Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
08/2002
08/08/2002WO2002018432A3 Protein extracted from the intestines of vertebrates, which absorbs cholesterol, and the use of this protein for identifying inhibitors of intestinal cholesterol transport
08/08/2002WO2002010140A3 Imidazolyl derivatives
08/08/2002WO2002000631A3 Benzhydryl derivatives
08/08/2002WO2001098268A3 Piperidine amides as modulators of chemokine receptor activity
08/08/2002WO2001094312A3 Indolinone derivatives as protein kinase/phosphatase inhibitors
08/08/2002WO2001093840A3 Ligands of integrin receptors
08/08/2002WO2001081334A3 Cyclic amidine compounds and their use as alpha4beta2 nicotinic acetylcholine receptor ligands
08/08/2002WO2001009090A3 Hydantoin, thiohydantoin, pyrimidinedione and thioxopyrimidinone derivatives, preparation method and use as medicines
08/08/2002US20020107398 Microbicides in crop protection
08/08/2002US20020107392 Quinolinone derivatives
08/08/2002US20020107275 Novel crystal and solvate forms of ondansetron hydrochloride and processes for their preparation
08/08/2002US20020107273 Aryl or heteroaryl fused imidazole compounds as anti-inflammatory and analgesic agents
08/08/2002US20020107263 Squaric acid derivatives
08/08/2002US20020107255 Potent and selective inhibitors of chemokine binding to its receptor CCR1 found on inflammatory and immunomodulatory cells (preferably leukocytes and lymphocytes).
08/08/2002CA2672805A1 Pyrimidine derivatives
08/08/2002CA2454215A1 Polymers
08/08/2002CA2438594A1 Diazocine derivatives and their use as tryptase inhibitors
08/08/2002CA2436133A1 Receptor selective cannabimimetic aminoalkylindoles
08/08/2002CA2436130A1 Substituted indoles and their use as integrin antagonists
08/07/2002EP1229035A1 Imine intermediates for the preparation of trisubstituted imidazole compounds with multiple therapeutic properties
08/07/2002EP1228760A2 5-membered heterocycle derivatives, production thereof and use thereof as medicaments
08/07/2002EP1228759A2 Pharmaceutical compositions containing a taxane having a furyl or thienyl substituted side-chain
08/07/2002EP1228071A1 Pharmaceutically active isoindoline derivatives
08/07/2002EP1228067A1 5-membered n-heterocyclic compounds with hypogylcemic and hypolipidemic activity
08/07/2002EP1228065A1 (indol-3-yl)-cycloalkyl]-3-substituted azetidines for the treatment of central nervous system disorders
08/07/2002EP1228064A1 N-aryl-(homopiperazinyl)-cyclohexyl amines as 5-ht transporters
08/07/2002EP1228063A2 Substituted pyridines and pyridazines with angiogenesis inhibiting activity
08/07/2002EP1228061A1 Dipeptidyl peptidase iv inhibitors and methods of making and using dipeptidyl peptidase iv inhibitors
08/07/2002EP1228060A1 Arylalkane, arylalkene and aryl azaalkane, medicaments containing said compounds and method for the production thereof
08/07/2002EP1228051A1 Semicarbazone derivatives and their use as thrombopoietin mimetics
08/07/2002EP1228044A2 Pyrrolo imidazole derivatives and their use as medicaments
08/07/2002EP1228041A2 Indole derivatives and their use as 5ht2a ligands
08/07/2002EP1227847A2 Inhibitors of the endothelin signalling pathway and alphavbeta3 integrin receptor antagonists for combination therapy
08/07/2002EP1227805A2 Mediators of hedgehog signaling pathways, compositions and uses related thereto
08/07/2002EP0874843B1 Substituted 4-(1h-benzimidazol-2-yl) 1,4]diazepanes useful for the treatment of allergic diseases
08/07/2002CN1362957A C17 heterosubustituted acetate taxanes as antitumor agents
08/07/2002CN1362954A Sulfamato hydroxamic acid metalloprotease inhibitor
08/07/2002CN1362953A Pyrazole compositions useful as inhibitors of ERK
08/07/2002CN1362640A Silver-halides photo-sensitive emulsion layer with reinforced photographic photosensibility
08/07/2002CN1088702C Disubstituted bicyclic heterocycles, their production and use as medicaments
08/06/2002US6429288 Peptides containing an arginine mimetic for the treatment of bone metabolic disorders, their production, and drugs containing these compounds
08/06/2002US6429205 Anticoagulants
08/01/2002WO2002059117A1 Piperazine- and piperidine-derivatives as melanocortin receptor agonists
08/01/2002WO2002059112A2 Pyrazole compounds useful as protein kinase inhibitors
08/01/2002WO2002059111A2 Pyrazole compounds useful as protein kinase inhibitors
08/01/2002WO2002059110A1 Pyrimidineamines as angiogenesis modulators
08/01/2002WO2002059109A2 Naphthostyril derivatives and their use as inhibitors of cyclin- dependent kinases
08/01/2002WO2002059108A1 Melanocortin receptor agonists
