Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
08/2002
08/22/2002WO2002064546A2 Acylated 6,7,8,9-tetrahydro-5h-benzocycloheptenyl amines and their use as pharmaceutical
08/22/2002WO2002064545A1 Acylated indanyl amines and their use as pharmaceuticals
08/22/2002WO2002064137A1 Use of l-2-oxothiazolidine-4-carboxylic acid for the treatment of type 2 diabetes
08/22/2002US20020115866 Reacting 2-chloropyridine with 2-methylaminoethanol, coupling product obtained with 4-fluorobenzaldehyde in a solvent and alkali hydroxide or alkoxide, recovering product, converting into the thiazolidine-2,4-dione and reacting with maleic acid
08/22/2002US20020115853 6-(3-nitrophenyl)-3H-benzooxazol-2-one for example; contraceptives, treating hormone dependent tumors, endometriosis; progesterone receptor agonists and antagonists
08/22/2002US20020115826 Enzyme inhibitor for use for use in the treatment of cell proliferative defects
08/22/2002US20020115700 Inhibiting telomerase activity with 5-(3-Isatinylidinyl)thiazolidineones and 3-(thiazolidinon-5-yl) indoles
08/22/2002US20020115671 Inhibitors of p38-a kinase
08/22/2002DE10114425C1 Diaminobenzol-Derivate und diese Verbindungen enthaltende Haarfärbemittel Diaminobenzene derivatives and compositions containing these compounds hair dye
08/22/2002CA2438105A1 Method for preparing compounds derived from thiazolidinedione, oxazolidinedione
08/22/2002CA2426535A1 Heteroaryl alkyl piperazine derivatives as fatty acid oxidation inhibitors
08/21/2002EP1232149A2 Fungicidal melithiazole derivatives
08/21/2002EP1231939A2 Oncolytic combinations for the treatment of cancer
08/21/2002EP1231919A2 Novel class of cytodifferentiating agents and histone deacetylase inhibitors, and methods of use thereof
08/21/2002EP0802179B1 Substituted amidinonaphthyl ester derivatives
08/20/2002US6437177 α-hydroxy, -amino, and halo derivatives of β-sulfonyl hydroxamic acids as matrix metallopropteinases inhibitors
08/20/2002US6437143 Thiazolidone-2 derivatives, 4-diketone substituted, method for obtaining them and pharmaceutical compositions containing same
08/20/2002US6437142 10,10,10-trifluoro-5,5-dimethyl-9-triethylsilanyloxy-9-trifluo romethyl-dec-7-enal reacted with triethyl phosphonoacetate or ethyl (trimethylsilyl) acetate and then coupling with 2-mercapto-benzothiazole
08/20/2002US6436989 Prodrugs of aspartyl protease inhibitors
08/20/2002US6436978 For preventing or treating disorders modulated by alpha-2 adrenoceptors
08/20/2002US6436976 Mixtures including tebuconazole, having synergistic effects, used as pesticides, insecticides and fungicides
08/20/2002US6436489 Commercial optical display devices.
08/20/2002CA2180378C Forms a and b of n-[[[2-[[[2-[(diaminomethylene)amino]-4-thiazolyl]methyl]thio]ethyl]amino]methylene]-4-bromo-benzenesulfonamide
08/15/2002WO2002062791A1 Hetaryl substituted homotetramic and homotetronic acids and the use thereof as pesticides
08/15/2002WO2002062783A1 Dyes for keratin fibres containing 1,3-diamino-4-heteroarylbenzene derivatives and novel 1,3-diamino-4-heteroarylbenzene derivatives
08/15/2002WO2002062776A1 2-amino-4-(pyridin-2-yl)-thiazole derivatives as transforming growth factor beta (tgf-beta) inhibitors
08/15/2002WO2002062775A1 2-acylaminothiazole derivative or its salt
08/15/2002WO2002062774A1 Thiazole derivatives for treating ppar related disorders
08/15/2002WO2002062337A1 Thiazolidinediones
08/15/2002WO2002062301A2 Method and composition for rejuvinating cells, tissues, organs, hair and nails
08/15/2002WO2002028434A3 Use of a ppar delta activator for treating inflammatory conditions
08/15/2002WO2002028433A3 Use of a ppar delta activator in the treatment of diseases related to no inhibit ion or tnf inhibition
08/15/2002WO2001072685B1 Polyamine analogues as cytotoxic agents
08/15/2002US20020111493 Amidino compounds useful as nitric oxide synthase inhibitors
08/15/2002US20020111373 Thiadiazolidin-2,4-dione compound
08/15/2002US20020111372 Fused heteroaromatic glucokinase activators
08/15/2002US20020111368 Amino acid hydroxyethylamino sulfonamide retroviral protease inhibitors
08/15/2002US20020111347 Nervous system disorders
08/15/2002US20020111273 Insecticides, fungicides, miticides, plant safening agents
08/15/2002US20020110560 Lowering elevated post-prandial blood glucose levels in mammals by increasing incretin half-life comprising administering inhibitor of Dipeptidyl Peptidase (DP IV) or enzymes having DP-IV-like activity
08/15/2002CA2436433A1 Dyes for keratin fibres containing 1,3-diamino-4-heteroarylbenzene derivatives and novel 1,3-diamino-4-heteroarylbenzene derivatives
08/15/2002CA2435844A1 Method and composition for rejuvinating cells, tissues, organs, hair and nails
08/15/2002CA2432188A1 Thiazole derivatives for treating ppar related disorders
08/14/2002EP1230230A1 Indeno-, naphtho-, and benzocyclohepta-dihydrothiazole derivatives, the production thereof and their use as anorectic medicaments
