Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
04/2006
04/20/2006US20060084658 Nitrogen-containing cyclic compound and pharmaceutical composition containing the compound
04/20/2006US20060084657 Piperazine derivative
04/20/2006US20060084641 IL-8 receptor antagonists
04/20/2006CA2582459A1 Substituted sulfones and methods of use
04/19/2006EP1646659A2 Improved pharmaceutical drug candidates and methods for preparation thereof
04/19/2006EP1646392A2 7 and 8 membered heterocyclic cyclopentyl benzylamide modulators of chemokine receptor activity
04/19/2006EP1253924B1 Nitrate salts of antimicrobial agents
04/19/2006EP1117698B1 Chelates comprising chinoid groups as photoinitiators
04/19/2006EP1112284B1 Piperazine-4-phenyl derivatives as inhibitors of the interaction between mdm2 and p53
04/19/2006EP1064274B1 Benzenesulfonamide derivatives and their use as medicaments
04/19/2006CN1761646A Cannabinoid receptor ligands
04/19/2006CN1252058C Phenoxy indenone compounds, process for preparing same and use thereof
04/19/2006CN1252040C Novel aryl, alkenyl and alkynl 4-dedimethylamino tetracycline derivatives
04/19/2006CN1252038C New derivatives of substituted anilines with herbicidal activity
04/19/2006CN1251671C Beta secretase inhibitors
04/18/2006US7030275 Cationic polymer; detergents, cleaning compounds
04/18/2006US7030247 Method for the production of biperidin
04/18/2006US7030242 Selective inhibition of aggrecanase in osteoarthritis treatment
04/18/2006US7030239 Compounds to treat Alzheimer's disease
04/18/2006US7030160 An agonist as beta-3 adrenergic receptors; chemical intermediates preparing through decyclization, hydroxylation; for treating gastrointestinal diseases, obesity, diabetics, psychotropic agents, nervous system disorders
04/18/2006US7030157 Hormone replacment therapy; anticancer agent; sexual disorders
04/18/2006US7030124 Method of treating depression with delta receptor agonist compounds
04/18/2006US7030122 1,4-disubstituted piperazine ligands for neurotransmitter receptors
04/18/2006US7030120 Nitrogen-containing heterocyclic compounds and benzamide compounds and drugs containing the same
04/18/2006US7030116 Compounds and compositions as cathepsin inhibitors
04/18/2006US7030115 Anticancer agents; autoimmune diseases; antiinflammatory agents
04/18/2006CA2360943C N2-phenylamidine derivatives
04/13/2006WO2006039383A2 Synthesis by chiral diamine-mediated asymmetric alkylation
04/13/2006WO2006038594A1 N-type calcium channel inhibitor
04/13/2006WO2006038039A1 Modulators of hcv replication
04/13/2006WO2006037982A2 Modulators of crth2 receptor activity for the treatment of prostaglandin d2 mediated diseases
04/13/2006WO2005007621A3 Ubiquitin ligase inhibitors
04/13/2006US20060079691 Ionic liquids having [n(cf3)2]-anions
04/13/2006US20060079561 Insecticidal anthranilamides
04/13/2006US20060079527 Compounds such as 1-[4-(3,4-difluoro-phenyl) -piperazin-1 -yl]-3-{methyl-[2-(9H-xanthen-9-yl)-ethyl]-amino}-propan-1 -one in free base or acid addition salt form, for therapy of depression, anxiety and bipolar disorders
04/13/2006US20060079506 Adamantyl acetamides as 11-beta hydroxysteroid dehydrogenase inhibitors
04/13/2006DE102004049728A1 Verfahren zur Herstellung von monosubstituierten Piperazinderivaten Process for the preparation of mono-substituted piperazine derivatives
04/13/2006CA2582760A1 Modulators of hcv replication
