Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
03/2001
03/08/2001WO1999063930A8 Novel angiotensin receptor modulators and their uses
03/08/2001WO1999019296A8 Aminobutanoic acid derivatives
03/08/2001DE19941650A1 New fluorothiophene, furan, isoxazole, thiazole, cyclopentane, cyclopentene and alkylfluorothiophenecarboxylic acid compounds are useful in liquid crystals mixtures and synthesis of liquid crystals, agrochemicals and pharmaceuticals
03/08/2001CA2384435A1 Bicyclic androgen and progesterone receptor modulator compounds and methods
03/08/2001CA2384194A1 Benzylidene-thiazolidinediones and analogues and their use in the treatment of inflammation
03/08/2001CA2383347A1 Benzylidene-thiazolidinediones and analogues and their use in the treatment of diabetes
03/08/2001CA2382966A1 Biaryl-oxa(thia)zole derivatives and their use as ppars modulators
03/07/2001EP1080086A1 Dihydropyrimidines
03/07/2001EP1080082A1 Intermediates for the synthesis of epothilones and methods for their preparation
03/07/2001EP1080080A1 Novel therapeutic agents that modulate neurokinin receptors
03/07/2001EP1079825A2 Compounds that inhibit the binding of integrins to their receptors
03/07/2001EP1079821A1 Protease inhibitors
03/07/2001EP1079819A1 Hydroxamic acid derivatives as antibacterials
03/07/2001CN1286254A Aromatic amino ether as analgesics
03/06/2001US6197970 Process for producing 2-hydroxybenzamide derivatives
03/06/2001US6197969 Reacting metal salt of 2-aminothiophenol with an amino acid-n-carboxylic anhydride; cyclization in acid
03/06/2001US6197968 Storage stability; colorless after solution treatment
03/06/2001US6197803 Heterocyclic carboxamide-containing thiourea inhibitors of herpes viruses containing phenylenediamine group
03/06/2001US6197802 For agriculture
03/06/2001US6197791 N-hdroxy-2-(alkyl, aryl, or heteroaryl, sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
03/06/2001US6197782 Therapy for sexual disorders
03/06/2001US6197778 Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
03/06/2001US6197748 Ketoheterocyclic inhibitors of factor Xa
03/06/2001CA2081113C Thiazolidine-2,4-dione derivative, salt thereof, and production of the same
03/06/2001CA2073673C Esters of 2-arylmethyl-1-naphthol derivatives as 5-lipoxygenase inhibitors
03/01/2001WO2001014372A2 Oxazole and thiazole derivatives as neurotrophin production/secretion promoting agent
03/01/2001WO2001014355A1 Substituted piperazine derivatives, the production thereof and their utilization as medicaments
03/01/2001WO2001014354A1 Substituted 2-arylbenzazole compounds and their use as antitumour agents
03/01/2001WO2001014353A1 Arylmethyl-carbonylamino-thiazole derivatives and their use as antitumor agents
03/01/2001WO2001014352A1 Substituted benzylthiazolidine-2,4-dione derivatives
03/01/2001WO2001014351A1 Substituted benzylthiazolidine-2,4-dione derivatives
03/01/2001WO2001014350A1 Substituted benzylthiazolidine-2,4-dione derivatives
03/01/2001WO2001014349A1 Substituted benzylthiazolidine-2,4-dione derivatives
03/01/2001WO2001014339A2 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
03/01/2001WO2001014334A1 Fluorenone compounds with modified 7-position substituents for treating and preventing brain and spinal injury
03/01/2001WO2001014324A1 Selective inhibitors of the urokinase plasminogene activators
03/01/2001WO2001014310A1 PLEUROMUTILIN β-KETOESTERS
03/01/2001DE19940389A1 Selektive Inhibitoren des Urokinase-Plasminogen Aktivators Selective inhibitors of urokinase plasminogen activator
03/01/2001CA2382582A1 Substituted benzylthiazolidine-2,4-dione derivatives
03/01/2001CA2382574A1 Substituted benzylthiazolidine-2,4-dione derivatives
03/01/2001CA2382311A1 Substituted piperazine derivatives, the preparation thereof and their use as medicaments
03/01/2001CA2376275A1 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
02/2001
02/28/2001EP1077977A1 Retroviral protease inhibiting compounds
02/28/2001EP1077961A1 Process for the manufacture of a sulfenimide
02/28/2001EP1077960A1 (2-acylaminothiazole-4-yl)acetic acid derivatives
02/28/2001EP1077958A1 Oxazole-aryl-carboxylic acids useful in the treatment of insulin resistance and hyperglycemia
02/28/2001EP1077957A1 Oxyiminoalkanoic acid derivatives with hypoglycemic and hypolipidemic activity
02/28/2001EP1077931A1 Benzamide derivatives for the treatment of diseases mediated by cytokines
02/28/2001CN1285820A Metabotropic glutamate receptor antagonists for treating central nervous system disease
02/27/2001US6194614 Process for the preparation of benzothiazolone compounds
