |
11/20/2002 | EP0925302B1 Palladium catalyzed indolization |
11/20/2002 | EP0826673B1 Acetamide derivatives, process for producing the same, and medicinal composition containing the same |
11/20/2002 | EP0721453B1 Process for the preparation of n-methyl-3-(1-methyl-4-piperidinyl)-14-indole-5-ethanesulphonamide |
11/20/2002 | CN1094491C 2-{4-[4-(4,5-methylimidazol-1-yl)butyl]-1-piperazinyl}-5-fluoropyrimiding, preparation and use thereof |
11/19/2002 | US6482956 Endothelin receptor antagonists |
11/19/2002 | US6482955 Organometallic reagent reacted with an activated carboxylic acid to produce a ketone reacted with carbon disulfide and dihalomethane, further reacting the dithietane product with a secondary amine, and condensing the thioamide with hydrazine |
11/19/2002 | US6482951 Isoindolin-1-one glucokinase activators |
11/19/2002 | US6482949 Colormetric sensor compositions and methods |
11/19/2002 | US6482920 Acryloyl substituted distamycin derivatives, process for preparing them, and their use as antitumor and antiviral agents |
11/19/2002 | US6482848 Prodrugs of 3-(pyrrol-2-ylmethylidene)-2-indolinone derivatives |
11/19/2002 | US6482847 3-(1-methyl-3-indolyl)-4-(1-methyl-6-nitro-3-indolyl)-1h -pyrrole-2,5-dione anticarcinogenic agents |
11/19/2002 | US6482834 Quinoline and quinoxaline compounds which inhibit platelet-derived growth factor and/or p56lck tyrosine kinases |
11/19/2002 | US6482832 Heterocyclically substituted amides, their production and their use |
11/19/2002 | US6482773 Pyridazin-3-one derivatives, their use, and intermediates for their production |
11/19/2002 | CA2138308C Preparation of hexahydroazepinones and hexahydroazepinoles |
11/18/2002 | WO2001087855A1 Triazole derivatives |
11/14/2002 | WO2002090355A1 N-aroyl cyclic amines |
11/14/2002 | WO2002090348A1 Sulfonamides |
11/14/2002 | WO2002090347A1 Amide compounds |
11/14/2002 | WO2002090335A1 Azole compounds, process for preparation of the same and use thereof |
11/14/2002 | WO2002089811A1 Benzo[d]azepine derivatives as 5-ht6 receptor antagonists. |
11/14/2002 | WO2002089804A1 Alpha-2-adrenergic agonist/fatty acid compositions |
11/14/2002 | WO2002089793A1 Sulfonamides |
11/14/2002 | WO2002089792A1 Sulfonamides |
11/14/2002 | WO2002081453A8 Thiohydantoins and use thereof for treating diabetes |
11/14/2002 | WO2002074764A3 Piperazine derivatives and their use as 5-ht1b ligands |
11/14/2002 | WO2002064550A8 Glucocorticoid receptor modulators |
11/14/2002 | US20020169322 Use of N-alkylamino-heterocylic compounds for the treatment of migraine |
11/14/2002 | US20020169313 Of carbonyl compounds with secondary amines in the presence of a water scavenger, preferably trifluoroacetic acid; preparation of imidazole-containing benzodiazepines, which are inhibitors of farnesyl protein transferase |
11/14/2002 | US20020169200 Antitumor, antiinflammatory and antiarthritic agents, treating metastasis, restenosis, osteoporosis, inflammation, macular degeneration, and diabetic retinopathy |
11/14/2002 | US20020169180 Quinoline or quinazoline derivatives; antitumor agent, treating respiratory tract and gastrointestinal disorders |
11/14/2002 | US20020169165 Substituted bicyclic derivatives for the treatment of abnormal cell growth |
11/14/2002 | US20020169159 An acetamide derivative is useful for treatment of inflammatory and immune conditions and diseases; modulates the expressin and/or function of a chemokine receptor |
11/14/2002 | US20020169113 Orally available peptidic thrombin inhibitors |
11/14/2002 | CA2446396A1 N-aroyl cyclic amines |
11/14/2002 | CA2446387A1 Azole compound, process for producing the same and use thereof |
11/14/2002 | CA2446365A1 Sulfonamides |
11/14/2002 | CA2446234A1 Alpha-2-adrenergic agonist/fatty acid compositions |
11/13/2002 | EP1256576A1 Fused imidazolium derivatives |
11/13/2002 | EP1256574A1 Nitrogen-containing compounds having kinase inhibitory activity and drugs containing the same |
11/13/2002 | EP1255753A2 Prodigiosin-derivatives as neoplastic and anti-viral agents |