04/12/2006EP1645556A1 Arylpiperazine-benzoylamide derivatives useful as pharmaceutical agents
04/12/2006EP1644347A1 N-PHENYL-PIPERAZINE DERIVATIVES AND METHODS OF PROPHYLAXIS OR TREATMENT OF 5HT sb 2C /sb RECEPTOR ASSOCIATED DISEASES
04/12/2006EP1644345A1 Urea derivatives of piperazines and piperidines as fatty acid oxidation inhibitors
04/12/2006EP1644340A1 N-{'4-substituted piperazine-1-sulfonylmethyl]alkyl}-n-hydroxyformamide compounds as metalloproteinase inhibitors
04/12/2006EP1644337A1 Melanocortin-4 receptor binding compounds and methods of use thereof
04/12/2006EP1644328A1 Sulfonamide derivatives as 5ht7 receptor antagonists
04/12/2006EP1644325A2 Methods and compositions for treating amyloid-related diseases
04/12/2006EP1644322A1 Aspartyl protease inhibitors
04/12/2006EP1644026A2 Sigma ligands for neuronal regeneration and functional recovery
04/12/2006EP1311499B1 Bicyclic compounds as h3 receptor ligands
04/12/2006EP1311471B1 Phenyl- and phenylalkyl-substituted ethanolamines and ethylenediamines
04/11/2006US7026510 Inhibitors of the chemotactic activation induced by the fraction C5a of complement and from other chemotactic proteins (chemokines) that y activate a 7-transmembrane-domain receptor; psoriasis, rheumatoid arthritis, ulcerative colitis, acute respiratory distress syndrome, fibrosis; antiischemic agents
04/11/2006US7026498 Coordination catalyst containing ligand
04/11/2006US7026357 Diphenylurea compounds
04/11/2006US7026323 N-(naphth-2-ylaminocarbonylacetyl)- or N-(naphth-2-ylcarbonylamino- acetyl)- piperazine derivatives, e.g., 2-[((4-(ethoxycarbonyl)piperazin-1-yl)carbonylmethyl)carbonyl]aminonaphthalene; useful as antithrombotic agents
04/11/2006US7026316 (optionally aza)cycloalkyl-N,N-optionally thia-, oxothia- or dioxothia-)alkyleneglycine derivatives, e.g., N-{4-[(1S)-1-amino-2-oxo-2-(1,3-thiazolidin-3-yl)ethyl]cyclohexyl}-N'-hexylureA; especially treating type 2 diabetes
04/11/2006CA2217030C Protease inhibiting succinic acid derivatives
04/11/2006CA2089440C Ortho-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic and medicaments containing them
04/11/2006CA2089439C 3,5-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic and medicament containing them
04/06/2006US20060074247 Improving storage stability by reacting with hydrogen sulfate lithium- containing compound; aspartyl protease inhibitors
04/06/2006US20060074238 Asymmetric process for the preparation of diarylethylpiperazines derivatives and novel asymmetric diarylmethylamines as intermediates
04/06/2006US20060074123 Cyclic AMP-specific phosphodiesterase inhibitors
04/06/2006US20060074110 Multicyclic compounds which inhibit leukocyte adhesion mediated by VLA-4
04/06/2006US20060074091 Nootropic effect enhancer
04/06/2006US20060074085 Bcl-XL inhibitors; N-{[4-({(1R)-5-(dimethylamino)-1-[(phenylthio)methyl]pentyl}amino)-3-nitrophenyl]sulfonyl}-4-(4-fluorophenyl)piperidine-1-carboxamide; useful for promoting apoptosis; Anticancer agents; autoimmune diseases; antiinflammatory agents
04/05/2006EP1642894A1 Quaternary ammonium salt, electrolyte, and electrochemical device
04/05/2006EP1642880A1 Hsp90 family protein inhibitors
04/05/2006EP1641771A1 Hydroxamate sulfonamides as cd23 shedding inhibitors
04/05/2006EP1641748A2 N-alkyl phenylcarboxamide beta-secretase inhibitors for the treatment of alzheimer s disease
04/05/2006EP1370544B1 Nitric oxide donors based on metallic centres