02/27/2001US6194575 Reacting 2-nitroimino-3,5-dimethyl-1,3, 5-triaza-cyclohexane derivative with urea in presence of diluent to form 1,3-di-substituted 2-nitroguanidine
02/27/2001US6194451 Prevent release tumor necrosis factor; antiinflammatory agents
02/27/2001US6194448 N, N-disubstituted amides that inhibit the binding of integrins to their receptors
02/27/2001US6194443 Aminophenol derivatives with fungicidal property
02/27/2001US6194396 Benzimidazole compounds as bradykinin antagonists
02/27/2001CA2316662A1 Use of crf antagonists and related compositions
02/22/2001WO2001012615A2 Fungicidal heteroaryl hepta-2,6-dienoic acid derivatives
02/22/2001WO2000071500A8 Halogen compounds
02/22/2001WO2000055126A3 N-cyanomethylamides as protease inhibitors
02/22/2001WO1999063996A8 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht2 receptors
02/22/2001DE19939645A1 New 1,3-bis(2,3-dihydroxybenzoylamino) substituted (hetero)aromatic siderophore compounds useful as bacterial growth factors and chemotherapeutic agents, e.g. for treatment of Alzheimer's disease
02/22/2001DE19939516A1 New 1-carboxyalkyl-4-(hetero)aryl-piperazine derivatives, as microsomal triglyceride transfer protein inhibitors useful for reducing plasma atherogenic lipoprotein levels, e.g. in treatment of hyperlipidemia
02/21/2001CN1284944A Integrin receptor antagonists
02/21/2001CN1062265C Method for producing triazine derivatives
02/20/2001US6191282 Derivatives of 5-membered nitrogen containing heterocyclic ring is used as anticarcinogenic agent and anticoagulant
02/20/2001US6191161 Prolylendopeptidase inhibitors
02/20/2001US6191154 Compositions and methods for the treatment of Alzheimer's disease, central nervous system injury, and inflammatory diseases
02/20/2001US6191153 Schizophrenia, parkinson's disease
02/20/2001US6191150 Formamide compounds as therapeutic agents
02/20/2001US6190923 Diethylenetriamine-N,N′,N″-triacetic acid derivatives
02/15/2001WO2001010854A1 Benzothiazole compounds and their use as optical brighteners
02/15/2001WO2001010853A1 Substituted 2-imino-thiazolines
02/15/2001WO2001010852A1 Process for the preparation of thiazole derivatives
02/15/2001WO2001010834A2 Antibacterial agents
02/15/2001WO2001010825A1 Carbamate derivatives and agricultural/horticultural bactericides
02/15/2001WO2001010798A1 Solid phase synthesis of oxa- and thiazoles
02/15/2001WO2001010383A2 Caspase inhibitors and uses thereof
02/15/2001WO2000054759A3 Lxr modulators
02/15/2001DE19937771A1 Substituierte 2-Imino-thiazoline Substituted 2-imino-thiazolines
02/15/2001CA2380838A1 Process for the preparation of thiazole derivatives
02/14/2001EP1076056A1 Novel spiro compounds or salts thereof and preventives/remedies for autoimmune diseases and ap-1 inhibitors containing the same
02/14/2001EP1076053A1 3-arylphenyl sulfide derivatives and insecticides and miticides
02/14/2001EP1075481A1 Monomeric, oligomeric and polymeric knoevenagel condensation products
02/14/2001CN1284071A Sulphona mide derivatives as prodrugs of aspartyl protease inhibitors
02/13/2001US6187944 A phenyl acrylonitrile compounds useful as active ingredients of an insecticide, a miticide, a nematicide, a soil pesticide, a fungicide and a marine antifouling agent
02/13/2001US6187933 Bind to retinoid receptors; treating skin disorders
02/13/2001US6187927 Process for preparing a 2-chloro-5-chloromethyl-thiazole compound
02/13/2001US6187812 For controlling animal pests or harmful fungi; (e,e,e)-2-methoxyimino-2-(2'-(1?-methyl, 1?-(1?'-ethoxyiminoethyl))iminooxymethyl)phenylacetic acid monomethylamide, for example
02/13/2001US6187802 Substituted 4-arylmethylene-2-imino-2,3-dihydrothiazoles and derivatives and their pharmaceutical use
02/13/2001US6187801 6-chloro-2-methyl-8h-indeno(1,2-d)-thiazole hydrochloride, for example; administering to treat obesity, diabetes; anorectics
02/13/2001US6187797 Phenyl-isoxazoles as factor XA Inhibitors
02/08/2001WO2001009108A1 Process for making n-alkyl bis(thiazolyl)sulfenimides
02/08/2001WO2001009088A1 Urea derivatives as inhibitors of ccr-3 receptor
02/08/2001WO2000044717A3 Synthesis of oligoketides
02/07/2001EP1073654A1 2,3-olefinic epothilone derivatives
02/07/2001EP1073648A1 12,13-Modified epothilone derivatives
02/07/2001EP1073647A1 12,13-cyclopropane epothilone derivatives
02/07/2001EP1073640A1 Naphthalene derivatives, their production and use
02/07/2001EP1073638A1 Heterocyclically substituted amides, their production and their use
02/07/2001EP1073633A2 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2