Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
01/2003
01/29/2003CN1100043C Sulfonamide derivative and process for preparing same
01/28/2003US6512125 A process for the preparation of a compound of the formula: H2NOSO3H for indole derivatives The synthesis of memory enhancing, analgetic, and antidepressant N-alkyl-N-pyridinyl-1H-indol-1-armines is described.
01/28/2003US6512001 D-proline derivatives
01/28/2003US6512000 Aminocarbonyl-substituted benzimidazoles having tryptase-inhibitory activity
01/28/2003US6511998 Pyrazole carboxamides useful for the treatment of obesity and other disorders
01/28/2003US6511997 For treatment of a disease associated with tumor necrosis factor alpha, interleukin 1, interleukin 6 or cyclooxygenase II; such as irritable bowel disease
01/28/2003US6511996 Suitable compounds for i.v.-administration due to their intrinsic properties, such as high stability and high solubility in water
01/28/2003US6511994 Modulators of CCR5 chemokine receptor activity
01/28/2003US6511993 Metalloprotease inhibitors
01/28/2003US6511978 Pyrrole derivatives useful for farnesyl transferase inhibitors and their preparations
01/28/2003US6511977 For preventing or treating cardiac arrhythmia or atrial arrhythmia
01/28/2003US6511976 Having antipsychotic, cardiovascular and gastrokinetic activity
01/28/2003US6511649 Vitronectin receptor antagonist pharmaceuticals
01/28/2003US6511648 Vitronectin receptor antagonist pharmaceuticals
01/28/2003CA2148839C Use of alpha-1c specific compounds to treat benign prostatic hyperplasia
01/24/2003CA2394209A1 1-diphenylmethyl-pyrazole derivatives as opioid receptor ligands
01/23/2003WO2003006988A1 Cardiovascular safety assay
01/23/2003WO2003006506A2 Protease inhibitor conjugates and antibodies useful in immunoassay
01/23/2003WO2003006459A1 Piperazine oxime derivatives having nk-1 receptor antagonistic activity
01/23/2003WO2003006458A1 Benzo [g] quinoline derivatives for treating glaucoma and myopia
01/23/2003WO2003006457A1 Variolin derivatives and their use as antitumor agents
01/23/2003WO2003006456A1 4-substituted-picolinic acid amide derivates useful as fungicides
01/23/2003WO2003006454A2 Heterocyclic carboxamides and their use as fungicides
01/23/2003WO2003006444A2 Substituted amides, sulfonamides and ureas useful for inhibiting kinase activity
01/23/2003WO2003006438A1 Benzimidazole derivatives for treating microglia-activation associated diseases such as inflammatory, allergic, infectious or autoimmune diseases
01/23/2003WO2003006437A1 Imidazole derivatives as adenosine deaminase inhibitors
01/23/2003WO2003006423A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003WO2003006020A1 Pyridin-2-yl-methlyamine derivatives for treating opioid dependence
01/23/2003WO2003006016A2 Use of nk-1 receptor antagonists with pyridinic structure, for the treatment of brain, spinal or nerve injury
01/23/2003WO2003005999A2 Methods of treating cytokine mediated diseases
01/23/2003WO2003005824A2 Substituted 3-heteroaryl (amino-or-oxy)-pyrrolidin-2-ones, method for the production thereof and use thereof as herbicides or as plant growth regulators
01/23/2003WO2002088088A9 Process for preparing 1-methyl-1,2,3,4-tetrahydroisoquinoline or a salt thereof
01/23/2003WO2002055491A3 1,2-DISUBSTITUTED CYCLIC INHIBITORS OF MATRIX METALLORPROTEASES AND TNF-$g(a)
01/23/2003WO2002053535A3 Process for making amlodipine, derivatives thereof, and precursors therefor
01/23/2003WO2002051808A3 Muscarinic antagonists
01/23/2003WO2002050066A3 Pyrazole compounds useful as protein kinase inhibitors
01/23/2003WO2002047456A3 Urotensin-ii receptor antagonists
01/23/2003WO2002046171A3 Anilinopyrimidine derivatives as ikk inhibitors and compositions and methods related thereto
01/23/2003WO2002041835A3 Estrogen receptor modulators
01/23/2003WO2002034760A3 Compounds and methods
01/23/2003WO2002008177A2 N-substituted-1-amino-1,1-dialkylcarboxylic acid derivatives
01/23/2003WO2001070669A3 Process for forming an amide bond
01/23/2003US20030018197 Administering a therapeutically effective amount of a pyrrazole sulfide or ether compound to treat the human immunodeficiency virus infection
01/23/2003US20030018193 Beta-alanine derivatives and their use as receptor anatgonists