08/01/2002WO2002059095A1 Melanocortin receptor agonists
08/01/2002WO2002058730A2 Compositions for treatment of ocular neovascularization
08/01/2002WO2002058704A1 Imidazolyl derivatives as corticotropin releasing factor inhibitors
08/01/2002WO2002058695A1 (halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents
08/01/2002WO2002058690A2 Methods for the treatment of diseases using malonyl-coa decarbox ylase inhibitors
08/01/2002WO2002028861A3 Methods and compounds for treating proliferative diseases
08/01/2002US20020103384 Therapeutically active and selective heterocyclic compounds that are inhibitors of the enzyme DPP-IV
08/01/2002US20020103381 Useful in pharmaceutical industry, such as antiinflammatory or antiarthritic agents; solid phase synthesis; esterification of a hydroxylated solid support, treating wtih trimethylsilyldiazomethane, deprotecting
08/01/2002US20020103247 Indole and dihydroindole derivatives
08/01/2002US20020103245 1-aryl or heteroaryl substituted 5-amino-4 carbonylpyrazole derivatives; antiinflammatory agents
08/01/2002US20020103243 Sulfamoyl compounds and agricultural and horticultural fungicides
08/01/2002US20020103235 Substituted imidazoles as dual histamine H1 and H3 agonists or antagonists
08/01/2002US20020103234 Heterocycl-containing carboxylic acid derivative and drug containing the same
08/01/2002US20020103229 Indazole derivatives as JNK inhibitors and compositions and methods related thereto
08/01/2002US20020103208 Useful in treatment of anxiety disorders, affective disorders such as depression, psychosis and schizophrenia, Parkinson's disease
08/01/2002US20020103205 Muscarinic antagonists
08/01/2002US20020103202 Heteroaryl-phenyl substituted factor Xa inhibitors
08/01/2002US20020103201 Selective NPY (Y5) antagonists (triazines)
08/01/2002US20020103198 Acylamino cyclopropane derivatives
08/01/2002US20020103197 For use in protecting human and animal hair and skin against damaging action of UV radiation
08/01/2002US20020103185 Pyrazole derivatives
08/01/2002US20020103184 Cyclic malonamides as inhibitors of a beta protein production
08/01/2002US20020103164 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith
08/01/2002US20020102608 Library of indolinone compounds for use in the treatment of cancer
08/01/2002US20020102597 Methods for selecting compounds for treating ischemia-related cellular damage
08/01/2002US20020102435 Electroluminescence device, cyclic azine compound and production process of cyclic azine dye
08/01/2002CA2434558A1 Imidazolyl derivatives as corticotropin releasing factor inhibitors
08/01/2002CA2432988A1 Melanocortin receptor agonists
08/01/2002CA2432985A1 Piperazine- and piperidine-derivatives as melanocortin receptor agonists
08/01/2002CA2431996A1 Melanocortin receptor agonists
08/01/2002CA2431904A1 (halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents
07/2002
07/31/2002EP1227093A2 Beta-lactams useful for preparation of taxanes having furyl or thienyl substituted side-chain
07/31/2002EP1227092A2 Isonitrile intermediates for the preparation of tri-substituted imidazole compounds with multiple therapeutic properties
07/31/2002EP1227091A2 Formamide intermediates for the preparation of tri-substituted imidazole compounds with multiple therapeutic properties
07/31/2002EP1226435A1 Axor35, a g-protein coupled receptor
07/31/2002EP1226141A1 Heterocyclic substituted pyrazolones
07/31/2002EP1226138A1 Fab i inhibitors
07/31/2002EP1226129A1 Methods and compositions utilizing quinazolinones
07/31/2002EP1226128A1 New pyrimidine-2,4,6-trione derivatives, processes for their production and pharmaceutical agents containing these compounds
07/31/2002EP1226126A1 Pyrimidine derivatives
07/31/2002EP1226123A1 Cyano compounds as factor xa inhibitors
07/31/2002EP1226122A1 Bicyclic vasopressin agonists
07/31/2002EP1226116A1 Processes for the preparation of sumatriptan and related compounds
07/31/2002EP1060165A4 Method for preparing n-substituted heterocyclic derivatives using a phase-transfer catalyst
07/31/2002CN1361773A Substituted 3-pyridyl-4-arylpyrroles, and related therapeutic and prophylactic methods
07/31/2002CN1361770A Heteroaromatic ring compounds
07/31/2002CN1361769A Substituted 2-aryl-1,2,4-triazine-3,5-di(thi) one
07/31/2002CN1088459C 1,4-disubstituted piperazines
07/30/2002US6426413 Inhibitors of caspases
07/30/2002CA2344707C N-substituted cycloalkyl and polycycloalkyl alpha-substituted trp-phe- and phenethylamine derivatives
07/30/2002CA2110806C 4-(1h-pyrrol-1-yl)imidazoles with angiotensin ii antagonist activity
07/25/2002WO2002057259A2 Pyrazole compounds useful as protein kinase inhibitors