Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
04/2003
04/10/2003WO2003028459A1 Nicotinic acid-heterocyclyl-amides and analogous pyrimidine derivatives serving as pesticides
04/10/2003WO2003028458A1 N-thio-nicotinamide derivatives and related compounds for use as pesticides
04/10/2003WO2003002974A3 Ecl labels having improved non-specific binding properties, methods of using and kits containing the same
04/10/2003WO2003000186A3 Novel phenylamino-pyrimidines and uses thereof
04/10/2003WO2003000175A3 Pediatric formulation of gatifloxacin
04/10/2003WO2002102793A3 Quinazolinediones as antibacterial agents
04/10/2003WO2002094203A3 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
04/10/2003WO2002078639A3 A method of treating proliferative diseases using eg5 inhibitors
04/10/2003WO2002070540A3 Peptide deformylase inhibitors
04/10/2003WO2002041889A3 Indolsulfonyl compounds useful in the treatment of cns disorders
04/10/2003WO2002030920A1 Benzimidazole compounds, process for producing the same and use thereof
04/10/2003US20030069430 Substituted oxindole derivatives as protein tyrosine and as protein serine/threonine kinase inhibitors and compositions and methods of treating chemotherapy and radiation therapy side effects
04/10/2003US20030069428 Pharmaceutically active isoindoline derivatives
04/10/2003US20030069425 Substituted pyrimidine compounds and methods of use
04/10/2003US20030069424 Indolylmaleimide derivatives
04/10/2003US20030069423 Novel processes for the preparation of adenosine compounds and intermediates thereto
04/10/2003US20030069422 Process for preparation of pyrazolo[4,3-d]pyrimidin-7-ones and intermediates thereof
04/10/2003US20030069418 Ligands for cellular receptors, including opiate receptors; side effect reduction; base structure is a saturated nitrogen-containing ring substituted with a tertiary amide that is N-substituted with an arylalkyl group
04/10/2003US20030069417 Reacting 2-amino-3-hydroxymethyl pyridine with N-methyl-1-phenyl-2,2'-iminodiethyl chloride to form 1-(3-hydroxymethylpyridyl-2-yl)-4-methyl-2-phenyl-piperazine, and then reacting with ring closing agent to form mirtazepine
04/10/2003US20030069416 Cycloalkylpyrrole-3-carboxylic acid derivatives and heterocycloalkylpyrrole-3-carboxylic acid derivatives
04/10/2003US20030069299 Substituted indolinones, preparation thereof and their use as pharmaceutical compositions
04/10/2003US20030069297 4-aryl substituted indolinones
04/10/2003US20030069287 Process for preparing prodrugs of benzenesulfonamide-containing cox-2 inhibitors
04/10/2003US20030069284 Anticancer agent
04/10/2003US20030069278 Heterocyclyloxy-, -thioxy- and -aminobenzazole derivatives as 5-hydroxytryptamine-6 ligands
04/10/2003US20030069276 Viricides; aids therapy
04/10/2003US20030069273 Substituted 3,5-diphenyl-1,2,4-triazoles and their use as pharmaceutical metal chelators
04/10/2003US20030069272 Prevent joint stiffness; adjust concentration of synovial fluid
04/10/2003US20030069266 Composition and antiviral activity of substituted azaindoleoxoacetic piperazine derivatives
04/10/2003US20030069261 Therapy for eating disorders, sexual disorders, psychological disorders
04/10/2003US20030069258 Novel guanidine mimics factor Xa inhibitors
04/10/2003US20030069257 Benzimidazole and pyridylimidazole derivatives
04/10/2003US20030069252 Viricides; antiinflammatory agents
04/10/2003US20030069250 Anticoagulants
04/10/2003US20030069249 Analgesics; central nervous system disorders
04/10/2003US20030069248 Antiinflammatory agents; controlling cell cycle
04/10/2003US20030069245 Aids therapy
04/10/2003US20030069243 Novel substituted imidazole compounds
04/10/2003US20030069241 Analgesics; central nervous system disorders; gastrointestinal disorder; therapy for drug abruse ; antiinflammatory agents
04/10/2003US20030069239 Anticancer agents
04/10/2003US20030069234 CXCR3 antagonists
04/10/2003US20030069230 Quinazolone derivatives as alpha 1A/B adrenergic receptor antagonists
04/10/2003US20030069224 Non-nucleoside reverse transcriptase inhibitors
04/10/2003US20030069223 Peptidyl deformylase inhibitors used for inhibiting bacteria or preventing bacterial contamination of a cell culture medium
04/10/2003US20030069210 Especially imidazolyl- or 1,2,4-triazolyl- pyrimidine derivatives
04/10/2003US20030069169 Co-administration of melanocortin receptor agonist and phosphodiesterase inhibitor for treatment of cyclic-AMP associated disorders
