Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
01/2003
01/23/2003WO2003005824A2 Substituted 3-heteroaryl (amino-or-oxy)-pyrrolidin-2-ones, method for the production thereof and use thereof as herbicides or as plant growth regulators
01/23/2003WO2002050066A3 Pyrazole compounds useful as protein kinase inhibitors
01/23/2003WO2002046171A3 Anilinopyrimidine derivatives as ikk inhibitors and compositions and methods related thereto
01/23/2003WO2002036562A3 1-aryl- or 1-alkylsulfonyl-heterocyclylbenzazoles as 5-hydroxytryptamine-6 ligands
01/23/2003US20030018197 Administering a therapeutically effective amount of a pyrrazole sulfide or ether compound to treat the human immunodeficiency virus infection
01/23/2003US20030018189 Cyclic polyamines having total 9-24 members which have activity in against HIV-infected cells as well as other biological activity related to binding of ligands to chemokine receptors
01/23/2003US20030018062 Deacetylase inhibitors
01/23/2003US20030018059 Antiinflammatory agents; antihistamines; antiallergens
01/23/2003US20030018051 Pyrazole derivatives - p38 MAP kinase inhibitors
01/23/2003US20030018035 Central nervous system disorders
01/23/2003US20030018034 Piperazine compounds and medicinal use thereof
01/23/2003US20030018029 Tyrosine kinase inhbitor; antiproliferative agents
01/23/2003US20030018025 Psychological disorders, antidepressants, Parkinson's disease
01/23/2003CA2453503A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003CA2453396A1 Compounds and methods for the inhibition of trypanosoma cruzi
01/23/2003CA2453175A1 Interaction inhibitors of tcf-4 with beta-catenin
01/23/2003CA2449243A1 Protease inhibitor conjugates and antibodies useful in immunoassay
01/23/2003CA2446726A1 Piperazine oxime derivatives having nk-1 receptor antagonistic activity
01/22/2003WO2002010131A1 Pyrrole derivatives
01/22/2003EP1277751A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277749A1 2- and 2,5-substituted phenylketo enols
01/22/2003EP1277741A1 Cyclic compounds
01/22/2003EP1277738A1 Condensed heteroaryl derivatives
01/22/2003EP1277735A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277734A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277733A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1276732A1 Amides of r-2-(aminoaryl)-propionic acids for use in theprevention of leucocyte activation"
01/22/2003EP1276727A1 Novel amino carboxy alkyl derivatives of barbituric acid
01/22/2003EP1276723A2 Pyrazole compounds having anti proliferative activity
01/22/2003EP1276721A2 Methylation of indole compounds using dimethyl carbonate
01/22/2003EP1107738A4 Novel pharmaceutical salt form
01/22/2003EP1006114B1 Pyrazole derivatives and cox inhibitors containing them
01/22/2003EP0898562B1 Hydroxamic acid derivatives for use with the treatment of diseases related to connective tissue degradation
01/22/2003EP0729465B1 Pyrone derivatives as protease inhibitors and antiviral agents
01/22/2003CN1392875A Condensed azepines as vasopressino agonists
01/22/2003CN1392874A Cyclic amidine compounds
01/22/2003CN1099413C Certain fused N-pyrrolylaniline: new class of GABA brain receptor ligand
01/22/2003CA2416946A1 Pyrrole derivatives
01/21/2003US6509341 The invention relates to carboxylic acid derivatives of formula (I), wherein the substituents have the meaning as commented in the description. It also relates to the production and use of same as endothelin receptor antagonists.
