Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587) |
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06/03/2003 | CA2223625C Substituted n-(indole-2-carbonyl-) amides and derivatives as glycogen phosphorylase inhibitors |
05/30/2003 | WO2003044016A1 3-SUBSTITUTED OXINDOLE β3 AGONISTS |
05/30/2003 | WO2003044014A1 Indole-2-carboxamides as factor xa inhibitors |
05/30/2003 | WO2003044010A1 Nitrogenous tetrahydropyridyl-alkyl-heterocycles with tnf activity |
05/30/2003 | WO2003043993A1 5-phenylpyrimidines, agents comprising the same, method for production and use thereof |
05/30/2003 | WO2003043985A1 Heterocyclic compounds and methods of use |
05/30/2003 | WO2003043983A1 Piperazine derivatives destabilising androgen receptors |
05/30/2003 | WO2003043981A1 2-(3-sulfonylamino-2-oxopyrrolidin-1-yl)propanamides as factor xa inhibitors |
05/30/2003 | WO2003043980A1 Azetidinyl diamines useful as ligands of the nociceptin receptor orl-1 |
05/30/2003 | WO2003043632A2 Use of bisindolmaleimide and gemcitabine for the treatment of cancer |
05/30/2003 | WO2003018552A3 Aromatic and heteroaromatic acid halides for synthesizing polyamides |
05/30/2003 | WO2003010141A3 Hepatitis c virus polymerase inhibitors with a heterobicyclic structure |
05/30/2003 | WO2003005824B1 Substituted 3-heteroaryl (amino-or-oxy)-pyrrolidin-2-ones, method for the production thereof and use thereof as herbicides or as plant growth regulators |
05/30/2003 | WO2002070739A3 Assay for identifying inhibitors of the rna dependent rna polymerase (ns5b) of hcv |
05/30/2003 | WO2002036116A9 Tripeptidyl peptidase inhibitors |
05/30/2003 | WO2002016313A3 Integrin receptor inhibitors |
05/30/2003 | CA2465807A1 Use of bisindolmaleimide and gemcitabine for the treatment of cancer |
05/29/2003 | US20030100770 D-proline derivatives |
05/29/2003 | US20030100769 Such s 2-(6-chloro-3-pyridyl)-2-imidazoline which has good affinity for and activate alpha-4-beta-2-nicotinic acetyl-choline receptors; for treatment and prevention of neuro-degenerative disorders (Alzheimer's/Parkinson's disease) |
05/29/2003 | US20030100757 2-(4-aryl or heteroaryl-piperazin-1-ylmethyl)-1H-indole derivatives interacting with the dopamine D4 receptor |
05/29/2003 | US20030100755 For example (2S, 3S, 5S)-2-(2,6-dimethylphenoxyacetyl)amino-3-hydroxy-5-(2S-(1-tetrahydro-pyrimid-2-onyl)-3-methyl butanoyl)amino-1,6-diphenylhexane; HIV therapy |
05/29/2003 | US20030100599 2-amino-fluorene derivatives useful for prophylactic and/or therapeutic treatment of diseases and conditions associated with alpha 4 intergrins or their ligands |
05/29/2003 | US20030100588 Indole-type inhibitors of p38 kinase |
05/29/2003 | US20030100582 Benzimidazole compounds for regulating IgE |
05/29/2003 | US20030100571 Such as 2-((6-(((4-(3,4-dimethoxyphenyl)methyl)amino)-7-ethyl-7H-purin-2-yl)amino) -4,5-methyl-N-phenyl-5-thiazole-carboxamide for treatment of lymphocyte mediated diseases such as transplant rejection and graft versus host disease |
05/29/2003 | US20030100558 Such as 4-(4-fluorophenyl)-5-(2-phenylmethylamino)pyrimidin-4-yl)-1-ethoxymethyl -(1,2,3)triazole for inhibition of release of inflammatory interleukins; for treatment of osteoarthritis, rheumatoid arthritis, and congestive heart failure |
05/29/2003 | US20030100555 Prodrugs of a 3-(pyrrol-2-ylmethylidene)-2-indolinone derivatives |
05/29/2003 | US20030100554 Pyrazole derivatives |
05/29/2003 | US20030100088 Protease inhibitor conjugates and antibodies useful in immunoassay |
