Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
02/2003
02/06/2003US20030027832 4-Phenyl-1-piperazinyl, -piperidinyl and -tetrahydropyridyl derivatives
02/06/2003US20030027823 N,N'-disubstituted benzimidazolone derivatives with affinity at the serotonin and dopamine receptors
02/06/2003US20030027812 Useful for treating or preventing a disorder or condition selected from hypertension, depression, anxiety, phobias, post trauma stress, sexual disfunction, eating disorder, obesity, Alzheimer's disease, Parkinson's disease etc.
02/06/2003US20030027797 For therapy of metabolic disorders related to insulin resistance or hyperglycemia
02/06/2003US20030027794 N-heterocyclic derivatives as NOS inhibitors
02/06/2003US20030026763 Using water soluble dyes
02/06/2003US20030026521 Optical interleaver
02/06/2003CA2454903A1 Substituted piperazines as modulators of the melanocortin receptor
02/06/2003CA2453106A1 Macrocyclic metal complexes and use thereof for production of conjugates with biomolecules
02/05/2003EP1282084A2 Method for preparing pyrimidone derivatives with antifungal activity
02/05/2003EP1281709A1 Novel heterocyclic compounds with anti-inflammatory activity
02/05/2003EP1280797A1 Inhibitors of dipeptidyl peptidase iv
02/05/2003EP1280796A1 Pyrimidinyl methyl indole derivatives with antibacterial activity
02/05/2003EP1280795A2 N-substituted carbamoyloxyalkyl-azolium derivatives
02/05/2003EP1280793A2 Cyclic amidine compounds and their use as alpha4beta2 nicotinic acetylcholine receptor ligands
02/05/2003EP1280781A1 5-ht 7 receptor antagonists
02/05/2003EP0984960B1 N-triazolyl-2-indolecarboxamides and their use as cck-a agonists
02/05/2003EP0848706B1 Substituted benzene-fused heterocyclics as neurokinin antagonists
02/05/2003EP0817632B1 Tricyclic carbamate compounds useful for inhibition of g-protein function and for treatment of proliferative diseases
02/05/2003CN1395568A 1,2-diaryl benzimidazole derivative for treating illnesses associated with microglia activation
02/05/2003CN1395563A Isatine derivatives with neurotrophic activity
02/05/2003CN1395562A Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
02/05/2003CN1395485A Water soluble prodrugs of azole compounds
02/05/2003CN1100777C N-heterocyclic derivatives as NOS inhibitor
02/05/2003CN1100761C Benzyloxy substituted aryl copounds and their use as fungicides and insecticides
02/05/2003CN1100540C Protein tyrosine kinase aryl and heteroaryl quinazoline compounds having selective inhibition of HER-2 autophosphorylation properties
02/04/2003US6515133 Certain diaryl imidazoles act as partial agonists or antagonists for NPY receptors, in particular NPY 5 receptors. They are of use, for example in treating loss of appetite. Such compounds bear aryl groups in the 2 position.
02/04/2003US6515124 Dehydroamino acids
02/04/2003US6515013 For diseases or conditions caused by or exacerbated by histamine-3 receptor activity
02/04/2003US6515011 Anticoagulants
02/04/2003US6515003 Useful in the treatment of diseases related to lipid and carbohydrate metabolism
02/04/2003US6514998 For controlling animal pests and harmful fungi
02/04/2003US6514993 Serotonin 5-HT1A and dopamin D2 receptor ligands
02/04/2003US6514990 Pharmaceutically active compounds and methods of use
02/04/2003US6514981 Methods of modulating tyrosine protein kinase function with indolinone compounds
02/04/2003US6514977 For treating p38 kinase mediated disorders
02/04/2003US6514975 Anti-inflammatory piperazinyl-benzyl-tetrazole derivatives and intermediates thereof
02/04/2003US6514974 Pyrido-, pyrimido-, pyridazo- and pyrazo- pyridazines having angiogenesis inhibiting activity
02/04/2003US6514971 Cinnoline derivatives and use as medicine
02/04/2003US6514970 Urotensin-II receptor antagonists
02/04/2003US6514968 Treating a disease or condition in a mammal wherein the 5-HT receptor is implicated and modulation of 5-HT function is desired comprising
02/04/2003US6514964 Treating diseases, conditions or disorders mediated by integrin receptors, such as vitronectin and fibronectin receptors
02/04/2003CA2271566C Substituted phenyl pyrimidines useful in the treatment of cns disorders
01/2003
01/31/2003CA2396020A1 Imidazolidinone derivatives
01/30/2003WO2003008410A2 Polypyrroles as agents for treating cancer, treating viral diseases and causing immunosuppression
01/30/2003WO2003008409A1 Quinoline derivatives and their use as tyrosine kinase inhibitors
01/30/2003WO2003008407A2 Phenylsulfonyl-1,3-dihydro-2h-indole-2-one derivatives, their preparation and their therapeutic use
01/30/2003WO2003008405A1 Compounds derived from diaminopyrazole substituted by a heteroaromatic radical and their use in oxidation dyeing of keratinous fibres
