Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
01/2003
01/08/2003EP1272185A2 Use of quinazoline derivatives as angiogenesis inhibitors
01/08/2003EP1196500B1 Reactive dye compounds
01/08/2003EP1121356B1 3-tetrahydropyridin-4-yl indoles for treatment of psychotic disorders
01/08/2003EP1119355B1 Naphthalenecarboxamides as tachykinin receptor antagonists
01/08/2003EP1077945B1 Isoquinolines as urokinase inhibitors
01/08/2003EP1021404B1 Azetidinone derivatives for the treatment of hcmv infections
01/08/2003EP0946175B1 USE OF A COMBINATION OF H+, K+ -ATPase INHIBITORS AND GLUCOCORTICOIDS IN THE TREATMENT OF NASAL POLYPS
01/08/2003EP0892795B1 Piperidinylpyramidine derivatives
01/08/2003EP0859768B1 Amine acid salt compounds and process for the production thereof
01/08/2003CN1390214A New phenylpiperazines
01/08/2003CN1390213A Aryloxy propanolamines for improving livestock production
01/08/2003CN1390206A Inhibitors of factor Xa
01/08/2003CN1390204A Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
01/08/2003CN1390203A Novel 5-pyrimidine carboxamide derivatives and the pharmaceutical compositions containing said derivatives
01/08/2003CN1390201A Cyclic amine compounds as CCR5-antagonists
01/08/2003CN1390200A Inhibitors of metalloproteinases
01/08/2003CN1390091A Use of polysiloxanes containing quaternary amino groups as formulation auxiliary agents, and composition containing the same
01/08/2003CN1389203A Method for treating hair-dropping using thyromimetic compound
01/08/2003CN1098264C Substituted 4-(1H-benzimidzol-2-yl-amino) piepridines useful for the treatment of allergic diseases
01/08/2003CN1098263C Pyridin-2-yl-methylaminederivatives, method of preparing and application as medicine
01/08/2003CN1098262C Acid-addition salts of optically active piperidine compound and process for producing the same
01/08/2003CN1098261C Process for optical purification of enantiomerically enriched benzimidazole derivatives
01/08/2003CN1098260C 2,4-diaminopyrimidine derivatives
01/08/2003CN1098259C Novel carboxy substituted cyclic carboxamide derivatives
01/08/2003CN1098256C Substd. benzenesulfonamide derivatives as prodrugs of COX-2 inhibitors
01/08/2003CN1098254C Sulfonamides
01/08/2003CN1098104C New oral pharmaceutical dosage form
01/07/2003US6504036 2- and 2.5-substituted phenylketoenols
01/07/2003US6504034 Cell antiproliferative agents; anticancer agents
01/07/2003US6504032 Forming 2,4'-, 2,3'- or 2,2'-dipyridyl's, by reacting 1,2,4-triazines, nitriles and hydrazines, then with glyoxal and finally with 2,5-norbornadiene; cylization; by product inhibition
01/07/2003US6503938 Treatment of estrogen related disease or tumor, including prostatic hyperplasia, breast cancer, endometrial carcinoma, anovulatory infertility, melanoma or osteoporosis
01/07/2003US6503935 Imidazoles and related compounds as α1A agonists
01/07/2003US6503933 Combating phytopathogenic fungi
01/07/2003US6503930 Pyrazole derivatives as p38 kinase inhibitors
01/07/2003US6503929 Nitrate salt of anti-ulcer medicine
01/07/2003US6503928 Central nervous system disorders; psychological disorders
01/07/2003US6503926 Nitrogen heterocycle compounds
01/07/2003US6503925 Treating anxiety, anesthesia, and epilepsy
01/07/2003US6503912 Substituted guanidine derivatives
01/07/2003US6503907 Indole and dihydroindole derivatives
01/07/2003US6503905 3,3-biarylpiperidine and 2,2-biarylmorpholine derivatives
01/07/2003US6503902 Treatment of neurological disorders related to beta -amyloid production such as Alzheimer's disease and Down's Syndrome.
