Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
08/2001
08/28/2001US6281212 Chemokine receptor antagonists and methods of use therefor
08/28/2001US6281206 Amidino and benzamidino compounds
08/28/2001CA2017252C Retroviral protease inhibiting compounds
08/23/2001WO2001060803A1 Fused imidazolium derivatives
08/23/2001WO2001007029A3 Substituted guanidines and the use thereof
08/23/2001WO2000071508A3 Inhibitors of factor Xa
08/23/2001US20010016659 Omega-carboxyaryl substituted diphenyl ureas as raf kinase inhibitors
08/23/2001US20010016207 Compounds such as N-(1-(cyanomethylcarbamoyl)cyclohexyl)-4-(piperazin-1-yl)-benzamide
08/23/2001DE10005631A1 Arginin-Mimetika als Faktor X¶a¶-Inhibitoren Arginine mimetics as inhibitors of factor X¶a¶
08/22/2001EP1125582A2 Use of estrogen agonists / antagonists for the treatment of sexual dysfunction
08/22/2001EP1124797A1 N-arylsulfonyl amino acid omega amides
08/22/2001EP1124795A1 Inhibitors of the egf-receptor tyrosine kinase and their use
08/22/2001EP1124552A1 Antitumor chrysene derivatives
08/22/2001EP0960093B1 Method for hydrogenating compounds from the group of imines or enamines
08/22/2001CN1309690A Amine reaction compounds comprising one or more active ingredient
08/22/2001CN1309654A Biphenyl derivs.
08/22/2001CN1309634A Hydrazine derivs.
08/22/2001CN1309116A Cyclic amine substd. phenylalkanone and preparing method thereof
08/21/2001US6277987 Sulfonylamino acid and sulfonylamino hydroxamic acid derivatives
08/21/2001US6277897 Photoinitiators and applications therefor
08/21/2001US6277840 Antiinflammatory agents
08/21/2001CA2236940C Processes and intermediates for preparing 3-(1-piperazinyl)-1,2-benzisothiazole
08/21/2001CA2205555C Use of nitric oxide-releasing agents for reducing metastasis risk
08/21/2001CA2196845C Hydroxamic acid compounds
08/16/2001WO2001059067A2 A group of anti-cancer compounds with specific structure and their production method
08/16/2001WO2001059000A1 New 3-arylbenzofuranones with electron-withdrawing substituents as stabilizers
08/16/2001WO2001058886A1 Dipeptide nitrile cathepsin k inhibitors
08/16/2001WO2001058859A1 ARGININE MIMETICS AS FACTOR Xa INHIBITORS
08/16/2001WO2001058855A1 Use of androgen receptor suppressors
08/16/2001WO2001058854A1 A topical antiandrogen for hair loss and other hyperandrogenic conditions
08/16/2001WO2001010842A3 Melanocortin-4 receptor binding compounds and methods of use thereof
08/16/2001WO2001007435A3 N-(indolcarbonyl-)piperazin derivatives als 5-ht2a-receptor ligands
08/16/2001EP1123926A1 Piperazine derivatives for treatment of CNS disorders
08/16/2001EP1123918A1 Aromatic amine derivatives, process for the preparation thereof and agents containing the same
08/16/2001EP1123276A1 N-(2-aryl-propionyl)-sulfonamides and pharmaceutical preparations containing them
08/16/2001EP0704439B1 Novel intermediate for synthetic use and process for producing aminopiperazine derivative
08/16/2001CA2400063A1 New 3-arylbenzofuranones with electron-withdrawing substituents as stabilizers
08/16/2001CA2398923A1 A group of anti-cancer compounds with specific structure and their production method
08/15/2001CN1308608A Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
08/15/2001CN1308606A Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use pharmaceutical preparations comprising them
08/15/2001CN1308604A 2,3,5-substituted biphenyls useful in the treatment of insulin resistance and hyperglycemia
08/15/2001CN1308602A Method for purifying hexamethylenediamine in mixtures of hexamethylenediamine and an unsaturated cyclic imine
08/15/2001CN1308534A Angiogenesis inhibitors
08/14/2001US6274618 Administering (-)-cis-6-phenyl-5-(4-(2-pyrrolidin-1-yl-ethoxy)-phenyl)-5,6,7,8 -tetrahydronphthalen-2-ol to treat vaginal dryness, itching, or painful intercourse
08/14/2001US6274588 4-phenyl-pyrimidine derivatives
08/14/2001US6274583 Alpha 1a adrenergic receptor antagonists
08/14/2001US6274336 Producing three-dimensional structure of active site using computer program, displaying and superimposing three-dimensional representation of test compound onto active site, preparing test compound, and testing in biological assay
08/14/2001CA2159640C Second messenger cell signaling inhibitors
08/14/2001CA2158484C Novel benzopyrane derivatives, process for their preparation and pharmaceutical compositions containing them
08/09/2001WO2001057947A1 Use of amidines
08/09/2001WO2001057008A1 2-benzothiazolyl urea derivatives and their use as protein kinase inhibitors