01/30/2003WO2003008387A1 Compounds useful for treatment or prevention of disease mediated by alpha-2b-adrenoceptor
01/30/2003WO2003008377A1 Prostaglandin analogues_as ep4 receptor agonists
01/30/2003WO2003007959A1 Quinoxaline derivatives which have parp inhibitory action
01/30/2003WO2003007958A1 Tetrahydroquinoxalines acting as bradykinin antagonists
01/30/2003WO2003007945A1 Viral polymerase inhibitors
01/30/2003WO2003007883A2 Acylsemicarbazides as cyclin dependent kinase inhibitors useful as anti-cancer and anti-proliferative agents
01/30/2003WO2002088079A3 Dual inhibitors of pde 7 and pde 4
01/30/2003US20030023098 Compounds and method of treatment having agonist-like activity selective at alpha 2B or 2B/2C adrenergic receptors
01/30/2003US20030023087 Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use
01/30/2003US20030023031 Acryloyl substituted distamycin derivatives, process for preparing them, and their use as antitumor and antiviral agents
01/30/2003US20030022927 Novel benzimidazole derivatives
01/30/2003US20030022907 Anxiolytic agents and analgesics
01/30/2003US20030022905 Prevention and/or therapy of ischaemia and reperfusion damage; poly(ADP-ribose)-synthetase inhibitors
01/30/2003US20030022885 Pyrazole compounds useful as protein kinase inhibitors
01/30/2003US20030022884 Heterocycle derivatives and drugs
01/30/2003US20030022794 Bioactive pesticides
01/30/2003US20030019050 Novel cationic 4-hydroxyindoles, their use for the oxidation dyeing of keratinous fibers, dyeing compositions, and methods of dyeing
01/30/2003CA2454187A1 Compounds useful for treatment or prevention of disease mediated by alpha-2b-adrenoceptor
01/30/2003CA2454007A1 Tetrahydroquinoxalines acting as bradykinin antagonists
01/30/2003CA2453636A1 Polypyrroles as agents for treating cancer, treating viral diseases and causing immunosuppression
01/30/2003CA2453594A1 Acylsemicarbazides as cyclin dependent kinase inhibitors useful as anti-cancer and anti-proliferative agents
01/30/2003CA2451392A1 Prostaglandin analogues as ep4 receptor agonists
01/30/2003CA2450437A1 1-phenylsulphonyl-1,3-dihydro-2h-indol-2-one derivatives, their preparation and their therapeutic application
01/29/2003EP1279673A1 Imidotriazine derivatives
01/29/2003EP1279666A1 1-diphenylmethyl-pyrazole derivatives as opioid receptor ligands
01/29/2003EP1278748A2 Inhibitors of human phosphatidyl-inositol 3-kinase delta
01/29/2003EP1278743A1 Novel anti-infectives
01/29/2003EP1278740A1 Hydroxyphenyl-piperazinyl-methyl-benzamide derivatives for the treatment of pain
01/29/2003EP1278735A1 2,4-di(hetero-)arylamino(-oxy)-5-substituted pyrimidines as antineoplastic agents
01/29/2003EP1278728A1 Pyrrolidine and piperidine derivatives and their use for the treatment of neurodegenerative disorders
01/29/2003EP1028948B1 Phenyl-alkyl-imidazoles as h3 receptor antagonists
01/29/2003CN1394205A Indazole compounds, pharmaceutical compositions, and their use for mediating or inhibiting cell proliferation
01/29/2003CN1393444A Compound for treating impotence
01/29/2003CN1100055C Piperazine and piperidine compounds
01/29/2003CN1100046C 喹唑啉衍生物 Quinazoline derivatives
01/28/2003WO2002010155A1 Substituted aryl ketones and their use as herbicides
01/28/2003US6512001 D-proline derivatives
01/28/2003US6512000 Aminocarbonyl-substituted benzimidazoles having tryptase-inhibitory activity
01/28/2003US6511998 Pyrazole carboxamides useful for the treatment of obesity and other disorders
01/28/2003US6511978 Pyrrole derivatives useful for farnesyl transferase inhibitors and their preparations
01/28/2003US6511941 Synergistic mixture
01/28/2003US6511663 Tri- and tetra-valent monospecific antigen-binding proteins
01/28/2003CA2417385A1 Substituted aryl ketones and their use as herbicides
01/28/2003CA2083534C Indolopyrrolocarbazole derivatives
01/24/2003CA2394209A1 1-diphenylmethyl-pyrazole derivatives as opioid receptor ligands
01/23/2003WO2003006506A2 Protease inhibitor conjugates and antibodies useful in immunoassay
01/23/2003WO2003006459A1 Piperazine oxime derivatives having nk-1 receptor antagonistic activity
01/23/2003WO2003006447A2 Interaction inhibitors of tcf-4 with beta-catenin
01/23/2003WO2003006443A2 2- 4-(naphtalin-2-yl)-thiazol-2-ylaminocarbonyl benzoic acid and 2- 4-(naphtalin-2-yl)-pyrimidin-2-ylaminocarbonyl benzoic acid and additional compounds serving as telomerase inhibitors for use in tumor therapy
01/23/2003WO2003006437A1 Imidazole derivatives as adenosine deaminase inhibitors
01/23/2003WO2003006423A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003WO2003006012A1 Compounds and methods for the inhibition of trypanosoma cruz i