05/29/2003 | US20030098440 Adhesion promoters containing benzotriazoles |
05/28/2003 | EP1314733A1 Indole-2-carboxamides as factor Xa inhibitors |
05/28/2003 | EP1314732A2 Substituted pyrimidine compounds and their use |
05/28/2003 | EP1314731A2 Substituted pyrimidine compounds and their use |
05/28/2003 | EP1314728A1 Pyridyl and pyrimidinyl imines as intermediates for imidazole derivatives |
05/28/2003 | EP1313713A2 4-pyrimidinamine derivatives, pharmaceutical compositions and related methods |
05/28/2003 | EP1313712A2 Process and intermediates for preparing retroviral protease inhibitors |
05/28/2003 | EP1313711A2 Indazole derivatives as jnk inhibitors |
05/28/2003 | EP1313710A1 Pyrazole derivatives and their use as protein kinase inhibitors |
05/28/2003 | EP1313704A2 Compounds useful as insecticides, compounds useful as acaricides, and processes to use and make same |
05/28/2003 | EP1161428B1 Pyrimidine compounds |
05/28/2003 | EP1100777B1 Sulfurated distamycin derivatives, process for preparing them, and their use as antitumor agents |
05/28/2003 | EP0973763B1 Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and pharmaceutical compositions containing same |
05/28/2003 | EP0966464B1 Substituted 2,4-diaminopyrimidines |
05/28/2003 | CN1420889A Pharmaceutically active isoindoline derivs. |
05/28/2003 | CN1420883A N-aryl-(homopiperazinyl) cyclohexyl amines as 5-HT transporters |
05/28/2003 | CN1420882A Substd. oxoazaheterocyclyl compounds |
05/28/2003 | CN1420879A Substd. pyridines and pyridazines with angiogenesis inhibiting activity |
05/28/2003 | CN1420873A Substd. phenyluracils |
05/28/2003 | CN1420114A 2,3-disubstd. -4(3H)-quinazolones |
05/28/2003 | CN1109675C Arylpyrimidine derivs. |
05/27/2003 | US6569880 Bis(benzimidazole) derivatives serving as potassium blocking agents |
05/27/2003 | US6569871 Substituted imidazole compounds |
05/27/2003 | US6569868 Imidazoly 2-indolinones as anticarcinogenic, -diabetic, -arthritic, -proliferative and inflammatory agents; fibrosis; autoimmune disorder, angiogenesis, restenosis, psoriasis, osteoarthritis and rheumatoid arthritis |
05/27/2003 | US6569856 Treatment of feeding disorders, obesity, bulimia nervosa, sexual/reproductive disorders, depression, epileptic seizure, cardiovascular disorders, sleep disturbances |
05/27/2003 | US6569855 Particularly zinc metalloprotease activity for treatment of variety of maladies involving inflammation and/or tissue integrity |
05/27/2003 | US6569851 Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting β-amyloid peptide release and/or its synthesis by use of such compounds |
05/27/2003 | US6569849 N-Substituted azaheterocyclic compounds |
05/27/2003 | US6569847 Inhibitors of cathepsins for treating muscular dystrophy, osteoporosis, rheumatoid arthritis, neuronal or cardiac ischaemia, allergy, or Chagas disease |
05/27/2003 | US6569402 Vitronectin receptor antagonist pharmaceuticals |
05/27/2003 | CA2213054C Novel bis(imido) derivatives, a process for their preparation and pharmaceutical compositions containing them |
05/27/2003 | CA2066104C Benzazepine derivatives as vasopressin antagonists |
05/22/2003 | WO2003042234A2 Non-peptide somatostatin receptor ligands |
05/22/2003 | WO2003042211A1 Phenyl substituted triazoles and their use as selective inhibors of akl5 kinase |
05/22/2003 | WO2003042208A1 Pyrazole derivatives as psychopharmaceuticals |