08/14/2002EP1230229A1 Method for producing 2-chloro-5-chloromethyl-1,3-thiazol
08/14/2002EP1230227A1 Benzoxa-and benzothiazolyl sulfamates and their use as steroid sulfatase inhibitors
08/14/2002EP0799215B1 Process for preparing benzyl-substituted rhodanine derivatives
08/14/2002EP0790974B1 Substituted 4-biarylbutyric or 5-biarylpentanoic acids and derivatives as matrix metalloprotease inhibitiors
08/14/2002CN1364168A Hydrochloride of fused-heterocycle compound
08/14/2002CN1364164A Method for producing 4-ayano-2-aminomethylthiazol
08/14/2002CN1364163A Method for producing 2-aminomethyl-4-cyano-thiazol
08/14/2002CN1364155A N-Cyanomethyl amides as protease inhibitors
08/14/2002CN1364153A Substituted phenoxyacetic acids
08/13/2002US6433188 Fused heteroaromatic glucokinase activators
08/13/2002US6432999 Pyrazole substituted hydroxamic acid derivatives as cyclooxygenase-2 and 5-lipoxygenase inhibitors
08/13/2002US6432989 Use of CRF antagonists to treat circadian rhythm disorders
08/13/2002US6432962 Antiinflammatory agents
08/13/2002US6432958 2-piperazinoalkylaminobenzoazole derivatives: dopamine receptor subtype specific ligands
08/13/2002US6432949 Amide derivatives useful as inhibitors of the production of cytokines
08/13/2002US6432921 Oligopeptides
08/08/2002WO2002060898A1 Thiazolyl-, oxazolyl-, pyrrolyl-, and imidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes
08/08/2002WO2002060896A1 Ether derivatives useful as inhibitors of pde4 isozymes
08/08/2002WO2002060858A1 Novel compound having maillard reaction inhibitory activity
08/08/2002WO2002060443A1 Thiazolidinediones
08/08/2002WO2002060374A2 Benz-1,3-azole derivatives and their uses as heparanase inhibitors
08/08/2002WO2002002518A3 Compounds to treat alzheimer's disease
08/08/2002WO2001093840A3 Ligands of integrin receptors
08/08/2002US20020107406 Calcium receptor-active compounds
08/08/2002US20020107396 3-cycloalkyl- or propyl-2-(3,4-dihalophenyl)-N-quinolinyl-, quinazolinyl-, or quinoxolinyl-propionamide.
08/08/2002US20020107269 Inhibiting cell proliferation and treating cancer
08/08/2002US20020107258 Inhibition of human telomerase by a G-quadruplex-interaction compound
08/08/2002US20020106762 Generating preerential compound for use as prophylactic agent; obtain chemical intermediate, incubate with enzyme, recover prophylactic agent
08/08/2002CA2436551A1 Thiazolyl-, oxazolyl-, pyrrolyl-, and imidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes
08/08/2002CA2436544A1 Ether derivatives useful as inhibitors of pde4 isozymes
08/07/2002EP1229037A1 Heterocyclic N-acetonylbenzamides and their use as fungicides
08/07/2002EP1229028A1 Heterocyclic N-acetonylbenzamides and their use as fungicides
08/07/2002EP1229027A1 Heterocyclic N-acetonylbenzamides and their use as fungicides
08/07/2002EP1228760A2 5-membered heterocycle derivatives, production thereof and use thereof as medicaments
08/07/2002EP1228087A1 Antibody catalysis of enantio- and diastereo-selective aldol reactions
08/07/2002EP1228061A1 Dipeptidyl peptidase iv inhibitors and methods of making and using dipeptidyl peptidase iv inhibitors
08/07/2002EP1228053A1 Substituted piperazine derivatives, the production and use thereof as inhibitors of the microsomal triglyceride transfer protein (mtp)
08/07/2002EP1228051A1 Semicarbazone derivatives and their use as thrombopoietin mimetics
08/07/2002EP1227847A2 Inhibitors of the endothelin signalling pathway and alphavbeta3 integrin receptor antagonists for combination therapy
08/07/2002EP1058679A4 Synthesis of epothilones, intermediates thereto and analogues therof
08/07/2002EP0975638B1 Epothilones with a modified side chain
08/07/2002EP0770599B1 Process for the preparation of aromatic or heteroaromatic sulfonyl halides
08/07/2002CN1362952A 2-arylimino-2,3-dihydothiazoles, and their use thereof as somatostain receptor ligands
08/07/2002CN1362951A Dihetero-substituted metalloprotease inhibitors
08/07/2002CN1362947A N-cyanomethylamides as protease inhibitors
08/07/2002CN1362640A Silver-halides photo-sensitive emulsion layer with reinforced photographic photosensibility
08/07/2002CN1088709C Amine compound and its acid addition salt
08/07/2002CN1088702C Disubstituted bicyclic heterocycles, their production and use as medicaments
08/07/2002CN1088701C Method to convert 5-carboxanilid-haloalkylthiazoles to single form
08/06/2002US6429207 Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases
08/06/2002US6429206 Using agonist of nicotinergic acetylcholine receptors
08/01/2002WO2002059114A1 Lfa-1 antagonist compounds
08/01/2002WO2002059100A1 Halogen compounds having thrombopoietin receptor agonism
08/01/2002WO2002059099A1 Cyclic compounds having thrombopoietin receptor agonism
08/01/2002WO2002059098A1 Thiazole and oxazole derivatives as activators of human peroxisome proliferator activated receptors
08/01/2002WO2002059086A1 Carboxamides as fungicides in agriculture