11/13/2002 | EP1255752A2 Pyrrole substituted 2-indolinone protein kinase inhibitors |
11/13/2002 | EP1255751A2 1,3-dihydro-2h-indol-2-one derivatives and their use as ligands for v1b or v1b and v1a arginine-vasopressin receptors |
11/13/2002 | EP1255740A2 Substituted arylpyrazines |
11/13/2002 | EP1255739A1 3-aminoquinazolin-2,4-dione antibacterial agents |
11/13/2002 | EP1255738A2 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto |
11/13/2002 | EP1255734A1 Isatine derivatives with neurotrophic activity |
11/13/2002 | EP1255536A2 Indolinone derivatives for modulation of c-kit tyrosine protein kinase |
11/13/2002 | EP1068199B1 N-aryloxyethyl-indoly-alkylamines for the treatment of depression |
11/13/2002 | CN1379775A Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
11/13/2002 | CN1379766A Benzoic acid derivatives for treatment of diabetes mellitus |
11/13/2002 | CN1379765A Benzodiazepine derivatives usable as parental metabolic glutamate receptor antagonist |
11/13/2002 | CN1379764A Benzodiazepine derivatives |
11/13/2002 | CN1379762A Beta substituted metalloprotease inhibitors |
11/13/2002 | CN1379668A 3(5)-ureido-pyrazole derivatives, process for their preparation and their use as antitumor agents |
11/12/2002 | US6479531 Gastrin and cholecystokinin receptor ligands |
11/12/2002 | US6479508 Viral polymerase inhibitors |
11/12/2002 | US6479505 6-arylphenanthridines with PDE-IV inhibiting activity |
11/12/2002 | US6479500 Alleviating side effects caused by use of an anti-tumor agent comprising administering 5-chloro-6-(2-iminopyrrolidin-1-yl)methyl-2,4(1h,3h)-pyrimidin edione |
11/12/2002 | US6479494 Arylalkanoyl pyridazines |
11/12/2002 | US6479492 Compounds which inhibit leukocyte adhesion mediated by VLA-4 |
11/12/2002 | US6479490 Treatment of diseases characterized by excess th2 cytokines and/ or an excess ige production. |
11/12/2002 | US6479480 1h-indole derivatives bearing an optionally substituted phenyl moiety at the 2-position of the indole ring system and a methylene-linked heterocyclic moiety at the 3-position of the indole ring system; schizophrenia treatment |
11/12/2002 | US6479479 Azetidine derivatives, their preparation and pharmaceutical compositions containing them |
11/12/2002 | US6479435 Or diaryl sulfides, 1-(4-chloro-2-fluoro-5-(2-pyrimidyloxy)phenyl)-4-difluoromethy l-3-methyl-1,4-dihydro-1,2,4-triazolin-5-one for example |
11/12/2002 | CA2324959C Phthalimido compounds as intermediates for producing substance p receptor antagonists |
11/12/2002 | CA2246839C Pharmaceutical compositions containing ampa receptor antagonists for treating dyskineslas associated with dopamine agonist therapy |
11/12/2002 | CA2144294C (pyrrolidinyl)phenyl carbamates and intermediate compounds, processes for their preparation and their use as medicaments |
11/07/2002 | WO2002088115A1 Novel sulfonamide derivatives, intermediate thereof, its preparation methods, and pharmaceutical composition comprising the same |
11/07/2002 | WO2002088114A2 Heteroaryl ofefinic azacyclic and heteroaryl acetylenic azacyclic compounds for the treatment of cns disorders |
11/07/2002 | WO2002088113A1 Triazole compounds useful in treating diseases associated with unwanted cytokine activity |
11/07/2002 | WO2002088112A1 Heterocyclic compound and antitumor agent containing the same as active ingredient |
11/07/2002 | WO2002088110A1 Quinoline derivative having azolyl group and quinazoline derivative |
11/07/2002 | WO2002088108A1 Triazole compounds useful in treating diseases associated with unwanted cytokine activity |
11/07/2002 | WO2002088107A1 Nitrogenous fused-ring compound having pyrazolyl group as substituent and medicinal composition thereof |
11/07/2002 | WO2002088101A2 Inhibitors of bace |
11/07/2002 | WO2002088097A1 Triazole-derived kinase inhibitors and uses thereof |
11/07/2002 | WO2002088095A1 Fused pyrimidines as antagonists of the corticotropin releasing factor (crf) |
11/07/2002 | WO2002088094A1 2-iminoimidazole derivatives (1) |