01/21/2003US6509340 Amide and urea derivatives as 5-HT reuptake inhibitors and as 5-HT1B/1D ligands
01/21/2003US6509336 Imidazolyl derivatives
01/21/2003US6509328 Glutamate receptor antagonists
01/21/2003US6508957 Fluorescent maleimides and uses thereof
01/21/2003CA2078106C Treatment of central nervous system disorders with imidazole angiotensin-ii receptor antagonists
01/16/2003WO2003004490A1 High molecular weight hydroxyphenylbenzotriazole uv-absorbers for thin film applications
01/16/2003WO2003004489A1 Compositions and methods for inhibiting prenyltransferases
01/16/2003WO2003004488A1 Indazole benzimidazole compounds as tyrosine and serine/threonine kinase inhibitors
01/16/2003WO2003004476A1 Aminoalkyl-substituted benzotriazoles and triazoles as metal deactivators
01/16/2003WO2003004027A1 Substituted anilinic piperidines as mch selective antagonists
01/16/2003WO2003004023A1 1-alkyl-2-aryl-benzimidazole derivatives, their use for producing medicaments and pharmaceutical preparations containing said derivatives
01/16/2003WO2003004020A1 Heteroaryl carboxylic acid amides, the production thereof and the use of the same as inhibitors of the microsomal triglyceride transfer protein (mtp)
01/16/2003WO2002051837A3 Heterocyclindazole and azaindazole compounds as 5-hydroxytryptamine-6 ligands
01/16/2003WO2002050062A3 Benzimidazole and pyridylimidazole derivatives as ligands for gaba receptors
01/16/2003WO2002012196A3 Lactam compounds and their use as inhibitors of serine proteases and method
01/16/2003US20030013886 Such as (E)-1-(2-Pyridyl)-2-styryl-1H-benzimidazole; antiinflammatory and analgesic agents; prostaglandin inhibitors
01/16/2003US20030013875 3-azabicyclo[3.1.0]hexane derivatives useful in therapy
01/16/2003US20030013724 Novel prolines as antimicrobial agents
01/16/2003US20030013721 Antiinflammatory agents; immunology; cardiovascular disorders; rheumatic disorders
01/16/2003US20030013712 Antiinflammatory agents
01/16/2003US20030013700 Thrombin inhibitors
01/16/2003CA2454613A1 Substituted anilinic piperidines as mch selective antagonists
01/15/2003EP1275646A1 Indolylpyrrole derivatives and cell death inhibitors
01/15/2003EP1275644A1 Benzenesulfonamide derivatives, process for their preparation and pharmaceutical compositions containing them
01/15/2003EP1275391A1 Pharmaceutical compositions containing irbesartan and a diuretic
01/15/2003EP1274706A1 Pyrazoles for inhibiting protein kinases
01/15/2003EP1274702A1 Process for the synthesis of a known tetrazol derivative
01/15/2003EP1274692A1 Quinazoline compounds
01/15/2003EP1274682A2 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
01/15/2003EP1274424A1 Compounds and methods
01/15/2003EP1023265B1 Azetidinone derivatives for the treatment of hcmv infections
01/15/2003EP0925287B1 Heterocyclic metalloprotease inhibitors
01/15/2003EP0851756B1 Use of ondansetron in the manufacture of a medicament for the treatment of tremor
01/15/2003EP0820451B1 Novel heterocyclic compounds
01/15/2003EP0729468B1 Non-peptide tachykinin receptor antagonists
01/15/2003EP0722442B1 Polyazacycloalkanes as dichelants
01/15/2003CN1391564A Chemical compounds
01/15/2003CN1391563A Therapeutic quinazoline derivatives
01/15/2003CN1391562A Quinazoline derivatives as pharmaceuticals
01/15/2003CN1391557A 6-position substituted indoline, production and use thereof as medicament
01/15/2003CN1391555A Benzamides and related inhibitors of factor Xa
01/15/2003CN1391474A 5-membered heterocycle derivatives, production thereof and use as medicaments
01/15/2003CN1391473A VLA-4 inhibitor compounds
01/15/2003CN1098838C Substituted N-(indole-2-carbonyl)-beta-alanimamides and derivatives as antidiabetic agents
01/14/2003US6506906 Preparation and use of bifunctional molecules having DNA sequence binding specificity
01/14/2003US6506901 1-(9H-Carbazol-4-yloxy)-3-((1-(7-trifluoromethyl-quinolin-4-yl) -piperidin-4-lmethyl)-amino)-propan-2-ol, for example; treating diabetes, urinary continence, atherosclerosis, gastrointestinal disorders, glaucoma
01/14/2003US6506787 Aids therapy
01/14/2003US6506779 Acetylene derivatives as anti-inflammatory/analgesic agents
01/14/2003US6506770 Antiviral compounds
01/14/2003US6506754 Compounds as anticoagulants
01/14/2003US6506748 Aromatic heterocyclic compounds as antiinflammatory agents
01/14/2003US6506747 Method of treating an inflammatory disease which comprises administering to a patient in need of such treatment-a N-(4-(5-Ethyl-3-pyridin-3-yl-pyrazol-1-yl)phenyl)pyridine-3-carboxamide;
01/14/2003US6506738 Treatment of viral infections. More particularly, the invention provides benzimidazolone derivatives for the treatment of respiratory syncytial virus infection.
01/09/2003WO2003002561A1 N-aroyl cyclic amine derivatives as orexin receptor antagonists
01/09/2003WO2003002558A1 Remedial agent for viral infectious disease
01/09/2003WO2003002553A2 Fluoropyrrolidines as dipeptidyl peptidase inhibitors
01/09/2003WO2003002552A1 Novel indole derivatives
01/09/2003WO2003002544A1 N-heterocyclic inhibitors of tnf-alpha expression
01/09/2003WO2003002542A1 N-heterocyclic inhibitors of tnf-alpha expression
01/09/2003WO2003002540A1 Cyclic diamine compound having five-membered cyclic group
01/09/2003WO2003002533A1 Triamide-substituted indoles, benzofuranes and benzothiophenes as inhibitors of microsomal triglyceride transfer protein (mtp) and/or apolipoprotein b (apo b) secretion