04/10/2003US20030069140 Herbicides
04/10/2003CA2462647A1 6-membered unsaturated heterocyclic compounds useful for selective inhibition of the coagulation cascade
04/10/2003CA2462601A1 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade
04/10/2003CA2462419A1 N-heterocyclyl hydrazides as neurotrophic agents
04/10/2003CA2462305A1 6-membered heterocyclic compounds useful for selective inhibition of the coagulation cascade
04/10/2003CA2462112A1 Spiro-hydantoin compounds useful as anti-inflammatory agents
04/10/2003CA2461919A1 Substituted 2,5-diamidoindoles as ece inhibitors for the treatment of cardiovascular diseases
04/10/2003CA2461034A1 Tetrahydroisochinolines, their production and the use thereof as analgesics
04/10/2003CA2460906A1 Insecticidal and acaricidal 3-substituted pyrazoles
04/10/2003CA2460594A1 Mch receptor antagonists
04/10/2003CA2460168A1 4¬piperidin-4-yliden-(3-carbamoylphenyl)methyl| benzamide derivatives and their use for the treatment of pain, spinal injuries or gastrointestinal disorders
04/10/2003CA2459825A1 Compounds useful as reversible inhibitors of cysteine proteases
04/10/2003CA2457798A1 Process for preparing heterocyclo-alkylsulfonyl pyrazole derivatives
04/10/2003CA2457647A1 Benzimidazolidinone derivatives as muscarinic agents
04/10/2003CA2425363A1 Benzimidazole compounds, process for producing the same and use thereof
04/09/2003EP1300406A1 Method for producing pyridine compound
04/09/2003EP1300399A1 Phenylpyridazine derivatives and drugs containing the same
04/09/2003EP1300398A1 Propane-1,3-dione derivatives
04/09/2003EP1300396A1 1,2-dihydropyridine compounds, process for preparation of the same and use thereof
04/09/2003EP1299388A1 Variolin derivatives as anti-cancer agents
04/09/2003EP1299383A1 Sulfonyl-pyrrolidine derivatives useful for the treatment of neurological disorders
04/09/2003EP1299382A1 Composition and antiviral activity of substituted indoleoxoacetic piperazine derivatives
04/09/2003EP1299380A1 Indole derivatives useful for the treatment of cns disorders
04/09/2003EP1299379A2 Lactam metalloprotease inhibitors
04/09/2003EP1299378A1 Tetrahydropyridino or piperidino heterocyclic derivatives
04/09/2003EP1299364A1 Benzodiazepines as inhibitors of hpv e1 helicase
04/09/2003EP1299362A1 Selective melanin concentrating hormone-1 (mch1) receptor antagonists and uses thereof
04/09/2003EP1299361A1 Pyrazole derivatives
04/09/2003EP1299358A2 Pyridoxine and pyridoxal analogues: cardiovascular therapeutics
04/09/2003EP1299357A1 Novel compounds
04/09/2003EP1299356A1 Novel compounds
04/09/2003EP1299346A2 Process for forming an amide bond
04/09/2003EP1220844B1 Aryl sulfonamide-substituted benzimidazol derivatives thereof as tryptase inhibitors
04/09/2003EP1149090B1 Novel crystalline form of the potassium salt of (s)-omeprazole
04/09/2003EP0993458B1 3-benzylpiperidine
04/09/2003EP0946547B1 A novel compound form
04/09/2003EP0946165B1 Integrin antagonists
04/09/2003EP0873123B1 Inhibitors of protein isoprenyl transferases
04/09/2003EP0850224B1 Radiation-activated cytotoxin therapy
04/09/2003EP0843663B1 4-aryl-thio-pyridin-2(1h)-ones, drugs containing same, and uses thereof for treating hiv-related diseases
04/09/2003EP0829474B1 Indazole derivatives having monocyclic amino group
04/09/2003EP0758327B1 Pyranone compounds useful to treat retroviral infections
04/09/2003EP0708768B1 Tri-substituted imidazoles having multiple therapeutic properties
04/09/2003EP0674623B1 Bicyclic fibrinogen antagonists
04/09/2003CN1409709A Substituted bisindolylmaleimides for inhibition of cell proliferation
04/09/2003CN1409708A 酪氨酸激酶抑制剂 Tyrosine kinase inhibitor
04/09/2003CN1409704A Heterocycle derivatives and drugs
04/09/2003CN1409703A 4-aminopiperidine derivatives and their use as medicine
04/09/2003CN1105114C Sulfonyl divalent aryl alpha-hydroxy-iso-hydroximic acid compounds
04/09/2003CN1105113C Fungicidal pyrimidinones
04/09/2003CN1105102C Amino-butenate compound and preparation method thereof
04/08/2003US6545162 Solid phase biosynthesis of viricide antibiotic
04/08/2003US6545161 Substituted benzene compounds, process for their preparation, and herbicidal and defoliant compositions containing them
04/08/2003US6545158 Such as N-(3,5-dichloropyridin-4-yl)-2-(1-(4-fluorobenzyl)-5-hydroxyindol-3-yl)-2 -oxoacetamide; for treatment of eosinophil-related disorders and chronic obstructive pulmonary disease