Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
02/2003
02/19/2003CN1398252A Dehydroamino acids compounds
02/19/2003CN1398189A Combination therapy of radiation and COX-2 inhibitor for treatment of neoplasia
02/19/2003CN1397556A Alkali-metal or alkali-earth metal salt of polyprotic acid delotadine and its medical composition
02/19/2003CN1397550A Novel benzene amine compound, its prepn. process and medicinal compsns. contg. them
02/19/2003CN1101816C Substituted purine derivatives, processes for their prepn. their use, and compsns. comprising them
02/18/2003WO2002016329A1 Novel phenylalanine derivatives
02/18/2003US6521681 Phenol-free stabilization of polyolefin fibres
02/18/2003US6521655 Substituted imidazoles useful in the treatment of inflammatory diseases
02/18/2003US6521653 Microbicidal benzotriazoles
02/18/2003US6521650 Amines as pharmaceutical agents
02/18/2003US6521643 Pyridine compounds and their pharmaceutical use
02/18/2003US6521638 2,3-dihydro-1H-isoindole derivatives useful as modulators of dopamine D3 receptors (antipsychotic agents)
02/18/2003US6521631 Heterocyclic sulfonamides
02/18/2003US6521630 Tetrahydroquinazoline-2,4-diones and therapeutic uses thereof
02/18/2003US6521629 2-amine substituted quinoline or quinozoline derivatives useful for treating benign prostatic hyperplasia
02/18/2003US6521625 Anticaogulants
02/18/2003US6521624 Synthesis and use of retinoid compounds having negative hormone and/or antagonist activities
02/18/2003US6521623 N,N'-disubstituted benzimidazolone derivatives with affinity at the serotonin and dopamine receptors
02/18/2003US6521622 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
02/18/2003US6521621 1-(1,2-disubstituted piperidinyl)-4-substituted piperazine derivatives
02/18/2003US6521618 Antineoplastic agents, agents for treatment of osteoporosis and polycystic kidney disease
02/18/2003US6521614 N-(amidinophenyl)cyclourea analogs as factor Xa inhibitors
02/18/2003US6521610 4-Haloalkyl-3-heterocyclylpyridines and 4-haloalkyl-5-heterocyclyl-pyrimidines, processes for their preparation, compositions comprising them, and their use as pesticides
02/18/2003US6521592 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
02/18/2003US6521256 Stabilized pharmaceutical composition
02/18/2003CA2264508C Substituted benzocycloheptapyridine derivatives useful for inhibition of farnesyl protein transferase
02/13/2003WO2003011876A1 Ligands and catalyst systems thereof for ethylene oligomerisation to linear alpha olefins
02/13/2003WO2003011872A1 Platelet adp receptor inhibitors
02/13/2003WO2003011858A1 Substituted isoindoles and e use thereof
02/13/2003WO2003011854A1 Pyrazole-derived kinase inhibitors and uses thereof
02/13/2003WO2003011853A1 6-aryl-4-aminopicolinates and their use as herbicides
02/13/2003WO2003011841A1 1,2,4-triazin-3,5-diones as gonadotropin-releasing hormone receptor (gnrh) antagonists
02/13/2003WO2003011839A1 1,3,5-triazine-2,4,6-triones, preparation and use as gonadotropin-releasing hormone receptor antagonists
02/13/2003WO2003011836A1 Tyrosine kinase inhibitors
02/13/2003WO2003011833A1 Indazole or indole derivatives, their use in human medicine and more particularly in cancerology
02/13/2003WO2003011829A1 Process for the production of quinazolines
02/13/2003WO2003011815A1 Bicyclic heteroaromatic alanines
02/13/2003WO2003011812A1 NOVEL AMINE DERIVATIVE HAVING HUMAN β-TRYPTASE INHIBITORY ACTIVITY AND DRUGS CONTAINING THE SAME
02/13/2003WO2003011799A1 Kinetic resolutions of chirat 3- and 3-substituted carboxylic acids
02/13/2003WO2003011302A1 Androgen receptor modulators and methods of use thereof
02/13/2003WO2003011297A1 N3-substituted 6-anilinopyrimidines and methods to treat gram-positive bacterial and mycoplasmal infections
02/13/2003WO2003011293A2 Pyridinone and pyridazinone derivatives as gonadotropin-releasing hormone receptor antagonists
02/13/2003WO2003011287A1 Pyrazolon derivatives as inhibitors of gsk-3
02/13/2003WO2002076974A3 Process for the preparation of tetrasubstituted imidazole derivatives and novel crystalline structures thereof
02/13/2003WO2002053556A3 Pyrrolidinylmethyl substituted decahydroisoquinolines as excitatory amino acid receptor antagonists
02/13/2003WO2002013830A1 Cytokine production inhibitors
02/13/2003US20030032812 Cyclobutaindolecarboxamide compounds
02/13/2003US20030032811 Sulfonyltriazol derivatives and their use for combating micro-organisms
02/13/2003US20030032803 Novel amide derivatives as inhibitors of matrix metalloproteinases, TNF-alpha, and aggrecanase
02/13/2003US20030032656 2-Amino-nicotinamide derivatives and their use as vegf-receptor tyrosine kinase inhibitors
02/13/2003US20030032654 Useful for the treatment or prevention of asthma and other allergic diseases.
