Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
01/2003
01/02/2003US20030004173 Pharmaceutically active compounds
01/02/2003US20030004166 Novel triazine compounds useful as sorbitol dehydrogenase inhibitors
01/02/2003US20030004164 Anticancer agents; autoimmune diseases
01/02/2003US20030004162 Antidiabetic agents; dietetics
01/02/2003US20030004161 Anticancer agents; autoimmune diseases
01/02/2003US20030004158 Kinase inhbitor; antiproliferative agents
01/02/2003US20030004137 Muscle relaxants, controlling immunology, strokes, antidiabetic agents
01/02/2003US20030003396 Reflection, protective or covering layers which can be written on or read by blue, red or infrared light
01/02/2003US20030003049 Simultaneous dual isotope imaging of cardiac perfusion and cardiac inflammation
01/02/2003EP1270567A1 Pyrazoline derivatives or tetrahydropyridazine derivatives and medicinal use thereof
01/02/2003EP1270560A1 Hiv replication inhibiting pyrimidines
01/02/2003EP1270557A1 Ethylenediamine derivatives
01/02/2003EP1270555A1 Method for oxidizing a thioether group into a sulfoxide group
01/02/2003EP1268479A1 Phenyl-substituted indolizine derivatives and their use as histamine h3 ligands
01/02/2003EP1268478A2 Phenyl-substituted imidazopyridines
01/02/2003EP1268469A1 N-(heterocyclyl)benzene or pyridine sulphonamides as antithrombotic agents and anticoagulants
01/02/2003EP1268468A1 4-amino-6,7-dimethoxy-2-(5-methanesulfonamido-1,2,3,4-tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazoline mesylat and polymorphs
01/02/2003EP1268467A1 Heteroaromatic compounds having two-photon absorption activity
01/02/2003EP1268466A1 Decahydro-isoquinolines
01/02/2003EP1268465A1 Triarylimidazole derivatives as cytokine inhibitors
01/02/2003EP1268455A2 Piperazine derivatives
01/02/2003EP1268454A1 Succinoylamino heterocycles as inhibitors of a-beta protein production
01/02/2003EP1268449A1 Substituted piperidines as melanocortin receptor agonists
01/02/2003EP1268445A1 4-amino-5-cyano-2-anilino-pyrimidine derivatives and their use as inhibitors of cell-cycle kinases
01/02/2003EP1268444A1 2,4-di(hetero-)arylamino(-oxy)-5-substituted pyrmidines as antineoplastic agents
01/02/2003EP1268437A1 Inhibitors of protein kinases
01/02/2003EP1268435A1 4,5-dihydro-1h-pyrazole derivatives having cb 1-antagonistic activity
01/02/2003EP1268433A1 Cyclic lactams as inhibitors of a-beta-protein production
01/02/2003EP1268432A1 ISOQUINOLONE INHIBITORS OF FACTOR Xa
01/02/2003EP1268431A1 3-cyanoquinolines,3-cyano-1,6-naphthyridines, and 3-cyano-1,7-naphthyridines as protein kinase inhibitors
01/02/2003EP1268429A1 Vitronectin receptor antagonist bicyclic compounds, preparation method and compositions containing same
01/02/2003EP1268428A2 Polycyclic aryl and heteroaryl substituted 4-pyridones useful for selective inhibition of the coagulation cascade
01/02/2003EP1268422A1 Indoles for treating diseases that can be treated using thyroid hormones
01/02/2003EP1268421A2 Phenyl-substituted indoles as histamine h3-receptor antagonists
01/02/2003EP1268419A1 Pyrrolidine derivatives useful as bax inhibitors
01/02/2003EP1268418A1 Pharmaceutically active pyrrolidine derivatives as bax inhibitors
01/02/2003EP1267878A2 Compounds with 5-ht activity useful for controlling visual field loss
01/02/2003EP1267876A1 Thrombin inhibitors
01/02/2003EP1267874A2 Therapeutic uses of ppar mediators
01/02/2003EP1267872A2 Farnesyl protein transferase inhibitor combinations with anti-tumor anthracycline derivatives
01/02/2003EP1267870A2 Inhibition of cytokine generation
01/02/2003EP1267848A1 Dosing regimen comprising a farnesyl protein transferase inhibitor for the treatment of cancer
01/02/2003EP1109785B1 Indole derivatives and their use in the treatment of malignant and other diseases caused by pathological cell proliferation
01/02/2003EP1083897A4 Hiv integrase inhibitors
01/02/2003EP0934265B1 Amidinophenyl-pyrrolidines, -pyrrolines, and -isoxazolidines and derivatives thereof
01/02/2003EP0925286B1 Substituted pyrimidine derivatives and their pharmaceutical use
01/02/2003EP0804431B9 GLYCOPROTEIN IIb/IIIa ANTAGONISTS
01/02/2003EP0751939B9 Naphthylamides as central nervous system agents
01/02/2003EP0705245B1 Novel intermediates for the preparation of antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives
01/02/2003CA2414726A1 Bicyclic lactams and sulfonamides with 5-ht1a-affinity and use thereof for preventing and treating cerebral ischaemia
01/01/2003CN1097592C Slfonic acid amide derivatives with herbicides activity