01/23/2003US20030018189 Cyclic polyamines having total 9-24 members which have activity in against HIV-infected cells as well as other biological activity related to binding of ligands to chemokine receptors
01/23/2003US20030018062 Deacetylase inhibitors
01/23/2003US20030018059 Antiinflammatory agents; antihistamines; antiallergens
01/23/2003US20030018057 Certain heteroaryl substituted thiol inhibitors of endothelin-converting enzyme
01/23/2003US20030018052 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
01/23/2003US20030018051 Pyrazole derivatives - p38 MAP kinase inhibitors
01/23/2003US20030018046 Chemokine receptor binding heterocyclic compounds
01/23/2003US20030018045 Heterocyclic beta-3 adrenergic receptor agonists
01/23/2003US20030018038 1,4 substituted piperidinyl NMDA/NR2B antagonists
01/23/2003US20030018035 Central nervous system disorders
01/23/2003US20030018034 Piperazine compounds and medicinal use thereof
01/23/2003US20030018029 Tyrosine kinase inhbitor; antiproliferative agents
01/23/2003US20030018025 Psychological disorders, antidepressants, Parkinson's disease
01/23/2003US20030018024 Biphenyl vasopressin agonists
01/23/2003US20030018012 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
01/23/2003CA2453503A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003CA2453169A1 Substituted amides, sulfonamides and ureas useful for inhibiting kinase activity
01/23/2003CA2453147A1 Methods of treating cytokine mediated diseases
01/23/2003CA2451566A1 Use of nk-1 receptor antagonists for the treatment of brain, spinal or nerve injury
01/23/2003CA2449243A1 Protease inhibitor conjugates and antibodies useful in immunoassay
01/23/2003CA2446726A1 Piperazine oxime derivatives having nk-1 receptor antagonistic activity
01/23/2003CA2418173A1 N-substituted-1-amino-1,1-dialkylcarboxylic acid derivatives
01/23/2003CA2417156A1 3,4-dihydroisoquinoline derivative compound and a pharmaceutical agent comprising it as active ingredient
01/22/2003WO2002010131A1 Pyrrole derivatives
01/22/2003EP1277752A1 Process for producing optically active sulfoxide derivative
01/22/2003EP1277751A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277749A1 2- and 2,5-substituted phenylketo enols
01/22/2003EP1277741A1 Cyclic compounds
01/22/2003EP1277738A1 Condensed heteroaryl derivatives
01/22/2003EP1277735A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277734A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277733A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277471A1 Stable liquid preparation
01/22/2003EP1276741A1 Phenyl substituted 4-hydroxy tetrahydropyridone
01/22/2003EP1276740A2 Novel epothilone derivatives, method for the preparation thereof and their pharmaceutical use
01/22/2003EP1276738A1 2-amino-3-(alkyl)-pyrimidone derivatives as gsk3.beta. inhibitors
01/22/2003EP1276737A1 Sodium-hydrogen exchanger type 1 inhibitor (nhe-1)
01/22/2003EP1276732A1 Amides of r-2-(aminoaryl)-propionic acids for use in theprevention of leucocyte activation"
01/22/2003EP1276726A2 Substituted phenyl farnesyltransferase inhibitors
01/22/2003EP1276725A2 5-substituted tetralones as inhibitors of ras farnesyl transferase
01/22/2003EP1276724A2 Dihydro-2h-naphthalene-1-one inhibitors of ras farnesyl transferase
01/22/2003EP1276723A2 Pyrazole compounds having anti proliferative activity
01/22/2003EP1276722A1 Naphthamidine urokinase inhibitors
01/22/2003EP1276720A2 2-acyl indol derivatives and their use as anti-tumour agents
01/22/2003EP1107738A4 Novel pharmaceutical salt form
01/22/2003EP1030838B1 Method of synthesis of pyrrole amides
01/22/2003EP0898562B1 Hydroxamic acid derivatives for use with the treatment of diseases related to connective tissue degradation
01/22/2003EP0844241B1 Inhibitor for narcotic analgetic dependence/resistance acquisition
01/22/2003EP0646115B1 Heterocyclic-cyclic amine derivatives
01/22/2003CN1392874A Cyclic amidine compounds
01/22/2003CN1099415C Pesticidal 1-arylpyrazoles
01/22/2003CN1099413C Certain fused N-pyrrolylaniline: new class of GABA brain receptor ligand
01/22/2003CA2416946A1 Pyrrole derivatives
01/21/2003US6509476 Process for preparing N-benzyl indoles
01/21/2003US6509469 Process for the production of pyridine derivatives
01/21/2003US6509468 FR 173657 used as an antiallergen, antiinflammatory agent, antishock agent, or analgesic; autoimmune diseases