08/09/2001WO2001056989A2 Inhibitors of factor xa
08/09/2001WO2001056979A1 Substituted cyanoacetamide derivatives and herbicides
08/09/2001WO2001056974A2 Inha inhibitors and their use as antibacterials
08/09/2001WO2001056563A1 Adamantyl derivatives as anti-cancer agents
08/09/2001WO2001010834A9 Antibacterial agents
08/09/2001WO2000071511A3 INHIBITORS OF FACTOR Xa
08/09/2001WO2000059878A3 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF
08/09/2001WO2000047554A3 INHIBITORS OF FACTOR Xa
08/09/2001US20010012857 Pharmaceutical for treatment of neurological and neuropsychiatric disorders
08/09/2001US20010012848 An indane-like compounds which can be useful for treating psychosis and other conditions associated with modulation of a muscarinic receptor
08/09/2001DE10004928A1 Use of perfluorinated two-five carbon carboxylic acid amides as solvent (component) for salt conductors in electrolytes, e.g. for rechargeable batteries
08/09/2001CA2398754A1 2-benzothiazolyl urea derivatives and their use as protein kinase inhibitors
08/08/2001EP1122242A1 Cyanophenyl derivatives
08/08/2001EP1121342A1 Diaminopropionic acid derivatives
08/08/2001EP1121118A1 Formamides as therapeutic agents
08/08/2001CN1307563A N-phenyl-N'-phenylpropylpiperazine derivatives and process for the preparation thereof
08/08/2001CN1069356C Process for purifying tertiary aminoxide aqueous solution
08/07/2001US6271395 Substituted with an N-methyl benzene-acetamide and 1-pyrrolidinyl
08/07/2001US6271235 HIV protease inhibitors
08/07/2001CA2297944A1 The groups with anticancer activity and the method of making their derivatives
08/02/2001WO2001055125A1 A process for the preparation of quetiapine and intermediates therefor
08/02/2001WO2001055111A1 Biaryl compounds, their preparation and their use in therapy
08/02/2001WO2001054691A1 Nitrate salts of antimicrobial agents
08/02/2001WO2000076971A3 Serine protease inhibitors
08/02/2001WO2000066175A3 Conjugates as therapies for cancer and prostate diseases
08/02/2001US20010011136 Anticancer agents
08/02/2001US20010011135 Anticancer agents
08/02/2001US20010011093 Arylgycinamide derivatives, methods of producing these substances and pharmaceutical compositions containing such compounds
08/02/2001CA2397754A1 Nitrate salts of antimicrobial agents
08/01/2001EP1120410A1 Nicotinic acid esters useful as CNS agents and having affinity for 5-HT receptors
08/01/2001EP1120114A2 Compositions and methods for treating conditions responsive to estrogen
08/01/2001EP0877737B1 Novel n-(arylsulphonyl)amino acid derivatives having bradykinin receptor affinity
08/01/2001CN1306526A Novel heterocyclically substituted amides with cysteine protease-inhibiting effect
08/01/2001CN1306509A Substituted benzamides, their prodn. and use as cysteine protease inhibitors
08/01/2001CN1306505A Substituted benzamides, their prodn. and use
08/01/2001CN1306428A Inhibitors of transcription factor NF-KB
08/01/2001CN1305989A Benzene sulfonamide compounds, its preparing method and medicinal compsns. contg. same
08/01/2001CN1305812A N-(aryloxy group alkyl) heteroaromatic guadine and heteroaromatic guazine used as medicines
07/2001
07/31/2001US6268504 Aryloxy-alkyl-dialkylamines
07/31/2001US6268367 Piperazine derivatives for treating bone deficit conditions
07/31/2001US6268361 Estrogen dependent disorders including cancer, enodmetriosis, etc
07/26/2001WO2001053280A1 Substituted phenylamidines medicaments containing said compounds and method for production thereof
07/26/2001WO2001053279A1 Urea compounds as inhibitors for vla-4
07/26/2001WO2001053260A1 Carboxamides useful as inhibitors of microsomal triglyceride transfer protein and of apolipoprotein b secretion
07/26/2001WO2001053258A1 Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
07/26/2001WO2000018750A9 Chelates comprising chinoid groups as photoinitiators
07/26/2001US20010009962 One pot process for preparing sildenafil (drug for erectile dysfunction) and derivatives by reacting for example 4-(2-methoxy-5-(4-methyl-1-piperazinylsulfonyl)benzamido)-1-methyl-3-propyl -1H-pyrazole-5-carboxamide with ethanol
07/26/2001US20010009915 Nitrogen oxide yielding and thromboxane A2 (TXA2) and serotonin (5HT2) receptor antagonist; treatment of atherothrombotic cardiovascular disorders
07/26/2001DE10002510A1 New phenylamidine compounds are useful for the treatment of thrombosis, cerebrovascular disorders, heart infarction, arteriosclerosis, osteoporosis, tumor metastasis, shock and diabetes