04/05/2006EP1140846B1 Aspartic protease inhibitors
04/05/2006EP0933993B1 Substituted cyclopentane compounds useful as neuraminidase inhibitors
04/05/2006CN1756551A New arylpiperazinyl compounds
04/05/2006CN1754873A Aryl sulfonamides and analogues thereof and their use in the treatment of neurodegenerative diseases
04/05/2006CN1249054C Process for preparation of aripiprazole
04/05/2006CN1249020C Aromatic diamide derivatives, chemicals for agricultural or horticultural use and usage thereof
04/04/2006US7022845 Monomethylation of nitrogeneous heterocycles
04/04/2006US7022707 such as S-4-[(2-propylamino)carbonyl]oxybenzyl piperazine-1-thiocarboxylate for treatment of obesity and/or diabetes
04/04/2006US7022703 Acetylenic compound useful in treating inflammatory disorders
04/04/2006CA2294624C Cationic monobenzene nitrophenylenediamines, their use in dying keratin fibres, dyeing compositions containing them and dyeing processes
04/04/2006CA2256492C Diarylalkyl cyclic diamine derivatives as chemokine receptor antagonists
03/2006
03/30/2006WO2006034441A1 Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors
03/30/2006WO2006032994A2 Muscarinic receptor antagonists
03/30/2006WO2005047899A3 Use of the lipoxin receptor, fprl1, as a tool for identifying compounds effective in the treatment of pain and inflammation
03/30/2006WO2004053071A3 Method for discovering neurogenic agents
03/30/2006US20060069257 Use of specific bidentate ligands, e.g., 2-dicyclohexylphosphino-2'-dimethylamino-biphenyl, in transition metal-catalyzed carbon-heteroatom and carbon-carbon bond-forming reactions including amination and arylation and with aryl halide reactants and amine, boronic acid, borane or ketone reactants
03/30/2006US20060069250 Synthesis by chiral diamine-mediated asymmetric alkylation
03/30/2006US20060069104 Neurotrophic factor production accelerator
03/30/2006US20060069103 17 Beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
03/30/2006US20060069100 Variously substituted derivatives of guanidine, and their use as medicines with anti-diabetes and/or anti-obesity activity
03/30/2006US20060069037 Peptide-containing alpha-ketoamide cysteine and serine protease inhibitors
03/30/2006CA2580860A1 Pyridine derivatives for inhibiting human stearoyl-coa-desaturase
03/30/2006CA2580856A1 Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors
03/29/2006EP1639029A2 Biodegradable poly(beta-amino esters) and uses thereof
03/29/2006EP1638549A2 Novel antibacterial agents
03/29/2006EP1379234B1 Halogenated aminobenzophenones and aminobenzoylpyridines as inhibitors of il-1 and tnf
03/29/2006CN1753866A Arylcycloalkyl derivatives having branched side chains used as ppar receptor regulator, processes for their preparation and their use as pharmaceuticals
03/29/2006CN1753676A Crystalline non-solvated 1-(4-(2-piperidinylethoxy)phenoxy)-2-(4-methanesulfonylphenyl)-6-hydroxynaphthalene hydrochloride
03/29/2006CN1247547C Piperidine and piperazine substituted N-hydroxyformamides as inhibitors of metalloproteinases
03/29/2006CN1247543C Method for the production of biperiden II
03/29/2006CN1247523C Substituted 1 and 2 naphthol mannich bases
03/28/2006US7019137 Alkylation of 2,3-dihydro-1,4-benzodioxin-5-amine in chlorobenzene using trifluoromethanesulfonic acid salts of N,N-bis(2-chloroethyl)-alanine methyl ester, to form serotonin receptor antagonists; nervous system disorders