05/22/2003 | WO2003042205A1 Piperidine derivatives and their use as modulators of chemokine receptor activity (especially ccr5) |
05/22/2003 | WO2003042188A1 Triazole derivative and medicinal composition containing the same |
05/22/2003 | WO2003042187A1 Serin protease inhibitors |
05/22/2003 | WO2003042181A1 4,4-difluoro-1,2,3,4-tetrahydro-5h-1-benzazepine derivatives or salts thereof |
05/22/2003 | WO2003042176A1 Azabicyclo compound, matrix metalloprotease inhibitor, and skin preparation |
05/22/2003 | WO2003042175A1 Sulphonamide derivatives, the preparation thereof and the application of same as medicaments |
05/22/2003 | WO2003042174A1 Cannabinoid receptor ligands |
05/22/2003 | WO2003042173A1 Nk1 antagonists |
05/22/2003 | WO2003041715A1 Substituted 1,4-benzodiazepines and uses thereof for the treatment of cancer |
05/22/2003 | WO2003041714A1 Benzotriazepines as gastrin and cholecystokinin receptor ligands |
05/22/2003 | WO2003041658A2 Process for the preparation of 3,7-disubstituted-2,3,4,5- tetrahydro-1h-1,4-benzodiazepine compounds |
05/22/2003 | WO2003041644A2 Method to treat cystic fibrosis |
05/22/2003 | WO2003022280A3 3-glyoxlylamideindoles for treating cancer |
05/22/2003 | WO2003007883A3 Acylsemicarbazides as cyclin dependent kinase inhibitors useful as anti-cancer and anti-proliferative agents |
05/22/2003 | WO2002100327A3 Substituted 1-benzazepines and derivatives thereof |
05/22/2003 | WO2002044168A3 Indole-type inhibitors of p38 kinase |
05/22/2003 | US20030097004 3,4-Di-substituted cyclobutene-1,2-diones as CXC chemokine receptor antagonists |
05/22/2003 | US20030096990 Reacting phenylisocyanate compound with substituted hydrazono ester compound to form phenyl-2,4(1H,3H)-pyrimidinedione derivatives |
05/22/2003 | US20030096852 Inhibiting binding interaction between hGH (human growth hormone) or a mutant thereof and an hGH binding protein or receptor in mammal administering benzimidazole compound |
05/22/2003 | US20030096836 2-Aroylimidazole compounds for treating cancer |
05/22/2003 | US20030096830 Pyrrolo(3,2-d)pyrimidin-7-yl)-1,4-imino-D-ribitol derivatives; for suppression of T-cell function |
05/22/2003 | US20030096827 Heterocyclic amine derivatives; for treating an inflammatory or immune disease, a cardiovascular disease, or a neurodegenerative condition |
05/22/2003 | US20030096825 Antiviral activity; treatment of HIV and AIDS |
05/22/2003 | US20030096820 Nitrogen containing heterobicycles as factor Xa inhibitors |
05/22/2003 | US20030095958 Inhibiting beta amyloid converting enzyme responsible for A beta peptide cleavage to treat Alzheimer's Disease, Down's Syndrome, etc. |
05/22/2003 | CA2467267A1 Phenyl substituted triazoles and their use as selective inhibors of akl5 kinase |
05/22/2003 | CA2467081A1 Pyrazole derivatives as psychopharmaceuticals |
05/22/2003 | CA2466955A1 Benzotriazepines as gastrin and cholecystokinin receptor ligands |
05/22/2003 | CA2466665A1 Method to treat cystic fibrosis |
05/22/2003 | CA2466465A1 Nk1 antagonists |
05/22/2003 | CA2466440A1 Cannabinoid receptor ligands |
05/22/2003 | CA2466055A1 Substituted 1,4-benzodiazepines and uses thereof for the treatment of cancer |
05/22/2003 | CA2464347A1 Piperidine derivatives and their use as modulators of chemokine receptor activity (especially ccr5) |
05/22/2003 | CA2464069A1 4,4-difluoro-1,2,3,4-tetrahydro-5h-1-benzazepine derivative or salt thereof |
05/21/2003 | EP1311501A1 Antithrombotic agents |
05/21/2003 | EP1311488A1 Substituted imidazoles as tafia inhibitors |