01/01/2003CN1097591C Process for preparing pyrimidine derivatives
12/2002
12/31/2002US6500959 Pyrrolidine derivatives and processes for preparing same
12/31/2002US6500956 Method for the catalytic production of substituted bipyridyl derivatives
12/31/2002US6500955 One pot synthesis of [2,8-Bis (trifluoromethyl)-4-quinolinyl]-2-pyridinylmethanone, a mefloquine intermediate
12/31/2002US6500950 Benzylidenepyrazolones, their preparation and use
12/31/2002US6500948 Metalloproteinase inhibitors-compositions, uses preparation and intermediates thereof
12/31/2002US6500855 Nitrogen containing aromatic heterocycles with ortho-substituted p1 groups; anticoagulants
12/31/2002US6500854 Chondrongenesis promotors and indolin-2-one derivatives
12/31/2002US6500852 Inhibitors of bacterial NAD synthetase
12/31/2002US6500851 Antithrombotic agents
12/31/2002US6500850 Pesticidal 1-arylpyrazoles
12/31/2002US6500846 2-(4-chlorophenyl)-7-methoxychromen-4-one, as cyclin-dependent kinase inhibitors, used as anticarcinogenic agents or for prophylaxis of neurodegenerative disease
12/31/2002US6500845 Activating cytokine release using immunosuppressants such as 2-(3-methyl-2-oxo-piperidin-3-yl)-benzo(d)isoselenazol-3-one, racemic mixtures or isomers having dimensional stability, prepared in the presence of reducing agent
12/31/2002US6500844 Cyclopentyl modulators of chemokine receptor activity
12/31/2002US6500842 N-((4-chlorophenyl)methyl)-8-hydroxy-7-quinolinecarboxamide administered as viricides against herpes virus
12/31/2002US6500823 Energy deficiency of the cell caused by parp inhibition, in diabetes complications, in oxygen deficient status of the heart and brain, in neurodegenerative diseases, in the treatment of autoimmune and/or viral diseases
12/31/2002US6500822 Benzocycloalkylenylamine derivatives as muscarinic receptor antagonists
12/31/2002US6500821 Treat various forms of epilepsies and of states of anxiety and tension.
12/31/2002US6500818 Naphthalenecarboxamides as tachykinin receptor antagonists
12/27/2002WO2002102793A2 Quinazolinediones as antibacterial agents
12/27/2002WO2002102792A1 Novel heterocyclic antibacterial compounds
12/27/2002WO2002102791A1 Pyrrolidine bicyclic compounds
12/27/2002WO2002102790A1 N-formyl hydroxylamine compounds as inhibitors of pdf
12/27/2002WO2002102787A2 Novel sulfonic acid derivatives
12/27/2002WO2002102782A2 QUINAZOLINE DERIVATIVES which PROMOTE THE RELEASE OF PARATHYROID_HORMONE
12/27/2002WO2002102778A1 Phenylpyridine carbonyl piperazine derivative
12/27/2002WO2002102380A1 Monocyclic or bicyclic carbocycles and heterocycles as factor xa inhibitors
12/27/2002WO2002102359A2 Alkylidene pyrazolidinedione derivatives and use for treating diabetes and obesity
12/27/2002WO2002102315A2 QUINAZOLINE AND PYRIDO[2,3-d]PYRIMIDINE INHIBITORS OF PHOSPHODIESTERASE (PDE) 7
12/27/2002WO2002102314A2 Purine inhibitors of phosphodiesterase (pde) 7
12/27/2002WO2002092565A3 3-aminoalkyl-2-aryl-indole derivatives and their use as gnrh antagonists
12/27/2002WO2002074753A3 5-phenylpyrimidine, methods and intermediate products for the production thereof and use of the same for controlling pathogenic fungi
12/27/2002WO2002056888A3 Assay method, tnf modulator and its use
12/27/2002WO2002055609A3 Indole/indoline based hybrid dyes and indole/indoline based hybrid dye intermediate products
12/27/2002WO2002046181A3 Abca-1 elevating compounds against coronary artery disease or atherosclerosis
12/27/2002WO2002009758A3 Inhibitors of cellular efflux pumps of microbes
12/27/2002WO2001085095B1 Chiral fluoroquinolizinone arginine salt forms
12/27/2002WO2001052855A8 Drug combination for the treatment of depression and related disorders comprising mirtazapine and gepirone
12/27/2002CA2450936A1 Purine inhibitors of phosphodiesterase (pde) 7
12/27/2002CA2450724A1 Quinazoline and pyrido¬2,3-d|pyrimidine inhibitors of phosphodiesterase (pde) 7
12/27/2002CA2449212A1 Alkylidene pyrazolidinedione derivatives and use for treating diabetes and obesity
12/27/2002CA2448526A1 N-formyl hydroxylamine compounds as inhibitors of pdf
12/27/2002CA2448298A1 Phenylpyridine carbonyl piperazine derivative
12/27/2002CA2446963A1 Quinazolinediones as antibacterial agents
12/27/2002CA2446931A1 Pyrrolidine bicyclic compounds
12/27/2002CA2429113A1 Monocyclic or bicyclic carbocycles and heterocycles as factor xa inhibitors
12/26/2002US20020198407 Antiallergy agents and bronchodilators
12/26/2002US20020198383 For use in regioselective and enantioselective alkylations of allylic substrates
12/26/2002US20020198381 Herbicidal pyridine compounds