01/07/2003US6503901 Amino lactam sulfonamides as inhibitors of Aβ protein production
01/07/2003US6503898 Administering 4,7-dibenzyl-5,6-dihydroxy-N,N*-di(m-aminobenzyl)--1,3-diazepin-2-one or salt to treat human immunodeficiency virus infection
01/07/2003CA2228524C Quinazolinone-containing pharmaceutical compositions for prevention of neovascularization and for treating human malignancies
01/07/2003CA2075684C 1-acylpiperidine compounds
01/07/2003CA2047531C 1-(substituted pyridinylamino)-1h-indol-5-yl substituted carbamates, a process and intermediates for their preparation and their use as medicaments
01/05/2003CA2392189A1 Heterocyclo-alkylsulfonyl pyrazoles as anti-inflammatory/analgesic agents
01/05/2003CA2390181A1 Sulfonyl aryl triazoles as anti-inflammatory/analgesic agents
01/03/2003WO2003000692A2 Oxytocin agonists
01/03/2003WO2003000681A1 Antibacterial having quinolinecarboxamide skeleton
01/03/2003WO2003000680A1 Diamine derivatives
01/03/2003WO2003000679A2 Herbicidal substituted pyridines, method for producing the same and their use as herbicidal agents and plant growth regulators
01/03/2003WO2003000678A1 Cyanoanthranilamide derivatives and the use thereof as medicaments
01/03/2003WO2003000677A1 Spiropiperidine compounds as ligands for orl-1 receptor
01/03/2003WO2003000666A1 5-ht receptor ligands and uses thereof
01/03/2003WO2003000665A1 Antibacterial uracil derivatives
01/03/2003WO2003000664A1 Uracil derivatives and the use thereof for treating bacterial diseases
01/03/2003WO2003000663A1 5-ht receptor ligands and uses thereof
01/03/2003WO2003000660A1 Quinoline derivative and quinazoline derivative inhibiting self-phosphorylation of hepatocytus proliferator receptor, and medicinal composition containing the same
01/03/2003WO2003000657A1 Diamine derivatives
01/03/2003WO2003000289A1 Composition comprising a pde-4 inhibitor and h1-receptor antagonist and the use thereof for the manufacture of a medicament for the treatment of respiratory diseases
01/03/2003WO2003000267A1 Amino nicotinate derivatives as glucokinase (glk) modulators
01/03/2003WO2003000262A1 Vinyl phenyl derivatives as glk activators
01/03/2003WO2003000251A1 Novel idolinones and uses thereof
01/03/2003WO2003000250A1 3-fluoro-pyrrolidines as antidiabetic agents
01/03/2003WO2003000186A2 Novel phenylamino-pyrimidines and uses thereof
01/03/2003WO2003000181A2 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/03/2003WO2003000180A2 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/03/2003WO2003000175A2 Pediatric formulation of gatifloxacin
01/03/2003WO2002088101A3 Inhibitors of bace
01/03/2003WO2002083656A3 5-membered heterocycles, preparation and use thereof as mao inhibitors and lipid peroxidation inhibitors, preparation thereof and use thereof as medicaments
01/03/2003WO2002060869A3 Use of p38 inhibitors for the treatment of inflammation-enhanced cough
01/03/2003WO2002046170A8 Anilinopyrimidine derivatives as jnk pathway inhibitors and compositions and methods related thereto
01/03/2003CA2455292A1 5-ht receptor ligands and uses thereof
01/03/2003CA2454538A1 Quinoline derivatives and quinazoline derivatives capable of inhibiting autophosphorylation of hepatocyte growth factor receptors, and pharmaceutical composition comprising the same
01/03/2003CA2451354A1 Herbicidal substituted pyridines, their preparation, and their use as herbicides and plant growth regulators
01/03/2003CA2451249A1 Amino nicotinate derivatives as glucokinase (glk) modulators
01/03/2003CA2450758A1 Composition comprising a pde-4 inhibitor and h1-receptor antagonist and the use thereof for the manufacture of a medicament for the treatment of respiratory diseases
01/03/2003CA2450742A1 Pediatric formulation of gatifloxacin
01/03/2003CA2450579A1 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/03/2003CA2450550A1 Spiropiperidine compounds as ligands for orl-1 receptor
01/03/2003CA2450491A1 5-ht receptor ligands and uses thereof
01/03/2003CA2450480A1 Oxytocin agonists
01/03/2003CA2450475A1 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/03/2003CA2449441A1 3-fluoro-pyrrolidines as antidiabetic agents
01/02/2003WO2002002529A1 Bicyclic lactams and sulfonamides with 5-ht1a-affinity and use thereof for preventing and treating cerebral ischaemia
01/02/2003US20030004353 Process for preparing integrin antagonist intermediates
01/02/2003US20030004351 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
01/02/2003US20030004344 Thrombin or factor Xa inhibitors
01/02/2003US20030004342 Imidazolyl derivatives
01/02/2003US20030004340 Skin disorders; gastrointestinal disorders
01/02/2003US20030004339 Therapy for benign prostatic hyperplasia
01/02/2003US20030004208 Squalene synthetase inhibitors; antilipemic agents, anticholesterol agents
01/02/2003US20030004192 Using cyanoguanidine compound; anticancer agents
01/02/2003US20030004190 Reacting potassium salt with magnesium compound
01/02/2003US20030004185 Viricides, organ transplants, antiarthritic agents
01/02/2003US20030004183 Quinoline-4-carboxamide derivatives as NK-2 and NK-3 receptor antagonists
01/02/2003US20030004181 Disubstituted bicyclic heterocycles, the preparation thereof, and their use as pharmaceutical compositions
01/02/2003US20030004174 Antiinflammatory agents, anticancer agents, antihistamines, central nervous system disorders