02/13/2003US20030032653 Crystal forms of 6-[(4-chloro-phenyl)-hydroxy-(3-methyl-3H-imidazol-4-yl)-methyl]-4-(3-ethynyl-phenyl)-1-methyl-1H-quinolin-2-one, 2,3-dihydroxybutanedioate salts and method of production
02/13/2003US20030032652 Hydroxamic and carboxylic acid derivatives
02/13/2003US20030032647 Aromatic nitrogen-containing 6-membered cyclic compounds
02/13/2003US20030032623 E.g., 1-(2-(1-adamantyl)ethyl)-1-pentyl-3-(3-(4-pyridyl)propyl)urea; useful as therapeutic agents for autoimmune diseases such as rheumatoid arthritis.
02/13/2003CA2468925A1 Platelet adp receptor inhibitors
02/13/2003CA2456187A1 Pyrazole-derived kinase inhibitors and uses thereof
02/13/2003CA2456166A1 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids
02/13/2003CA2456096A1 Novel amine derivative having human .beta.-tryptase inhibitory activity and medecine containing the same
02/13/2003CA2455853A1 Ligands and catalyst systems thereof for ethylene oligomerisation to linear alpha olefins
02/13/2003CA2455833A1 1,3,5-triazine-2,4,6-triones, preparation and use as gonadotropin-releasing hormone receptor antagonists
02/13/2003CA2455772A1 Substituted isoindoles and their use
02/13/2003CA2455235A1 1,2,4-triazin-3,5-diones as gonadotropin-releasing hormone receptor (gnrh) antagonists
02/13/2003CA2455179A1 Androgen receptor modulators and methods of use thereof
02/13/2003CA2451075A1 Process for the production of quinazolines
02/12/2003EP1283199A1 Melanin-concentrating hormone antagonist
02/12/2003EP1283055A1 Soluble beta amyloid precursor protein secretion promoters
02/12/2003EP1282630A1 Hydroxylamine esters as polymerization initiators
02/12/2003EP1282617A1 Hydantoin derivatives with affinity for somatostatin receptors
02/12/2003EP1282616A1 Hydroxyphenyl-piperidin-4-ylidene-methyl-benzamide derivatives for the treatement of pain
02/12/2003EP1282614A1 Hydroxamic acid derivatives
02/12/2003EP1282612A2 Alkynyl phenyl heteroaromatic glucokinase activators
02/12/2003EP1282609A2 Piperazinedione compounds
02/12/2003EP1282607A2 Prodrugs of hiv replication inhibiting pyrimidines
02/12/2003EP1282606A2 Hiv replication inhibiting pyrimidines and triazines
02/12/2003EP1282602A1 Propanoic acid derivatives as integrin receptor antagonists
02/12/2003EP1282600A1 Inhibitors of dipeptidyl peptidase iv
02/12/2003EP1282418A2 Use of pyrazole derivatives for treating infertility
02/12/2003EP1189899B1 Pyrazinone thrombin inhibitors
02/12/2003EP1064262B1 Substituted isoindolones and their use as cyclic gmp modulators in medicaments
02/12/2003EP1003724B1 Substituted quinoline derivatives with antiviral action
02/12/2003EP0995744B1 Cis-substituted fluoromethylpyrrolidine derivatives
02/12/2003EP0988292B1 Piperazine derivatives and their use as anti-inflammatory agents
02/12/2003EP0941112B1 Methods and compositions for stimulating neurite growth using compounds with affinity for fkbp12 in combination with neurotrophic factors
02/12/2003EP0871623B1 3-azetidinylalkylpiperidines or -pyrrolidines as tachykinin antagonists
02/12/2003EP0816338B1 3-(bis-substituted-phenylmethylene)oxindole derivatives
02/12/2003CN1396920A 1,3-disubstituted pyrrolidines as alpha-2-adrenoceptor antagonists
02/12/2003CN1396912A 2-amino-nicotinamide derivative sand their use as VEGF-receptor tyrosine kinase inhibitors
02/12/2003CN1396833A Integrin expression inhibitors
02/12/2003CN1396807A 除草组合物 Herbicidal compositions
02/12/2003CN1396164A Rusuan Jiatishaxing and its usage
02/12/2003CN1396159A 2,4,6-trisubstituent-sym-triazine compound and its synthesizing process
02/12/2003CN1101392C Farnesyl protein transferase inhibiting (imidazol-5-yl)methyl-2-quindinone derivatives
02/12/2003CN1101391C Farnesyl transferase inhibiting 2-quinolone derivatives
02/12/2003CN1101390C Heterocyclyl uracils
02/12/2003CN1101384C Process for preparing 1-biphenylmethylmidazole derivatives
02/12/2003CN1101380C 4-mercaptopyrrolidine derivatives as farnesyl transferase inhibitors
02/12/2003CN1101190C HIV protease inhibitor combination medicine
02/11/2003US6518429 Anticancer agents, treating restenosis, atherosclerosis and hepatitis virus
02/11/2003US6518296 Substituted 3-thiocarbamoylpyrazoles